Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 10

Results: 25

Polyamine Drug Discovery. Edited by Patrick Woster and Robert A. Casero, Jr.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1859, doi. 10.1002/cmdc.201200294

By:

Tripier, Raphaël

Publication type:

Article

Ion Channel Phosphorylopathy: a Link between Genomic Variation and Human Disease.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1757, doi. 10.1002/cmdc.201200236

By:

Gentile, Saverio

Publication type:

Article

Advances in Targeting Voltage-Gated Sodium Channels with Small Molecules.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1712, doi. 10.1002/cmdc.201200298

By:

Nardi, Antonio;
Damann, Nils;
Hertrampf, Torsten;
Kless, Achim

Publication type:

Article

Back Cover: Selective Modification of the N-Terminal Structure of Polytheonamide B Significantly Changes its Cytotoxicity and Activity as an Ion Channel (ChemMedChem 10/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1864, doi. 10.1002/cmdc.201290052

By:

Shinohara, Naoki;
Itoh, Hiroaki;
Matsuoka, Shigeru;
Inoue, Masayuki

Publication type:

Article

Design and Synthesis of 3-Carbamoylbenzoic Acid Derivatives as Inhibitors of Human Apurinic/Apyrimidinic Endonuclease 1 (APE1).

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1825, doi. 10.1002/cmdc.201200334

By:

Aiello, Francesca;
Shabaik, Yumna;
Esqueda, Adrian;
Sanchez, Tino W.;
Grande, Fedora;
Garofalo, Antonio;
Neamati, Nouri

Publication type:

Article

Kinase Drug Discovery. Edited by Richard A. Ward and Frederick W. Goldberg.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1858, doi. 10.1002/cmdc.201200231

By:

Engh, Richard

Publication type:

Article

Graphical Abstract: ChemMedChem 10/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 10, p. 1699, doi. 10.1002/cmdc.201290049
Publication type:: Article

2-Aminopyridine Derivatives as Potential σ2 Receptor Antagonists.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1847, doi. 10.1002/cmdc.201200246

By:

Abate, Carmen;
Ferorelli, Savina;
Niso, Mauro;
Lovicario, Cesarea;
Infantino, Vittoria;
Convertini, Paolo;
Perrone, Roberto;
Berardi, Francesco

Publication type:

Article

Identification of Selective Inhibitors of the Potassium Channel Kv1.1-1.2(3) by High-Throughput Virtual Screening and Automated Patch Clamp.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1775, doi. 10.1002/cmdc.201100600

By:

Wacker, Sören J.;
Jurkowski, Wiktor;
Simmons, Katie J.;
Fishwick, Colin W. G.;
Johnson, A. Peter;
Madge, David;
Lindahl, Erik;
Rolland, Jean-Francois;
de Groot, Bert L.

Publication type:

Article

Synthesis and Biological Evaluation of ortho-Aryl N-Hydroxycinnamides as Potent Histone Deacetylase (HDAC) 8 Isoform-Selective Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1815, doi. 10.1002/cmdc.201200300

By:

Huang, Wei-Jan;
Wang, Yi-Ching;
Chao, Shi-Wei;
Yang, Chen-Yui;
Chen, Liang-Chieh;
Lin, Mei-Hsiang;
Hou, Wen-Chi;
Chen, Mei-Yu;
Lee, Tai-Lin;
Yang, Ping;
Chang, Chung-I

Publication type:

Article

Asymmetric 4-Aryl-1,4-dihydropyridines Potentiate Mutant Cystic Fibrosis Transmembrane Conductance Regulator (CFTR).

