Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 9

Results: 29

The Inverse Type II β-Turn on D-Trp-Phe, a Pharmacophoric Motif for MOR Agonists.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1640, doi. 10.1002/cmdc.201100169
By:
- Gentilucci, Luca;
- Tolomelli, Alessandra;
- De Marco, Rossella;
- Spampinato, Santi;
- Bedini, Andrea;
- Artali, Roberto
Publication type:
Article
Spotlights on our sister journals: ChemMedChem 9/2011.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1546, doi. 10.1002/cmdc.201190040
Publication type:
Article
The Evolution of Drug Discovery: From Traditional Medicines to Modern Drugs. By Enrique Raviña.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1746, doi. 10.1002/cmdc.201100321
By:
- Steinhagen, Henning
Publication type:
Article
Small Molecule Binding to Proteins: Affinity and Binding/Unbinding Dynamics from Atomistic Simulations.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1578, doi. 10.1002/cmdc.201100237
By:
- Huang, Danzhi;
- Caflisch, Amedeo
Publication type:
Article
A Partial Convergence in Action of Methylene Blue and Artemisinins: Antagonism with Chloroquine, a Reversal with Verapamil, and an Insight into the Antimalarial Activity of Chloroquine.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1603, doi. 10.1002/cmdc.201100184
By:
- Haynes, Richard K.;
- Cheu, Kwan-Wing;
- Li, Ka-Yan;
- Tang, Maggie Mei-Ki;
- Wong, Ho-Ning;
- Chen, Min-Jiao;
- Guo, Zu-Feng;
- Guo, Zhi-Hong;
- Coghi, Paolo;
- Monti, Diego
Publication type:
Article
Identification of a Glycogen Synthase Kinase-3β Inhibitor that Attenuates Hyperactivity in CLOCK Mutant Mice.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1593, doi. 10.1002/cmdc.201100188
By:
- Kozikowski, Alan P.;
- Gunosewoyo, Hendra;
- Guo, Songpo;
- Gaisina, Irina N.;
- Walter, Richard L.;
- Ketcherside, Ariel;
- McClung, Colleen A.;
- Mesecar, Andrew D.;
- Caldarone, Barbara
Publication type:
Article
Preview: ChemMedChem 10/2011.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1751, doi. 10.1002/cmdc.201190041
Publication type:
Article
Structure-Guided Design of a Highly Selective Glycogen Synthase Kinase-3β Inhibitor: a Superior Neuroprotective Pyrazolone Showing Antimania Effects.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1587, doi. 10.1002/cmdc.201100231
By:
- Chen, Wenwen;
- Gaisina, Irina N.;
- Gunosewoyo, Hendra;
- Malekiani, Sam A.;
- Hanania, Taleen;
- Kozikowski, Alan P.
Publication type:
Article
Inside Cover: Light-Activated Release of Nitric Oxide with Fluorescence Reporting in Living Cells (ChemMedChem 9/2011).
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1534, doi. 10.1002/cmdc.201190038
By:
- Vittorino, Elisa;
- Sciortino, Maria Teresa;
- Siracusano, Gabriel;
- Sortino, Salvatore
Publication type:
Article
Camptothecin and Thiocamptothecin: the Role of Sulfur in Shifting the Hydrolysis Equilibrium towards the Closed Lactone Form.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1706, doi. 10.1002/cmdc.201100206
By:
- Pistolozzi, Marco;
- Varchi, Greta;
- Degli Esposti, Alessandra;
- Guerrini, Andrea;
- Sotgiu, Giovanna;
- Ballestri, Marco;
- Ferroni, Claudia;
- Venturini, Alessandro;
- Bertucci, Carlo
Publication type:
Article
