Works matching IS 18607179 AND DT 2008 AND VI 3 AND IP 12

Results: 23

Design and Synthesis of Potent and Selective Azaindole-Based Rho Kinase (ROCK) Inhibitors.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1893, doi. 10.1002/cmdc.200800211

By:

Schirok, Hartmut;
Kast, Raimund;
Figueroa-Pérez, Santiago;
Bennabi, Samir;
Gnoth, Mark J.;
Feurer, Achim;
Heckroth, Heike;
Thutewohl, Michael;
Paulsen, Holger;
Knorr, Andreas;
Hütter, Joachim;
Lobell, Mario;
Münter, Klaus;
Geiß, Volker;
Ehmke, Heimo;
Lang, Dieter;
Radtke, Martin;
Mittendorf, Joachim;
Stasch, Johannes-Peter

Publication type:

Article

Reduction of Alzheimer's Disease Amyloid Plaque Load in Transgenic Mice by D3, a D-Enantiomeric Peptide Identified by Mirror Image Phage Display.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1848, doi. 10.1002/cmdc.200800273

By:

van Groen, Thomas;
Wiesehan, Katja;
Funke, Susanne A.;
Kadish, Inga;
Nagel-Steger, Luitgard;
Willbold, Dieter

Publication type:

Article

Graphical Abstract: ChemMedChem 12/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 12, p. 1799, doi. 10.1002/cmdc.200890047
Publication type:: Article

Bisphosphonated Benzoxazinorifamycin Prodrugs for the Prevention and Treatment of Osteomyelitis.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1863, doi. 10.1002/cmdc.200800255

By:

Reddy, Ranga;
Dietrich, Evelyne;
Lafontaine, Yanick;
Houghton, Tom J.;
Belanger, Odette;
Dubois, Anik;
Arhin, Francis F.;
Sarmiento, Ingrid;
Fadhil, Ibtihal;
Laquerre, Karine;
Ostiguy, Valerie;
Lehoux, Dario;
Moeck, Gregory;
Parr, Thomas R.;
Rafai Far, Adel

Publication type:

Article

Norcantharidin Analogues: Synthesis, Anticancer Activity and Protein Phosphatase 1 and 2A Inhibition.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1878, doi. 10.1002/cmdc.200800192

By:

Hill, Timothy A.;
Stewart, Scott G.;
Gordon, Christopher P.;
Ackland, Stephen P.;
Gilbert, Jayne;
Sauer, Benjamin;
Sakoff, Jennette A.;
McCluskey, Adam

Publication type:

Article

Ground State, Intermediate, and Multivalent Nucleotide Analogue Inhibitors of Cytidine 5′-Triphosphate Synthase.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1853, doi. 10.1002/cmdc.200800236

By:

Taylor, Scott D.;
Lunn, Faylene A.;
Bearne, Stephen L.

Publication type:

Article

Thiobarbiturates as Sirtuin Inhibitors: Virtual Screening, Free-Energy Calculations, and Biological Testing.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1965, doi. 10.1002/cmdc.200800104

By:

Uciechowska, Urszula;
Schemies, Jörg;
Neugebauer, Robert C.;
Huda, Elisabeth-Maria;
Schmitt, Martin L.;
Meier, Rene;
Verdin, Eric;
Jung, Manfred;
Sippl, Wolfgang

Publication type:

Article

Differences in Paclitaxel and Docetaxel Interactions with Tubulin Detected by Mutagenesis of Yeast Tubulin.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1844, doi. 10.1002/cmdc.200800288

By:

Winefield, Robert D.;
Entwistle, Ruth A.;
Foland, Travis B.;
Lushington, Gerald H.;
Himes, Richard H.

Publication type:

Article

The Handbook of Nanomedicine. By Kewal K. Jain.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1977, doi. 10.1002/cmdc.200800397

By:

Amiji, Mansoor M.

Publication type:

Article

Natural-Product-Like Spiroketals and Fused Bicyclic Acetals as Potential Therapeutic Agents for B-Cell Chronic Lymphocytic Leukaemia.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1922, doi. 10.1002/cmdc.200800265

By:

Milroy, Lech-Gustav;
Zinzalla, Giovanna;
Loiseau, François;
Qian, Zizheng;
Prencipe, Giuseppe;
Pepper, Chris;
Fegan, Chris;
Ley, Steven V.

Publication type:

Article

HER-2-Targeted Nanoparticle-Affibody Bioconjugates for Cancer Therapy.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1839, doi. 10.1002/cmdc.200800122

By:

Alexis, Frank;
Basto, Pamela;
Levy-Nissenbaum, Etgar;
Radovic-Moreno, Aleksandar F.;
Zhang, Liangfang;
Pridgen, Eric;
Wang, Andrew Z.;
Marein, Shawn L.;
Westerhof, Katrina;
Molnar, Linda K.;
Farokhzad, Omid C.

