Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 1

Results: 29

In vivo Enhancement in Bioavailability of Atazanavir in the Presence of Proton-Pump Inhibitors using Mesoporous Materials.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 43, doi. 10.1002/cmdc.201100500

By:

Xia, Xin;
Zhou, Chunfang;
Ballell, Lluís;
Garcia-Bennett, Alfonso E.

Publication type:

Article

Specific Targeting of Hypoxic Tumor Tissue with Nitroimidazole-Peptide Conjugates.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 57, doi. 10.1002/cmdc.201100401

By:

Splith, Katrin;
Bergmann, Ralf;
Pietzsch, Jens;
Neundorf, Ines

Publication type:

Article

Identification of 1,3-Diiminoisoindoline Carbohydrazides as Potential Antimalarial Candidates.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 151, doi. 10.1002/cmdc.201100441

By:

Mombelli, Paolo;
Witschel, Matthias C.;
van Zijl, Anthoni W.;
Geist, Julie G.;
Rottmann, Matthias;
Freymond, Céline;
Röhl, Franz;
Kaiser, Marcel;
Illarionova, Victoria;
Fischer, Markus;
Siepe, Isabella;
Schweizer, W. Bernd;
Brun, Reto;
Diederich, François

Publication type:

Article

Concise Notice to Authors: ChemMedChem 1/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 1, p. 19, doi. 10.1002/cmdc.201190060
Publication type:: Article

Rofecoxib Analogues Possessing a Nitric Oxide Donor Sulfohydroxamic Acid (SO2NHOH) Cyclooxygenase-2 Pharmacophore: Synthesis, Molecular Modeling, and Biological Evaluation as Anti-inflammatory Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 62, doi. 10.1002/cmdc.201100393

By:

Bhardwaj, Atul;
Huang, Zhangjian;
Kaur, Jatinder;
Knaus, Edward E.

Publication type:

Article

Cover Picture: Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E-4031 Analogues (ChemMedChem 1/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 1, doi. 10.1002/cmdc.201190057

By:

Vilums, Maris;
Overman, Jeroen;
Klaasse, Elisabeth;
Scheel, Olaf;
Brussee, Johannes;
IJzerman, Adriaan P.

Publication type:

Article

Editorial: Quality Research. Outstanding Publications.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 3, doi. 10.1002/cmdc.201100462

By:

Ortúzar, Natalia;
Williams, Scott D.

Publication type:

Article

Quaternary Ammonium Salts and Their Antimicrobial Potential: Targets or Nonspecific Interactions?

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 22, doi. 10.1002/cmdc.201100404

By:

Tischer, Maximilian;
Pradel, Gabriele;
Ohlsen, Knut;
Holzgrabe, Ulrike

Publication type:

Article

Back Cover: Identification and Characterization of Inhibitors of the Aminoglycoside Resistance Acetyltransferase Eis from Mycobacterium tuberculosis (ChemMedChem 1/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 176, doi. 10.1002/cmdc.201190063

By:

Green, Keith D.;
Chen, Wenjing;
Garneau-Tsodikova, Sylvie

Publication type:

Article

Development of Improved PPAR β/ δ Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 159, doi. 10.1002/cmdc.201100408

By:

Toth, Philipp M.;
Naruhn, Simone;
Pape, Veronika F. S.;
Dörr, Stefanie M. A.;
Klebe, Gerhard;
Müller, Rolf;
Diederich, Wibke E.

Publication type:

Article

Nocodazole is a High-Affinity Ligand for the Cancer-Related Kinases ABL, c-KIT, BRAF, and MEK.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 53, doi. 10.1002/cmdc.201100410

By:

Park, Hwangseo;
Hong, Seunghee;
Hong, Sungwoo

Publication type:

Article

Antiviral Drugs: From Basic Discovery Through Clinical Trials. Edited by Wieslaw M. Kazmierski.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 172, doi. 10.1002/cmdc.201100421

By:

Rowley, Michael

Publication type:

Article

Discovery of a Pharmacologically Active Antagonist of the Two-Pore-Domain Potassium Channel K2P9.1 (TASK-3).

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 123, doi. 10.1002/cmdc.201100351

By:

Coburn, Craig A.;
Luo, Yunfu;
Cui, Mingxiang;
Wang, Jiabing;
Soll, Richard;
Dong, Jingchao;
Hu, Bin;
Lyon, Michael A.;
Santarelli, Vincent P.;
Kraus, Richard L.;
Gregan, Yun;
Wang, Yi;
Fox, Steven V.;
Binns, Jacquelyn;
Doran, Scott M.;
Reiss, Duane R.;
Tannenbaum, Pamela L.;
Gotter, Anthony L.;
Meinke, Peter T.;
Renger, John J.

