Works matching IS 18607179 AND DT 2009 AND VI 4 AND IP 3

Results: 26

1,3-Dioxolane-Based Ligands as Rigid Analogues of Naftopidil: Structure-Affinity/Activity Relationships at α1 and 5-HT1A Receptors.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 393, doi. 10.1002/cmdc.200800277

By:

Sorbi, Claudia;
Franchini, Silvia;
Tait, Annalisa;
Prandi, Adolfo;
Gallesi, Rossella;
Angeli, Piero;
Marucci, Gabriella;
Pirona, Lorenza;
Poggesi, Elena;
Brasili, Livio

Publication type:

Article

Cover Picture: Exploring the Implications of Vitamin B12 Conjugation to Insulin on Insulin Receptor Binding (ChemMedChem 3/2009).

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 297, doi. 10.1002/cmdc.200990010

By:

Petrus, Amanda K.;
Allis, Damian G.;
Smith, Robert P.;
Fairchild, Timothy J.;
Doyle, Robert P.

Publication type:

Article

Unsaturated Mannich Bases Active Against Multidrug-Resistant Trypanosoma brucei brucei Strains.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 339, doi. 10.1002/cmdc.200800360

By:

Wenzel, I. Nicole;
Wong, Pui E.;
Maes, Louis;
Müller, Thomas J. J.;
Krauth-Siegel, R. Luise;
Barrett, Michael P.;
Davioud-Charvet, Elisabeth

Publication type:

Article

Recent Approaches to Antifungal Therapy for Invasive Mycoses.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 310, doi. 10.1002/cmdc.200800353

By:

Mathew, Bijoy P.;
Nath, Mahendra

Publication type:

Article

Preview: ChemMedChem 4/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 3, p. 479, doi. 10.1002/cmdc.200990014
Publication type:: Article

Synthesis, SAR, and Biological Evaluation of α-Sulfonylphosphonic Acids as Selective Matrix Metalloproteinase Inhibitors.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 352, doi. 10.1002/cmdc.200800324

By:

Rubino, Maria Teresa;
Agamennone, Mariangela;
Campestre, Cristina;
Fracchiolla, Giuseppe;
Laghezza, Antonio;
Loiodice, Fulvio;
Nuti, Elisa;
Rossello, Armando;
Tortorella, Paolo

Publication type:

Article

In Silico Screening for PTPN22 Inhibitors: Active Hits from an Inactive Phosphatase Conformation.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 440, doi. 10.1002/cmdc.200800375

By:

Wu, Shuangding;
Bottini, Massimo;
Rickert, Robert C.;
Mustelin, Tomas;
Tautz, Lutz

Publication type:

Article

Exploring the Implications of Vitamin B12 Conjugation to Insulin on Insulin Receptor Binding.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 421, doi. 10.1002/cmdc.200800346

By:

Petrus, Amanda K.;
Allis, Damian G.;
Smith, Robert P.;
Fairchild, Timothy J.;
Doyle, Robert P.

Publication type:

Article

DNA Binding Ellipticine Analogues: Synthesis, Biological Evaluation, and Structure-Activity Relationships.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 363, doi. 10.1002/cmdc.200800368

By:

Ferlin, Maria Grazia;
Marzano, Christine;
Gandin, Valentina;
Dall'Acqua, Stefano;
Dalla Via, Lisa

Publication type:

Article

Cytotoxicities and Structure-Activity Relationships of Natural and Unnatural Lamellarins toward Cancer Cell Lines.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 457, doi. 10.1002/cmdc.200800339

By:

Chittchang, Montakarn;
Batsomboon, Paratchata;
Ruchirawat, Somsak;
Ploypradith, Poonsakdi

Publication type:

Article

Efficient Synthesis of Highly Active Phospha-Isosteres of the Influenza Neuraminidase Inhibitor Oseltamivir.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 335, doi. 10.1002/cmdc.200800379

By:

Carbain, Benoit;
Collins, Patrick J.;
Callum, Lori;
Martin, Stephen R.;
Hay, Alan J.;
McCauley, John;
Streicher, Hansjörg

Publication type:

Article

Systems Biological Approaches in Infectious Diseases. Edited by Helen I. Boshoff and Clifton E. Barry, III.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 473, doi. 10.1002/cmdc.200900039

By:

Chan, Christina;
Wang, Xuewei

Publication type:

