Works matching IS 18607179 AND DT 2008 AND VI 3 AND IP 5

Results: 22

Carba-nucleosides as Potent Antagonists of the Adenosine 5′-Diphosphate (ADP) Purinergic Receptor (P2Y12) on Human Platelets.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 732, doi. 10.1002/cmdc.200700310

By:

Ye, Hong;
Chen, Cailin;
Zhang, Han-Cheng;
Haertlein, Barbara;
Parry, Tom J.;
Damiano, Bruce P.;
Maryanoff, Bruce E.

Publication type:

Article

A Dual Selective Antitumor Agent and Fluorescence Probe: the Binary BMVC-Porphyrin Photosensitizer.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 725, doi. 10.1002/cmdc.200700336

By:

Kang, Chi-Chih;
Chen, Chin-Tin;
Cho, Chih-Chien;
Lin, Yu-Chen;
Chang, Cheng-Chung;
Chang, Ta-Chau

Publication type:

Article

Competitive Inhibitors of Helicobacter pylori Type II Dehydroquinase: Synthesis, Biological Evaluation, and NMR Studies.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 756, doi. 10.1002/cmdc.200700307

By:

Sánchez-Sixto, Cristina;
Prazeres, Verónica F. V.;
Castedo, Luis;
Suh, Se Won;
Lamb, Heather;
Hawkins, Alastair R.;
Cañada, Francisco Javier;
Jiménez-Barbero, Jesús;
González-Bello, Concepción

Publication type:

Article

Graphical Abstract: ChemMedChem 5/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 5, p. 679, doi. 10.1002/cmdc.200890019
Publication type:: Article

A Study of the Binding Energies of Efavirenz to Wild-Type and K103N/Y181C HIV-1 Reverse Transcriptase Based on the ONIOM Method.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 803, doi. 10.1002/cmdc.200700181

By:

Srivab, Pensri;
Hannongbua, Supa

Publication type:

Article

Preview: ChemMedChem 6/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 5, p. 846, doi. 10.1002/cmdc.200890021
Publication type:: Article

Oxali-Titanocene Y: A Potent Anticancer Drug.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 729, doi. 10.1002/cmdc.200700302

By:

Claffey, James;
Hogan, Megan;
Müller-Bunz, Helge;
Pampillón, Clara;
Tacke, Matthias

Publication type:

Article

The First Potent Subtype-Selective Retinoid X Receptor (RXR) Agonist Possessing a 3-Isopropoxy-4-isopropylphenylamino Moiety, NEt-3IP (RXRα/β-dual agonist).

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 780, doi. 10.1002/cmdc.200700313

By:

Takamatsu, Kayo;
Takano, Atsushi;
Yakushiji, Nobumasa;
Morohashi, Kazunori;
Morishita, Ken-ichi;
Matsuura, Nobuyasu;
Makishima, Makoto;
Tai, Akihiro;
Sasaki, Kenji;
Kakuta, Hiroki

Publication type:

Article

pH Effects on the Conformational Preferences of Amyloid β-Peptide (1-40) in HFIP Aqueous Solution by NMR Spectroscopy.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 833, doi. 10.1002/cmdc.200700324

By:

Valerio, Mariacristina;
Porcelli, Fernando;
Zbilut, Joseph P.;
Giuliani, Alessandro;
Manetti, Cesare;
Conti, Filippo

Publication type:

Article

Zinc-Binding Groups Modulate Selective Inhibition of MMPs.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 812, doi. 10.1002/cmdc.200700290

By:

Agrawal, Arpita;
Romero-Perez, Diego;
Jacobsen, Jennifer A.;
Villarreal, Francisco J.;
Cohen, Seth M.

Publication type:

Article

Rapid Identification of a Putative Interaction between β2-Adrenoreceptor Agonists and ATF4 using a Chemical Genomics Approach.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 742, doi. 10.1002/cmdc.200700317

By:

Ladwa, Sweta R.;
Dilly, Suzanne J.;
Clark, Andrew J.;
Marsh, Andrew;
Taylor, Paul C.

Publication type:

Article

Cover Picture: Rapid Identification of a Putative Interaction between β2-Adrenoreceptor Agonists and ATF4 using a Chemical Genomics Approach (ChemMedChem 5/2008).

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 677, doi. 10.1002/cmdc.200890018

By:

Ladwa, Sweta R.;
Dilly, Suzanne J.;
Clark, Andrew J.;
Marsh, Andrew;
Taylor, Paul C.

Publication type:

Article

Development of Pyrrolo[2,1- c][1,4]benzodiazepine β-Galactoside Prodrugs for Selective Therapy of Cancer by ADEPT and PMT.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 794, doi. 10.1002/cmdc.200700328

By:

Kamal, Ahmed;
Tekumalla, Venkatesh;
Krishnan, Anita;
Pal-Bhadra, Manika;
Bhadra, Utpal

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 5/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 5, p. 686, doi. 10.1002/cmdc.200890020
Publication type:: Article

SyGMa: Combining Expert Knowledge and Empirical Scoring in the Prediction of Metabolites.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 821, doi. 10.1002/cmdc.200700312

By:

Ridder, Lars;
Wagener, Markus

Publication type:

Article

Click Chemistry and Medicinal Chemistry: A Case of 'Cyclo- Addiction'.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 715, doi. 10.1002/cmdc.200700334

By:

Moorhouse, A. D.;
Moses, J. E.

