Works matching IS 18607179 AND DT 2010 AND VI 5 AND IP 9

Results: 27

Spotlights on our sister journals: ChemMedChem 9/2010.

Published in:: ChemMedChem, 2010, v. 5, n. 9, p. 1416, doi. 10.1002/cmdc.201090040
Publication type:: Article

Synthesis of Bioactive 2-Aza-Analogues of Ipecac and Alangium Alkaloids.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1456, doi. 10.1002/cmdc.201000230

By:

Kölzer, Michael;
Weitzel, Kerstin;
Göringer, H. Ulrich;
Thines, Eckhard;
Opatz, Till

Publication type:

Article

Inside Cover: Improved 2,4-Diarylthiazole-Based Antiprion Agents: Switching the Sense of the Amide Group at C5 Leads to an Increase in Potency (ChemMedChem 9/2010).

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1406, doi. 10.1002/cmdc.201090037

By:

Thompson, Mark J.;
Louth, Jennifer C.;
Greenwood, Gemma K.;
Sorrell, Fiona J.;
Knight, Sandra G.;
Adams, Nathan B. P.;
Chen, Beining

Publication type:

Article

Heme Oxygenase Inhibition by 1-Aryl-2-(1 H-imidazol-1-yl/1 H-1,2,4-triazol-1-yl)ethanones and Their Derivatives.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1541, doi. 10.1002/cmdc.201000120

By:

Roman, Gheorghe;
Vlahakis, Jason Z.;
Vukomanovic, Dragic;
Nakatsu, Kanji;
Szarek, Walter A.

Publication type:

Article

Specific Inhibitors of the Breast Cancer Resistance Protein (BCRP).

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1498, doi. 10.1002/cmdc.201000216

By:

Pick, Anne;
Klinkhammer, Werner;
Wiese, Michael

Publication type:

Article

Prediction of the Three-Dimensional Structure for the Rat Urotensin II Receptor, and Comparison of the Antagonist Binding Sites and Binding Selectivity between Human and Rat Receptors from Atomistic Simulations.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1594, doi. 10.1002/cmdc.201000175

By:

Kim, Soo-Kyung;
Li, Youyong;
Park, Changmoon;
Abrol, Ravinder;
Goddard, William A.

Publication type:

Article

Bidentate Zinc Chelators for α-Carbonic Anhydrases that Produce a Trigonal Bipyramidal Coordination Geometry.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1609, doi. 10.1002/cmdc.201000200

By:

Schulze Wischeler, Johannes;
Innocenti, Alessio;
Vullo, Daniela;
Agrawal, Arpita;
Cohen, Seth M.;
Heine, Andreas;
Supuran, Claudiu T.;
Klebe, Gerhard

Publication type:

Article

Cover Picture: Ease of Synthesis, Controllable Sizes, and In Vivo Large-Animal-Lymph Migration of Polymeric Nanoparticles (ChemMedChem 9/2010).

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1405, doi. 10.1002/cmdc.201090036

By:

Zubris, Kimberly Ann V.;
Khullar, Onkar V.;
Griset, Aaron P.;
Gibbs-Strauss, Summer;
Frangioni, John V.;
Colson, Yolonda L.;
Grinstaff, Mark W.

Publication type:

Article

Erythroid Induction of Chronic Myelogenous Leukemia K562 Cells Following Treatment with a Photoproduct Derived from the UV-A Irradiation of 5-Methoxypsoralen.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1506, doi. 10.1002/cmdc.201000204

By:

Salvador, Alessia;
Dall'Acqua, Stefano;
Sardo, Manlio Sutera;
Caffieri, Sergio;
Vedaldi, Daniela;
Dall'Acqua, Francesco;
Borgatti, Monica;
Zuccato, Cristina;
Bianchi, Nicoletta;
Gambari, Roberto

Publication type:

Article

Ease of Synthesis, Controllable Sizes, and In Vivo Large-Animal-Lymph Migration of Polymeric Nanoparticles.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1435, doi. 10.1002/cmdc.201000250

By:

Zubris, Kimberly Ann V.;
Khullar, Onkar V.;
Griset, Aaron P.;
Gibbs-Strauss, Summer;
Frangioni, John V.;
Colson, Yolonda L.;
Grinstaff, Mark W.

