Works in ChemMedChem, 2015, Vol 10, Issue 11

Results: 23

pH-Cleavable Nucleoside Lipids: A New Paradigm for Controlling the Stability of Lipid-Based Delivery Systems.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1797, doi. 10.1002/cmdc.201500381
By:
- Oumzil, Khalid;
- Benizri, Sébastien;
- Tonelli, Giovanni;
- Staedel, Cathy;
- Appavoo, Ananda;
- Chaffanet, Max;
- Navailles, Laurence;
- Barthélémy, Philippe
Publication type:
Article
Inside Cover: Tetrazolylhydrazides as Selective Fragment-Like Inhibitors of the JumonjiC-Domain-Containing Histone Demethylase KDM4A (ChemMedChem 11/2015).
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1770, doi. 10.1002/cmdc.201500459
By:
- Rüger, Nicole;
- Roatsch, Martin;
- Emmrich, Thomas;
- Franz, Henriette;
- Schüle, Roland;
- Jung, Manfred;
- Link, Andreas
Publication type:
Article
6-Methyluracil Derivatives as Bifunctional Acetylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1863, doi. 10.1002/cmdc.201500334
By:
- Semenov, Vyacheslav E.;
- Zueva, Irina V.;
- Mukhamedyarov, Marat A.;
- Lushchekina, Sofya V.;
- Kharlamova, Alexandra D.;
- Petukhova, Elena O.;
- Mikhailov, Anatoly S.;
- Podyachev, Sergey N.;
- Saifina, Lilya F.;
- Petrov, Konstantin A.;
- Minnekhanova, Oksana A.;
- Zobov, Vladimir V.;
- Nikolsky, Evgeny E.;
- Masson, Patrick;
- Reznik, Vladimir S.
Publication type:
Article
Tetrazolylhydrazides as Selective Fragment-Like Inhibitors of the JumonjiC-Domain-Containing Histone Demethylase KDM4A.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1875, doi. 10.1002/cmdc.201500335
By:
- Rüger, Nicole;
- Roatsch, Martin;
- Emmrich, Thomas;
- Franz, Henriette;
- Schüle, Roland;
- Jung, Manfred;
- Link, Andreas
Publication type:
Article
Multicomponent Crystal Systems of Known Antimalarial Drug Molecules.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1786, doi. 10.1002/cmdc.201500337
By:
- Clements, Monica;
- le Roex, Tanya;
- Blackie, Margaret
Publication type:
Article
Discovery of Novel Allosteric Non-Bisphosphonate Inhibitors of Farnesyl Pyrophosphate Synthase by Integrated Lead Finding.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1884, doi. 10.1002/cmdc.201500338
By:
- Marzinzik, Andreas L.;
- Amstutz, René;
- Bold, Guido;
- Bourgier, Emmanuelle;
- Cotesta, Simona;
- Glickman, J. Fraser;
- Götte, Marjo;
- Henry, Christelle;
- Lehmann, Sylvie;
- Hartwieg, J. Constanze D.;
- Ofner, Silvio;
- Pellé, Xavier;
- Roddy, Thomas P.;
- Rondeau, Jean‐Michel;
- Stauffer, Frédéric;
- Stout, Steven J.;
- Widmer, Armin;
- Zimmermann, Johann;
- Zoller, Thomas;
- Jahnke, Wolfgang
Publication type:
Article
Phototoxic Activity and DNA Interactions of Water-Soluble Porphyrins and Their Rhenium(I) Conjugates.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1901, doi. 10.1002/cmdc.201500288
By:
- Mion, Giuliana;
- Gianferrara, Teresa;
- Bergamo, Alberta;
- Gasser, Gilles;
- Pierroz, Vanessa;
- Rubbiani, Riccardo;
- Vilar, Ramon;
- Leczkowska, Anna;
- Alessio, Enzo
Publication type:
Article
MS Binding Assays for D<sub>1</sub> and D<sub>5</sub> Dopamine Receptors.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1924, doi. 10.1002/cmdc.201500355
By:
- Neiens, Patrick;
- Höfner, Georg;
- Wanner, Klaus Theodor
Publication type:
Article
Discovery of Inhibitors of Trypanosoma brucei by Phenotypic Screening of a Focused Protein Kinase Library.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1809, doi. 10.1002/cmdc.201500300
By:
- Woodland, Andrew;
- Thompson, Stephen;
- Cleghorn, Laura A. T.;
- Norcross, Neil;
- De Rycker, Manu;
- Grimaldi, Raffaella;
- Hallyburton, Irene;
- Rao, Bhavya;
- Norval, Suzanne;
- Stojanovski, Laste;
- Brun, Reto;
- Kaiser, Marcel;
- Frearson, Julie A.;
- Gray, David W.;
- Wyatt, Paul G.;
- Read, Kevin D.;
- Gilbert, Ian H.
Publication type:
Article
Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1821, doi. 10.1002/cmdc.201500301
By:
- Spinks, Daniel;
- Smith, Victoria;
- Thompson, Stephen;
- Robinson, David A.;
- Luksch, Torsten;
- Smith, Alasdair;
- Torrie, Leah S.;
- McElroy, Stuart;
- Stojanovski, Laste;
- Norval, Suzanne;
- Collie, Iain T.;
- Hallyburton, Irene;
- Rao, Bhavya;
- Brand, Stephen;
- Brenk, Ruth;
- Frearson, Julie A.;
- Read, Kevin D.;
- Wyatt, Paul G.;
- Gilbert, Ian H.