Article

Synthesis, Chiral Resolution and Pharmacological Evaluation of a 2,3-Benzodiazepine-Derived Noncompetitive AMPA Receptor Antagonist.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 415, doi. 10.1002/cmdc.200800341

By:

Calabrò, Maria Luisa;
Raneri, Daniela;
Ficarra, Paola;
Mennini, Tiziana;
Colleoni, Simona;
Grazioso, Giovanni;
Micale, Nicola;
Zappalà, Maria;
Grasso, Silvana

Publication type:

Article

High-Throughput Analysis in the Pharmaceutical Industry. Edited by Perry G. Wang.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 474, doi. 10.1002/cmdc.200900001

By:

Kyranos, James N.

Publication type:

Article

SHOP: A Method For Structure-Based Fragment and Scaffold Hopping.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 427, doi. 10.1002/cmdc.200800355

By:

Fontaine, Fabien;
Cross, Simon;
Plasencia, Guillem;
Pastor, Manuel;
Zamora, Ismael

Publication type:

Article

Concerning Cytochromes P450: Role in the Metabolism and Toxicity of Drugs and other Xenobiotics . Edited by Costas Ioannides.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 473, doi. 10.1002/cmdc.200900005

By:

Ingelman-Sundberg, Magnus

Publication type:

Article

Glycosylated Neurotensin Analogues Exhibit Sub-picomolar Anticonvulsant Potency in a Pharmacoresistant Model of Epilepsy.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 400, doi. 10.1002/cmdc.200800421

By:

Lee, Hee-Kyoung;
Zhang, Liuyin;
Smith, Misty D.;
White, H. Steve;
Bulaj, Grzegorz

Publication type:

Article

Graphical Abstract: ChemMedChem 3/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 3, p. 299, doi. 10.1002/cmdc.200990012
Publication type:: Article

Spotlights on our sister journals: ChemMedChem 3/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 3, p. 308, doi. 10.1002/cmdc.200990013
Publication type:: Article

The Azulene Framework as a Novel Arene Bioisostere: Design of Potent Dopamine D4 Receptor Ligands Inducing Penile Erection.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 325, doi. 10.1002/cmdc.200800395

By:

Löber, Stefan;
Tschammer, Nuska;
Hübner, Harald;
Melis, Maria Rosaria;
Argiolas, Antonio;
Gmeiner, Peter

Publication type:

Article

Structurally Minimized μ-Conotoxin Analogues as Sodium Channel Blockers: Implications for Designing Conopeptide-Based Therapeutics.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 406, doi. 10.1002/cmdc.200800292

By:

Han, Tiffany S.;
Zhang, Min-Min;
Walewska, Aleksandra;
Gruszczynski, Pawel;
Robertson, Charles R.;
Cheatham, Thomas E.;
Yoshikami, Doju;
Olivera, Baldomero M.;
Bulaj, Grzegorz

Publication type:

Article

The Synthesis and in vivo Evaluation of 2′,2′-Difluoro KRN7000.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 329, doi. 10.1002/cmdc.200800348

By:

Leung, Leo;
Tomassi, Cyrille;
Van Beneden, Katrien;
Decruy, Tine;
Trappeniers, Matthias;
Elewaut, Dirk;
Gao, Yifang;
Elliott, Tim;
Al-Shamkhani, Aymen;
Ottensmeier, Christian;
Werner, Jörn M.;
Williams, Anthony;
Van Calenbergh, Serge;
Linclau, Bruno

Publication type:

Article

Characterization of New PPARγ Agonists: Analysis of Telmisartan's Structural Components.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 445, doi. 10.1002/cmdc.200800285

By:

Goebel, Matthias;
Clemenz, Markus;
Staels, Bart;
Unger, Thomas;
Kintscher, Ulrich;
Gust, Ronald

Publication type:

Article

Design, Synthesis, and Biological Evaluation of Enantiomeric β- N-Acetylhexosaminidase Inhibitors LABNAc and DABNAc as Potential Agents against Tay-Sachs and Sandhoff Disease.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 378, doi. 10.1002/cmdc.200800350

By:

Rountree, J. S. Shane;
Butters, Terry D.;
Wormald, Mark R.;
Boomkamp, Stephanie D.;
Dwek, Raymond A.;
Asano, Naoki;
Ikeda, Kyoko;
Evinson, Emma L.;
Nash, Robert J.;
Fleet, George W. J.

