Works matching IS 18607179 AND DT 2010 AND VI 5 AND IP 11

Results: 24

Inhibition of HIV-1 Entry: Multiple Keys to Close the Door.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1825, doi. 10.1002/cmdc.201000292
By:
- Hertje, Maria;
- Zhou, Mingkui;
- Dietrich, Ursula
Publication type:
Article
Towards the Discovery of New Hypnotic Agents: Synthesis and Preliminary Pharmacological Evaluation of a Novel Class of Dibenzo[ a, d]cycloheptene Derivatives.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1843, doi. 10.1002/cmdc.201000280
By:
- Castiglioni, Emiliano;
- Di Fabio, Romano;
- Togninelli, Andrea;
- Brough, Stephen;
- Brown, Fiona;
- Cin, Michele Dal;
- Gianotti, Massimo;
- Marchioro, Carla;
- Merlo, Giancarlo;
- Spinosa, Raffaella;
- Wigglesworth, Mark J.;
- Botta, Maurizio
Publication type:
Article
Toward the First Nonpeptidic Molecular Tong Inhibitor of Wild-Type and Mutated HIV-1 Protease Dimerization.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1899, doi. 10.1002/cmdc.201000308
By:
- Vidu, Anamaria;
- Dufau, Laure;
- Bannwarth, Ludovic;
- Soulier, Jean-Louis;
- Sicsic, Sames;
- Piarulli, Umberto;
- Reboud-Ravaux, Michèle;
- Ongeri, Sandrine
Publication type:
Article
Development of Peptide and Small-Molecule HIV-1 Fusion Inhibitors that Target gp41.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1813, doi. 10.1002/cmdc.201000289
By:
- Cai, Lifeng;
- Jiang, Shibo
Publication type:
Article
Enzyme Inhibition in Drug Discovery and Development: The Good and the Bad. Edited by Chuang Lu and Albert P. Li.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1949, doi. 10.1002/cmdc.201000315
By:
- Costi, Maria Paola
Publication type:
Article
Hypoxia-Selective Growth Inhibition of Cancer Cells by Furospinosulin-1, a Furanosesterterpene Isolated from an Indonesian Marine Sponge.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1919, doi. 10.1002/cmdc.201000302
By:
- Arai, Masayoshi;
- Kawachi, Takashi;
- Setiawan, Andi;
- Kobayashi, Motomasa
Publication type:
Article
Fusion Intermediates of HIV-1 gp41 as Targets for Antibody Production: Design, Synthesis, and HR1-HR2 Complex Purification and Characterization of Generated Antibodies.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1907, doi. 10.1002/cmdc.201000313
By:
- Mzoughi, Olfa;
- Gaston, Fabrice;
- Granados, Giovana C.;
- Lakhdar-Ghazal, Faouzi;
- Giralt, Ernest;
- Bahraoui, Elmostafa
Publication type:
Article
Preview: ChemMedChem 12/2010.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1955, doi. 10.1002/cmdc.201090053
Publication type:
Article
Synthesis of Imidazothiazole-Chalcone Derivatives as Anticancer and Apoptosis Inducing Agents.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1937, doi. 10.1002/cmdc.201000346
By:
- Kamal, Ahmed;
- Dastagiri, D.;
- Ramaiah, M. Janaki;
- Reddy, J. Surendranadha;
- Bharathi, E. Vijaya;
- Srinivas, Chatla;
- Pushpavalli, S. N. C. V. L.;
- Pal, Dhananjaya;
- Pal-Bhadra, Manika
Publication type:
Article
Feeding the Antimalarial Pipeline.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1837, doi. 10.1002/cmdc.201000341
By:
- Schlitzer, Martin;
- Ortmann, Regina
Publication type:
Article
Synthesis, In Vitro and In Vivo Release Kinetics, and Anti-HIV Activity of A Sustained-Release Prodrug (mPEG-AZT) of 3′-Azido-3′-deoxythymidine (AZT, Zidovudine).
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1893, doi. 10.1002/cmdc.201000352
By:
- Li, Wenjun;
- Chang, Yu;
- Zhan, Peng;
- Zhang, Na;
- Liu, Xinyong;
- Pannecouque, Christophe;
- De Clercq, Erik
Publication type:
Article
Spotlights on our sister journals: ChemMedChem 11/2010.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1810, doi. 10.1002/cmdc.201090052
Publication type:
Article
A Turning Point in The Fight against HIV.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1799, doi. 10.1002/cmdc.201000338
By:
- Williams, Scott D.
Publication type:
Article
Cover Picture: Probing Multidrug-Resistance and Protein-Ligand Interactions with Oxatricyclic Designed Ligands in HIV-1 Protease Inhibitors (ChemMedChem 11/2010).