Publication type:

Article

18F-Labeled FAUC 346 and BP 897 Derivatives as Subtype-Selective Potential PET Radioligands for the Dopamine D3 Receptor.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 788, doi. 10.1002/cmdc.200700327

By:

Hocke, Carsten;
Prante, Olaf;
Salama, Ismael;
Hübner, Harald;
Löber, Stefan;
Kuwert, Torsten;
Gmeiner, Peter

Publication type:

Article

Inhibition of HIV-1 by a Peptide Ligand of the Genomic RNA Packaging Signal Ψ.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 749, doi. 10.1002/cmdc.200700194

By:

Dietz, Julia;
Koch, Joachim;
Kaur, Ajit;
Raja, Chinnappan;
Stein, Stefan;
Grez, Manuel;
Pustowka, Anette;
Mensch, Sarah;
Ferner, Jan;
Möller, Lars;
Bannert, Norbert;
Tampé, Robert;
Divita, Gilles;
Mély, Yves;
Schwalbe, Harald;
Dietrich, Ursula

Publication type:

Article

G-Quadruplexes: Targets in Anticancer Drug Design.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 690, doi. 10.1002/cmdc.200700300

By:

Ou, Tian-miao;
Lu, Yu-jing;
Tan, Jia-heng;
Huang, Zhi-shu;
Wong, Kwok-Yin;
Gu, Lian-quan

Publication type:

Article

Synthesis and Biological Evaluation of Isosteric Analogues of FK866, an Inhibitor of NAD Salvage.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 771, doi. 10.1002/cmdc.200700311

By:

Galli, Ubaldina;
Ercolano, Emanuela;
Carraro, Lorenzo;
Blasi Roman, Cintia R.;
Sorba, Giovanni;
Canonico, Pier Luigi;
Genazzani, Armando A.;
Tron, Gian Cesare;
Billington, Richard A.

Publication type:

Article

Towards a Self-Adjuvanting Multivalent B and T cell Epitope Containing Synthetic Glycolipopeptide Cancer Vaccine.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 737, doi. 10.1002/cmdc.200700315

By:

Renaudet, Olivier;
BenMohamed, Lbachir;
Dasgupta, Gargi;
Bettahi, Ilham;
Dumy, Pascal

Publication type:

Article

Synthesis of an Original Oxygenated Taxuspine X Analogue: a Versatile 'Non-Natural' Natural Product with Remarkable P-gp Modulating Activity.

Published in:

ChemMedChem, 2008, v. 3, n. 5, p. 745, doi. 10.1002/cmdc.200700337

By:

Avramova, Stanislava I.;
Galletti, Elena;
Renzulli, Michela L.;
Giorgi, Gianluca;
Sgaragli, Gianpietro;
Alderighi, Daniela;
Ghiron, Chiara;
Corelli, Federico;
Radi, Marco;
Botta, Maurizio

Publication type:

Article

Works matching IS 18607179 AND DT 2008 AND VI 3 AND IP 5

Carba-nucleosides as Potent Antagonists of the Adenosine 5′-Diphosphate (ADP) Purinergic Receptor (P2Y<sub>12</sub>) on Human Platelets.

A Dual Selective Antitumor Agent and Fluorescence Probe: the Binary BMVC-Porphyrin Photosensitizer.

Competitive Inhibitors of Helicobacter pylori Type II Dehydroquinase: Synthesis, Biological Evaluation, and NMR Studies.

Graphical Abstract: ChemMedChem 5/2008.

A Study of the Binding Energies of Efavirenz to Wild-Type and K103N/Y181C HIV-1 Reverse Transcriptase Based on the ONIOM Method.

Preview: ChemMedChem 6/2008.

Oxali-Titanocene Y: A Potent Anticancer Drug.

The First Potent Subtype-Selective Retinoid X Receptor (RXR) Agonist Possessing a 3-Isopropoxy-4-isopropylphenylamino Moiety, NEt-3IP (RXRα/β-dual agonist).

pH Effects on the Conformational Preferences of Amyloid β-Peptide (1-40) in HFIP Aqueous Solution by NMR Spectroscopy.

Zinc-Binding Groups Modulate Selective Inhibition of MMPs.

Rapid Identification of a Putative Interaction between β<sub>2</sub>-Adrenoreceptor Agonists and ATF4 using a Chemical Genomics Approach.

Cover Picture: Rapid Identification of a Putative Interaction between β<sub>2</sub>-Adrenoreceptor Agonists and ATF4 using a Chemical Genomics Approach (ChemMedChem 5/2008).

Development of Pyrrolo[2,1- c][1,4]benzodiazepine β-Galactoside Prodrugs for Selective Therapy of Cancer by ADEPT and PMT.

Spotlights on our sister journals: ChemMedChem 5/2008.

SyGMa: Combining Expert Knowledge and Empirical Scoring in the Prediction of Metabolites.

Click Chemistry and Medicinal Chemistry: A Case of 'Cyclo- Addiction'.

<sup>18</sup>F-Labeled FAUC 346 and BP 897 Derivatives as Subtype-Selective Potential PET Radioligands for the Dopamine D3 Receptor.

Inhibition of HIV-1 by a Peptide Ligand of the Genomic RNA Packaging Signal Ψ.

G-Quadruplexes: Targets in Anticancer Drug Design.

Synthesis and Biological Evaluation of Isosteric Analogues of FK866, an Inhibitor of NAD Salvage.

Towards a Self-Adjuvanting Multivalent B and T cell Epitope Containing Synthetic Glycolipopeptide Cancer Vaccine.

Synthesis of an Original Oxygenated Taxuspine X Analogue: a Versatile 'Non-Natural' Natural Product with Remarkable P-gp Modulating Activity.