Works matching IS 18607179 AND DT 2007 AND VI 2 AND IP 7

Results: 19

Cover Picture: Design and Synthesis of 2,3,5-Substituted Imidazolidin-4-one Inhibitors of BACE-1 (ChemMedChem 7/2007).

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 909, doi. 10.1002/cmdc.200790022

By:

Barrow, James C.;
Rittle, Kenneth E.;
Ngo, Phung L.;
Selnick, Harold G.;
Graham, Samuel L.;
Pitzenberger, Steven M.;
McGaughey, Georgia B.;
Colussi, Dennis;
Lai, Ming-Tain;
Huang, Qian;
Tugusheva, Katherine;
Espeseth, Amy S.;
Simon, Adam J.;
Munshi, Sanjeev K.;
Vacca, Joseph P.

Publication type:

Article

Malaria Chemotherapeutics Part I: History of Antimalarial Drug Development, Currently Used Therapeutics, and Drugs in Clinical Development.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 944, doi. 10.1002/cmdc.200600240

By:

Schlitzer, Martin

Publication type:

Article

Apparent Asymmetry in Fingerprint Similarity Searching is a Direct Consequence of Differences in Bit Densities and Molecular Size.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1037, doi. 10.1002/cmdc.200700050

By:

Wang, Yuan;
Eckert, Hanna;
Bajorath, Jürgen

Publication type:

Article

Aminocyclitols as Pharmacological Chaperones for Glucocerebrosidase, a Defective Enzyme in Gaucher Disease.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 992, doi. 10.1002/cmdc.200700061

By:

Egido-Gabás, Meritxell;
Canals, Daniel;
Casas, Josefina;
Llebaria, Amadeu;
Delgado, Antonio

Publication type:

Article

Rational Design, Synthesis, and Evaluation of Nanomolar Type II Dehydroquinase Inhibitors.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1015, doi. 10.1002/cmdc.200700032

By:

Payne, Richard J.;
Peyrot, Fabienne;
Kerbarh, Olivier;
Abell, Andrew D.;
Abell, Chris

Publication type:

Article

7-Azamelatonin: Efficient Synthetic Routes, Excited-State Double Proton Transfer Properties and Biomedical Implications.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1071, doi. 10.1002/cmdc.200700043

By:

Wu, Pei-Wen;
Cheng, Yi-Ming;
Hsieh, Wan-Ting;
Wang, Yu-Hsiu;
Wei, Ching-Yen;
Chou, Pi-Tai

Publication type:

Article

Synthesis and Structure-Activity Relationship of Cytotoxic Marine Cyclodepsipeptide IB-01212 Analogues.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1076, doi. 10.1002/cmdc.200700025

By:

Cruz, Luis J.;
Francesch, Andres;
Cuevas, Carmen;
Albericio, Fernando

Publication type:

Article

1,2-Mannobioside Mimic: Synthesis, DC-SIGN Interaction by NMR and Docking, and Antiviral Activity.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1030, doi. 10.1002/cmdc.200700047

By:

Reina, José J.;
Sattin, Sara;
Invernizzi, Donatella;
Mari, Silvia;
Martínez-Prats, Lorena;
Tabarani, Georges;
Fieschi, Franck;
Delgado, Rafael;
Nieto, Pedro M.;
Rojo, Javier;
Bernardi, Anna

Publication type:

Article

Preview: ChemMedChem 8/2007.

Published in:: ChemMedChem, 2007, v. 2, n. 7, p. 1086, doi. 10.1002/cmdc.200790021
Publication type:: Article

Highly Potent and Selective Substrate Analogue Factor Xa Inhibitors Containing D-Homophenylalanine Analogues as P3 Residue: Part 2.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1043, doi. 10.1002/cmdc.200700031

By:

Stürzebecher, Anne;
Dönnecke, Daniel;
Schweinitz, Andrea;
Schuster, Oliver;
Steinmetzer, Peter;
Stürzebecher, Uta;
Kotthaus, Joscha;
Clement, Bernd;
Stürzebecher, Jörg;
Steinmetzer, Torsten

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 7/2007.

Published in:: ChemMedChem, 2007, v. 2, n. 7, p. 918, doi. 10.1002/cmdc.200790024
Publication type:: Article

Synthesis and Biological Validation of Novel Synthetic Histone/Protein Methyltransferase Inhibitors.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 987, doi. 10.1002/cmdc.200700023

By:

Mai, Antonello;
Valente, Sergio;
Cheng, Donghang;
Perrone, Andrea;
Ragno, Rino;
Simeoni, Silvia;
Sbardella, Gianluca;
Brosch, Gerald;
Nebbioso, Angela;
Conte, Mariarosaria;
Altucci, Lucia;
Bedford, Mark T.

Publication type:

Article

GPCR Targeted Library Design: Novel Dopamine D<sub>3</sub> Receptor Ligands.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1000, doi. 10.1002/cmdc.200700067

By:

Böcker, A.;
Sasse, B. C.;
Nietert, M.;
Stark, H.;
Schneider, G.

Publication type:

Article

Design and Synthesis of 2,3,5-Substituted Imidazolidin-4-one Inhibitors of BACE-1.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 995, doi. 10.1002/cmdc.200700038

By:

Barrow, James C.;
Rittle, Kenneth E.;
Ngo, Phung L.;
Selnick, Harold G.;
Graham, Samuel L.;
Pitzenberger, Steven M.;
McGaughey, Georgia B.;
Colussi, Dennis;
Lai, Ming-Tain;
Huang, Qian;
Tugusheva, Katherine;
Espeseth, Amy S.;
Simon, Adam J.;
Munshi, Sanjeev K.;
Vacca, Joseph P.

Publication type:

Article

Graphical Abstract: ChemMedChem 7/2007.

Published in:: ChemMedChem, 2007, v. 2, n. 7, p. 911, doi. 10.1002/cmdc.200790023
Publication type:: Article

Paclitaxel And Docetaxel Resistance: Molecular Mechanisms and Development of New Generation Taxanes.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 920, doi. 10.1002/cmdc.200600308

By:

Galletti, Elena;
Magnani, Matteo;
Renzulli, Michela L.;
Botta, Maurizio

Publication type:

Article

Fragment-Based Synthesis and SAR of Modified FKBP Ligands: Influence of Different Linking on Binding Affinity.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1054, doi. 10.1002/cmdc.200600296

By:

Röhrig, Christoph H.;
Loch, Caroline;
Guan, Jia-Ying;
Siegal, Gregg;
Overhand, Mark

Publication type:

Article

Importance of Interaction between C1 Domain and Lipids in Protein Kinase Cα Activation: Hydrophobic Side Chain Direction in Isobenzofuranone Ligands Controls Enzyme Activation Level.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1006, doi. 10.1002/cmdc.200700080

By:

Hirai, Go;
Shimizu, Tadashi;
Watanabe, Toru;
Ogoshi, Yosuke;
Ohkubo, Megumi;
Sodeoka, Mikiko

Publication type:

Article

Design, Synthesis, and Structural Studies on Potent Biaryl Inhibitors of Type II Dehydroquinases.

Published in:

ChemMedChem, 2007, v. 2, n. 7, p. 1010, doi. 10.1002/cmdc.200700062

By:

Payne, Richard J.;
Riboldi-Tunnicliffe, Alan;
Kerbarh, Olivier;
Abell, Andrew D.;
Lapthorn, Adrian J.;
Abell, Chris

Publication type:

Article