Publication type:

Article

Inside Cover: Cytotoxicities and Structure-Activity Relationships of Natural and Unnatural Lamellarins toward Cancer Cell Lines (ChemMedChem 3/2009).

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 298, doi. 10.1002/cmdc.200990011

By:

Chittchang, Montakarn;
Batsomboon, Paratchata;
Ruchirawat, Somsak;
Ploypradith, Poonsakdi

Publication type:

Article

Fluorescent Benzofurazan-Cholic Acid Conjugates for in vitro Assessment of Bile Acid Uptake and Its Modulation by Drugs.

Published in:

ChemMedChem, 2009, v. 4, n. 3, p. 466, doi. 10.1002/cmdc.200800383

By:

Rohacova, Jana;
Marín, M. Luisa;
Martinez-Romero, Alicia;
Diaz, Laura;
O'Connor, José-Enrique;
Gomez-Lechon, M. Jose;
Donato, M. Teresa;
Castell, José V.;
Miranda, Miguel A.

Publication type:

Article

Works matching IS 18607179 AND DT 2009 AND VI 4 AND IP 3

1,3-Dioxolane-Based Ligands as Rigid Analogues of Naftopidil: Structure-Affinity/Activity Relationships at α<sub>1</sub> and 5-HT<sub>1A</sub> Receptors.

Cover Picture: Exploring the Implications of Vitamin B<sub>12</sub> Conjugation to Insulin on Insulin Receptor Binding (ChemMedChem 3/2009).

Unsaturated Mannich Bases Active Against Multidrug-Resistant Trypanosoma brucei brucei Strains.

Recent Approaches to Antifungal Therapy for Invasive Mycoses.

Preview: ChemMedChem 4/2009.

Synthesis, SAR, and Biological Evaluation of α-Sulfonylphosphonic Acids as Selective Matrix Metalloproteinase Inhibitors.

In Silico Screening for PTPN22 Inhibitors: Active Hits from an Inactive Phosphatase Conformation.

Exploring the Implications of Vitamin B<sub>12</sub> Conjugation to Insulin on Insulin Receptor Binding.

DNA Binding Ellipticine Analogues: Synthesis, Biological Evaluation, and Structure-Activity Relationships.

Cytotoxicities and Structure-Activity Relationships of Natural and Unnatural Lamellarins toward Cancer Cell Lines.

Efficient Synthesis of Highly Active Phospha-Isosteres of the Influenza Neuraminidase Inhibitor Oseltamivir.

Systems Biological Approaches in Infectious Diseases. Edited by Helen I. Boshoff and Clifton E. Barry, III.

Synthesis, Chiral Resolution and Pharmacological Evaluation of a 2,3-Benzodiazepine-Derived Noncompetitive AMPA Receptor Antagonist.

High-Throughput Analysis in the Pharmaceutical Industry. Edited by Perry G. Wang.

SHOP: A Method For Structure-Based Fragment and Scaffold Hopping.

Concerning Cytochromes P450: Role in the Metabolism and Toxicity of Drugs and other Xenobiotics . Edited by Costas Ioannides.

Glycosylated Neurotensin Analogues Exhibit Sub-picomolar Anticonvulsant Potency in a Pharmacoresistant Model of Epilepsy.

Graphical Abstract: ChemMedChem 3/2009.

Spotlights on our sister journals: ChemMedChem 3/2009.

The Azulene Framework as a Novel Arene Bioisostere: Design of Potent Dopamine D4 Receptor Ligands Inducing Penile Erection.

Structurally Minimized μ-Conotoxin Analogues as Sodium Channel Blockers: Implications for Designing Conopeptide-Based Therapeutics.

The Synthesis and in vivo Evaluation of 2′,2′-Difluoro KRN7000.

Characterization of New PPARγ Agonists: Analysis of Telmisartan's Structural Components.

Design, Synthesis, and Biological Evaluation of Enantiomeric β- N-Acetylhexosaminidase Inhibitors LABNAc and DABNAc as Potential Agents against Tay-Sachs and Sandhoff Disease.

Inside Cover: Cytotoxicities and Structure-Activity Relationships of Natural and Unnatural Lamellarins toward Cancer Cell Lines (ChemMedChem 3/2009).

Fluorescent Benzofurazan-Cholic Acid Conjugates for in vitro Assessment of Bile Acid Uptake and Its Modulation by Drugs.