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Serpin A1 C-Terminal Peptides as Collagen Turnover Modulators.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1850, doi. 10.1002/cmdc.201500472
By:
- Pascarella, Simona;
- Tiberi, Caterina;
- Sabatino, Giuseppina;
- Nuti, Francesca;
- Papini, Anna Maria;
- Giovannelli, Lisa;
- Rovero, Paolo
Publication type:
Article
Reactivity, Selectivity, and Reaction Mechanisms of Aminoguanidine, Hydralazine, Pyridoxamine, and Carnosine as Sequestering Agents of Reactive Carbonyl Species: A Comparative Study.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1778, doi. 10.1002/cmdc.201500552
By:
- Colzani, Mara;
- De Maddis, Danilo;
- Casali, Gaia;
- Carini, Marina;
- Vistoli, Giulio;
- Aldini, Giancarlo
Publication type:
Article
Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1709, doi. 10.1002/cmdc.201600015
By:
- Corona, Angela;
- Desantis, Jenny;
- Massari, Serena;
- Distinto, Simona;
- Masaoka, Takashi;
- Sabatini, Stefano;
- Esposito, Francesca;
- Manfroni, Giuseppe;
- Maccioni, Elias;
- Cecchetti, Violetta;
- Pannecouque, Christophe;
- Le Grice, Stuart F. J.;
- Tramontano, Enzo;
- Tabarrini, Oriana
Publication type:
Article
Albumin Nanoparticles for Brain Delivery: A Comparison of Chemical versus Thermal Methods and in vivo Behavior.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1840, doi. 10.1002/cmdc.201600080
By:
- Bergonzi, Maria C.;
- Guccione, Clizia;
- Grossi, Cristina;
- Piazzini, Vieri;
- Torracchi, Andrea;
- Luccarini, Ilaria;
- Casamenti, Fiorella;
- Bilia, Anna R.
Publication type:
Article
The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A2A Adenosine Receptor.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1829, doi. 10.1002/cmdc.201500595
By:
- Thomas, Ajiroghene;
- Buccioni, Michela;
- Dal Ben, Diego;
- Lambertucci, Catia;
- Marucci, Gabriella;
- Santinelli, Claudia;
- Spinaci, Andrea;
- Kachler, Sonja;
- Klotz, Karl‐Norbert;
- Volpini, Rosaria
Publication type:
Article
Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position 9.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1856, doi. 10.1002/cmdc.201500607
By:
- Merlino, Francesco;
- Brancaccio, Diego;
- Yousif, Ali M.;
- Piras, Linda;
- Campiglia, Pietro;
- Gomez‐Monterrey, Isabel;
- Santicioli, Paolo;
- Meini, Stefania;
- Maggi, Carlo A.;
- Novellino, Ettore;
- Carotenuto, Alfonso;
- Grieco, Paolo
Publication type:
Article
Enhanced Efficacy of Artemisinin Loaded in Transferrin-Conjugated Liposomes versus Stealth Liposomes against HCT-8 Colon Cancer Cells.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1745, doi. 10.1002/cmdc.201500586
By:
- Leto, Isabella;
- Coronnello, Marcella;
- Righeschi, Chiara;
- Bergonzi, Maria Camilla;
- Mini, Enrico;
- Bilia, Anna Rita
Publication type:
Article
A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1819, doi. 10.1002/cmdc.201600022
By:
- Mammoli, Valerio;
- Bonifazi, Alessandro;
- Dal Ben, Diego;
- Giannella, Mario;
- Giorgioni, Gianfabio;
- Piergentili, Alessandro;
- Pigini, Maria;
- Quaglia, Wilma;
- Thomas, Ajiroghene;
- Newman, Amy H.;
- Ferré, Sergi;
- Sanchez‐Soto, Marta;
- Keck, Thomas M.;
- Del Bello, Fabio
Publication type:
Article
In Vivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1812, doi. 10.1002/cmdc.201500596
By:
- Bruno, Elvira;
- Buemi, Maria R.;
- De Luca, Laura;
- Ferro, Stefania;
- Monforte, Anna‐Maria;
- Supuran, Claudiu T.;
- Vullo, Daniela;
- De Sarro, Giovambattista;
- Russo, Emilio;
- Gitto, Rosaria
Publication type:
Article
Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1721, doi. 10.1002/cmdc.201600053
By:
- Rocca, Roberta;
- Costa, Giosuè;
- Artese, Anna;
- Parrotta, Lucia;
- Ortuso, Francesco;
- Maccioni, Elias;
- Pinato, Odra;
- Greco, Maria Laura;
- Sissi, Claudia;
- Alcaro, Stefano;
- Distinto, Simona;
- Moraca, Federica
Publication type:
Article
Targeting Steroidogenic Cytochromes P450 (CYPs) with 6-Substituted 1-Imidazolylmethylxanthones.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1770, doi. 10.1002/cmdc.201600078
By:
- Gobbi, Silvia;
- Hu, Qingzhong;
- Zimmer, Christina;
- Belluti, Federica;
- Rampa, Angela;
- Hartmann, Rolf W.;
- Bisi, Alessandra
Publication type:
Article
Cationic Supramolecular Vesicular Aggregates for Pulmonary Tissue Selective Delivery in Anticancer Therapy.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1734, doi. 10.1002/cmdc.201600070
By:
- Licciardi, Mariano;
- Paolino, Donatella;
- Mauro, Nicolò;
- Cosco, Donato;
- Giammona, Gaetano;
- Fresta, Massimo;
- Cavallaro, Gennara;
- Celia, Christian
Publication type:
Article
Design, Synthesis, and Evaluation of Acrylamide Derivatives as Direct NLRP3 Inflammasome Inhibitors.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1790, doi. 10.1002/cmdc.201600055
By:
- Cocco, Mattia;
- Miglio, Gianluca;
- Giorgis, Marta;
