Works matching IS 18607179 AND DT 2008 AND VI 3 AND IP 10

Results: 22

Spotlights on our sister journals: ChemMedChem 10/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 10, p. 1474, doi. 10.1002/cmdc.200890040
Publication type:: Article

Structure-Based Optimization of Protein Tyrosine Phosphatase-1 B Inhibitors: Capturing Interactions with Arginine 24.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1525, doi. 10.1002/cmdc.200800188

By:

Wan, Zhao-Kui;
Lee, Jinbo;
Hotchandani, Rajeev;
Moretto, Alessandro;
Binnun, Eva;
Wilson, Douglas P.;
Kirincich, Steve J.;
Follows, Bruce C.;
Ipek, Manus;
Xu, Weixin;
Joseph-McCarthy, Diane;
Zhang, Yan-Ling;
Tam, May;
Erbe, David V.;
Tobin, James F.;
Li, Wei;
Tam, Steve Y.;
Mansour, Tarek S.;
Wu, Junjun

Publication type:

Article

Integrating Structure- and Ligand-Based Virtual Screening: Comparison of Individual, Parallel, and Fused Molecular Docking and Similarity Search Calculations on Multiple Targets.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1566, doi. 10.1002/cmdc.200800129

By:

Tan, Lu;
Geppert, Hanna;
Sisay, Mihiret T.;
Gütschow, Michael;
Bajorath, Jürgen

Publication type:

Article

Preview: ChemMedChem 11/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 10, p. 1618, doi. 10.1002/cmdc.200890041
Publication type:: Article

Apoptosis-Inducing High <sup>.</sup>NO Concentrations Are Not Sustained Either in Nascent or in Developed Cancers.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1493, doi. 10.1002/cmdc.200800257

By:

Heller, Adam

Publication type:

Article

Biomedical Potentials of Crown Ethers: Prospective Antitumor Agents.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1478, doi. 10.1002/cmdc.200800118

By:

Kralj, Marijeta;
Tušek-Božić, Ljerka;
Frkanec, Leo

Publication type:

Article

Discovery of NMDA Glycine Site Inhibitors from the Chemical Universe Database GDB.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1520, doi. 10.1002/cmdc.200800198

By:

Nguyen, Kong Thong;
Syed, Salahuddin;
Urwyler, Stephan;
Bertrand, Sonia;
Bertrand, Daniel;
Reymond, Jean-Louis

Publication type:

Article

Cover Picture: Computational Studies to Discover a New NR2B/NMDA Receptor Antagonist and Evaluation of Pharmacological Profile (ChemMedChem 10/2008).

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1465, doi. 10.1002/cmdc.200890038

By:

Gitto, Rosaria;
De Luca, Laura;
Ferro, Stefania;
Occhiuto, Francesco;
Samperi, Stefania;
De Sarro, Giovanbattista;
Russo, Emilio;
Ciranna, Lucia;
Costa, Lara;
Chimirri, Alba

Publication type:

Article

A Potent Integrin Antagonist from a Small Library of Cyclic RGD Pentapeptide Mimics Including Benzyl-Substituted Azabicycloalkane Amino Acids.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1589, doi. 10.1002/cmdc.200800143

By:

Arosio, Daniela;
Belvisi, Laura;
Colombo, Lino;
Colombo, Matteo;
Invernizzi, Donatella;
Manzoni, Leonardo;
Potenza, Donatella;
Serra, Massimo;
Castorina, Massimo;
Pisano, Claudio;
Scolastico, Carlo

Publication type:

Article

Anti-Inflammatory Activity of a New Class of Nitric Oxide Synthase Inhibitors That Release Nitric Oxide.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1580, doi. 10.1002/cmdc.200800201

By:

Botta, Maurizio;
Distrutti, Eleonora;
Mencarelli, Andrea;
Parlato, Maria Cristina;
Raffi, Francesco;
Cipriani, Sabrina;
Fiorucci, Stefano

Publication type:

Article

Synthesis, Antiproliferative Evaluation, and Structure-Activity Relationships of 3-Arylquinolines.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1516, doi. 10.1002/cmdc.200800160

By:

Xiao, Zhu-Ping;
Lv, Peng-cheng;
Xu, Suo-Ping;
Zhu, Tao-Tao;
Zhu, Hai-Liang

Publication type:

Article

Scaffold-Hopping Cascade Yields Potent Inhibitors of 5-Lipoxygenase.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1535, doi. 10.1002/cmdc.200800153

