Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 1

Results: 28

Symmetry Complementarity-Guided Design of Anthrax Toxin Inhibitors Based on β-Cyclodextrin: Synthesis and Relative Activities of Face-Selective Functionalized Polycationic Clusters.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 181, doi. 10.1002/cmdc.201000419

By:

Díaz-Moscoso, Alejandro;
Méndez-Ardoy, Alejandro;
Ortega-Caballero, Fernando;
Benito, Juan M.;
Ortiz Mellet, Carmen;
Defaye, Jacques;
Robinson, Tanisha M.;
Yohannes, Adiamseged;
Karginov, Vladimir A.;
García Fernández, José M.

Publication type:

Article

Integrated Synthetic, Pharmacological, and Computational Investigation of cis-2-(3,5-Dichlorophenylcarbamoyl)cyclohexanecarboxylic Acid Enantiomers As Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 4.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 131, doi. 10.1002/cmdc.201000378

By:

Christov, Christo;
González-Bulnes, Patricia;
Malhaire, Fanny;
Karabencheva, Tatyana;
Goudet, Cyril;
Pin, Jean-Philippe;
Llebaria, Amadeu;
Giraldo, Jesús

Publication type:

Article

Tetrakisphosphates and Bispyrophosphates of myo-Inositol Derivatives as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Oxygen Release.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 169, doi. 10.1002/cmdc.201000421

By:

Koumbis, Alexandros E.;
Duarte, Carolina D.;
Nicolau, Claude;
Lehn, Jean-Marie

Publication type:

Article

Palmitoylated SDF1 α Shows Increased Resistance against Proteolytic Degradation in Liver Homogenates.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 193, doi. 10.1002/cmdc.201000403

By:

Bellmann-Sickert, Kathrin;
Beck-Sickinger, Annette G.

Publication type:

Article

Inside Cover: 1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ8-Δ7 Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity (ChemMedChem 1/2011).

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 2, doi. 10.1002/cmdc.201090062

By:

Abate, Carmen;
Niso, Mauro;
Contino, Marialessandra;
Colabufo, Nicola Antonio;
Ferorelli, Savina;
Perrone, Roberto;
Berardi, Francesco

Publication type:

Article

Discovery of 4-Benzylamino-Substituted α-Carbolines as a Novel Class of Receptor Tyrosine Kinase Inhibitors.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 63, doi. 10.1002/cmdc.201000384

By:

Krug, Martin;
Wichapong, Kanin;
Erlenkamp, German;
Sippl, Wolfgang;
Schächtele, Christoph;
Totzke, Frank;
Hilgeroth, Andreas

Publication type:

Article

Polyphosphates and Pyrophosphates of Hexopyranoses as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Effect on Oxygen Release.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 153, doi. 10.1002/cmdc.201000366

By:

Fylaktakidou, Konstantina C.;
Duarte, Carolina D.;
Koumbis, Alexandros E.;
Nicolau, Claude;
Lehn, Jean-Marie

Publication type:

Article

Chemotherapeutic Evaluation of a Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing Mice.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 49, doi. 10.1002/cmdc.201000377

By:

Floyd, William C.;
Datta, Gopal K.;
Imamura, Shinichi;
Kieler-Ferguson, Heidi M.;
Jerger, Katherine;
Patterson, Andrew W.;
Fox, Megan E.;
Szoka, Francis C.;
Fréchet, Jean M. J.;
Ellman, Jonathan A.

Publication type:

Article

Cover Picture: Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1 (ChemMedChem 1/2011).

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 1, doi. 10.1002/cmdc.201090059

By:

Lluis, Matthew;
Wang, Yun;
Monzingo, Arthur F.;
Fast, Walter;
Robertus, Jon D.

Publication type:

Article

The Winds of Change.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 3, doi. 10.1002/cmdc.200000493

By:

Ortúzar, Natalia

Publication type:

Article

Preview: ChemMedChem 2/2011.

