Works matching IS 18607179 AND DT 2008 AND VI 3 AND IP 6

Results: 23

Discovery of a Drug-Like G-Quadruplex Binding Ligand by High-Throughput Docking.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 881, doi. 10.1002/cmdc.200700342

By:

Ma, Dik-Lung;
Lai, Tat-Shing;
Chan, Fung-Yi;
Chung, Wai-Hong;
Abagyan, R.;
Leung, Yun-Chung;
Wong, Kwok-Yin

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 6/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 6, p. 858, doi. 10.1002/cmdc.200890025
Publication type:: Article

Conformationally Restricted Hydantoin-Based Peptidomimetics as Inhibitors of Caspase-3 with Basic Groups Allowed at the S3 Enzyme Subsite.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 979, doi. 10.1002/cmdc.200800020

By:

Vázquez, Jesús;
García-Jareño, Alicia;
Mondragón, Laura;
Rubio-Martinez, Jaime;
Pérez-Payá, Enrique;
Albericio, Fernando

Publication type:

Article

Graphical Abstract: ChemMedChem 6/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 6, p. 851, doi. 10.1002/cmdc.200890024
Publication type:: Article

Herceptin-Platinum(II) Binding Complexes: Novel Cancer-Cell-Specific Agents.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 954, doi. 10.1002/cmdc.200700349

By:

Gao, Jian;
Liu, Ya Guang;
Liu, Renbin;
Zingaro, Ralph A.

Publication type:

Article

Molecular Recognition of Small-Cell Lung Cancer Cells Using Aptamers.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 991, doi. 10.1002/cmdc.200800030

By:

Chen, Hui William;
Medley, Colin D.;
Sefah, Kwame;
Shangguan, Dihua;
Tang, Zhiwen;
Meng, Ling;
Smith, Josh E.;
Tan, Weihong

Publication type:

Article

Prodrugs: Challenges and Rewards. Parts 1 and 2. Edited by Valentino J. Stella, Ronald T. Borchardt, Michael J. Hageman, Reza Oliyai, Hans Maag, and Jefferson W. Tilley.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 1003, doi. 10.1002/cmdc.200800115

By:

Kubinyi, Hugo

Publication type:

Article

Dipeptide Derivatives of AZT: Synthesis, Chemical Stability, Activation in Human Plasma, hPEPT1 Affinity, and Antiviral Activity.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 970, doi. 10.1002/cmdc.200800012

By:

Santos, Cledir;
Morais, José;
Gouveia, Luís;
de Clercq, Erik;
Pannecouque, Christophe;
Nielsen, Carsten Uhd;
Steffansen, Bente;
Moreira, Rui;
Gomes, Paula

Publication type:

Article

Drug Discovery Research: New Frontiers in the Post-Genomic Era. Edited by Ziwei Huang.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 1003, doi. 10.1002/cmdc.200800016

By:

Barton, William A.

Publication type:

Article

Cover Picture: Herceptin-Platinum(II) Binding Complexes: Novel Cancer-Cell-Specific Agents (ChemMedChem 6/2008).

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 849, doi. 10.1002/cmdc.200890023

By:

Gao, Jian;
Liu, Ya Guang;
Liu, Renbin;
Zingaro, Ralph A.

Publication type:

Article

A Combinatorial Approach to 2,4,6-Trisubstituted Triazines with Potent Antimalarial Activity: Combining Conventional Synthesis and Microwave-Assistance.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 873, doi. 10.1002/cmdc.200700344

By:

Melato, Sergio;
Prosperi, Davide;
Coghi, Paolo;
Basilico, Nicoletta;
Monti, Diego

Publication type:

Article

Substituted Pyrazolo[3,4- b]pyridines as Potent A1 Adenosine Antagonists: Synthesis, Biological Evaluation, and Development of an A1 Bovine Receptor Model.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 898, doi. 10.1002/cmdc.200700355

By:

Tuccinardi, Tiziano;
Schenone, Silvia;
Bondavalli, Francesco;
Brullo, Chiara;
Bruno, Olga;
Mosti, Luisa;
Zizzari, Alessandra Tania;
Tintori, Cristina;
Manetti, Fabrizio;
Ciampi, Osele;
Trincavelli, Maria Letizia;
Martini, Claudia;
Martinelli, Adriano;
Botta, Maurizio

Publication type:

Article

Discovery of VHR Phosphatase Inhibitors with Micromolar Activity based on Structure-Based Virtual Screening.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 877, doi. 10.1002/cmdc.200700348

By:

Park, Hwangseo;
Jung, Suk-Kyeong;
Jeong, Dae Gwin;
Ryu, Seong Eon;
Kim, Seung Jun

Publication type:

Article

Towards an Integrated Description of Hydrogen Bonding and Dehydration: Decreasing False Positives in Virtual Screening with the HYDE Scoring Function.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 885, doi. 10.1002/cmdc.200700319

By:

Reulecke, Ingo;
Lange, Gudrun;
Albrecht, Jürgen;
Klein, Robert;
Rarey, Matthias

Publication type:

Article

Inhibitors of Inducible NO Synthase Expression: Total Synthesis of ( S)-Curvularin and Its Ring Homologues.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 924, doi. 10.1002/cmdc.200800022

By:

Elzner, Stephan;
Schmidt, Denise;
Schollmeyer, Dieter;
Erkel, Gerhard;
Anke, Timm;
Kleinert, Hartmut;
Förstermann, Ulrich;
Kunz, Horst

Publication type:

Article

The Art of Drug Synthesis. Edited by Douglas S. Johnson and Jie Jack Li.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 1002, doi. 10.1002/cmdc.200800015

By:

Peukert, Stefan;
Radetich, Branko

Publication type:

Article

Naphthoxazepine Inhibitors of HIV-1 Integrase: Synthesis and Biological Evaluation.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 986, doi. 10.1002/cmdc.200800026

By:

Garofalo, Antonio;
Grande, Fedora;
Brizzi, Antonella;
Aiello, Francesca;
Dayam, Raveendra;
Neamati, Nouri

Publication type:

Article

Investigating Amine Derivatives of Ambruticin VS-5 and VS-4.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 963, doi. 10.1002/cmdc.200800008

By:

Tian, Zong-Qiang;
Wang, Zhan;
Xu, Yuan;
Tran, Chau Q.;
Myles, David C.;
Zhong, Ziyang;
Simmons, Jessica;
Vetcher, Leandro;
Katz, Leonard;
Li, Yong;
Shaw, Simon J.

