Works matching IS 18607179 AND DT 2009 AND VI 4 AND IP 9

Results: 25

Synthesis and in vitro Evaluation of Trifluoroethylamine Analogues of Enkephalins.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1416, doi. 10.1002/cmdc.200900158

By:

Sinisi, Roberta;
Ghilardi, Alessandra;
Ruiu, Stefania;
Lazzari, Paolo;
Malpezzi, Luciana;
Sani, Monica;
Pani, Luca;
Zanda, Matteo

Publication type:

Article

Design, Synthesis, and SAR of Naphthyl-Substituted Diarylpyrimidines as Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1537, doi. 10.1002/cmdc.200900212

By:

Liang, Yong-Hong;
Feng, Xiao-Qing;
Zeng, Zhao-Sen;
Chen, Fen-Er;
Balzarini, Jan;
Pannecouque, Christophe;
De Clercq, Erik

Publication type:

Article

Preview: ChemMedChem 10/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 9, p. 1551, doi. 10.1002/cmdc.200990045
Publication type:: Article

MS Binding Assays-with MALDI toward High Throughput.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1523, doi. 10.1002/cmdc.200900201

By:

Höfner, Georg;
Merkel, Dietrich;
Wanner, Klaus Theodor

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 9/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 9, p. 1396, doi. 10.1002/cmdc.200990044
Publication type:: Article

Cover Picture: Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability / A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo (ChemMedChem 9/2009)

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1385, doi. 10.1002/cmdc.200990041

By:

Vacondio, Federica;
Silva, Claudia;
Lodola, Alessio;
Fioni, Alessandro;
Rivara, Silvia;
Duranti, Andrea;
Tontini, Andrea;
Sanchini, Silvano;
Clapper, Jason R.;
Piomelli, Daniele;
Mor, Marco;
Tarzia, Giorgio;
King, Alvin R.

Publication type:

Article

Chemoinformatics Approaches to Virtual Screening. Edited by Alexandre Varnek and Alexander Tropsha.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1546, doi. 10.1002/cmdc.200900223

By:

Wegscheid-Gerlach, Christof

Publication type:

Article

Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1495, doi. 10.1002/cmdc.200900120

By:

Vacondio, Federica;
Silva, Claudia;
Lodola, Alessio;
Fioni, Alessandro;
Rivara, Silvia;
Duranti, Andrea;
Tontini, Andrea;
Sanchini, Silvano;
Clapper, Jason R.;
Piomelli, Daniele;
Mor, Marco;
Tarzia, Giorgio

Publication type:

Article

A Consistent Dataset of Kinetic Solubilities for Early-Phase Drug Discovery.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1529, doi. 10.1002/cmdc.200900205

By:

Kramer, Christian;
Heinisch, Tilmann;
Fligge, Thilo;
Beck, Bernd;
Clark, Timothy

Publication type:

Article

Structure-Based and in silico Design of Hsp90 Inhibitors.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1399, doi. 10.1002/cmdc.200900256

By:

Sgobba, Miriam;
Rastelli, Giulio

Publication type:

Article

Inhibition of Human Leukocyte Elastase by Brunsvicamides A-C: Cyanobacterial Cyclic Peptides.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1425, doi. 10.1002/cmdc.200900139

By:

Sisay, Mihiret T.;
Hautmann, Stephanie;
Mehner, Christian;
König, Gabriele M.;
Bajorath, Jürgen;
Gütschow, Michael

Publication type:

Article

Docking Studies of Structurally Diverse Antimalarial Drugs Targeting PfATP6: No Correlation between in silico Binding Affinity and in vitro Antimalarial Activity.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1469, doi. 10.1002/cmdc.200900200

By:

Garah, Fatima Bousejra-El;
Stigliani, Jean-Luc;
Coslédan, Frédéric;
Meunier, Bernard;
Robert, Anne

Publication type:

Article

Graphical Abstract: ChemMedChem 9/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 9, p. 1387, doi. 10.1002/cmdc.200990043
Publication type:: Article

Systematic Extraction of Structure-Activity Relationship Information from Biological Screening Data.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1431, doi. 10.1002/cmdc.200900222

By:

Wawer, Mathias;
Bajorath, Jürgen

Publication type:

Article

Discovery of Ligands for the Human Intestinal Di-/Tripeptide Transporter (hPEPT1) Using a QSAR-Assisted Virtual Screening Strategy.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1439, doi. 10.1002/cmdc.200900145

By:

Larsen, Simon Birksø;
Omkvist, Diana Højmark;
Brodin, Birger;
Nielsen, Carsten Uhd;
Steffansen, Bente;
Olsen, Lars;
Jørgensen, Flemming Steen

Publication type:

Article

Pyrrole-Based Hydroxamates and 2-Aminoanilides: Histone Deacetylase Inhibition and Cellular Activities.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1411, doi. 10.1002/cmdc.200900082

By:

Valente, Sergio;
Conte, Mariarosaria;
Tardugno, Maria;
Massa, Silvio;
Nebbioso, Angela;
Altucci, Lucia;
Mai, Antonello

Publication type:

Article

Synthesis, Crystal Structure and Immunosuppressive Activity of Acylamide Derivatives Containing 1,4-Benzodioxan.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1421, doi. 10.1002/cmdc.200900167

By:

Lv, Peng-Cheng;
Wang, Kai-Rui;
Mao, Wen-Jun;
Xiong, Jing;
Li, Huan-Qiu;
Yang, Ying;
Shi, Lei;
Zhu, Hai-Liang

Publication type:

Article

Indoloquinolizidine-Peptide Hybrids as Multiple Agonists for D1 and D2 Dopamine Receptors.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1514, doi. 10.1002/cmdc.200900149

By:

Vendrell, Marc;
Soriano, Aroa;
Casadó, Vicent;
Díaz, José Luis;
Lavilla, Rodolfo;
Canela, Enric I.;
Lluís, Carme;
Franco, Rafael;
Albericio, Fernando;
Royo, Miriam

Publication type:

Article

Inside Cover: Docking Studies of Structurally Diverse Antimalarial Drugs Targeting PfATP6: No Correlation between in silico Binding Affinity and in vitro Antimalarial Activity. (ChemMedChem 9/2009).

