Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 8

Results: 27

Synthesis, Structural Characterization, and Pro-apoptotic Activity of 1-Indanone Thiosemicarbazone Platinum(II) and Palladium(II) Complexes: Potential as Antileukemic Agents.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1485, doi. 10.1002/cmdc.201100060

By:

Gómez, Natalia;
Santos, Diego;
Vázquez, Ramiro;
Suescun, Leopoldo;
Mombrú, Álvaro;
Vermeulen, Monica;
Finkielsztein, Liliana;
Shayo, Carina;
Moglioni, Albertina;
Gambino, Dinorah;
Davio, Carlos

Publication type:

Article

Aromatase and Dual Aromatase-Steroid Sulfatase Inhibitors from the Letrozole and Vorozole Templates.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1423, doi. 10.1002/cmdc.201100145

By:

Wood, Paul M.;
Woo, L. W. Lawrence;
Thomas, Mark P.;
Mahon, Mary F.;
Purohit, Atul;
Potter, Barry V. L.

Publication type:

Article

Novel Silicon-Containing Analogues of the Retinoid Agonist Bexarotene: Syntheses and Biological Effects on Human Pluripotent Stem Cells.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1509, doi. 10.1002/cmdc.201100156

By:

Bauer, Jennifer B.;
Lippert, W. Peter;
Dörrich, Steffen;
Tebbe, David;
Burschka, Christian;
Christie, Victoria B.;
Tams, Daniel M.;
Henderson, Andrew P.;
Murray, Bridgid A.;
Marder, Todd B.;
Przyborski, Stefan A.;
Tacke, Reinhold

Publication type:

Article

Antimalarial Mannoxanes: Hybrid Antimalarial Drugs with Outstanding Oral Activity Profiles and A Potential Dual Mechanism of Action.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1357, doi. 10.1002/cmdc.201100196

By:

Chadwick, James;
Amewu, Richard K.;
Marti, Francesc;
Garah, Fatima Bousejra-El;
Sharma, Raman;
Berry, Neil G.;
Stocks, Paul A.;
Burrell-Saward, Hollie;
Wittlin, Sergio;
Rottmann, Matthias;
Brun, Reto;
Taramelli, Donatella;
Parapini, Silvia;
Ward, Stephen A.;
O'Neill, Paul M.

Publication type:

Article

Warfarin Glycosylation Invokes a Switch from Anticoagulant to Anticancer Activity.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1347, doi. 10.1002/cmdc.201100178

By:

Peltier-Pain, Pauline;
Timmons, Shannon C.;
Grandemange, Agnès;
Benoit, Etienne;
Thorson, Jon S.

Publication type:

Article

R. K. Haynes.

Published in:: ChemMedChem, 2011, v. 6, n. 8, p. 1333, doi. 10.1002/cmdc.201100313
Publication type:: Article

Spotlights on our sister journals: ChemMedChem 8/2011.

Published in:: ChemMedChem, 2011, v. 6, n. 8, p. 1330, doi. 10.1002/cmdc.201190035
Publication type:: Article

Discovery of Adamantyl Heterocyclic Ketones as Potent 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1439, doi. 10.1002/cmdc.201100144

By:

Su, Xiangdong;
Vicker, Nigel;
Thomas, Mark P.;
Pradaux-Caggiano, Fabienne;
Halem, Heather;
Culler, Michael D.;
Potter, Barry V. L.

