Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 1

Results: 28

Symmetry Complementarity-Guided Design of Anthrax Toxin Inhibitors Based on β-Cyclodextrin: Synthesis and Relative Activities of Face-Selective Functionalized Polycationic Clusters.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 181, doi. 10.1002/cmdc.201000419
By:
- Díaz-Moscoso, Alejandro;
- Méndez-Ardoy, Alejandro;
- Ortega-Caballero, Fernando;
- Benito, Juan M.;
- Ortiz Mellet, Carmen;
- Defaye, Jacques;
- Robinson, Tanisha M.;
- Yohannes, Adiamseged;
- Karginov, Vladimir A.;
- García Fernández, José M.
Publication type:
Article
Integrated Synthetic, Pharmacological, and Computational Investigation of cis-2-(3,5-Dichlorophenylcarbamoyl)cyclohexanecarboxylic Acid Enantiomers As Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 4.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 131, doi. 10.1002/cmdc.201000378
By:
- Christov, Christo;
- González-Bulnes, Patricia;
- Malhaire, Fanny;
- Karabencheva, Tatyana;
- Goudet, Cyril;
- Pin, Jean-Philippe;
- Llebaria, Amadeu;
- Giraldo, Jesús
Publication type:
Article
Chemotherapeutic Evaluation of a Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing Mice.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 49, doi. 10.1002/cmdc.201000377
By:
- Floyd, William C.;
- Datta, Gopal K.;
- Imamura, Shinichi;
- Kieler-Ferguson, Heidi M.;
- Jerger, Katherine;
- Patterson, Andrew W.;
- Fox, Megan E.;
- Szoka, Francis C.;
- Fréchet, Jean M. J.;
- Ellman, Jonathan A.
Publication type:
Article
Palmitoylated SDF1 α Shows Increased Resistance against Proteolytic Degradation in Liver Homogenates.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 193, doi. 10.1002/cmdc.201000403
By:
- Bellmann-Sickert, Kathrin;
- Beck-Sickinger, Annette G.
Publication type:
Article
Inside Cover: 1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ8-Δ7 Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity (ChemMedChem 1/2011).
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 2, doi. 10.1002/cmdc.201090062
By:
- Abate, Carmen;
- Niso, Mauro;
- Contino, Marialessandra;
- Colabufo, Nicola Antonio;
- Ferorelli, Savina;
- Perrone, Roberto;
- Berardi, Francesco
Publication type:
Article
Discovery of 4-Benzylamino-Substituted α-Carbolines as a Novel Class of Receptor Tyrosine Kinase Inhibitors.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 63, doi. 10.1002/cmdc.201000384
By:
- Krug, Martin;
- Wichapong, Kanin;
- Erlenkamp, German;
- Sippl, Wolfgang;
- Schächtele, Christoph;
- Totzke, Frank;
- Hilgeroth, Andreas
Publication type:
Article
Polyphosphates and Pyrophosphates of Hexopyranoses as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Effect on Oxygen Release.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 153, doi. 10.1002/cmdc.201000366
By:
- Fylaktakidou, Konstantina C.;
- Duarte, Carolina D.;
- Koumbis, Alexandros E.;
- Nicolau, Claude;
- Lehn, Jean-Marie
Publication type:
Article
Tetrakisphosphates and Bispyrophosphates of myo-Inositol Derivatives as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Oxygen Release.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 169, doi. 10.1002/cmdc.201000421
By:
- Koumbis, Alexandros E.;
- Duarte, Carolina D.;
- Nicolau, Claude;
- Lehn, Jean-Marie
Publication type:
Article
Cover Picture: Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1 (ChemMedChem 1/2011).
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 1, doi. 10.1002/cmdc.201090059
By:
- Lluis, Matthew;
- Wang, Yun;
- Monzingo, Arthur F.;
- Fast, Walter;
- Robertus, Jon D.
Publication type:
Article
The Winds of Change.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 3, doi. 10.1002/cmdc.200000493
By:
- Ortúzar, Natalia
Publication type:
Article
Preview: ChemMedChem 2/2011.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 207, doi. 10.1002/cmdc.201090061
Publication type:
Article
Structure-Activity Relationship Refinement and Further Assessment of Indole-3-glyoxylamides as a Lead Series against Prion Disease.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 115, doi. 10.1002/cmdc.201000383
By:
- Thompson, Mark J.;
- Louth, Jennifer C.;
- Ferrara, Steven;
- Sorrell, Fiona J.;
- Irving, Benjamin J.;
- Cochrane, Edward J.;