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1797, doi. 10.1002/cmdc.201090049
By:
- Ghosh, Arun K.;
- Xu, Chun-Xiao;
- Rao, Kalapala Venkateswara;
- Baldridge, Abigail;
- Agniswamy, Johnson;
- Wang, Yuan-Fang;
- Weber, Irene T.;
- Aoki, Manabu;
- Miguel, Salcedo Gomez Pedro;
- Amano, Masayuki;
- Mitsuya, Hiroaki
Publication type:
Article
Graphical Abstract: ChemMedChem 11/2010.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1804, doi. 10.1002/cmdc.201090051
Publication type:
Article
Novel Huprine Derivatives with Inhibitory Activity toward β-Amyloid Aggregation and Formation as Disease-Modifying Anti-Alzheimer Drug Candidates.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1855, doi. 10.1002/cmdc.201000322
By:
- Viayna, Elisabet;
- Gómez, Tània;
- Galdeano, Carles;
- Ramírez, Lorena;
- Ratia, Míriam;
- Badia, Albert;
- Clos, M. Victòria;
- Verdaguer, Ester;
- Junyent, Félix;
- Camins, Antoni;
- Pallàs, Mercè;
- Bartolini, Manuela;
- Mancini, Francesca;
- Andrisano, Vincenza;
- Arce, Mariana P.;
- Rodríguez-Franco, María Isabel;
- Bidon-Chanal, Axel;
- Luque, F. Javier;
- Camps, Pelayo;
- Muñoz-Torrero, Diego
Publication type:
Article
Phosphoramidate Prodrugs Deliver with Potency Against Hepatitis C Virus.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1841, doi. 10.1002/cmdc.201000310
By:
- Mehellou, Youcef
Publication type:
Article
Inside Cover: Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives (ChemMedChem 11/2010).
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1798, doi. 10.1002/cmdc.201090050
By:
- Tabarrini, Oriana;
- Massari, Serena;
- Daelemans, Dirk;
- Meschini, Francesco;
- Manfroni, Giuseppe;
- Bottega, Laura;
- Gatto, Barbara;
- Palumbo, Manlio;
- Pannecouque, Christophe;
- Cecchetti, Violetta
Publication type:
Article
Target Profiling of a Small Library of Phosphodiesterase 5 (PDE5) Inhibitors using Chemical Proteomics.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1927, doi. 10.1002/cmdc.201000303
By:
- Raijmakers, Reinout;
- Dadvar, Poupak;
- Pelletier, Sarah;
- Gouw, Joost;
- Rumpel, Klaus;
- Heck, Albert J. R.
Publication type:
Article
Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1880, doi. 10.1002/cmdc.201000267
By:
- Tabarrini, Oriana;
- Massari, Serena;
- Daelemans, Dirk;
- Meschini, Francesco;
- Manfroni, Giuseppe;
- Bottega, Laura;
- Gatto, Barbara;
- Palumbo, Manlio;
- Pannecouque, Christophe;
- Cecchetti, Violetta
Publication type:
Article
The Active Core in a Triazole Peptide Dual-Site Antagonist of HIV-1 gp120.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1871, doi. 10.1002/cmdc.201000222
By:
- Umashankara, Muddegowda;
- McFadden, Karyn;
- Zentner, Isaac;
- Schön, Arne;
- Rajagopal, Srivats;
- Tuzer, Ferit;
- Kuriakose, Syna A.;
- Contarino, Mark;
- LaLonde, Judith;
- Freire, Ernesto;
- Chaiken, Irwin
Publication type:
Article
Probing Multidrug-Resistance and Protein-Ligand Interactions with Oxatricyclic Designed Ligands in HIV-1 Protease Inhibitors.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1850, doi. 10.1002/cmdc.201000318
By:
- Ghosh, Arun K.;
- Xu, Chun-Xiao;
- Rao, Kalapala Venkateswara;
- Baldridge, Abigail;
- Agniswamy, Johnson;
- Wang, Yuan-Fang;
- Weber, Irene T.;
- Aoki, Manabu;
- Miguel, Salcedo Gomez Pedro;
- Amano, Masayuki;
- Mitsuya, Hiroaki
Publication type:
Article
A Novel Synthetic Route for the Anti-HIV Drug MC-1220 and its Analogues.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1847, doi. 10.1002/cmdc.201000244
By:
- Loksha, Yasser M.;
- Globisch, Daniel;
- Loddo, Roberta;
- Collu, Gabriella;
- La Colla, Paolo;
- Pedersen, Erik B.
Publication type:
Article
Targeting Protein Kinases for Cancer Therapy. By David J. Matthews and Mary E. Gerritsen.
Published in:
ChemMedChem, 2010, v. 5, n. 11, p. 1948, doi. 10.1002/cmdc.201000398
By:
- Kuhn, Daniel
Publication type:
Article