Works matching IS 18607179 AND DT 2009 AND VI 4 AND IP 11

Results: 27

4,4-Dimethyl- and Diastereomeric 4-Hydroxy-4-methyl- (2 S)-Glutamate Analogues Display Distinct Pharmacological Profiles at Ionotropic Glutamate Receptors and Excitatory Amino Acid Transporters.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1925, doi. 10.1002/cmdc.200900258

By:

Bunch, Lennart;
Pickering, Darryl S.;
Gefflaut, Thierry;
Vinatier, Virginie;
Helaine, Virgil;
Amir, Ahmad;
Nielsen, Birgitte;
Jensen, Anders A.

Publication type:

Article

Cancer Proteomics: From Bench to Bedside. Edited by Sayed S. Daoud.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1950, doi. 10.1002/cmdc.200900298

By:

Prokai, Laszlo

Publication type:

Article

Inside Cover: From Structure-Activity to Structure-Selectivity Relationships: Quantitative Assessment, Selectivity Cliffs, and Key Compounds (ChemMedChem 11/2009).

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1766, doi. 10.1002/cmdc.200990052

By:

Peltason, Lisa;
Hu, Ye;
Bajorath, Jürgen

Publication type:

Article

2-Acylaminopyridin-4-ylimidazoles as p38 MAP Kinase Inhibitors: Design, Synthesis, and Biological and Metabolic Evaluations.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1939, doi. 10.1002/cmdc.200900242

By:

Ziegler, Katharina;
Hauser, Dominik R. J.;
Unger, Anke;
Albrecht, Wolfgang;
Laufer, Stefan A.

Publication type:

Article

Combined Pharmacophore Modeling, Docking, and 3D QSAR Studies of ABCB1 and ABCC1 Transporter Inhibitors.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1883, doi. 10.1002/cmdc.200900282

By:

Pajeva, Ilza K.;
Globisch, Christoph;
Wiese, Michael

Publication type:

Article

Identification and Validation of a Potent Type II Inhibitor of Inactive Polo-like Kinase 1.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1806, doi. 10.1002/cmdc.200900338

By:

Keppner, Sarah;
Proschak, Ewgenij;
Schneider, Gisbert;
Spänkuch, Birgit

Publication type:

Article

The Cannabinoid Receptors. Edited by Patricia H. Reggio.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1949, doi. 10.1002/cmdc.200900286

By:

Selwood, David

Publication type:

Article

Synthesis and Pharmacological Characterization of Disila-AM80 (Disila-tamibarotene) and Disila-AM580, Silicon Analogues of the RARα-Selective Retinoid Agonists AM80 (Tamibarotene) and AM580.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1797, doi. 10.1002/cmdc.200900257

By:

Tacke, Reinhold;
Müller, Volker;
Büttner, Matthias W.;
Lippert, W. Peter;
Bertermann, Rüdiger;
Daiß, Jürgen O.;
Khanwalkar, Harshal;
Furst, Audrey;
Gaudon, Claudine;
Gronemeyer, Hinrich

Publication type:

Article

From Structure-Activity to Structure-Selectivity Relationships: Quantitative Assessment, Selectivity Cliffs, and Key Compounds.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1864, doi. 10.1002/cmdc.200900300

By:

Peltason, Lisa;
Hu, Ye;
Bajorath, Jürgen

Publication type:

Article

Cover Picture: Classification of Organic Molecules by Molecular Quantum Numbers (ChemMedChem 11/2009).

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1765, doi. 10.1002/cmdc.200990051

By:

Nguyen, Kong T.;
Blum, Lorenz C.;
van Deursen, Ruud;
Reymond, Jean-Louis

Publication type:

Article

High-Speed Microwave-Assisted Synthesis of the Trifluoromethylpyrazol-Derived Canonical Transient Receptor Potential (TRPC) Channel Inhibitor Pyr3.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1816, doi. 10.1002/cmdc.200900304

By:

Glasnov, Toma N.;
Groschner, Klaus;
Kappe, C. Oliver

Publication type:

Article

Chemical and Structural Biology to Direct the Repurposing of Sulindac.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1793, doi. 10.1002/cmdc.200900384

By:

Simard, Jeffrey R.;
Rauh, Daniel

Publication type:

Article

Preview: ChemMedChem 12/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 11, p. 1955, doi. 10.1002/cmdc.200990055
Publication type:: Article

Studies on the Synthesis and Activity of Three Tripalladium Complexes Containing Planaramine Ligands.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1841, doi. 10.1002/cmdc.200900267

By:

Farhad, Mohammad;
Yu, Jun Qing;
Beale, Philip;
Fisher, Keith;
Huq, Fazlul

Publication type:

Article

Aryloxy Phosphoramidate Triesters: a Technology for Delivering Monophosphorylated Nucleosides and Sugars into Cells.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1779, doi. 10.1002/cmdc.200900289

By:

Mehellou, Youcef;
Balzarini, Jan;
McGuigan, Christopher

Publication type:

Article

The Roles of 3′ and 4′ Hydroxy Groups in α-Galactosylceramide Stimulation of Invariant Natural Killer T Cells.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1810, doi. 10.1002/cmdc.200900350

By:

Xia, Chengfeng;
Zhang, Wenpeng;
Zhang, Yalong;
Chen, Wenlan;
Nadas, Janos;
Severin, Ryan;
Woodward, Robert;
Wang, Bin;
Wang, Xin;
Kronenberg, Mitchell;
Wang, Peng G.

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 11/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 11, p. 1776, doi. 10.1002/cmdc.200990054
Publication type:: Article

Synthesis and Evaluation of Imidazo[2,1- b]thiazoles as Iodide Efflux Inhibitors in Thyrocytes.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1819, doi. 10.1002/cmdc.200900365

By:

Lecat-Guillet, Nathalie;
Ambroise, Yves

Publication type:

Article

Synthesis and Biological Evaluation of Chromium Bioorganometallics Based on the Antibiotic Platensimycin Lead Structure.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1930, doi. 10.1002/cmdc.200900347

By:

Patra, Malay;
Gasser, Gilles;
Pinto, Antonio;
Merz, Klaus;
Ott, Ingo;
Bandow, Julia E.;
Metzler-Nolte, Nils

Publication type:

Article

3,5-Bis(benzylidene)-4-oxo-1-phosphonopiperidines and Related Diethyl Esters: Potent Cytotoxins with Multi-Drug-Resistance Reverting Properties.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1831, doi. 10.1002/cmdc.200900288

By:

Das, Swagatika;
Das, Umashankar;
Selvakumar, Ponniah;
Sharma, Rajendra K.;
Balzarini, Jan;
De Clercq, Erik;
Molnár, Joseph;
Serly, Julianna;
Baráth, Zoltán;
Schatte, Gabriele;
Bandy, Brian;
Gorecki, Dennis K. J.;
Dimmock, Jonathan R.

Publication type:

Article

Structural Model for the Binding Sites of Allosterically Potentiating Ligands on Nicotinic Acetylcholine Receptors.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1874, doi. 10.1002/cmdc.200900320

By:

Luttmann, Edgar;
Ludwig, Jürgen;
Höffle-Maas, Anja;
Samochocki, Marek;
Maelicke, Alfred;
Fels, Gregor

Publication type:

Article

Graphical Abstract: ChemMedChem 11/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 11, p. 1767, doi. 10.1002/cmdc.200990053
Publication type:: Article

Synthesis, Biological Evaluation of 1,1-Diarylethylenes as a Novel Class of Antimitotic Agents.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1912, doi. 10.1002/cmdc.200900290

By:

Hamze, Abdallah;
Giraud, Anne;
Messaoudi, Samir;
Provot, Olivier;
Peyrat, Jean-François;
Bignon, Jérôme;
Liu, Jian-Miao;
Wdzieczak-Bakala, Joanna;
Thoret, Sylviane;
Dubois, Joëlle;
Brion, Jean-Daniel;
Alami, Mouad

Publication type:

Article

Synthesis of Modified 4 H-1,2,4-Benzothiadiazine-1,1-dioxides and Determination of their Affinity and Selectivity for Different Types of K<sub>ATP</sub> Channels.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1850, doi. 10.1002/cmdc.200900261

By:

Lachenicht, Stefan;
Fischer, Andreas;
Schmidt, Claas;
Winkler, Marcus;
Rood, Achim;
Lemoine, Horst;
Braun, Manfred

Publication type:

Article

Classification of Organic Molecules by Molecular Quantum Numbers.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1803, doi. 10.1002/cmdc.200900317

By:

Nguyen, Kong T.;
Blum, Lorenz C.;
van Deursen, Ruud;
Reymond, Jean-Louis

Publication type:

Article

Molecular Fingerprint Recombination: Generating Hybrid Fingerprints for Similarity Searching from Different Fingerprint Types.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1859, doi. 10.1002/cmdc.200900243

By:

Nisius, Britta;
Bajorath, Jürgen

Publication type:

Article

Activators of P-glycoprotein: Structure-Activity Relationships and Investigation of their Mode of Action.

Published in:

ChemMedChem, 2009, v. 4, n. 11, p. 1897, doi. 10.1002/cmdc.200900283

By:

Sterz, Katja;
Möllmann, Lars;
Jacobs, Anna;
Baumert, Dieter;
Wiese, Michael

Publication type:

Article