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1386, doi. 10.1002/cmdc.200990042

By:

Garah, Fatima Bousejra-El;
Stigliani, Jean-Luc;
Coslédan, Frédéric;
Meunier, Bernard;
Robert, Anne

Publication type:

Article

A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1505, doi. 10.1002/cmdc.200900210

By:

Clapper, Jason R.;
Vacondio, Federica;
King, Alvin R.;
Duranti, Andrea;
Tontini, Andrea;
Silva, Claudia;
Sanchini, Silvano;
Tarzia, Giorgio;
Mor, Marco;
Piomelli, Daniele

Publication type:

Article

Drugs: From Discovery to Approval (2nd ed.). By Rick Ng.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1546, doi. 10.1002/cmdc.200900232

By:

Müller, Klaus

Publication type:

Article

Synthesis and Evaluation of New Antagonists of Bacterial Quorum Sensing in Vibrio harveyi.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1457, doi. 10.1002/cmdc.200900180

By:

Peng, Hanjing;
Cheng, Yunfeng;
Ni, Nanting;
Li, Minyong;
Choudhary, Gaurav;
Chou, Han Ting;
Lu, Chung-Dar;
Tai, Phang C.;
Wang, Binghe

Publication type:

Article

Retro-Enantio N-Methylated Peptides as β-Amyloid Aggregation Inhibitors.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1488, doi. 10.1002/cmdc.200900191

By:

Grillo-Bosch, Dolors;
Carulla, Natàlia;
Cruz, Montse;
Sánchez, Laia;
Pujol-Pina, Rosa;
Madurga, Sergio;
Rabanal, Francesc;
Giralt, Ernest

Publication type:

Article

Induced-Fit Docking Approach Provides Insight into the Binding Mode and Mechanism of Action of HIV-1 Integrase Inhibitors.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1446, doi. 10.1002/cmdc.200900166

By:

Barreca, Maria Letizia;
Iraci, Nunzio;
De Luca, Laura;
Chimirri, Alba

Publication type:

Article

Ex vivo and in vivo Evaluation of [18F]PR04.MZ in Rodents: A Selective Dopamine Transporter Imaging Agent.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1480, doi. 10.1002/cmdc.200900177

By:

Riss, Patrick J.;
Debus, Fabian;
Hummerich, René;
Schmidt, Ulrich;
Schloss, Patrick;
Lueddens, Hartmut;
Roesch, Frank

Publication type:

Article

Works matching IS 18607179 AND DT 2009 AND VI 4 AND IP 9

Synthesis and in vitro Evaluation of Trifluoroethylamine Analogues of Enkephalins.

Design, Synthesis, and SAR of Naphthyl-Substituted Diarylpyrimidines as Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase.

Preview: ChemMedChem 10/2009.

MS Binding Assays-with MALDI toward High Throughput.

Spotlights on our sister journals: ChemMedChem 9/2009.

Cover Picture: Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability / A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo (ChemMedChem 9/2009)

Chemoinformatics Approaches to Virtual Screening. Edited by Alexandre Varnek and Alexander Tropsha.

Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability.

A Consistent Dataset of Kinetic Solubilities for Early-Phase Drug Discovery.

Structure-Based and in silico Design of Hsp90 Inhibitors.

Inhibition of Human Leukocyte Elastase by Brunsvicamides A-C: Cyanobacterial Cyclic Peptides.

Docking Studies of Structurally Diverse Antimalarial Drugs Targeting PfATP6: No Correlation between in silico Binding Affinity and in vitro Antimalarial Activity.

Graphical Abstract: ChemMedChem 9/2009.

Systematic Extraction of Structure-Activity Relationship Information from Biological Screening Data.

Discovery of Ligands for the Human Intestinal Di-/Tripeptide Transporter (hPEPT1) Using a QSAR-Assisted Virtual Screening Strategy.

Pyrrole-Based Hydroxamates and 2-Aminoanilides: Histone Deacetylase Inhibition and Cellular Activities.

Synthesis, Crystal Structure and Immunosuppressive Activity of Acylamide Derivatives Containing 1,4-Benzodioxan.

Indoloquinolizidine-Peptide Hybrids as Multiple Agonists for D<sub>1</sub> and D<sub>2</sub> Dopamine Receptors.

Inside Cover: Docking Studies of Structurally Diverse Antimalarial Drugs Targeting PfATP6: No Correlation between in silico Binding Affinity and in vitro Antimalarial Activity. (ChemMedChem 9/2009).

A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo.

Drugs: From Discovery to Approval (2nd ed.). By Rick Ng.

Synthesis and Evaluation of New Antagonists of Bacterial Quorum Sensing in Vibrio harveyi.

Retro-Enantio N-Methylated Peptides as β-Amyloid Aggregation Inhibitors.

Induced-Fit Docking Approach Provides Insight into the Binding Mode and Mechanism of Action of HIV-1 Integrase Inhibitors.

Ex vivo and in vivo Evaluation of [<sup>18</sup>F]PR04.MZ in Rodents: A Selective Dopamine Transporter Imaging Agent.