- Meijer, Anthony J. H. M.;
- Chen, Beining
Publication type:
Article
Authors Profile.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 21, doi. 10.1002/cmdc.201000497
By:
- Kozikowski, Alan P.
Publication type:
Article
A Combined Ligand- and Structure-Based Virtual Screening Protocol Identifies Submicromolar PPARγ Partial Agonists.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 94, doi. 10.1002/cmdc.201000428
By:
- Vidović, Dušica;
- Busby, Scott A.;
- Griffin, Patrick R.;
- Schürer, Stephan C.
Publication type:
Article
Small-Molecule Inhibitors of the ERK Signaling Pathway: Towards Novel Anticancer Therapeutics.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 38, doi. 10.1002/cmdc.201000354
By:
- Yap, Jeremy L.;
- Worlikar, Shilpa;
- MacKerell, Alexander D.;
- Shapiro, Paul;
- Fletcher, Steven
Publication type:
Article
Modern Drug Synthesis. Edited by Jie Jack Li and Douglas S. Johnson.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 202, doi. 10.1002/cmdc.201000394
By:
- Schall, Andreas;
- Haning, Helmut
Publication type:
Article
Fluorine-Protein Interactions and 19F NMR Isotropic Chemical Shifts: An Empirical Correlation with Implications for Drug Design.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 104, doi. 10.1002/cmdc.201000412
By:
- Dalvit, Claudio;
- Vulpetti, Anna
Publication type:
Article
Spotlights on our sister journals: ChemMedChem 1/2011.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 18, doi. 10.1002/cmdc.201090060
Publication type:
Article
Solid-State Perturbation for Solubility Improvement: A Proof of Concept.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 60, doi. 10.1002/cmdc.201000405
By:
- Briggner, Lars-Erik;
- Hendrickx, Ramon;
- Kloo, Lars;
- Rosdahl, Jan;
- Svensson, Per H.
Publication type:
Article
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ8-Δ7 Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 73, doi. 10.1002/cmdc.201000371
By:
- Abate, Carmen;
- Niso, Mauro;
- Contino, Marialessandra;
- Colabufo, Nicola Antonio;
- Ferorelli, Savina;
- Perrone, Roberto;
- Berardi, Francesco
Publication type:
Article
BACE: Lead Target for Orchestrated Therapy of Alzheimer's Disease. Edited by Varghese John.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 201, doi. 10.1002/cmdc.201000427
By:
- Stamford, Andrew
Publication type:
Article
The Legumain Protease-Activated Auristatin Prodrugs Suppress Tumor Growth and Metastasis without Toxicity.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 54, doi. 10.1002/cmdc.201000478
By:
- Bajjuri, Krishna Mohan;
- Liu, Yuan;
- Liu, Cheng;
- Sinha, Subhash C.
Publication type:
Article
Asborin Inhibits Aldo/Keto Reductase 1A1.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 89, doi. 10.1002/cmdc.201000368
By:
- Scholz, Matthias;
- Steinhagen, Max;
- Heiker, John T.;
- Beck-Sickinger, Annette G.;
- Hey-Hawkins, Evamarie
Publication type:
Article
Monoclonal Antibody and Peptide-Targeted Radiotherapy of Cancer. Edited by Raymond M. Reilly.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 202, doi. 10.1002/cmdc.201000400
By:
- Mindt, Thomas L.;
- Forrer, Flavio
Publication type:
Article
New cis-Configured Aziridine-2-carboxylates as Aspartic Acid Protease Inhibitors.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 141, doi. 10.1002/cmdc.201000370
By:
- Büchold, Christian;
- Hemberger, Yasmin;
- Heindl, Cornelia;
- Welker, Armin;
- Degel, Björn;
- Pfeuffer, Thomas;
- Staib, Peter;
- Schneider, Sabrina;
- Rosenthal, Philip J.;
- Gut, Jiri;
- Morschhäuser, Joachim;
- Bringmann, Gerhard;
- Schirmeister, Tanja
Publication type:
Article
Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 81, doi. 10.1002/cmdc.201000392
By:
- Lluis, Matthew;
- Wang, Yun;
- Monzingo, Arthur F.;
- Fast, Walter;
- Robertus, Jon D.
Publication type:
Article
Graphical Abstract: ChemMedChem 1/2011.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 8, doi. 10.1002/cmdc.201090063
Publication type:
Article
Synthesis and Bioactivity of Carbohydrate Derivatives of Indigo, Its Isomers and Heteroanalogues.
Published in:
ChemMedChem, 2011, v. 6, n. 1, p. 25, doi. 10.1002/cmdc.201000374
By:
- Karapetyan, Gnuni;
- Chakrabarty, Kuheli;
- Hein, Martin;
- Langer, Peter
Publication type:
Article

Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 1

Symmetry Complementarity-Guided Design of Anthrax Toxin Inhibitors Based on β-Cyclodextrin: Synthesis and Relative Activities of Face-Selective Functionalized Polycationic Clusters.

Integrated Synthetic, Pharmacological, and Computational Investigation of cis-2-(3,5-Dichlorophenylcarbamoyl)cyclohexanecarboxylic Acid Enantiomers As Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 4.

Chemotherapeutic Evaluation of a Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing Mice.

Palmitoylated SDF1 α Shows Increased Resistance against Proteolytic Degradation in Liver Homogenates.

Inside Cover: 1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ<sub>8</sub>-Δ<sub>7</sub> Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity (ChemMedChem 1/2011).

Discovery of 4-Benzylamino-Substituted α-Carbolines as a Novel Class of Receptor Tyrosine Kinase Inhibitors.

Polyphosphates and Pyrophosphates of Hexopyranoses as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Effect on Oxygen Release.

Tetrakisphosphates and Bispyrophosphates of myo-Inositol Derivatives as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Oxygen Release.

Cover Picture: Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1 (ChemMedChem 1/2011).

The Winds of Change.

Preview: ChemMedChem 2/2011.

Structure-Activity Relationship Refinement and Further Assessment of Indole-3-glyoxylamides as a Lead Series against Prion Disease.

Authors Profile.

A Combined Ligand- and Structure-Based Virtual Screening Protocol Identifies Submicromolar PPARγ Partial Agonists.

Small-Molecule Inhibitors of the ERK Signaling Pathway: Towards Novel Anticancer Therapeutics.

Modern Drug Synthesis. Edited by Jie Jack Li and Douglas S. Johnson.

Fluorine-Protein Interactions and <sup>19</sup>F NMR Isotropic Chemical Shifts: An Empirical Correlation with Implications for Drug Design.

Spotlights on our sister journals: ChemMedChem 1/2011.

Solid-State Perturbation for Solubility Improvement: A Proof of Concept.

1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ<sub>8</sub>-Δ<sub>7</sub> Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity.

BACE: Lead Target for Orchestrated Therapy of Alzheimer's Disease. Edited by Varghese John.

The Legumain Protease-Activated Auristatin Prodrugs Suppress Tumor Growth and Metastasis without Toxicity.

Asborin Inhibits Aldo/Keto Reductase 1A1.

Monoclonal Antibody and Peptide-Targeted Radiotherapy of Cancer. Edited by Raymond M. Reilly.

New cis-Configured Aziridine-2-carboxylates as Aspartic Acid Protease Inhibitors.

Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1.

Graphical Abstract: ChemMedChem 1/2011.

Synthesis and Bioactivity of Carbohydrate Derivatives of Indigo, Its Isomers and Heteroanalogues.