Publication type:

Article

Design and Synthesis of Novel Dual-Action Compounds Targeting the Adenosine A2A Receptor and Adenosine Transporter for Neuroprotection.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1390, doi. 10.1002/cmdc.201100126

By:

Chen, Jhih-Bin;
Liu, Eric Minwei;
Chern, Ting-Rong;
Yang, Chieh-Wen;
Lin, Chia-I;
Huang, Nai-Kuei;
Lin, Yun-Lian;
Chern, Yijuang;
Lin, Jung-Hsin;
Fang, Jim-Min

Publication type:

Article

Toward the Discovery of Novel Anti-HIV Drugs. Second-Generation Inhibitors of the Cellular ATPase DDX3 with Improved Anti-HIV Activity: Synthesis, Structure-Activity Relationship Analysis, Cytotoxicity Studies, and Target Validation.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1371, doi. 10.1002/cmdc.201100166

By:

Maga, Giovanni;
Falchi, Federico;
Radi, Marco;
Botta, Lorenzo;
Casaluce, Gianni;
Bernardini, Martina;
Irannejad, Hamid;
Manetti, Fabrizio;
Garbelli, Anna;
Samuele, Alberta;
Zanoli, Samantha;
Esté, José A.;
Gonzalez, Emmanuel;
Zucca, Elisa;
Paolucci, Stefania;
Baldanti, Fausto;
De Rijck, Jan;
Debyser, Zeger;
Botta, Maurizio

Publication type:

Article

Cell-Free HIV-1 Virucidal Action by Modified Peptide Triazole Inhibitors of Env gp120.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1335, doi. 10.1002/cmdc.201100177

By:

Bastian, Arangassery R.;
Kantharaju;
McFadden, Karyn;
Duffy, Caitlin;
Rajagopal, Srivats;
Contarino, Mark R.;
Papazoglou, Elisabeth;
Chaiken, Irwin

Publication type:

Article

A 18F-Labeled Fluorobutyl-Substituted Spirocyclic Piperidine Derivative as a Selective Radioligand for PET Imaging of Sigma1 Receptors.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1401, doi. 10.1002/cmdc.201100108

By:

Maisonial, Aurélie;
Große Maestrup, Eva;
Fischer, Steffen;
Hiller, Achim;
Scheunemann, Matthias;
Wiese, Christian;
Schepmann, Dirk;
Steinbach, Jörg;
Deuther-Conrad, Winnie;
Wünsch, Bernhard;
Brust, Peter

Publication type:

Article

Graphical Abstract: ChemMedChem 8/2011.

Published in:: ChemMedChem, 2011, v. 6, n. 8, p. 1319, doi. 10.1002/cmdc.201190034
Publication type:: Article

Polyphosphates and Pyrophosphates of Pentopyranoses and Pentofuranoses as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Oxygen Release.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1495, doi. 10.1002/cmdc.201100110

By:

Fylaktakidou, Konstantina C.;
Duarte, Carolina D.;
Jogireddy, Rajamalleswaramma;
Koumbis, Alexandros E.;
Nicolau, Claude;
Lehn, Jean-Marie

Publication type:

Article

Chemokine Receptors as Drug Targets. Edited by Martine J. Smit, Sergio A. Lira and Rob Leurs.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1530, doi. 10.1002/cmdc.201100257

By:

Merritt, J. Robert

Publication type:

Article

Antagonism of the Stat3-Stat3 Protein Dimer with Salicylic Acid Based Small Molecules.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1459, doi. 10.1002/cmdc.201100194

By:

Fletcher, Steven;
Page, Brent D. G.;
Zhang, Xialoei;
Yue, Peibin;
Li, Zhi Hua;
Sharmeen, Sumaiya;
Singh, Jagdeep;
Zhao, Wei;
Schimmer, Aaron D.;
Trudel, Suzanne;
Turkson, James;
Gunning, Patrick T.

Publication type:

Article

Inside Cover: Cell-Free HIV-1 Virucidal Action by Modified Peptide Triazole Inhibitors of Env gp120 (ChemMedChem 8/2011).