Publication type:
Article
Applied RNAi. From Fundamental Research to Therapeutic Applications. Edited by Patrick Arbuthnot and Marc S. Weinberg.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1934, doi. 10.1002/cmdc.201500305
By:
- Brown, Stephen
Publication type:
Article
Development of Potent Adenosine Monophosphate Activated Protein Kinase (AMPK) Activators.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1915, doi. 10.1002/cmdc.201500371
By:
- Dokla, Eman M. E.;
- Fang, Chun‐Sheng;
- Lai, Po‐Ting;
- Kulp, Samuel K.;
- Serya, Rabah A. T.;
- Ismail, Nasser S. M.;
- Abouzid, Khaled A. M.;
- Chen, Ching‐Shih
Publication type:
Article
Cardiovascular and Metabolic Disease: Scientific Discoveries and New Therapies. Edited by Philip Peplow, James Adams, Tim Young.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1933, doi. 10.1002/cmdc.201500373
By:
- Plowright, Alleyn T.
Publication type:
Article
Green Chemistry Strategies for Drug Discovery. Edited by Emily A. Peterson and Julie B. Manley.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1932, doi. 10.1002/cmdc.201500377
By:
- Nitsche, Christoph
Publication type:
Article
Salicylketoximes That Target Glucose Transporter 1 Restrict Energy Supply to Lung Cancer Cells.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1892, doi. 10.1002/cmdc.201500320
By:
- Granchi, Carlotta;
- Qian, Yanrong;
- Lee, Hyang Yeon;
- Paterni, Ilaria;
- Pasero, Carolina;
- Iegre, Jessica;
- Carlson, Kathryn E.;
- Tuccinardi, Tiziano;
- Chen, Xiaozhuo;
- Katzenellenbogen, John A.;
- Hergenrother, Paul J.;
- Minutolo, Filippo
Publication type:
Article
Cover Picture: Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode (ChemMedChem 11/2015).
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1769, doi. 10.1002/cmdc.201500397
By:
- Spinks, Daniel;
- Smith, Victoria;
- Thompson, Stephen;
- Robinson, David A.;
- Luksch, Torsten;
- Smith, Alasdair;
- Torrie, Leah S.;
- McElroy, Stuart;
- Stojanovski, Laste;
- Norval, Suzanne;
- Collie, Iain T.;
- Hallyburton, Irene;
- Rao, Bhavya;
- Brand, Stephen;
- Brenk, Ruth;
- Frearson, Julie A.;
- Read, Kevin D.;
- Wyatt, Paul G.;
- Gilbert, Ian H.
Publication type:
Article
Discovery of Quinoline-Derived Trifluoromethyl Alcohols, Determination of Their in vivo Toxicity and Anticancer Activity in a Zebrafish Embryo Model.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1802, doi. 10.1002/cmdc.201500341
By:
- Sittaramane, Vinoth;
- Padgett, Jihan;
- Salter, Philip;
- Williams, Ashley;
- Luke, Shauntelle;
- McCall, Rebecca;
- Arambula, Jonathan F.;
- Graves, Vincent B.;
- Blocker, Mark;
- Van Leuven, David;
- Bowe, Keturah;
- Heimberger, Julia;
- Cade, Hannah C.;
- Immaneni, Supriya;
- Shaikh, Abid
Publication type:
Article
Design, Synthesis, and Photophysical Properties of Pyrroloquinoline-Based Compounds Showing Strong Blue Fluorescence as Potential Dyes for Biomedical Applications.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1846, doi. 10.1002/cmdc.201500366
By:
- Carta, Davide;
- Balasso, Anna;
- Caliceti, Paolo;
- Ferlin, Maria Grazia
Publication type:
Article
Back Cover: pH-Cleavable Nucleoside Lipids: A New Paradigm for Controlling the Stability of Lipid-Based Delivery Systems (ChemMedChem 11/2015).
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1940, doi. 10.1002/cmdc.201500438
By:
- Oumzil, Khalid;
- Benizri, Sébastien;
- Tonelli, Giovanni;
- Staedel, Cathy;
- Appavoo, Ananda;
- Chaffanet, Max;
- Navailles, Laurence;
- Barthélémy, Philippe
Publication type:
Article
The Role of Target Binding Kinetics in Drug Discovery.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1793, doi. 10.1002/cmdc.201500310
By:
- Guo, Dong;
- Heitman, Laura H.;
- IJzerman, Adriaan P.
Publication type:
Article
Isocyanides as Influenza A Virus Subtype H5N1 Wild-Type M2 Channel Inhibitors.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1837, doi. 10.1002/cmdc.201500318
By:
- Wu, Shuwen;
- Huang, Jing;
- Gazzarrini, Sabrina;
- He, Si;
- Chen, Lihua;
- Li, Jun;
- Xing, Li;
- Li, Chufang;
- Chen, Ling;
- Neochoritis, Constantinos G.;
- Liao, George P.;
- Zhou, Haibing;
- Dömling, Alexander;
- Moroni, Anna;
- Wang, Wei
Publication type:
Article
Graphical Abstract: ChemMedChem 11/2015.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1771, doi. 10.1002/cmdc.201581111
Publication type:
Article
Spotlights on our sister journals: ChemMedChem 11/2015.
Published in:
ChemMedChem, 2015, v. 10, n. 11, p. 1780, doi. 10.1002/cmdc.201581113
Publication type:
Article