By:

Hofmann, Bettina;
Franke, Lutz;
Proschak, Ewgenij;
Tanrikulu, Yusuf;
Schneider, Petra;
Steinhilber, Dieter;
Schneider, Gisbert

Publication type:

Article

Computational Studies to Discover a New NR2B/NMDA Receptor Antagonist and Evaluation of Pharmacological Profile.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1539, doi. 10.1002/cmdc.200800124

By:

Gitto, Rosaria;
De Luca, Laura;
Ferro, Stefania;
Occhiuto, Francesco;
Samperi, Stefania;
De Sarro, Giovanbattista;
Russo, Emilio;
Ciranna, Lucia;
Costa, Lara;
Chimirri, Alba

Publication type:

Article

Discovery of Water-Soluble Antioxidant Flavonols without Vasorelaxant Activity.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1572, doi. 10.1002/cmdc.200800146

By:

Yap, Suwan;
Loft, Karen J.;
Woodman, Owen L.;
Williams, Spencer J.

Publication type:

Article

Graphical Abstract: ChemMedChem 10/2008.

Published in:: ChemMedChem, 2008, v. 3, n. 10, p. 1467, doi. 10.1002/cmdc.200890039
Publication type:: Article

New DNA Polymerase IIIC Inhibitors: 3-Subtituted Anilinouracils with Potent Antibacterial Activity in vitro and in vivo.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1604, doi. 10.1002/cmdc.200800117

By:

Svenstrup, Niels;
Ehlert, Kerstin;
Ladel, Christoph;
Kuhl, Alexander;
Häbich, Dieter

Publication type:

Article

Inhibition of hERG Channel Trafficking: An Under-Explored Mechanism for Drug-Induced QT Prolongation.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1501, doi. 10.1002/cmdc.200800170

By:

Yeung, Kap-Sun;
Meanwell, Nicholas A.

Publication type:

Article

Benzimidazolium Salts as Small, Nonpeptidic and BBB-Permeable Human Prolyl Oligopeptidase Inhibitors.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1558, doi. 10.1002/cmdc.200800152

By:

Tarragó, Teresa;
Masdeu, Carme;
Gómez, Elena;
Isambert, Nicolás;
Lavilla, Rodolfo;
Giralt, Ernest

Publication type:

Article

Discovery of Novel Non-Cyclam Polynitrogenated CXCR4 Coreceptor Inhibitors.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1549, doi. 10.1002/cmdc.200800145

By:

Pettersson, Sofia;
Pérez-Nueno, Violeta I.;
Ros-Blanco, Laia;
Puig de La Bellacasa, Raimon;
Rabal, María Obdulia;
Batllori, Xavier;
Clotet, Bonaventura;
Clotet-Codina, Imma;
Armand-Ugón, Mercedes;
Esté, José;
Borrell, José I.;
Teixidó, Jordi

Publication type:

Article

On the Art of Compiling and Using 'Drug-Like' Chemical Fragment Spaces.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1503, doi. 10.1002/cmdc.200800178

By:

Degen, Jörg;
Wegscheid-Gerlach, Christof;
Zaliani, Andrea;
Rarey, Matthias

Publication type:

Article

The Discovery of Pyrano[3,4- b]indole-Based Allosteric Inhibitors of HCV NS5B Polymerase with In Vivo Activity.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1508, doi. 10.1002/cmdc.200800168

By:

LaPorte, Matthew G.;
Jackson, Randy W.;
Draper, Tandy L.;
Gaboury, Janet A.;
Galie, Kristin;
Herbertz, Torsten;
Hussey, Alison R.;
Rippin, Susan R.;
Benetatos, Christopher A.;
Chunduru, Srinivas K.;
Christensen, Joel S.;
Coburn, Glen A.;
Rizzo, Christopher J.;
Rhodes, Gerry;
O'Connell, John;
Howe, Anita Y. M.;
Mansour, Tarek S.;
Collett, Marc S.;
Pevear, Daniel C.;
Young, Dorothy C.

Publication type:

Article

α-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors.

Published in:

ChemMedChem, 2008, v. 3, n. 10, p. 1530, doi. 10.1002/cmdc.200800162

By:

Asso, Valentina;
Ghilardi, Elisa;
Bertini, Simone;
Digiacomo, Maria;
Granchi, Carlotta;
Minutolo, Filippo;
Rapposelli, Simona;
Bortolato, Andrea;
Moro, Stefano;
Macchia, Marco

Publication type:

Article