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1318, doi. 10.1002/cmdc.201190033

By:

Bastian, Arangassery R.;
Kantharaju;
McFadden, Karyn;
Duffy, Caitlin;
Rajagopal, Srivats;
Contarino, Mark R.;
Papazoglou, Elisabeth;
Chaiken, Irwin

Publication type:

Article

Identification of Benzopyran-4-one Derivatives (Isoflavones) as Positive Modulators of GABAA Receptors.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1340, doi. 10.1002/cmdc.201100120

By:

Gavande, Navnath;
Karim, Nasiara;
Johnston, Graham A. R.;
Hanrahan, Jane R.;
Chebib, Mary

Publication type:

Article

Identification of Xanthones as Selective Killers of Cancer Cells Overexpressing the ABC Transporter MRP1.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1478, doi. 10.1002/cmdc.201100102

By:

Genoux-Bastide, Estelle;
Lorendeau, Doriane;
Nicolle, Edwige;
Yahiaoui, Samir;
Magnard, Sandrine;
Di Pietro, Attilio;
Baubichon-Cortay, Hélène;
Boumendjel, Ahcène

Publication type:

Article

Orally Active, Antimetastatic, Nontoxic Diphenyl Ether-Derived Carbamoylphosphonate Matrix Metalloproteinase Inhibitors.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1471, doi. 10.1002/cmdc.201100153

By:

Frant, Julia;
Veerendhar, Ainelly;
Chernilovsky, Tamir;
Nedvetzki, Shlomo;
Vaksman, Olga;
Hoffman, Amnon;
Breuer, Eli;
Reich, Reuven

Publication type:

Article

Discovery, Structure-Activity Relationship Studies, and Crystal Structure of Nonpeptide Inhibitors Bound to the Shank3 PDZ Domain.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1411, doi. 10.1002/cmdc.201100094

By:

Saupe, Jörn;
Roske, Yvette;
Schillinger, Christian;
Kamdem, Nestor;
Radetzki, Silke;
Diehl, Anne;
Oschkinat, Hartmut;
Krause, Gerd;
Heinemann, Udo;
Rademann, Jörg

Publication type:

Article

Delineation of the Molecular Mechanisms of Nucleoside Recognition by Cytidine Deaminase through Virtual Screening.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1452, doi. 10.1002/cmdc.201100139

By:

Costanzi, Stefano;
Vilar, Santiago;
Micozzi, Daniela;
Carpi, Francesco M.;
Ferino, Giulio;
Vita, Alberto;
Vincenzetti, Silvia

Publication type:

Article

Design and Stereoselective Synthesis of Retinoids with Ferrocene or N-Butylcarbazole Pharmacophores that Induce Post-Differentiation Apoptosis in Acute Promyelocytic Leukemia Cells.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1518, doi. 10.1002/cmdc.201100065

By:

Ivanova, Diana;
Gronemeyer, Hinrich;
de Lera, Angel R.

Publication type:

Article

Novel Mechanism of Cathepsin B Inhibition by Antibiotic Nitroxoline and Related Compounds.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1351, doi. 10.1002/cmdc.201100098

By:

Mirković, Bojana;
Renko, Miha;
Turk, Samo;
Sosič, Izidor;
Jevnikar, Zala;
Obermajer, Nataša;
Turk, Dušan;
Gobec, Stanislav;
Kos, Janko

Publication type:

Article

Cover Picture: Identification of Benzopyran-4-one Derivatives (Isoflavones) as Positive Modulators of GABAA Receptors (ChemMedChem 8/2011).

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1317, doi. 10.1002/cmdc.201190032

By:

Gavande, Navnath;
Karim, Nasiara;
Johnston, Graham A. R.;
Hanrahan, Jane R.;
Chebib, Mary

Publication type:

Article

Oxime-Based Click Chemistry in the Development of 3-Isoxazolecarboxylic Acid Containing Inhibitors of Yersinia pestis Protein Tyrosine Phosphatase, YopH.

Published in:

ChemMedChem, 2011, v. 6, n. 8, p. 1363, doi. 10.1002/cmdc.201100200

By:

Bahta, Medhanit;
Burke, Terrence R.