Synthesis and Structure-Activity Relationships of Constrained Heterocyclic Analogues of Combretastatin A4.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1693, doi. 10.1002/cmdc.201100154
By:
- Arthuis, Martin;
- Pontikis, Renée;
- Chabot, Guy G.;
- Seguin, Johanne;
- Quentin, Lionel;
- Bourg, Stéphane;
- Morin-Allory, Luc;
- Florent, Jean-Claude
Publication type:
Article
Light-Activated Release of Nitric Oxide with Fluorescence Reporting in Living Cells.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1551, doi. 10.1002/cmdc.201100198
By:
- Vittorino, Elisa;
- Sciortino, Maria Teresa;
- Siracusano, Gabriel;
- Sortino, Salvatore
Publication type:
Article
Application of the Guanidine-Acylguanidine Bioisosteric Approach to Argininamide-Type NPY Y2 Receptor Antagonists.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1727, doi. 10.1002/cmdc.201100241
By:
- Pluym, Nikola;
- Brennauer, Albert;
- Keller, Max;
- Ziemek, Ralf;
- Pop, Nathalie;
- Bernhardt, Günther;
- Buschauer, Armin
Publication type:
Article
From Activity Cliffs to Target-Specific Scoring Models and Pharmacophore Hypotheses.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1630, doi. 10.1002/cmdc.201100179
By:
- Seebeck, Birte;
- Wagener, Markus;
- Rarey, Matthias
Publication type:
Article
Acetamide Scanning around Bicyclic Thiazoles: SAR at the H3 Receptor.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1559, doi. 10.1002/cmdc.201100248
By:
- Denonne, Frédéric;
- Célanire, Sylvain;
- Christophe, Bernard;
- Defays, Sabine;
- Delaunoy, Christel;
- Delporte, Marie-Laure;
- Detrait, Eric;
- Durieu, Véronique;
- Gillard, Michel;
- Lamberty, Yves;
- Lorent, Geneviève;
- Nicolas, Jean-Marie;
- Vanbellinghen, Alain;
- Van Houtvin, Nathalie;
- Provins, Laurent
Publication type:
Article
Bromophycolide A Targets Heme Crystallization in the Human Malaria Parasite Plasmodium falciparum.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1572, doi. 10.1002/cmdc.201100252
By:
- Stout, E. Paige;
- Cervantes, Serena;
- Prudhomme, Jacques;
- France, Stefan;
- La Clair, James J.;
- Le Roch, Karine;
- Kubanek, Julia
Publication type:
Article
Cover Picture: From Activity Cliffs to Target-Specific Scoring Models and Pharmacophore Hypotheses (ChemMedChem 9/2011).
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1533, doi. 10.1002/cmdc.201190037
By:
- Seebeck, Birte;
- Wagener, Markus;
- Rarey, Matthias
Publication type:
Article
Adamantyl Ethanone Pyridyl Derivatives: Potent and Selective Inhibitors of Human 11β-Hydroxysteroid Dehydrogenase Type 1.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1616, doi. 10.1002/cmdc.201100182
By:
- Su, Xiangdong;
- Pradaux-Caggiano, Fabienne;
- Vicker, Nigel;
- Thomas, Mark P.;
- Halem, Heather;
- Culler, Michael D.;
- Potter, Barry V. L.
Publication type:
Article
Unexpected Opioid Activity Profiles of Analogues of the Novel Peptide Kappa Opioid Receptor Ligand CJ-15,208.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1739, doi. 10.1002/cmdc.201100113
By:
- Aldrich, Jane V.;
- Kulkarni, Santosh S.;
- Senadheera, Sanjeewa N.;
- Ross, Nicolette C.;
- Reilley, Kate J.;
- Eans, Shainnel O.;
- Ganno, Michelle L.;
- Murray, Thomas F.;
- McLaughlin, Jay P.
Publication type:
Article
