Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 2

Results: 26

Design, Synthesis and Biological Evaluation of Noncovalent Inhibitors of Human CD38 NADase.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 223, doi. 10.1002/cmdc.201100487

By:

Zhou, Yi;
Ting, Kai Yiu;
Lam, Connie Mo Ching;
Kwong, Anna Ka Yee;
Xia, Jie;
Jin, Hongwei;
Liu, Zhenming;
Zhang, Liangren;
Cheung Lee, Hon;
Zhang, Lihe

Publication type:

Article

A Decade of the Human Genome Sequence-How Does the Medicinal Chemist Benefit?

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 194, doi. 10.1002/cmdc.201100498

By:

Brunschweiger, Andreas;
Hall, Jonathan

Publication type:

Article

Galloflavin (CAS 568-80-9): A Novel Inhibitor of Lactate Dehydrogenase.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 311, doi. 10.1002/cmdc.201100471

By:

Manerba, Marcella;
Vettraino, Marina;
Fiume, Luigi;
Di Stefano, Giuseppina;
Sartini, Andrea;
Giacomini, Elisa;
Buonfiglio, Rosa;
Roberti, Marinella;
Recanatini, Maurizio

Publication type:

Article

Application of Barluenga Boronic Coupling (BBC) to the Parallel Synthesis of Drug-like and Drug Fragment-like Molecules.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 233, doi. 10.1002/cmdc.201100339

By:

Nakagawa, Shoko;
Bainbridge, Katie A.;
Butcher, Ken;
Ellis, Dave;
Klute, Wolfgang;
Ryckmans, Thomas

Publication type:

Article

Back Cover: Discovery of Novel Stem Cell Mobilizers That Target the CXCR4 Receptor (ChemMedChem 2/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 336, doi. 10.1002/cmdc.201290005

By:

Wu, Chien-Huang;
Chang, Chun-Ping;
Song, Jen-Shin;
Jan, Jiing-Jyh;
Chou, Ming-Chen;
Wu, Szu-Huei;
Yeh, Kai-Chia;
Wong, Ying-Chieh;
Hsieh, Chieh-Jui;
Chen, Chiung-Tong;
Kao, Tzu-Ting;
Wu, Su-Ying;
Yeh, Ching-Fang;
Tseng, Chen-Tso;
Chao, Yu-Sheng;
Shia, Kak-Shan

Publication type:

Article

Discovery of Novel Stem Cell Mobilizers That Target the CXCR4 Receptor.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 209, doi. 10.1002/cmdc.201100525

By:

Wu, Chien-Huang;
Chang, Chun-Ping;
Song, Jen-Shin;
Jan, Jiing-Jyh;
Chou, Ming-Chen;
Wu, Szu-Huei;
Yeh, Kai-Chia;
Wong, Ying-Chieh;
Hsieh, Chieh-Jui;
Chen, Chiung-Tong;
Kao, Tzu-Ting;
Wu, Su-Ying;
Yeh, Ching-Fang;
Tseng, Chen-Tso;
Chao, Yu-Sheng;
Shia, Kak-Shan

Publication type:

Article

M. Alami.

Published in:: ChemMedChem, 2012, v. 7, n. 2, p. 193, doi. 10.1002/cmdc.201100495
Publication type:: Article

Graphical Abstract: ChemMedChem 2/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 2, p. 179, doi. 10.1002/cmdc.201290002
Publication type:: Article

A Synthetic C34 Trimer of HIV-1 gp41 Shows Significant Increase in Inhibition Potency.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 205, doi. 10.1002/cmdc.201100542

By:

Nomura, Wataru;
Hashimoto, Chie;
Ohya, Aki;
Miyauchi, Kosuke;
Urano, Emiko;
Tanaka, Tomohiro;
Narumi, Tetsuo;
Nakahara, Toru;
Komano, Jun A.;
Yamamoto, Naoki;
Tamamura, Hirokazu

Publication type:

Article

Experimental and Computational Active Site Mapping as a Starting Point to Fragment-Based Lead Discovery.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 248, doi. 10.1002/cmdc.201100490

By:

Behnen, Jürgen;
Köster, Helene;
Neudert, Gerd;
Craan, Tobias;
Heine, Andreas;
Klebe, Gerhard

Publication type:

Article

Study of the Anticancer Properties of Tin(IV) Carboxylate Complexes on a Panel of Human Tumor Cell Lines.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 301, doi. 10.1002/cmdc.201100432

By:

Rocamora-Reverte, Lourdes;
Carrasco-García, Estefanía;
Ceballos-Torres, Jesús;
Prashar, Sanjiv;
Kaluđerović, Goran N.;
Ferragut, José A.;
Gómez-Ruiz, Santiago

Publication type:

Article

Intermolecular and Intramolecular Hydrogen Bonds Involving Fluorine Atoms: Implications for Recognition, Selectivity, and Chemical Properties.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 262, doi. 10.1002/cmdc.201100483

By:

Dalvit, Claudio;
Vulpetti, Anna

Publication type:

Article

A Synthetic Lipid A Mimetic Modulates Human TLR4 Activity.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 213, doi. 10.1002/cmdc.201100494

By:

