Works in ChemMedChem, 2016, Vol 11, Issue 17

Results: 13

Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1904, doi. 10.1002/cmdc.201600180

By:

Annunziato, Giannamaria;
Angeli, Andrea;
D'Alba, Francesca;
Bruno, Agostino;
Pieroni, Marco;
Vullo, Daniela;
De Luca, Viviana;
Capasso, Clemente;
Supuran, Claudiu T.;
Costantino, Gabriele

Publication type:

Article

Synthesis and in vivo Evaluation of Fluorine-18 and Iodine-123 Pyrazolo[4,3- e]-1,2,4-triazolo[1,5- c]pyrimidine Derivatives as PET and SPECT Radiotracers for Mapping A<sub>2A</sub> Receptors.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1936, doi. 10.1002/cmdc.201600219

By:

Vala, Christine;
Morley, Thomas J.;
Zhang, Xuechun;
Papin, Caroline;
Tavares, Adriana Alexandre S.;
Lee, H. Sharon;
Constantinescu, Cristian;
Barret, Olivier;
Carroll, Vincent M.;
Baldwin, Ronald M.;
Tamagnan, Gilles D.;
Alagille, David

Publication type:

Article

Synthesis of Albicidin Derivatives: Assessing the Role of N-terminal Acylation on the Antibacterial Activity.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1899, doi. 10.1002/cmdc.201600231

By:

Kerwat, Dennis;
Grätz, Stefan;
Kretz, Julian;
Seidel, Maria;
Kunert, Maria;
Weston, John B.;
Süssmuth, Roderich D.

Publication type:

Article

Fragment Screening of RORγt Using Cocktail Crystallography: Identification of Simultaneous Binding of Multiple Fragments.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1881, doi. 10.1002/cmdc.201600242

By:

Xue, Yafeng;
Guo, Hongwei;
Hillertz, Per

Publication type:

Article

Substrate Fragmentation for the Design of M. tuberculosis CYP121 Inhibitors.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1924, doi. 10.1002/cmdc.201600248

By:

Kavanagh, Madeline E.;
Gray, Janine L.;
Gilbert, Sophie H.;
Coyne, Anthony G.;
McLean, Kirsty J.;
Davis, Holly J.;
Munro, Andrew W.;
Abell, Chris

Publication type:

Article

16-Membered Macrolide Lactone Derivatives Bearing a Triazole-Functionalized Arm at the Aglycone C13 Position as Antibacterial and Anticancer Agents.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1886, doi. 10.1002/cmdc.201600250

By:

Domagalska, Joanna;
Janas, Anna;
Pyta, Krystian;
Pecyna, Paulina;
Ruszkowski, Piotr;
Celewicz, Lech;
Gajecka, Marzena;
Bartl, Franz;
Przybylski, Piotr

Publication type:

Article

Dioxonaphthoimidazoliums are Potent and Selective Rogue Stem Cell Clearing Agents with SOX2-Suppressing Properties.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1944, doi. 10.1002/cmdc.201600262

By:

Ho, Si‐Han Sherman;
Ali, Azhar;
Ng, Yi‐Cheng;
Lam, Kuen‐Kuen Millie;
Wang, Shu;
Chan, Woon‐Khiong;
Chin, Tan‐Min;
Go, Mei‐Lin

Publication type:

Article

Fragment-Based Discovery of 5-Arylisatin-Based Inhibitors of Matrix Metalloproteinases 2 and 13.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1892, doi. 10.1002/cmdc.201600266

By:

Agamennone, Mariangela;
Belov, Dmitry S.;
Laghezza, Antonio;
Ivanov, Vladimir N.;
Novoselov, Anton M.;
Andreev, Ivan A.;
Ratmanova, Nina K.;
Altieri, Andrea;
Tortorella, Paolo;
Kurkin, Alexander V.

Publication type:

Article

Structure, Function, and Inhibition of Staphylococcus aureus Heptaprenyl Diphosphate Synthase.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1915, doi. 10.1002/cmdc.201600311

By:

Desai, Janish;
Liu, Yi‐Liang;
Wei, Hongli;
Liu, Weidong;
Ko, Tzu‐Ping;
Guo, Rey‐Ting;
Oldfield, Eric

Publication type:

Article

BODIPY-Appended 2-(2-Pyridyl)benzimidazole Platinum(II) Catecholates for Mitochondria-Targeted Photocytotoxicity.

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1956, doi. 10.1002/cmdc.201600320

By:

Mitra, Koushambi;
Gautam, Srishti;
Kondaiah, Paturu;
Chakravarty, Akhil R.

Publication type:

Article

Cover Picture: Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches (ChemMedChem 17/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1876, doi. 10.1002/cmdc.201600429

By:

Annunziato, Giannamaria;
Angeli, Andrea;
D'Alba, Francesca;
Bruno, Agostino;
Pieroni, Marco;
Vullo, Daniela;
De Luca, Viviana;
Capasso, Clemente;
Supuran, Claudiu T.;
Costantino, Gabriele

Publication type:

Article

Back Cover: Structure, Function, and Inhibition of Staphylococcus aureus Heptaprenyl Diphosphate Synthase (ChemMedChem 17/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 17, p. 1968, doi. 10.1002/cmdc.201600430

By:

Desai, Janish;
Liu, Yi‐Liang;
Wei, Hongli;
Liu, Weidong;
Ko, Tzu‐Ping;
Guo, Rey‐Ting;
Oldfield, Eric

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 17/2016.

Published in:: ChemMedChem, 2016, v. 11, n. 17, p. 1877, doi. 10.1002/cmdc.201681713
Publication type:: Article