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1799, doi. 10.1002/cmdc.201200311

By:

Giampieri, Michele;
Vanthuyne, Nicolas;
Nieddu, Erika;
Mazzei, Marco T.;
Anzaldi, Maria;
Pedemonte, Nicoletta;
Galietta, Luis J. V.;
Roussel, Christian;
Mazzei, Mauro

Publication type:

Article

Neglected Diseases and Drug Discovery. Edited by Michael J. Palmer and Timothy N. C. Wells.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1859, doi. 10.1002/cmdc.201200232

By:

Gilbert, Ian

Publication type:

Article

Preview: ChemMedChem 11/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 10, p. 1863, doi. 10.1002/cmdc.201290051
Publication type:: Article

Selective Modification of the N-Terminal Structure of Polytheonamide B Significantly Changes its Cytotoxicity and Activity as an Ion Channel.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1770, doi. 10.1002/cmdc.201200142

By:

Shinohara, Naoki;
Itoh, Hiroaki;
Matsuoka, Shigeru;
Inoue, Masayuki

Publication type:

Article

Synthesis and Cytotoxicity of Three trans-Palladium Complexes Containing Planaramine Ligands in Human Ovarian Tumor Models.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1840, doi. 10.1002/cmdc.201200310

By:

Mazumder, Mohammed Ehsanul Hoque;
Beale, Philip;
Chan, Charles;
Yu, Jun Qing;
Huq, Fazlul

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 10/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 10, p. 1708, doi. 10.1002/cmdc.201290050
Publication type:: Article

Structure-Activity Relationships of a Novel Group of Large-Conductance Ca2+-Activated K+ (BK) Channel Modulators: The GoSlo-SR Family.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1763, doi. 10.1002/cmdc.201200321

By:

Roy, Subhrangsu;
Morayo Akande, Adebola;
Large, Roddy J.;
Webb, Tim I.;
Camarasu, Costin;
Sergeant, Gerard P.;
McHale, Noel G.;
Thornbury, Keith D.;
Hollywood, Mark A.

Publication type:

Article

Inside Cover: Structure-Activity Relationships of a Novel Group of Large-Conductance Ca2+-Activated K+ (BK) Channel Modulators: The GoSlo-SR Family (ChemMedChem 10/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1694, doi. 10.1002/cmdc.201290048

By:

Roy, Subhrangsu;
Morayo Akande, Adebola;
Large, Roddy J.;
Webb, Tim I.;
Camarasu, Costin;
Sergeant, Gerard P.;
McHale, Noel G.;
Thornbury, Keith D.;
Hollywood, Mark A.

Publication type:

Article

Structural and Pharmacological Characterization of Phenylalanine-Based AMPA Receptor Antagonists at Kainate Receptors.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1793, doi. 10.1002/cmdc.201100599

By:

Venskutonytė, Raminta;
Frydenvang, Karla;
Valadés, Elena Antón;
Szymańska, Ewa;
Johansen, Tommy N.;
Kastrup, Jette S.;
Pickering, Darryl S.

Publication type:

Article

Trafficking of Intermediate (KCa3.1) and Small (KCa2.x) Conductance, Ca2+-Activated K+ Channels: a Novel Target for Medicinal Chemistry Efforts?

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1741, doi. 10.1002/cmdc.201200226

By:

Balut, Corina M.;
Hamilton, Kirk L.;
Devor, Daniel C.

Publication type:

Article

Editorial: Channeling Drug Discovery.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1695, doi. 10.1002/cmdc.201200416

By:

Steinhagen, Henning;
Damann, Nils

Publication type:

Article

Calcium- and Voltage-Gated Potassium (BK) Channel Activators in the 5β-Cholanic Acid-3α-ol Analogue Series with Modifications in the Lateral Chain.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1784, doi. 10.1002/cmdc.201200290

By:

Bukiya, Anna N.;
Patil, Shivaputra A.;
Li, Wei;
Miller, Duane D.;
Dopico, Alex M.

Publication type:

Article

Gram-Scale Solution-Phase Synthesis of Selective Sodium Bicarbonate Co-transport Inhibitor S0859: in vitro Efficacy Studies in Breast Cancer Cells.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1808, doi. 10.1002/cmdc.201200335

By:

Larsen, Ann M.;
Krogsgaard-Larsen, Niels;
Lauritzen, Gitte;
Olesen, Christina W.;
Honoré Hansen, Steen;
Boedtkjer, Ebbe;
Pedersen, Stine F.;
Bunch, Lennart

Publication type:

Article

Cover Picture: Identification of Selective Inhibitors of the Potassium Channel Kv1.1-1.2(3) by High-Throughput Virtual Screening and Automated Patch Clamp (ChemMedChem 10/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1693, doi. 10.1002/cmdc.201290047

By:

Wacker, Sören J.;
Jurkowski, Wiktor;
Simmons, Katie J.;
Fishwick, Colin W. G.;
Johnson, A. Peter;
Madge, David;
Lindahl, Erik;
Rolland, Jean-Francois;
de Groot, Bert L.