Publication type:

Article

Asymmetric Synthesis and Biological Evaluation of Glycosidic Prodrugs for a Selective Cancer Therapy.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1946, doi. 10.1002/cmdc.200800250

By:

Tietze, Lutz F.;
von Hof, J. Marian;
Krewer, Birgit;
Müller, Michael;
Major, Felix;
Schuster, Heiko J.;
Schuberth, Ingrid;
Alves, Frauke

Publication type:

Article

Cover Picture: Design and Synthesis of Potent and Selective Azaindole-Based Rho Kinase (ROCK) Inhibitors (ChemMedChem 12/2008).

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1797, doi. 10.1002/cmdc.200890046

By:

Schirok, Hartmut;
Kast, Raimund;
Figueroa-Pérez, Santiago;
Bennabi, Samir;
Gnoth, Mark J.;
Feurer, Achim;
Heckroth, Heike;
Thutewohl, Michael;
Paulsen, Holger;
Knorr, Andreas;
Hütter, Joachim;
Lobell, Mario;
Münter, Klaus;
Geiß, Volker;
Ehmke, Heimo;
Lang, Dieter;
Radtke, Martin;
Mittendorf, Joachim;
Stasch, Johannes-Peter

Publication type:

Article

Novel Acyl Phosphate Mimics that Target PlsY, an Essential Acyltransferase in Gram-Positive Bacteria.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1936, doi. 10.1002/cmdc.200800218

By:

Grimes, Kimberly D.;
Lu, Ying-Jie;
Zhang, Yong-Mei;
Luna, Vicki A.;
Hurdle, Julian G.;
Carson, Elizabeth I.;
Qi, Jianjun;
Kudrimoti, Sucheta;
Rock, Charles O.;
Lee, Richard E.

Publication type:

Article

Modeling of the Intestinal Peptide Transporter hPepT1 and Analysis of Its Transport Capacities by Docking and Pharmacophore Mapping.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1913, doi. 10.1002/cmdc.200800184

By:

Pedretti, Alessandro;
De Luca, Laura;
Marconi, Cristina;
Negrisoli, Gianpaolo;
Aldini, Giancarlo;
Vistoli, Giulio

Publication type:

Article

Small-Molecule Inhibitors of PDK1.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1810, doi. 10.1002/cmdc.200800195

By:

Peifer, Christian;
Alessi, Dario R.

Publication type:

Article

Dopamides, Vanillylamides, Ethanolamides, and Arachidonic Acid Amides of Anti-inflammatory and Analgesic Drug Substances as TRPV1 Ligands.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1956, doi. 10.1002/cmdc.200800271

By:

Sinning, Christian;
Watzer, Bernhard;
De Petrocellis, Luciano;
Di Marzo, Vincenzo;
Imming, Peter

Publication type:

Article

Preview: ChemMedChem 1/2009.

Published in:: ChemMedChem, 2008, v. 3, n. 12, p. 1980, doi. 10.1002/cmdc.200890049
Publication type:: Article

Three-Dimensional Database Mining Identifies a Unique Chemotype that Unites Structurally Diverse Botulinum Neurotoxin Serotype A Inhibitors in a Three-Zone Pharmacophore.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1905, doi. 10.1002/cmdc.200800241

By:

Hermone, Ann R.;
Burnett, James C.;
Nuss, Jonathan E.;
Tressler, Lyal E.;
Nguyen, Tam L.;
Šolaja, Bogdan A.;
Vennerstrom, Jonathan L.;
Schmidt, James J.;
Wipf, Peter;
Bavari, Sina;
Gussio, Rick

Publication type:

Article

Index 2008.

Published in:: ChemMedChem, 2008, v. 3, n. 12, p. 1981, doi. 10.1002/cmdc.200812345
Publication type:: Article

Efficient Cellular Labeling by CD44 Receptor-Mediated Uptake of Cationic Liposomes Functionalized with Hyaluronic Acid and Loaded with MRI Contrast Agents.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1858, doi. 10.1002/cmdc.200800234

By:

Esposito, Giovanna;
Geninatti Crich, Simonetta;
Aime, Silvio

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 12/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 12, p. 1808, doi. 10.1002/cmdc.200890048
Publication type:: Article

Hemisuccinate of 21-Hydroxy-6,19-Epoxyprogesterone: A Tissue-Specific Modulator of the Glucocorticoid Receptor.

Published in:

ChemMedChem, 2008, v. 3, n. 12, p. 1869, doi. 10.1002/cmdc.200800256

By:

Álvarez, Lautaro D.;
Martí, Marcelo A.;
Veleiro, Adriana S.;
Misico, Rosana I.;
Estrin, Darío A.;
Pecci, Adalí;
Burton, Gerardo

Publication type:

Article