Hepatitis C: Antiviral Drug Discovery and Development. Edited by Seng-Lai Tan and Yupeng He.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1748, doi. 10.1002/cmdc.201100238
By:
- Beaulieu, Pierre L.
Publication type:
Article
Design, Synthesis, and Biological Evaluation of Ring-Opened Bengamide Analogues.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1555, doi. 10.1002/cmdc.201100164
By:
- Tai, Wan-Yi;
- Zhang, Run-Tao;
- Ma, Yi-Ming;
- Gu, Min;
- Liu, Gang;
- Li, Jia;
- Nan, Fa-Jun
Publication type:
Article
Tissue Uptake Study and Photodynamic Therapy of Melanoma-Bearing Mice with a Nontoxic, Effective Chlorin.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1715, doi. 10.1002/cmdc.201100186
By:
- Dąbrowski, Janusz M.;
- Krzykawska, Martyna;
- Arnaut, Luis G.;
- Pereira, Mariette M.;
- Monteiro, Carlos J. P.;
- Simões, Sérgio;
- Urbańska, Krystyna;
- Stochel, Grażyna
Publication type:
Article
[3H]UR-MK136: A Highly Potent and Selective Radioligand for Neuropeptide Y Y1 Receptors.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1566, doi. 10.1002/cmdc.201100197
By:
- Keller, Max;
- Bernhardt, Günther;
- Buschauer, Armin
Publication type:
Article
Design, Synthesis, and Biological Activity of Urea Derivatives as Anaplastic Lymphoma Kinase Inhibitors.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1680, doi. 10.1002/cmdc.201100168
By:
- Boije af Gennäs, Gustav;
- Mologni, Luca;
- Ahmed, Shaheen;
- Rajaratnam, Mohanathas;
- Marin, Oriano;
- Lindholm, Niko;
- Viltadi, Michela;
- Gambacorti-Passerini, Carlo;
- Scapozza, Leonardo;
- Yli-Kauhaluoma, Jari
Publication type:
Article
Development of Antitrypanosomal and Antiplasmodial Nonpeptidic Cysteine Protease Inhibitors based on N-Protected-Guanidino-Furan and -Pyrrole Building Blocks.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1581, doi. 10.1002/cmdc.201100189
By:
- Langolf, Sebastian;
- Machon, Uwe;
- Ehlers, Martin;
- Sicking, Wilhelm;
- Schirmeister, Tanja;
- Büchhold, Christian;
- Gelhaus, Christoph;
- Rosenthal, Philip J.;
- Schmuck, Carsten
Publication type:
Article
New Frontiers in Chemical Biology: Enabling Drug Discovery. Edited by Mark E. Bunnage.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1747, doi. 10.1002/cmdc.201100254
By:
- Kritzer, Joshua
Publication type:
Article
Graphical Abstract: ChemMedChem 9/2011.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1535, doi. 10.1002/cmdc.201190039
Publication type:
Article
Synthesis of Aryl-Substituted Naphthalene-Linked Pyrrolobenzodiazepine Conjugates as Potential Anticancer Agents with Apoptosis-Inducing Ability.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1665, doi. 10.1002/cmdc.201100207
By:
- Kamal, Ahmed;
- Reddy, M. Kashi;
- Ramaiah, M. Janaki;
- Srikanth, Y. V. V.;
- Rajender;
- Reddy, V. Santosh;
- Kumar, G. Bharath;
- Pushpavalli, S. N. C. V. L.;
- Bag, Indira;
- Juvekar, Aarti;
- Sen, Subrata;
- Zingde, Surekha M.;
- Pal-Bhadra, Manika
Publication type:
Article
An Amphiphilic Conjugate Approach toward the Design and Synthesis of Betulinic Acid-Polyphenol Conjugates as Inhibitors of the HIV-1 gp41 Fusion Core Formation.
Published in:
ChemMedChem, 2011, v. 6, n. 9, p. 1654, doi. 10.1002/cmdc.201100149
By:
- Liu, Yan;
- Ke, Zhuofeng;
- Wu, Kwok Yiu;
- Liu, Shuwen;
- Chen, Wen-Hua;
- Jiang, Shibo;
- Jiang, Zhi-Hong
Publication type:
Article

Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 9

The Inverse Type II β-Turn on D-Trp-Phe, a Pharmacophoric Motif for MOR Agonists.

Spotlights on our sister journals: ChemMedChem 9/2011.

The Evolution of Drug Discovery: From Traditional Medicines to Modern Drugs. By Enrique Raviña.

Small Molecule Binding to Proteins: Affinity and Binding/Unbinding Dynamics from Atomistic Simulations.

A Partial Convergence in Action of Methylene Blue and Artemisinins: Antagonism with Chloroquine, a Reversal with Verapamil, and an Insight into the Antimalarial Activity of Chloroquine.

Identification of a Glycogen Synthase Kinase-3β Inhibitor that Attenuates Hyperactivity in CLOCK Mutant Mice.

Preview: ChemMedChem 10/2011.

Structure-Guided Design of a Highly Selective Glycogen Synthase Kinase-3β Inhibitor: a Superior Neuroprotective Pyrazolone Showing Antimania Effects.

Inside Cover: Light-Activated Release of Nitric Oxide with Fluorescence Reporting in Living Cells (ChemMedChem 9/2011).

Camptothecin and Thiocamptothecin: the Role of Sulfur in Shifting the Hydrolysis Equilibrium towards the Closed Lactone Form.

Synthesis and Structure-Activity Relationships of Constrained Heterocyclic Analogues of Combretastatin A4.

Light-Activated Release of Nitric Oxide with Fluorescence Reporting in Living Cells.

Application of the Guanidine-Acylguanidine Bioisosteric Approach to Argininamide-Type NPY Y<sub>2</sub> Receptor Antagonists.

From Activity Cliffs to Target-Specific Scoring Models and Pharmacophore Hypotheses.

Acetamide Scanning around Bicyclic Thiazoles: SAR at the H<sub>3</sub> Receptor.

Bromophycolide A Targets Heme Crystallization in the Human Malaria Parasite Plasmodium falciparum.

Cover Picture: From Activity Cliffs to Target-Specific Scoring Models and Pharmacophore Hypotheses (ChemMedChem 9/2011).

Adamantyl Ethanone Pyridyl Derivatives: Potent and Selective Inhibitors of Human 11β-Hydroxysteroid Dehydrogenase Type 1.

Unexpected Opioid Activity Profiles of Analogues of the Novel Peptide Kappa Opioid Receptor Ligand CJ-15,208.

Hepatitis C: Antiviral Drug Discovery and Development. Edited by Seng-Lai Tan and Yupeng He.

Design, Synthesis, and Biological Evaluation of Ring-Opened Bengamide Analogues.

Tissue Uptake Study and Photodynamic Therapy of Melanoma-Bearing Mice with a Nontoxic, Effective Chlorin.

[<sup>3</sup>H]UR-MK136: A Highly Potent and Selective Radioligand for Neuropeptide Y Y<sub>1</sub> Receptors.

Design, Synthesis, and Biological Activity of Urea Derivatives as Anaplastic Lymphoma Kinase Inhibitors.

Development of Antitrypanosomal and Antiplasmodial Nonpeptidic Cysteine Protease Inhibitors based on N-Protected-Guanidino-Furan and -Pyrrole Building Blocks.

New Frontiers in Chemical Biology: Enabling Drug Discovery. Edited by Mark E. Bunnage.

Graphical Abstract: ChemMedChem 9/2011.

Synthesis of Aryl-Substituted Naphthalene-Linked Pyrrolobenzodiazepine Conjugates as Potential Anticancer Agents with Apoptosis-Inducing Ability.

An Amphiphilic Conjugate Approach toward the Design and Synthesis of Betulinic Acid-Polyphenol Conjugates as Inhibitors of the HIV-1 gp41 Fusion Core Formation.