Publication type:

Article

Graphical Abstract: ChemMedChem 1/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 1, p. 7, doi. 10.1002/cmdc.201190062
Publication type:: Article

From a Library of MAG Antagonists to Nanomolar CD22 Ligands.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 134, doi. 10.1002/cmdc.201100407

By:

Mesch, Stefanie;
Lemme, Katrin;
Wittwer, Matthias;
Koliwer-Brandl, Hendrik;
Schwardt, Oliver;
Kelm, Sørge;
Ernst, Beat

Publication type:

Article

Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E-4031 Analogues.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 107, doi. 10.1002/cmdc.201100366

By:

Vilums, Maris;
Overman, Jeroen;
Klaasse, Elisabeth;
Scheel, Olaf;
Brussee, Johannes;
IJzerman, Adriaan P.

Publication type:

Article

Preview: ChemMedChem 2/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 1, p. 175, doi. 10.1002/cmdc.201190059
Publication type:: Article

Design, Synthesis and Biological Evaluation of Trypanosoma brucei Trypanothione Synthetase Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 95, doi. 10.1002/cmdc.201100420

By:

Spinks, Daniel;
Torrie, Leah S.;
Thompson, Stephen;
Harrison, Justin R.;
Frearson, Julie A.;
Read, Kevin D.;
Fairlamb, Alan H.;
Wyatt, Paul G.;
Gilbert, Ian H.

Publication type:

Article

Aspirin Analogues as Dual Cyclooxygenase-2/5-Lipoxygenase Inhibitors: Synthesis, Nitric Oxide Release, Molecular Modeling, and Biological Evaluation as Anti-Inflammatory Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 144, doi. 10.1002/cmdc.201100460

By:

Kaur, Jatinder;
Bhardwaj, Atul;
Huang, Zhangjian;
Knaus, Edward E.

Publication type:

Article

Platinum(II) Phenanthroimidazoles for Targeting Telomeric G-Quadruplexes.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 85, doi. 10.1002/cmdc.201100453

By:

Castor, Katherine J.;
Mancini, Johanna;
Fakhoury, Johans;
Weill, Nathanael;
Kieltyka, Roxanne;
Englebienne, Pablo;
Avakyan, Nicole;
Mittermaier, Anthony;
Autexier, Chantal;
Moitessier, Nicolas;
Sleiman, Hanadi F.

Publication type:

Article

Insights into Matriptase-2 Substrate Binding and Inhibition Mechanisms by Analyzing Active-Site-Mutated Variants.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 68, doi. 10.1002/cmdc.201100350

By:

Maurer, Eva;
Sisay, Mihiret T.;
Stirnberg, Marit;
Steinmetzer, Torsten;
Bajorath, Jürgen;
Gütschow, Michael

Publication type:

Article

The Tubulin Colchicine Domain: a Molecular Modeling Perspective.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 33, doi. 10.1002/cmdc.201100361

By:

Massarotti, Alberto;
Coluccia, Antonio;
Silvestri, Romano;
Sorba, Giovanni;
Brancale, Andrea

Publication type:

Article

Inside Cover: Insights into Matriptase-2 Substrate Binding and Inhibition Mechanisms by Analyzing Active-Site-Mutated Variants (ChemMedChem 1/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 2, doi. 10.1002/cmdc.201190061

By:

Maurer, Eva;
Sisay, Mihiret T.;
Stirnberg, Marit;
Steinmetzer, Torsten;
Bajorath, Jürgen;
Gütschow, Michael

Publication type:

Article

Identification and Characterization of Inhibitors of the Aminoglycoside Resistance Acetyltransferase Eis from Mycobacterium tuberculosis.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 73, doi. 10.1002/cmdc.201100332

By:

Green, Keith D.;
Chen, Wenjing;
Garneau-Tsodikova, Sylvie

Publication type:

Article

A Novel Aptamer Developed for Breast Cancer Cell Internalization.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 79, doi. 10.1002/cmdc.201100457

By:

Zhang, Kejing;
Sefah, Kwame;
Tang, Lili;
Zhao, Zilong;
Zhu, Guizhi;
Ye, Mao;
Sun, Weijia;
Goodison, Steve;
Tan, Weihong

Publication type:

