Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 11

Results: 29

Corrigendum: Advances in Targeting Voltage-Gated Sodium Channels with Small Molecules.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1874, doi. 10.1002/cmdc.201200443

By:

Nardi, Antonio;
Damann, Nils;
Hertrampf, Torsten;
Kless, Achim

Publication type:

Article

Beyond Heparinization: Design of Highly Potent Thrombin Inhibitors Suitable for Surface Coupling.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1965, doi. 10.1002/cmdc.201200292

By:

Steinmetzer, Torsten;
Baum, Bernhard;
Biela, Adam;
Klebe, Gerhard;
Nowak, Götz;
Bucha, Elke

Publication type:

Article

Partial Inhibition of Aldose Reductase by Nitazoxanide and Its Molecular Basis.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1921, doi. 10.1002/cmdc.201200333

By:

Zheng, Xuehua;
Zhang, Liping;
Chen, Weijia;
Chen, Yunyun;
Xie, Wei;
Hu, Xiaopeng

Publication type:

Article

Graphical Abstract: ChemMedChem 11/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 11, p. 1867, doi. 10.1002/cmdc.201290055
Publication type:: Article

Characterization of Telmisartan-Derived PPARγ Agonists: Importance of Moiety Shift from Position 6 to 5 on Potency, Efficacy and Cofactor Recruitment.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1935, doi. 10.1002/cmdc.201200337

By:

Herbst, Lena;
Goebel, Matthias;
Bandholtz, Sebastian;
Gust, Ronald;
Kintscher, Ulrich

Publication type:

Article

Synthesis and Antiproliferative Activity of the Ring System [1,2]Oxazolo[4,5- g]indole.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1901, doi. 10.1002/cmdc.201200296

By:

Barraja, Paola;
Caracausi, Libero;
Diana, Patrizia;
Spanò, Virginia;
Montalbano, Alessandra;
Carbone, Anna;
Parrino, Barbara;
Cirrincione, Girolamo

Publication type:

Article

Proteinases as Drug Targets. Edited by Ben M. Dunn.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 2040, doi. 10.1002/cmdc.201200179

By:

Sedrani, Richard

Publication type:

Article

Corrigendum: An Efficient Synthesis of a Hydroxyethylamine (HEA) Isostere and Its α-Aminophosphonate and Phosphoramidate Derivatives as Potential Anti-HIV Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1874, doi. 10.1002/cmdc.201200442

By:

Bhattacharya, Asish K.;
Rana, Kalpeshkumar C.;
Pannecouque, Christophe;
De Clercq, Eric

Publication type:

Article

Structural Studies on 4,5-Disubstituted 2-Aminoimidazole-Based Biofilm Modulators that Suppress Bacterial Resistance to β-Lactams.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 2030, doi. 10.1002/cmdc.201200350

By:

Su, Zhaoming;
Yeagley, Andrew A.;
Su, Rui;
Peng, Lingling;
Melander, Christian

Publication type:

Article

Back Cover: Discovery of a New Class of Liver Receptor Homolog-1 (LRH-1) Antagonists: Virtual Screening, Synthesis and Biological Evaluation (ChemMedChem 11/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 2044, doi. 10.1002/cmdc.201290058

By:

Rey, Jullien;
Hu, Haipeng;
Kyle, Fiona;
Lai, Chun-Fui;
Buluwela, Laki;
Coombes, R. Charles;
Ortlund, Eric A.;
Ali, Simak;
Snyder, James P.;
Barrett, Anthony G. M.

Publication type:

Article

( R)-α-Lipoyl-Glycyl- L-Prolyl- L-Glutamyl Dimethyl Ester Codrug as a Multifunctional Agent with Potential Neuroprotective Activities.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 2021, doi. 10.1002/cmdc.201200320

By:

Cacciatore, Ivana;
Baldassarre, Leonardo;
Fornasari, Erika;
Cornacchia, Catia;
Di Stefano, Antonio;
Sozio, Piera;
Cerasa, Laura Serafina;
Fontana, Antonella;
Fulle, Stefania;
Di Filippo, Ester Sara;
La Rovere, Rita Maria Laura;
Pinnen, Francesco

Publication type:

Article

Synthesis, Cytotoxicity, Induction of Apoptosis, and Interaction with DNA of Dinuclear Platinum(II) Complexes.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 2004, doi. 10.1002/cmdc.201200332

By:

Xu, Gang;
Gao, Chuanzhu;
Gou, Shaohua;
Cao, Zhe

Publication type:

Article

Inhibition of Bacterial Dihydrofolate Reductase by 6-Alkyl-2,4-diaminopyrimidines.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1974, doi. 10.1002/cmdc.201200291

By:

Nammalwar, Baskar;
Bourne, Christina R.;
Bunce, Richard A.;
Wakeham, Nancy;
Bourne, Philip C.;
Ramnarayan, Kal;
Mylvaganam, Shankari;
Berlin, K. Darrell;
Barrow, Esther W.;
Barrow, William W.

Publication type:

Article

Discovery of a New Class of Liver Receptor Homolog-1 (LRH-1) Antagonists: Virtual Screening, Synthesis and Biological Evaluation.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1909, doi. 10.1002/cmdc.201200307

By:

Rey, Jullien;
Hu, Haipeng;
Kyle, Fiona;
Lai, Chun-Fui;
Buluwela, Laki;
Coombes, R. Charles;
Ortlund, Eric A.;
Ali, Simak;
Snyder, James P.;
Barrett, Anthony G. M.