- Garella, Davide;
- Marini, Elisabetta;
- Costale, Annalisa;
- Regazzoni, Luca;
- Vistoli, Giulio;
- Orioli, Marica;
- Massulaha‐Ahmed, Raïhane;
- Détraz‐Durieux, Isabelle;
- Groslambert, Marine;
- Py, Bénédicte F.;
- Bertinaria, Massimo
Publication type:
Article
A Series of COX-2 Inhibitors Endowed with NO-Releasing Properties: Synthesis, Biological Evaluation, and Docking Analysis.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1804, doi. 10.1002/cmdc.201600086
By:
- Consalvi, Sara;
- Poce, Giovanna;
- Ragno, Rino;
- Sabatino, Manuela;
- La Motta, Concettina;
- Sartini, Stefania;
- Calderone, Vincenzo;
- Martelli, Alma;
- Ghelardini, Carla;
- Di Cesare Mannelli, Lorenzo;
- Biava, Mariangela
Publication type:
Article
Targeting Different Transthyretin Binding Sites with Unusual Natural Compounds.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1865, doi. 10.1002/cmdc.201600092
By:
- Ortore, Gabriella;
- Orlandini, Elisabetta;
- Braca, Alessandra;
- Ciccone, Lidia;
- Rossello, Armando;
- Martinelli, Adriano;
- Nencetti, Susanna
Publication type:
Article
Synthesis and Biological Evaluation of N2-Substituted 2,4-Diamino-6-cyclohexylmethoxy-5-nitrosopyrimidines and Related 5-Cyano-NNO-azoxy Derivatives as Cyclin-Dependent Kinase 2 (CDK2) Inhibitors.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1705, doi. 10.1002/cmdc.201600108
By:
- Cortese, Daniela;
- Chegaev, Konstantin;
- Guglielmo, Stefano;
- Wang, Lan Z.;
- Golding, Bernard T.;
- Cano, Céline;
- Fruttero, Roberta
Publication type:
Article
TRPV1-FAAH-COX: The Couples Game in Pain Treatment.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1686, doi. 10.1002/cmdc.201600111
By:
- Aiello, Francesca;
- Carullo, Gabriele;
- Badolato, Mariateresa;
- Brizzi, Antonella
Publication type:
Article
Indazole, Pyrazole, and Oxazole Derivatives Targeting Nitric Oxide Synthases and Carbonic Anhydrases.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1695, doi. 10.1002/cmdc.201600204
By:
- Maccallini, Cristina;
- Di Matteo, Mauro;
- Vullo, Daniela;
- Ammazzalorso, Alessandra;
- Carradori, Simone;
- De Filippis, Barbara;
- Fantacuzzi, Marialuigia;
- Giampietro, Letizia;
- Pandolfi, Assunta;
- Supuran, Claudiu T.;
- Amoroso, Rosa
Publication type:
Article
Molecular Basis for Differential Recognition of G-Quadruplex versus Double-Helix DNA by Bis-Phenanthroline Metal Complexes.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1762, doi. 10.1002/cmdc.201600129
By:
- Rigo, Riccardo;
- Bianco, Sara;
- Musetti, Caterina;
- Palumbo, Manlio;
- Sissi, Claudia
Publication type:
Article
Back Cover: Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement (ChemMedChem 16/2016).
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1875, doi. 10.1002/cmdc.201600393
By:
- Rocca, Roberta;
- Costa, Giosuè;
- Artese, Anna;
- Parrotta, Lucia;
- Ortuso, Francesco;
- Maccioni, Elias;
- Pinato, Odra;
- Greco, Maria Laura;
- Sissi, Claudia;
- Alcaro, Stefano;
- Distinto, Simona;
- Moraca, Federica
Publication type:
Article
3-Arylidene- N-hydroxyoxindoles: A New Class of Compounds Endowed with Antitumor Activity.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1700, doi. 10.1002/cmdc.201600225
By:
- Musso, Loana;
- Cincinelli, Raffaella;
- Zuco, Valentina;
- De Cesare, Michelandrea;
- Zunino, Franco;
- Fallacara, Anna Lucia;
- Botta, Maurizio;
- Dallavalle, Sabrina
Publication type:
Article
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1680, doi. 10.1002/cmdc.201600272
By:
- Milite, Ciro;
- Feoli, Alessandra;
- Viviano, Monica;
- Rescigno, Donatella;
- Mai, Antonello;
- Castellano, Sabrina;
- Sbardella, Gianluca
Publication type:
Article
Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1752, doi. 10.1002/cmdc.201600140
By:
- Granchi, Carlotta;
- Lapillo, Margherita;
- Spena, Concetta Russo;
- Rizzolio, Flavio;
- Tuccinardi, Tiziano;
- Martin, Teresa A.;
- Carlson, Kathryn E.;
- Katzenellenbogen, John A.;
- Minutolo, Filippo
Publication type:
Article
Cover Picture: Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors (ChemMedChem 16/2016).
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1669, doi. 10.1002/cmdc.201600392
By:
- Corona, Angela;
- Desantis, Jenny;
- Massari, Serena;
- Distinto, Simona;
- Masaoka, Takashi;
- Sabatini, Stefano;
- Esposito, Francesca;
- Manfroni, Giuseppe;
- Maccioni, Elias;
- Cecchetti, Violetta;
- Pannecouque, Christophe;
- Le Grice, Stuart F. J.;
- Tramontano, Enzo;
- Tabarrini, Oriana
Publication type:
Article
The 23rd National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015).
Published in:
2016
By:
- Campiglia, Pietro;
- Sbardella, Gianluca
Publication type:
Editorial
Spotlights on our sister journals: ChemMedChem 16/2016.
Published in:
ChemMedChem, 2016, v. 11, n. 16, p. 1676, doi. 10.1002/cmdc.201681613
Publication type:
Article