Publication type:

Article

Discovery Process and Characterization of Novel Carbohydrazide Derivatives as Potent and Selective GHSR1a Antagonists.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1450, doi. 10.1002/cmdc.201000185

By:

Sabbatini, Fabio Maria;
Di Fabio, Romano;
Corsi, Mauro;
Cavanni, Paolo;
Bromidge, Steve M.;
St-Denis, Yves;
D'Adamo, Lucilla;
Contini, Stefania;
Rinaldi, Marilisa;
Guery, Sebastien;
Savoia, Chiara;
Mundi, Claudia;
Perini, Benedetta;
Carpenter, Andrew J.;
Dal Forno, Giovanna;
Faggioni, Federico;
Tessari, Michela;
Pavone, Francesca;
Di Francesco, Carla;
Buson, Alberto

Publication type:

Article

Novel Peptidyl Aryl Vinyl Sulfones as Highly Potent and Selective Inhibitors of Cathepsins L and B.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1556, doi. 10.1002/cmdc.201000109

By:

Mendieta, Laura;
Picó, Anna;
Tarragó, Teresa;
Teixidó, Meritxell;
Castillo, Marcos;
Rafecas, Llorenç;
Moyano, Albert;
Giralt, Ernest

Publication type:

Article

Corrigendum: Pentalysine β-Carbonylphthalocyanine Zinc: An Effective Tumor-Targeting Photosensitizer for Photodynamic Therapy.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1414, doi. 10.1002/cmdc.201090042

By:

Chen, Zhuo;
Zhou, Shanyong;
Chen, Jincan;
Deng, Yicai;
Luo, Zhipu;
Chen, Hongwei;
Hamblin, Michael R.;
Huang, Mingdong

Publication type:

Article

Design, Synthesis, and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1616, doi. 10.1002/cmdc.201000210

By:

Pisani, Leonardo;
Catto, Marco;
Giangreco, Ilenia;
Leonetti, Francesco;
Nicolotti, Orazio;
Stefanachi, Angela;
Cellamare, Saverio;
Carotti, Angelo

Publication type:

Article

Synthesis, Cytotoxicity, and Insight into the Mode of Action of Re(CO)<sub>3</sub> Thymidine Complexes.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1513, doi. 10.1002/cmdc.201000196

By:

Bartholomä, Mark D.;
Vortherms, Anthony R.;
Hillier, Shawn;
Ploier, Birgit;
Joyal, John;
Babich, John;
Doyle, Robert P.;
Zubieta, Jon

Publication type:

Article

Bicyclic Derivatives of the Potent Dual Aromatase-Steroid Sulfatase Inhibitor 2-Bromo-4-{[(4-cyanophenyl)(4 H-1,2,4-triazol-4-yl)amino]methyl}phenylsulfamate: Synthesis, SAR, Crystal Structure, and in vitro and in vivo Activities.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1577, doi. 10.1002/cmdc.201000203

By:

Wood, Paul M.;
Woo, L. W. Lawrence;
Labrosse, Jean-Robert;
Thomas, Mark P.;
Mahon, Mary F.;
Chander, Surinder K.;
Purohit, Atul;
Reed, Michael J.;
Potter, Barry V. L.

Publication type:

Article

Probing the Peptidylglycine α-Hydroxylating Monooxygenase Active Site with Novel 4-Phenyl-3-butenoic Acid Based Inhibitors.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1568, doi. 10.1002/cmdc.201000214

By:

Langella, Emma;
Pierre, Sébastien;
Ghattas, Wadih;
Giorgi, Michel;
Réglier, Marius;
Saviano, Michele;
Esposito, Luciana;
Hardré, Renaud

Publication type:

Article

Corrigendum: Cover Picture: Discovery of a Class of Diketopiperazines as Antiprion Compounds (ChemMedChem 8/2010).