Publication type:

Article

Preview: ChemMedChem 7/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 6, p. 1006, doi. 10.1002/cmdc.200890022
Publication type:: Article

Synthesis and Biological Activity of a Novel Inhibitor of Dihydroceramide Desaturase.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 946, doi. 10.1002/cmdc.200700325

By:

Munoz-Olaya, Jose M.;
Matabosch, Xavier;
Bedia, Carmen;
Egido-Gabás, Meritxell;
Casas, Josefina;
Llebaria, Amadeu;
Delgado, Antonio;
Fabriàs, Gemma

Publication type:

Article

Towards Small-Molecule CXCR3 Ligands with Clinical Potential.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 861, doi. 10.1002/cmdc.200700365

By:

Wijtmans, Maikel;
Verzijl, Dennis;
Leurs, Rob;
de Esch, Iwan J. P.;
Smit, Martine J.

Publication type:

Article

Targeted RNA Interference of Cyclin A2 Mediated by Functionalized Single-Walled Carbon Nanotubes Induces Proliferation Arrest and Apoptosis in Chronic Myelogenous Leukemia K562 Cells.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 940, doi. 10.1002/cmdc.200700329

By:

Wang, Xiaohui;
Ren, Jinsong;
Qu, Xiaogang

Publication type:

Article

On the Way to Selective PARP-2 Inhibitors. Design, Synthesis, and Preliminary Evaluation of a Series of Isoquinolinone Derivatives.

Published in:

ChemMedChem, 2008, v. 3, n. 6, p. 914, doi. 10.1002/cmdc.200800010

By:

Pellicciari, Roberto;
Camaioni, Emidio;
Costantino, Gabriele;
Formentini, Laura;
Sabbatini, Paola;
Venturoni, Francesco;
Eren, Gökçen;
Bellocchi, Daniele;
Chiarugi, Alberto;
Moroni, Flavio

Publication type:

Article

Works matching IS 18607179 AND DT 2008 AND VI 3 AND IP 6

Discovery of a Drug-Like G-Quadruplex Binding Ligand by High-Throughput Docking.

Spotlights on our sister journals: ChemMedChem 6/2008.

Conformationally Restricted Hydantoin-Based Peptidomimetics as Inhibitors of Caspase-3 with Basic Groups Allowed at the S<sub>3</sub> Enzyme Subsite.

Graphical Abstract: ChemMedChem 6/2008.

Herceptin-Platinum(II) Binding Complexes: Novel Cancer-Cell-Specific Agents.

Molecular Recognition of Small-Cell Lung Cancer Cells Using Aptamers.

Prodrugs: Challenges and Rewards. Parts 1 and 2. Edited by Valentino J. Stella, Ronald T. Borchardt, Michael J. Hageman, Reza Oliyai, Hans Maag, and Jefferson W. Tilley.

Dipeptide Derivatives of AZT: Synthesis, Chemical Stability, Activation in Human Plasma, hPEPT1 Affinity, and Antiviral Activity.

Drug Discovery Research: New Frontiers in the Post-Genomic Era. Edited by Ziwei Huang.

Cover Picture: Herceptin-Platinum(II) Binding Complexes: Novel Cancer-Cell-Specific Agents (ChemMedChem 6/2008).

A Combinatorial Approach to 2,4,6-Trisubstituted Triazines with Potent Antimalarial Activity: Combining Conventional Synthesis and Microwave-Assistance.

Substituted Pyrazolo[3,4- b]pyridines as Potent A<sub>1</sub> Adenosine Antagonists: Synthesis, Biological Evaluation, and Development of an A<sub>1</sub> Bovine Receptor Model.

Discovery of VHR Phosphatase Inhibitors with Micromolar Activity based on Structure-Based Virtual Screening.

Towards an Integrated Description of Hydrogen Bonding and Dehydration: Decreasing False Positives in Virtual Screening with the HYDE Scoring Function.

Inhibitors of Inducible NO Synthase Expression: Total Synthesis of ( S)-Curvularin and Its Ring Homologues.

The Art of Drug Synthesis. Edited by Douglas S. Johnson and Jie Jack Li.

Naphthoxazepine Inhibitors of HIV-1 Integrase: Synthesis and Biological Evaluation.

Investigating Amine Derivatives of Ambruticin VS-5 and VS-4.

Preview: ChemMedChem 7/2008.

Synthesis and Biological Activity of a Novel Inhibitor of Dihydroceramide Desaturase.

Towards Small-Molecule CXCR3 Ligands with Clinical Potential.

Targeted RNA Interference of Cyclin A<sub>2</sub> Mediated by Functionalized Single-Walled Carbon Nanotubes Induces Proliferation Arrest and Apoptosis in Chronic Myelogenous Leukemia K562 Cells.

On the Way to Selective PARP-2 Inhibitors. Design, Synthesis, and Preliminary Evaluation of a Series of Isoquinolinone Derivatives.