Article

Analogue-Based Drug Discovery II. Edited by János Fischer and C. Robin Ganellin.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 171, doi. 10.1002/cmdc.201100479

By:

Burks, Heather E.;
Peukert, Stefan

Publication type:

Article

A Comparison of Linear and Cyclic Peptoid Oligomers as Potent Antimicrobial Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 114, doi. 10.1002/cmdc.201100358

By:

Huang, Mia Lace;
Shin, Sung Bin Y.;
Benson, Meredith A.;
Torres, Victor J.;
Kirshenbaum, Kent

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 1/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 1, p. 16, doi. 10.1002/cmdc.201190058
Publication type:: Article

Exhaustive Fluorine Scanning toward Potent p53-Mdm2 Antagonists.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 49, doi. 10.1002/cmdc.201100428

By:

Huang, Yijun;
Wolf, Siglinde;
Koes, David;
Popowicz, Grzegorz M.;
Camacho, Carlos J.;
Holak, Tad A.;
Dömling, Alexander

Publication type:

Article

Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 1

In vivo Enhancement in Bioavailability of Atazanavir in the Presence of Proton-Pump Inhibitors using Mesoporous Materials.

Specific Targeting of Hypoxic Tumor Tissue with Nitroimidazole-Peptide Conjugates.

Identification of 1,3-Diiminoisoindoline Carbohydrazides as Potential Antimalarial Candidates.

Concise Notice to Authors: ChemMedChem 1/2012.

Rofecoxib Analogues Possessing a Nitric Oxide Donor Sulfohydroxamic Acid (SO<sub>2</sub>NHOH) Cyclooxygenase-2 Pharmacophore: Synthesis, Molecular Modeling, and Biological Evaluation as Anti-inflammatory Agents.

Cover Picture: Understanding of Molecular Substructures that Contribute to hERG K<sup>+</sup> Channel Blockade: Synthesis and Biological Evaluation of E-4031 Analogues (ChemMedChem 1/2012).

Editorial: Quality Research. Outstanding Publications.

Quaternary Ammonium Salts and Their Antimicrobial Potential: Targets or Nonspecific Interactions?

Back Cover: Identification and Characterization of Inhibitors of the Aminoglycoside Resistance Acetyltransferase Eis from Mycobacterium tuberculosis (ChemMedChem 1/2012).

Development of Improved PPAR β/ δ Inhibitors.

Nocodazole is a High-Affinity Ligand for the Cancer-Related Kinases ABL, c-KIT, BRAF, and MEK.

Antiviral Drugs: From Basic Discovery Through Clinical Trials. Edited by Wieslaw M. Kazmierski.

Discovery of a Pharmacologically Active Antagonist of the Two-Pore-Domain Potassium Channel K<sub>2P</sub>9.1 (TASK-3).

Graphical Abstract: ChemMedChem 1/2012.

From a Library of MAG Antagonists to Nanomolar CD22 Ligands.

Understanding of Molecular Substructures that Contribute to hERG K<sup>+</sup> Channel Blockade: Synthesis and Biological Evaluation of E-4031 Analogues.

Preview: ChemMedChem 2/2012.

Design, Synthesis and Biological Evaluation of Trypanosoma brucei Trypanothione Synthetase Inhibitors.

Aspirin Analogues as Dual Cyclooxygenase-2/5-Lipoxygenase Inhibitors: Synthesis, Nitric Oxide Release, Molecular Modeling, and Biological Evaluation as Anti-Inflammatory Agents.

Platinum(II) Phenanthroimidazoles for Targeting Telomeric G-Quadruplexes.

Insights into Matriptase-2 Substrate Binding and Inhibition Mechanisms by Analyzing Active-Site-Mutated Variants.

The Tubulin Colchicine Domain: a Molecular Modeling Perspective.

Inside Cover: Insights into Matriptase-2 Substrate Binding and Inhibition Mechanisms by Analyzing Active-Site-Mutated Variants (ChemMedChem 1/2012).

Identification and Characterization of Inhibitors of the Aminoglycoside Resistance Acetyltransferase Eis from Mycobacterium tuberculosis.

A Novel Aptamer Developed for Breast Cancer Cell Internalization.

Analogue-Based Drug Discovery II. Edited by János Fischer and C. Robin Ganellin.

A Comparison of Linear and Cyclic Peptoid Oligomers as Potent Antimicrobial Agents.

Spotlights on our sister journals: ChemMedChem 1/2012.

Exhaustive Fluorine Scanning toward Potent p53-Mdm2 Antagonists.