Found: 26

Serpin A1 C-Terminal Peptides as Collagen Turnover Modulators.

Reactivity, Selectivity, and Reaction Mechanisms of Aminoguanidine, Hydralazine, Pyridoxamine, and Carnosine as Sequestering Agents of Reactive Carbonyl Species: A Comparative Study.

Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors.

Albumin Nanoparticles for Brain Delivery: A Comparison of Chemical versus Thermal Methods and in vivo Behavior.

The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A<sub>2A</sub> Adenosine Receptor.

Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position 9.

Enhanced Efficacy of Artemisinin Loaded in Transferrin-Conjugated Liposomes versus Stealth Liposomes against HCT-8 Colon Cancer Cells.

A Novel Class of Dopamine D<sub>4</sub> Receptor Ligands Bearing an Imidazoline Nucleus.

In Vivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents.

Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement.

Targeting Steroidogenic Cytochromes P450 (CYPs) with 6-Substituted 1-Imidazolylmethylxanthones.

Cationic Supramolecular Vesicular Aggregates for Pulmonary Tissue Selective Delivery in Anticancer Therapy.

Design, Synthesis, and Evaluation of Acrylamide Derivatives as Direct NLRP3 Inflammasome Inhibitors.

A Series of COX-2 Inhibitors Endowed with NO-Releasing Properties: Synthesis, Biological Evaluation, and Docking Analysis.

Targeting Different Transthyretin Binding Sites with Unusual Natural Compounds.

Synthesis and Biological Evaluation of N<sup>2</sup>-Substituted 2,4-Diamino-6-cyclohexylmethoxy-5-nitrosopyrimidines and Related 5-Cyano-NNO-azoxy Derivatives as Cyclin-Dependent Kinase 2 (CDK2) Inhibitors.

TRPV1-FAAH-COX: The Couples Game in Pain Treatment.

Indazole, Pyrazole, and Oxazole Derivatives Targeting Nitric Oxide Synthases and Carbonic Anhydrases.

Molecular Basis for Differential Recognition of G-Quadruplex versus Double-Helix DNA by Bis-Phenanthroline Metal Complexes.

Back Cover: Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement (ChemMedChem 16/2016).

3-Arylidene- N-hydroxyoxindoles: A New Class of Compounds Endowed with Antitumor Activity.

Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors.

Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.

Cover Picture: Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors (ChemMedChem 16/2016).

The 23<sup>rd</sup> National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015).

Spotlights on our sister journals: ChemMedChem 16/2016.