Published in:: ChemMedChem, 2011, v. 6, n. 1, p. 207, doi. 10.1002/cmdc.201090061
Publication type:: Article

Structure-Activity Relationship Refinement and Further Assessment of Indole-3-glyoxylamides as a Lead Series against Prion Disease.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 115, doi. 10.1002/cmdc.201000383

By:

Thompson, Mark J.;
Louth, Jennifer C.;
Ferrara, Steven;
Sorrell, Fiona J.;
Irving, Benjamin J.;
Cochrane, Edward J.;
Meijer, Anthony J. H. M.;
Chen, Beining

Publication type:

Article

Authors Profile.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 21, doi. 10.1002/cmdc.201000497

By:

Kozikowski, Alan P.

Publication type:

Article

A Combined Ligand- and Structure-Based Virtual Screening Protocol Identifies Submicromolar PPARγ Partial Agonists.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 94, doi. 10.1002/cmdc.201000428

By:

Vidović, Dušica;
Busby, Scott A.;
Griffin, Patrick R.;
Schürer, Stephan C.

Publication type:

Article

Small-Molecule Inhibitors of the ERK Signaling Pathway: Towards Novel Anticancer Therapeutics.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 38, doi. 10.1002/cmdc.201000354

By:

Yap, Jeremy L.;
Worlikar, Shilpa;
MacKerell, Alexander D.;
Shapiro, Paul;
Fletcher, Steven

Publication type:

Article

Modern Drug Synthesis. Edited by Jie Jack Li and Douglas S. Johnson.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 202, doi. 10.1002/cmdc.201000394

By:

Schall, Andreas;
Haning, Helmut

Publication type:

Article

Fluorine-Protein Interactions and 19F NMR Isotropic Chemical Shifts: An Empirical Correlation with Implications for Drug Design.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 104, doi. 10.1002/cmdc.201000412

By:

Dalvit, Claudio;
Vulpetti, Anna

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 1/2011.

Published in:: ChemMedChem, 2011, v. 6, n. 1, p. 18, doi. 10.1002/cmdc.201090060
Publication type:: Article

Solid-State Perturbation for Solubility Improvement: A Proof of Concept.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 60, doi. 10.1002/cmdc.201000405

By:

Briggner, Lars-Erik;
Hendrickx, Ramon;
Kloo, Lars;
Rosdahl, Jan;
Svensson, Per H.

Publication type:

Article

1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ8-Δ7 Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 73, doi. 10.1002/cmdc.201000371

By:

Abate, Carmen;
Niso, Mauro;
Contino, Marialessandra;
Colabufo, Nicola Antonio;
Ferorelli, Savina;
Perrone, Roberto;
Berardi, Francesco

Publication type:

Article

BACE: Lead Target for Orchestrated Therapy of Alzheimer's Disease. Edited by Varghese John.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 201, doi. 10.1002/cmdc.201000427

By:

Stamford, Andrew

Publication type:

Article

The Legumain Protease-Activated Auristatin Prodrugs Suppress Tumor Growth and Metastasis without Toxicity.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 54, doi. 10.1002/cmdc.201000478

By:

Bajjuri, Krishna Mohan;
Liu, Yuan;
Liu, Cheng;
Sinha, Subhash C.

Publication type:

Article

Asborin Inhibits Aldo/Keto Reductase 1A1.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 89, doi. 10.1002/cmdc.201000368

By:

Scholz, Matthias;
Steinhagen, Max;
Heiker, John T.;
Beck-Sickinger, Annette G.;
Hey-Hawkins, Evamarie

Publication type:

Article

Monoclonal Antibody and Peptide-Targeted Radiotherapy of Cancer. Edited by Raymond M. Reilly.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 202, doi. 10.1002/cmdc.201000400

By:

Mindt, Thomas L.;
Forrer, Flavio

Publication type:

Article

New cis-Configured Aziridine-2-carboxylates as Aspartic Acid Protease Inhibitors.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 141, doi. 10.1002/cmdc.201000370

By:

Büchold, Christian;
Hemberger, Yasmin;
Heindl, Cornelia;
Welker, Armin;
Degel, Björn;
Pfeuffer, Thomas;
Staib, Peter;
Schneider, Sabrina;
Rosenthal, Philip J.;
Gut, Jiri;
Morschhäuser, Joachim;
Bringmann, Gerhard;
Schirmeister, Tanja

Publication type:

Article

Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 81, doi. 10.1002/cmdc.201000392

By:

Lluis, Matthew;
Wang, Yun;
Monzingo, Arthur F.;
Fast, Walter;
Robertus, Jon D.