Publication type:

Article

Carprofen Analogues as Sirtuin Inhibitors: Enzyme and Cellular Studies.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1905, doi. 10.1002/cmdc.201200318

By:

Mellini, Paolo;
Carafa, Vincenzo;
Di Rienzo, Barbara;
Rotili, Dante;
De Vita, Daniela;
Cirilli, Roberto;
Gallinella, Bruno;
Provvisiero, Donatella Paola;
Di Maro, Salvatore;
Novellino, Ettore;
Altucci, Lucia;
Mai, Antonello

Publication type:

Article

MT<sub>1</sub>-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-{[(3- O-Substituted)anilino]alkyl}amides.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1954, doi. 10.1002/cmdc.201200303

By:

Rivara, Silvia;
Pala, Daniele;
Lodola, Alessio;
Mor, Marco;
Lucini, Valeria;
Dugnani, Silvana;
Scaglione, Francesco;
Bedini, Annalida;
Lucarini, Simone;
Tarzia, Giorgio;
Spadoni, Gilberto

Publication type:

Article

Inside Cover: Inhibition of Bacterial Dihydrofolate Reductase by 6-Alkyl-2,4-diaminopyrimidines (ChemMedChem 11/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1866, doi. 10.1002/cmdc.201290054

By:

Nammalwar, Baskar;
Bourne, Christina R.;
Bunce, Richard A.;
Wakeham, Nancy;
Bourne, Philip C.;
Ramnarayan, Kal;
Mylvaganam, Shankari;
Berlin, K. Darrell;
Barrow, Esther W.;
Barrow, William W.

Publication type:

Article

Discovery of Tyrosine Kinase Inhibitors by Docking into an Inactive Kinase Conformation Generated by Molecular Dynamics.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1983, doi. 10.1002/cmdc.201200331

By:

Zhao, Hongtao;
Huang, Danzhi;
Caflisch, Amedeo

Publication type:

Article

Cover Picture: Identification of Drugs Inducing Phospholipidosis by Novel in vitro Data (ChemMedChem 11/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1865, doi. 10.1002/cmdc.201290053

By:

Muehlbacher, Markus;
Tripal, Philipp;
Roas, Florian;
Kornhuber, Johannes

Publication type:

Article

Identification of Drugs Inducing Phospholipidosis by Novel in vitro Data.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1925, doi. 10.1002/cmdc.201200306

By:

Muehlbacher, Markus;
Tripal, Philipp;
Roas, Florian;
Kornhuber, Johannes

Publication type:

Article

Synthesis and Structure-Activity Relationships of Lansine Analogues as Antileishmanial Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1895, doi. 10.1002/cmdc.201200346

By:

Pieroni, Marco;
Girmay, Sisay;
Sun, Dianqing;
Sahu, Rajnish;
Tekwani, Babu L.;
Tan, Ghee T.

Publication type:

Article

Preview: ChemMedChem 12/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 11, p. 2043, doi. 10.1002/cmdc.201290057
Publication type:: Article

A Case Study of Single-Pill Combination Therapy: The Ezetimibe/Simvastatin Combination for Treatment of Hyperlipidemia.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1882, doi. 10.1002/cmdc.201200287

By:

Huang, Xianhai;
Chen, David Y.-K.

Publication type:

Article

Arene-Ru<sup>II</sup> Complexes of Curcumin Exert Antitumor Activity via Proteasome Inhibition and Apoptosis Induction.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 2010, doi. 10.1002/cmdc.201200341

By:

Bonfili, Laura;
Pettinari, Riccardo;
Cuccioloni, Massimiliano;
Cecarini, Valentina;
Mozzicafreddo, Matteo;
Angeletti, Mauro;
Lupidi, Giulio;
Marchetti, Fabio;
Pettinari, Claudio;
Eleuteri, Anna Maria

Publication type:

Article

A Facile Synthesis of Novel Bis-(indolyl)-1,3,4-oxadiazoles as Potent Cytotoxic Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1915, doi. 10.1002/cmdc.201200363

By:

Kumar, Dalip;
Arun, V.;
Maruthi Kumar, N.;
Acosta, Glen;
Noel, Brett;
Shah, Kavita

Publication type:

Article

HPLC Methods for Clinical Pharmaceutical Analysis: A User's Guide. By Herrmann Mascher.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 2040, doi. 10.1002/cmdc.201200374

By:

Jira, Thomas

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 11/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 11, p. 1878, doi. 10.1002/cmdc.201290056
Publication type:: Article

Fluorine-18 Radiolabeling and Radiopharmacological Characterization of a Benzodioxolylpyrimidine-based Radiotracer Targeting the Receptor Tyrosine Kinase EphB4.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1991, doi. 10.1002/cmdc.201200264

By:

Mamat, Constantin;
Mosch, Birgit;
Neuber, Christin;
Köckerling, Martin;
Bergmann, Ralf;
Pietzsch, Jens

Publication type:

Article

Systematic Structure-Activity Study on Potential Chaperone Lead Compounds for Acid α-Glucosidase.

Published in:

ChemMedChem, 2012, v. 7, n. 11, p. 1943, doi. 10.1002/cmdc.201200309

By:

Bruckmann, Chiara;
Repo, Heidi;
Kuokkanen, Elina;
Xhaard, Henri;
Heikinheimo, Pirkko

Publication type:

Article