Publication type:

Article

Drug Delivery in Oncology. Edited by Felix Kratz, Peter Senter and Henning Steinhagen.

Published in:

ChemMedChem, 2012, v. 7, n. 10, p. 1860, doi. 10.1002/cmdc.201200357

By:

Olmo López, Rosa María

Publication type:

Article

Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 10

Polyamine Drug Discovery. Edited by Patrick Woster and Robert A. Casero, Jr.

Ion Channel Phosphorylopathy: a Link between Genomic Variation and Human Disease.

Advances in Targeting Voltage-Gated Sodium Channels with Small Molecules.

Back Cover: Selective Modification of the N-Terminal Structure of Polytheonamide B Significantly Changes its Cytotoxicity and Activity as an Ion Channel (ChemMedChem 10/2012).

Design and Synthesis of 3-Carbamoylbenzoic Acid Derivatives as Inhibitors of Human Apurinic/Apyrimidinic Endonuclease 1 (APE1).

Kinase Drug Discovery. Edited by Richard A. Ward and Frederick W. Goldberg.

Graphical Abstract: ChemMedChem 10/2012.

2-Aminopyridine Derivatives as Potential σ<sub>2</sub> Receptor Antagonists.

Identification of Selective Inhibitors of the Potassium Channel Kv1.1-1.2<sub>(3)</sub> by High-Throughput Virtual Screening and Automated Patch Clamp.

Synthesis and Biological Evaluation of ortho-Aryl N-Hydroxycinnamides as Potent Histone Deacetylase (HDAC) 8 Isoform-Selective Inhibitors.

Asymmetric 4-Aryl-1,4-dihydropyridines Potentiate Mutant Cystic Fibrosis Transmembrane Conductance Regulator (CFTR).

Neglected Diseases and Drug Discovery. Edited by Michael J. Palmer and Timothy N. C. Wells.

Preview: ChemMedChem 11/2012.

Selective Modification of the N-Terminal Structure of Polytheonamide B Significantly Changes its Cytotoxicity and Activity as an Ion Channel.

Synthesis and Cytotoxicity of Three trans-Palladium Complexes Containing Planaramine Ligands in Human Ovarian Tumor Models.

Spotlights on our sister journals: ChemMedChem 10/2012.

Structure-Activity Relationships of a Novel Group of Large-Conductance Ca<sup>2+</sup>-Activated K<sup>+</sup> (BK) Channel Modulators: The GoSlo-SR Family.

Inside Cover: Structure-Activity Relationships of a Novel Group of Large-Conductance Ca<sup>2+</sup>-Activated K<sup>+</sup> (BK) Channel Modulators: The GoSlo-SR Family (ChemMedChem 10/2012).

Structural and Pharmacological Characterization of Phenylalanine-Based AMPA Receptor Antagonists at Kainate Receptors.

Trafficking of Intermediate (KCa3.1) and Small (KCa2.x) Conductance, Ca<sup>2+</sup>-Activated K<sup>+</sup> Channels: a Novel Target for Medicinal Chemistry Efforts?

Editorial: Channeling Drug Discovery.

Calcium- and Voltage-Gated Potassium (BK) Channel Activators in the 5β-Cholanic Acid-3α-ol Analogue Series with Modifications in the Lateral Chain.

Gram-Scale Solution-Phase Synthesis of Selective Sodium Bicarbonate Co-transport Inhibitor S0859: in vitro Efficacy Studies in Breast Cancer Cells.

Cover Picture: Identification of Selective Inhibitors of the Potassium Channel Kv1.1-1.2<sub>(3)</sub> by High-Throughput Virtual Screening and Automated Patch Clamp (ChemMedChem 10/2012).

Drug Delivery in Oncology. Edited by Felix Kratz, Peter Senter and Henning Steinhagen.