Publication type:

Article

Graphical Abstract: ChemMedChem 1/2011.

Published in:: ChemMedChem, 2011, v. 6, n. 1, p. 8, doi. 10.1002/cmdc.201090063
Publication type:: Article

Synthesis and Bioactivity of Carbohydrate Derivatives of Indigo, Its Isomers and Heteroanalogues.

Published in:

ChemMedChem, 2011, v. 6, n. 1, p. 25, doi. 10.1002/cmdc.201000374

By:

Karapetyan, Gnuni;
Chakrabarty, Kuheli;
Hein, Martin;
Langer, Peter

Publication type:

Article

Works matching IS 18607179 AND DT 2011 AND VI 6 AND IP 1

Symmetry Complementarity-Guided Design of Anthrax Toxin Inhibitors Based on β-Cyclodextrin: Synthesis and Relative Activities of Face-Selective Functionalized Polycationic Clusters.

Integrated Synthetic, Pharmacological, and Computational Investigation of cis-2-(3,5-Dichlorophenylcarbamoyl)cyclohexanecarboxylic Acid Enantiomers As Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 4.

Tetrakisphosphates and Bispyrophosphates of myo-Inositol Derivatives as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Oxygen Release.

Palmitoylated SDF1 α Shows Increased Resistance against Proteolytic Degradation in Liver Homogenates.

Inside Cover: 1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ<sub>8</sub>-Δ<sub>7</sub> Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity (ChemMedChem 1/2011).

Discovery of 4-Benzylamino-Substituted α-Carbolines as a Novel Class of Receptor Tyrosine Kinase Inhibitors.

Polyphosphates and Pyrophosphates of Hexopyranoses as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Effect on Oxygen Release.

Chemotherapeutic Evaluation of a Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing Mice.

Cover Picture: Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1 (ChemMedChem 1/2011).

The Winds of Change.

Preview: ChemMedChem 2/2011.

Structure-Activity Relationship Refinement and Further Assessment of Indole-3-glyoxylamides as a Lead Series against Prion Disease.

Authors Profile.

A Combined Ligand- and Structure-Based Virtual Screening Protocol Identifies Submicromolar PPARγ Partial Agonists.

Small-Molecule Inhibitors of the ERK Signaling Pathway: Towards Novel Anticancer Therapeutics.

Modern Drug Synthesis. Edited by Jie Jack Li and Douglas S. Johnson.

Fluorine-Protein Interactions and <sup>19</sup>F NMR Isotropic Chemical Shifts: An Empirical Correlation with Implications for Drug Design.

Spotlights on our sister journals: ChemMedChem 1/2011.

Solid-State Perturbation for Solubility Improvement: A Proof of Concept.

1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ<sub>8</sub>-Δ<sub>7</sub> Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity.

BACE: Lead Target for Orchestrated Therapy of Alzheimer's Disease. Edited by Varghese John.

The Legumain Protease-Activated Auristatin Prodrugs Suppress Tumor Growth and Metastasis without Toxicity.

Asborin Inhibits Aldo/Keto Reductase 1A1.

Monoclonal Antibody and Peptide-Targeted Radiotherapy of Cancer. Edited by Raymond M. Reilly.

New cis-Configured Aziridine-2-carboxylates as Aspartic Acid Protease Inhibitors.

Characterization of C-Alkyl Amidines as Bioavailable Covalent Reversible Inhibitors of Human DDAH-1.

Graphical Abstract: ChemMedChem 1/2011.

Synthesis and Bioactivity of Carbohydrate Derivatives of Indigo, Its Isomers and Heteroanalogues.