Publication type:

Article

Preview: ChemMedChem 9/2011.

Published in:: ChemMedChem, 2011, v. 6, n. 8, p. 1531, doi. 10.1002/cmdc.201190036
Publication type:: Article

Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 8

Synthesis, Structural Characterization, and Pro-apoptotic Activity of 1-Indanone Thiosemicarbazone Platinum(II) and Palladium(II) Complexes: Potential as Antileukemic Agents.

Aromatase and Dual Aromatase-Steroid Sulfatase Inhibitors from the Letrozole and Vorozole Templates.

Novel Silicon-Containing Analogues of the Retinoid Agonist Bexarotene: Syntheses and Biological Effects on Human Pluripotent Stem Cells.

Antimalarial Mannoxanes: Hybrid Antimalarial Drugs with Outstanding Oral Activity Profiles and A Potential Dual Mechanism of Action.

Warfarin Glycosylation Invokes a Switch from Anticoagulant to Anticancer Activity.

R. K. Haynes.

Spotlights on our sister journals: ChemMedChem 8/2011.

Discovery of Adamantyl Heterocyclic Ketones as Potent 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors.

Design and Synthesis of Novel Dual-Action Compounds Targeting the Adenosine A<sub>2A</sub> Receptor and Adenosine Transporter for Neuroprotection.

Toward the Discovery of Novel Anti-HIV Drugs. Second-Generation Inhibitors of the Cellular ATPase DDX3 with Improved Anti-HIV Activity: Synthesis, Structure-Activity Relationship Analysis, Cytotoxicity Studies, and Target Validation.

Cell-Free HIV-1 Virucidal Action by Modified Peptide Triazole Inhibitors of Env gp120.

A <sup>18</sup>F-Labeled Fluorobutyl-Substituted Spirocyclic Piperidine Derivative as a Selective Radioligand for PET Imaging of Sigma<sub>1</sub> Receptors.

Graphical Abstract: ChemMedChem 8/2011.

Polyphosphates and Pyrophosphates of Pentopyranoses and Pentofuranoses as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Oxygen Release.

Chemokine Receptors as Drug Targets. Edited by Martine J. Smit, Sergio A. Lira and Rob Leurs.

Antagonism of the Stat3-Stat3 Protein Dimer with Salicylic Acid Based Small Molecules.

Inside Cover: Cell-Free HIV-1 Virucidal Action by Modified Peptide Triazole Inhibitors of Env gp120 (ChemMedChem 8/2011).

Identification of Benzopyran-4-one Derivatives (Isoflavones) as Positive Modulators of GABA<sub>A</sub> Receptors.

Identification of Xanthones as Selective Killers of Cancer Cells Overexpressing the ABC Transporter MRP1.

Orally Active, Antimetastatic, Nontoxic Diphenyl Ether-Derived Carbamoylphosphonate Matrix Metalloproteinase Inhibitors.

Discovery, Structure-Activity Relationship Studies, and Crystal Structure of Nonpeptide Inhibitors Bound to the Shank3 PDZ Domain.

Delineation of the Molecular Mechanisms of Nucleoside Recognition by Cytidine Deaminase through Virtual Screening.

Design and Stereoselective Synthesis of Retinoids with Ferrocene or N-Butylcarbazole Pharmacophores that Induce Post-Differentiation Apoptosis in Acute Promyelocytic Leukemia Cells.

Novel Mechanism of Cathepsin B Inhibition by Antibiotic Nitroxoline and Related Compounds.

Cover Picture: Identification of Benzopyran-4-one Derivatives (Isoflavones) as Positive Modulators of GABA<sub>A</sub> Receptors (ChemMedChem 8/2011).

Oxime-Based Click Chemistry in the Development of 3-Isoxazolecarboxylic Acid Containing Inhibitors of Yersinia pestis Protein Tyrosine Phosphatase, YopH.

Preview: ChemMedChem 9/2011.