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1414, doi. 10.1002/cmdc.201090039

By:

Bolognesi, Maria Laura;
Ai Tran, Hoang Ngoc;
Staderini, Matteo;
Monaco, Alessandra;
López-Cobeñas, Alberto;
Bongarzone, Salvatore;
Biarnés, Xevi;
López-Alvarado, Pilar;
Cabezas, Nieves;
Caramelli, Maria;
Carloni, Paolo;
Menéndez, J. Carlos;
Legname, Giuseppe

Publication type:

Article

Novel 3-Carboxy- and 3-Phosphonopyrazoline Amino Acids as Potent and Selective NMDA Receptor Antagonists: Design, Synthesis, and Pharmacological Characterization.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1465, doi. 10.1002/cmdc.201000184

By:

Conti, Paola;
Pinto, Andrea;
Tamborini, Lucia;
Madsen, Ulf;
Nielsen, Birgitte;
Bräuner-Osborne, Hans;
Hansen, Kasper B.;
Landucci, Elisa;
Pellegrini-Giampietro, Domenico E.;
De Sarro, Giovambattista;
Donato Di Paola, Eugenio;
De Micheli, Carlo

Publication type:

Article

Preview: ChemMedChem 10/2010.

Published in:: ChemMedChem, 2010, v. 5, n. 9, p. 1635, doi. 10.1002/cmdc.201090041
Publication type:: Article

Praziquantel and Schistosomiasis.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1420, doi. 10.1002/cmdc.201000202

By:

Dömling, Alexander;
Khoury, Kareem

Publication type:

Article

Graphical Abstract: ChemMedChem 9/2010.

Published in:: ChemMedChem, 2010, v. 5, n. 9, p. 1407, doi. 10.1002/cmdc.201090038
Publication type:: Article

Discovery of 1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(2-(4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)- N-(piperidin-1-yl)-1 H-pyrazole-3-carboxamide as a Potential Peripheral Cannabinoid-1 Receptor Inverse Agonist.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1439, doi. 10.1002/cmdc.201000246

By:

Hung, Ming-Shiu;
Chang, Chun-Ping;
Li, Ting-Chieh;
Yeh, Teng-Kuang;
Song, Jen-Shin;
Lin, Yinchiu;
Wu, Chien-Huang;
Kuo, Po-Chu;
Amancha, Prashanth K.;
Wong, Ying-Chieh;
Hsiao, Wen-Chi;
Chao, Yu-Sheng;
Shia, Kak-Shan

Publication type:

Article

Improved 2,4-Diarylthiazole-Based Antiprion Agents: Switching the Sense of the Amide Group at C5 Leads to an Increase in Potency.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1476, doi. 10.1002/cmdc.201000217

By:

Thompson, Mark J.;
Louth, Jennifer C.;
Greenwood, Gemma K.;
Sorrell, Fiona J.;
Knight, Sandra G.;
Adams, Nathan B. P.;
Chen, Beining

Publication type:

Article

New Anacardic Acid-Inspired Benzamides: Histone Lysine Acetyltransferase Activators.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1530, doi. 10.1002/cmdc.201000158

By:

Souto, José A.;
Benedetti, Rosaria;
Otto, Katharina;
Miceli, Marco;
Álvarez, Rosana;
Altucci, Lucia;
de Lera, Angel R.

Publication type:

Article

Multitarget Drugs: Synthesis and Preliminary Pharmacological Characterization of Zileuton Analogues Endowed with Dual 5-LO Inhibitor and NO-Dependent Activities.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1444, doi. 10.1002/cmdc.201000198

By:

Boschi, Donatella;
Giorgis, Marta;
Cena, Clara;
Talniya, Naveen Chandra;
Di Stilo, Antonella;
Morini, Giuseppina;
Coruzzi, Gabriella;
Guaita, Elena;
Fruttero, Roberta;
Gasco, Alberto

Publication type:

Article

Synthesis of Anti-Microtubule N-(2-Arylindol-7-yl)benzenesulfonamide Derivatives and Their Antitumor Mechanisms.

Published in:

ChemMedChem, 2010, v. 5, n. 9, p. 1489, doi. 10.1002/cmdc.201000228

By:

Chiou, Chun-Tang;
Chen, Grace Shiahuy;
Chen, Meng-Ling;
Li, Huoming;
Shi, Lei;
Huang, Xiang-Hong;
Dai, Wei-Ming;
Chern, Ji-Wang

Publication type:

Article