Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 12


Results: 24
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    Lead Optimization of Thiazolo[5,4- c]piperidines: 3-Cyclobutoxy Linker as a Key Spacer for H<sub>3</sub>R Inverse Agonists.

    Published in:
    ChemMedChem, 2012, v. 7, n. 12, p. 2087, doi. 10.1002/cmdc.201200406
    By:
    • Provins, Laurent;
    • Denonne, Frédéric;
    • Célanire, Sylvain;
    • Christophe, Bernard;
    • Defays, Sabine;
    • Delaunoy, Christel;
    • Delporte, Marie-Laure;
    • Demaude, Thierry;
    • Durieu, Véronique;
    • Gillard, Michel;
    • Hubert, Delphine;
    • Lamberty, Yves;
    • Lorent, Geneviève;
    • Valade, Anne;
    • Vanbellinghen, Alain;
    • Van houtvin, Nathalie
    Publication type:
    Article
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    Camptothecin-7-yl-methanthiole: Semisynthesis and Biological Evaluation.

    Published in:
    ChemMedChem, 2012, v. 7, n. 12, p. 2134, doi. 10.1002/cmdc.201200322
    By:
    • Christodoulou, Michael S.;
    • Zunino, Franco;
    • Zuco, Valentina;
    • Borrelli, Stella;
    • Comi, Daniela;
    • Fontana, Gabriele;
    • Martinelli, Marisa;
    • Lorens, James B.;
    • Evensen, Lasse;
    • Sironi, Maurizio;
    • Pieraccini, Stefano;
    • Dalla Via, Lisa;
    • Gia, Ornella Maria;
    • Passarella, Daniele
    Publication type:
    Article
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    Aromatic Core Extension in the Series of N-Cyclic Bay-Substituted Perylene G-Quadruplex Ligands: Increased Telomere Damage, Antitumor Activity, and Strong Selectivity for Neoplastic over Healthy Cells.

    Published in:
    ChemMedChem, 2012, v. 7, n. 12, p. 2144, doi. 10.1002/cmdc.201200348
    By:
    • Franceschin, Marco;
    • Rizzo, Angela;
    • Casagrande, Valentina;
    • Salvati, Erica;
    • Alvino, Antonello;
    • Altieri, Alessandro;
    • Ciammaichella, Alina;
    • Iachettini, Sara;
    • Leonetti, Carlo;
    • Ortaggi, Giancarlo;
    • Porru, Manuela;
    • Bianco, Armandodoriano;
    • Biroccio, Annamaria
    Publication type:
    Article
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