Piazza, Matteo;
Calabrese, Valentina;
Damore, Gaetana;
Cighetti, Roberto;
Gioannini, Theresa;
Weiss, Jerrold;
Peri, Francesco

Publication type:

Article

Inside Cover: RAFT-Derived Polymer-Drug Conjugates: Poly(hydroxypropyl methacrylamide) (HPMA)-7-Ethyl-10-hydroxycamptothecin (SN-38) Conjugates (ChemMedChem 2/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 178, doi. 10.1002/cmdc.201290001

By:

Williams, Charlotte C.;
Thang, San H.;
Hantke, Tina;
Vogel, Uwe;
Seeberger, Peter H.;
Tsanaktsidis, John;
Lepenies, Bernd

Publication type:

Article

Cover Picture: Engineering and Functionalization of the Disulfide-Constrained Miniprotein Min-23 as a Scaffold for Diagnostic Application (ChemMedChem 2/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 177, doi. 10.1002/cmdc.201290000

By:

Zoller, Frederic;
Schwaebel, Thimon;
Markert, Annette;
Haberkorn, Uwe;
Mier, Walter

Publication type:

Article

Preview: ChemMedChem 3/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 2, p. 335, doi. 10.1002/cmdc.201290004
Publication type:: Article

Discovery and Characterization of Atropisomer PH-797804, a p38 MAP Kinase Inhibitor, as a Clinical Drug Candidate.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 273, doi. 10.1002/cmdc.201100439

By:

Xing, Li;
Devadas, Balekudru;
Devraj, Rajesh V.;
Selness, Shaun R.;
Shieh, Huey;
Walker, John K.;
Mao, Michael;
Messing, Dean;
Samas, Brian;
Yang, Jerry Z.;
Anderson, Gary D.;
Webb, Elizabeth G.;
Monahan, Joseph B.

Publication type:

Article

3-Substituted 2-Phenylimidazo[2,1- b]benzothiazoles: Synthesis, Anticancer Activity, and Inhibition of Tubulin Polymerization.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 292, doi. 10.1002/cmdc.201100511

By:

Kamal, Ahmed;
Sultana, Farheen;
Ramaiah, M. Janaki;
Srikanth, Y. V. V.;
Viswanath, A.;
Kishor, Chandan;
Sharma, Pranjal;
Pushpavalli, S. N. C. V. L.;
Addlagatta, Anthony;
Pal-Bhadra, Manika

Publication type:

Article

Elucidation of the Structure-Activity Relationships of Apelin: Influence of Unnatural Amino Acids on Binding, Signaling, and Plasma Stability.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 318, doi. 10.1002/cmdc.201100492

By:

Murza, Alexandre;
Parent, Alexandre;
Besserer-Offroy, Elie;
Tremblay, Hugo;
Karadereye, Félix;
Beaudet, Nicolas;
Leduc, Richard;
Sarret, Philippe;
Marsault, Éric

Publication type:

Article

Engineering and Functionalization of the Disulfide-Constrained Miniprotein Min-23 as a Scaffold for Diagnostic Application.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 237, doi. 10.1002/cmdc.201100497

By:

Zoller, Frederic;
Schwaebel, Thimon;
Markert, Annette;
Haberkorn, Uwe;
Mier, Walter

Publication type:

Article

Antiviral Drug Strategies. Edited by Erik De Clercq.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 334, doi. 10.1002/cmdc.201100548

By:

Gosselin, Gilles

Publication type:

Article

RAFT-Derived Polymer-Drug Conjugates: Poly(hydroxypropyl methacrylamide) (HPMA)-7-Ethyl-10-hydroxycamptothecin (SN-38) Conjugates.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 281, doi. 10.1002/cmdc.201100456

By:

Williams, Charlotte C.;
Thang, San H.;
Hantke, Tina;
Vogel, Uwe;
Seeberger, Peter H.;
Tsanaktsidis, John;
Lepenies, Bernd

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 2/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 2, p. 190, doi. 10.1002/cmdc.201290003
Publication type:: Article

Remarkable Stability and Cytostatic Effect of a Quercetin Conjugate, 3,7-Bis- O-Pivaloxymethyl (POM) Quercetin.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 229, doi. 10.1002/cmdc.201100478

By:

Kim, Mi Kyoung;
Park, Kwang-Su;
Chong, Youhoon

Publication type:

Article

Immunosuppressive Effects of Subglutinol Derivatives.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 218, doi. 10.1002/cmdc.201100409

By:

Lee, Won-Gil;
Kim, Woo-Seok;
Park, Sung-Gyoo;
Kim, Hyoungsu;
Hong, Jiyong;
Ko, Hyojin;
Kim, Yong-Chul

Publication type:

Article

Synthesis and Functional Characterization of Tridegin and Its Analogues: Inhibitors and Substrates of Factor XIIIa.

Published in:

ChemMedChem, 2012, v. 7, n. 2, p. 326, doi. 10.1002/cmdc.201100405

By:

Böhm, Miriam;
Kühl, Toni;
Hardes, Kornelia;
Coch, Richard;
Arkona, Christoph;
Schlott, Bernhard;
Steinmetzer, Torsten;
Imhof, Diana

Publication type:

Article