Works in Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, Vol 39, Issue 1

Results: 90

Evaluation of hydrazone and N-acylhydrazone derivatives of vitamin B6 and pyridine-4-carbaldehyde as potential drugs against Alzheimer's disease.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2431832

By:

Bartolić, Marija;
Matošević, Ana;
Maraković, Nikola;
Bušić, Valentina;
Roca, Sunčica;
Vikić-Topić, Dražen;
Sabljić, Antonio;
Bosak, Anita;
Gašo-Sokač, Dajana

Publication type:

Article

Antifungal and anti-biofilm effects of hydrazone derivatives on Candida spp.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2429109

By:

Popczyk, Pierre;
Ghinet, Alina;
Bortolus, Clovis;
Kamus, Laure;
Lensink, Marc F.;
de Ruyck, Jérôme;
Sendid, Boualem;
Dubar, Faustine

Publication type:

Article

Investigation of the inhibitory properties of azo-dyes on chorismate synthase from Paracoccidioides brasiliensis.

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2427175

By:

Fuchs, Katharina;
Totaro, Massimo G.;
Toplak, Marina;
Bijelic, Aleksandar;
Macheroux, Peter

Publication type:

Article

Discovery of novel 2,4-diarylaminopyrimidine hydrazone derivatives as potent anti-thyroid cancer agents capable of inhibiting FAK.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2423875

By:

Li, Hongting;
Jia, Mei-Qi;
Qin, Zhao-Long;
Lu, Changliang;
Chu, Weili;
Zhang, Ze;
Niu, Jinbo;
Song, Jian;
Zhang, Sai-Yang;
Fu, Lijun

Publication type:

Article

Structure optimization and molecular dynamics studies of new tumor-selective s-triazines targeting DNA and MMP-10/13 for halting colorectal and secondary liver cancers.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2423174

By:

Morcos, Christine A.;
Haiba, Nesreen S.;
Bassily, Rafik W.;
Abu-Serie, Marwa M.;
El-Yazbi, Amira F.;
Soliman, Omar A.;
Khattab, Sherine N.;
Teleb, Mohamed

Publication type:

Article

Exploring structural and biological insights of TEAD through rational design and synthesis of niflumic acid derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2419925

By:

Choi, Yong-Sung;
Kim, Yoon-Jung;
Jeon, Yeram;
Kang, Jong Soon;
Lee, Juhee;
Hong, Eunmi;
Park, Young-Hoon;
Kim, Wantae;
Cha, Boksik;
Jeon, Raok

Publication type:

Article

Discovering a novel dual specificity tyrosine-phosphorylation-regulated kinase 1A (DYRK1A) inhibitor and its impact on tau phosphorylation and amyloid-β formation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2418470

By:

Tu, Huang-Ju;
Chao, Min-Wu;
Lee, Cheng-Chung;
Peng, Chao-Shiang;
Wu, Yi-Wen;
Lin, Tony Eight;
Chang, Yu-Wei;
Yen, Shih-Chung;
Hsu, Kai-Cheng;
Pan, Shiow-Lin;
HuangFu, Wei-Chun

Publication type:

Article

Bacillus lipopeptides inhibit lipase activity and promote 3T3-L1 preadipocyte differentiation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2417915

By:

Chen, Meichun;
Chen, Deju;
Xiao, Rongfeng;
Zheng, Xuefang;
Liu, Bo;
Wang, Jieping

Publication type:

Article

Synthesis and biological evaluation of quinoxaline derivatives as ASK1 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2414382

By:

Han, Xiaorui;
Lan, Pingping;
Chen, Qianfeng;
Liu, Hua;
Chen, Zhongwen;
Wang, Tiantian;
Wang, Zengtao

Publication type:

Article

Expanding the antiprotozoal activity and the mechanism of action of n-butyl and iso-butyl ester of quinoxaline-1,4-di-N-oxide derivatives against Giardia lamblia, Trichomonas vaginalis, and Entamoeba histolytica. An in vitro and in silico approach.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2413018

By:

González-González, Alonzo;
Sánchez-Sánchez, Oscar;
Yépez-Mulia, Lilián;
Delgado-Maldonado, Timoteo;
Vázquez-Jiménez, Lenci K.;
López-Velázquez, Gabriel;
de la Mora-de la Mora, José Ignacio;
Pacheco-Gutierrez, Sebastian;
Chino-Ríos, Laura;
Arias, Diego;
Moreno-Rodríguez, Adriana;
Paz-González, Alma;
Ortíz-Pérez, Eyra;
Rivera, Gildardo

Publication type:

Article

Design, synthesis and biological evaluation of marine naphthoquinone-naphthol derivatives as potential anticancer agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2412865

By:

Li, Yujuan;
Yelv, Luyou;
Wu, Xiaoqiu;
Liu, Ning;
Zhu, Yamin

Publication type:

Article

Structure-guided discovery of novel dUTPase inhibitors with anti-Nocardia activity by computational design.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2411573

By:

Wang, Zhi-Zheng;
Weng, Jun;
Qi, Jing;
Fu, Xin-Xin;
Xing, Ban-Bin;
Hu, Yang;
Huang, Chun-Hsiang;
Chen, Chin-Yu;
Wei, Zigong

Publication type:

Article

Synthesis and biological evaluation of ortho-phenyl phenylhydroxamic acids containing phenothiazine with improved selectivity for class IIa histone deacetylases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2406025

By:

Hsu, Kai-Cheng;
Huang, Yun-Yi;
Chu, Jung-Chun;
Huang, Yu-Wen;
Hu, Jing-Lan;
Lin, Tony Eight;
Yen, Shih-Chung;
Weng, Jing-Ru;
Huang, Wei-Jan

Publication type:

Article

Novel hybrids of 1,2,3-triazole-benzoxazole: design, synthesis, and assessment of DprE1 enzyme inhibitors using fluorometric assay and computational analysis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2403744

By:

Singh, Manisha;
Batt, Sarah M.;
Canales, Christian S. C.;
Pavan, Fernando R.;
Kumar, Sethu Arun;
Akshatha, Handattu S.;
Bhagyalalitha, Meduri;
Pujar, Karthik G.;
Bidye, Durgesh;
Pujar, Gurubasavaraj V.;
Besra, Gurdyal S.

Publication type:

Article

Design, synthesis, and biological activity evaluation of dihydromyricetin derivatives against SARS-CoV-2-Omicron virus.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2390909

By:

Wu, Cong;
Jiang, Qi;
Zhong, Hui;
Zhou, Xudong;
Liu, Leping;
Pan, Tong;
Liu, Chao;
Wang, Wei;
Sheng, Wenbing

Publication type:

Article

Discovery of selective ACAT2 antagonist via a combination strategy based on deep docking, pharmacophore modelling, and molecular dynamics simulation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2403736

By:

Liu, Yanfeng;
Ding, Feng;
Deng, Liangying;
Zhang, Shuran;
Wu, Lixing;
Tong, Huangjin

Publication type:

Article

Discovery of natural anthraquinones as potent inhibitors against pancreatic lipase: structure-activity relationships and inhibitory mechanism.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2398561

By:

Chen, Zi-Qiang;
He, Wen-Yao;
Yang, Si-Yuan;
Ma, Hong-Hong;
Zhou, Jing;
Li, Hao;
Zhu, Ya-Di;
Qian, Xing-Kai;
Zou, Li-Wei

Publication type:

Article

Novel alloxazine analogues: design, synthesis, and antitumour efficacy enhanced by kinase screening, molecular docking, and ADME studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2398551

By:

Samaha, Doaa;
Mahmoud, Sawsan;
Mohamed, Mosaad Sayed;
Abdullah, Rokaia S.;
A. Abou Taleb, Nageh;
Nagamatsu, Tomohisa;
Ali, Hamed I.

Publication type:

Article

Synthesis, molecular modelling, and biological evaluation of novel quinoxaline derivatives for treating type II diabetes.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2395985

By:

Alasmary, Fatmah Ali S.;
Abdullah, Dalal A.;
Masand, Vijay H.;
Ben Bacha, Abir;
Omar Ebeid, Abdelsattar Mansour;
El-Araby, Moustafa E.;
Alafeefy, Ahmed M

Publication type:

Article

Synthesis and in vitro evaluation of benzo[b]thiophene-3-carboxylic acid 1,1-dioxide derivatives as anticancer agents targeting the RhoA/ROCK pathway.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2390911

By:

Liang, Jinhao;
Huang, Jin;
Yang, Jianzhan;
Liang, Weihong;
Li, Haoxiang;
Wu, Yunshan;
Liu, Bo

Publication type:

Article

Discovery of 1,3-disubstituted prop-2-en-1-one derivatives as inhibitors of neutrophilic inflammation via modulation of MAPK and Akt pathways.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2402988

By:

Abdel-Halim, Mohammad;
El-Gamil, Dalia S.;
Hammam, Mennatallah A.;
El-Shazly, Mohamed;
Wang, Yi-Hsuan;
Kung, Po-Hsiung;
Chen, Yu-Cheng;
Korinek, Michal;
Abadi, Ashraf H.;
Engel, Matthias;
Hwang, Tsong-Long

Publication type:

Article

Non-small cell lung cancer sensitisation to platinum chemotherapy via new thiazole-triazole hybrids acting as dual T-type CCB/MMP-9 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2388209

By:

Gamal, Hassan;
Ismail, Khadiga A.;
Omar, A-Mohsen M. E.;
Teleb, Mohamed;
Abu-Serie, Marwa M.;
Huang, Sun;
Abdelsattar, Abdalla S.;
Zamponi, Gerald W.;
Fahmy, Hesham

Publication type:

Article

Crystal structure of dihydroneopterin aldolase from Mycobacterium tuberculosis associated with 8-mercaptoguanine, and development of novel S8-functionalized analogues as inhibitors: Synthesis, enzyme inhibition, in vitro toxicity and antitubercular activity

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2388207

By:

Czeczot, Alexia de Matos;
Muniz, Mauro Neves;
Perelló, Marcia Alberton;
Silva, Éverton Edésio Dinis;
Timmers, Luís Fernando Saraiva Macedo;
Berger, Andresa;
Gonzalez, Laura Calle;
Arraché Gonçalves, Guilherme;
Moura, Sidnei;
Machado, Pablo;
Bizarro, Cristiano Valim;
Basso, Luiz Augusto

Publication type:

Article

In-cell bioluminescence resonance energy transfer (BRET)-based assay uncovers ceritinib and CA-074 as SARS-CoV-2 papain-like protease inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2387417

By:

Li, Mei;
Bei, Zhu-Chun;
Yuan, Yongtian;
Wang, Baogang;
Zhang, Dongna;
Xu, Likun;
Zhao, Liangliang;
Xu, Qin;
Song, Yabin

Publication type:

Article

Design, synthesis, and biological evaluation of (thio)urea derivatives as potent Escherichia coli β-glucuronidase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2387415

By:

Xu, Keren;
Ying, Leyi;
Ying, Titi;
Wu, Qihao;
Du, Lin;
Yu, Yanlei;
Ying, Youmin;
Wei, Bin;
Wang, Hong;
Yang, Zhikun

Publication type:

Article

Challenging the Biginelli scaffold to surpass the first line antitubercular drugs: Mycobacterium tuberculosis thymidine monophosphate kinase (TMPKmt) inhibition activity and molecular modelling studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2386668

By:

El-Shoukrofy, Mai S.;
Atta, Amal;
Fahmy, Salwa;
Sriram, Dharmarajan;
Shehat, Michael G.;
Labouta, Ibrahim M.;
Mahran, Mona A.

Publication type:

Article

Statement of Retraction: Dihydroartemisinin enhances the anti-tumor effect of photodynamic therapy by targeting PKM2-mediated glycolysis in esophageal cancer cell.

Published in:: 2024
Publication type:: Correction Notice

Design, synthesis, and evaluation of novel stilbene derivatives that degrade acidic nucleoplasmic DNA-binding protein 1 (And1) and synergize with PARP1 inhibitor in NSCLC cells.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2383886

By:

Chen, Leyuan;
Ren, Zhonghao;
Zhang, Yunze;
Hou, Wenbin;
Li, Yiliang

Publication type:

Article

The repertoire of iron superoxide dismutases from Leishmania infantum as targets in the search for therapeutic agents against leishmaniasis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2377586

By:

García-Soriano, Juan Carlos;
de Lucio, Héctor;
Elvira-Blázquez, Daniel;
Alcón-Calderón, Mercedes;
Sanz del Olmo, Natalia;
Sánchez-Murcia, Pedro A.;
Ortega, Paula;
de la Mata, Francisco Javier;
Jiménez-Ruiz, Antonio

Publication type:

Article

Correction.

Published in:: 2024
Publication type:: Correction Notice

Vitamin B6 inhibits activity of Helicobacter pylori adenylosuccinate synthetase and growth of reference and clinical, antibiotic-resistant H. pylori strains.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2372734

By:

Wojtyś, Marta Ilona;
Maksymiuk, Weronika;
Narczyk, Marta;
Bubić, Ante;
Ašler, Ivana Leščić;
Krzyżek, Paweł;
Gościniak, Grażyna;
Jagusztyn-Krynicka, Elżbieta Katarzyna;
Bzowska, Agnieszka

Publication type:

Article

A comprehensive investigation of the anion inhibition profile of a β-carbonic anhydrase from Acinetobacter baumannii for crafting innovative antimicrobial treatments.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2372731

By:

De Luca, Viviana;
Giovannuzzi, Simone;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Click estradiol dimers with novel aromatic bridging units: synthesis and anticancer evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2367139

By:

Řehulka, Jiří;
Jurášek, Michal;
Dráber, Pavel;
Ivanová, Aleksandra;
Gurská, Soňa;
Ječmeňová, Kateřina;
Mokshyna, Olena;
Hajdúch, Marián;
Polishchuk, Pavel;
Drašar, Pavel B.;
Džubák, Petr

Publication type:

Article

Targeting the glutamine-arginine-proline metabolism axis in cancer.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2367129

By:

Wang, Di;
Duan, Jiang-jie;
Guo, Yu-feng;
Chen, Jun-jie;
Chen, Tian-qing;
Wang, Jun;
Yu, Shi-cang

Publication type:

Article

Fluorinated indeno-quinoxaline bearing thiazole moieties as hypoglycaemic agents targeting α-amylase, and α-glucosidase: synthesis, molecular docking, and ADMET studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2367128

By:

Gohar, Nirvana A.;
Fayed, Eman A.;
A. Ammar, Yousry;
A. Abu Ali, Ola;
Ragab, Ahmed;
Mahfoz, Amal M.;
Abusaif, Moustafa S.

Publication type:

Article

Anilino-1,4-naphthoquinones as potent mushroom tyrosinase inhibitors: in vitro and in silico studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2357174

By:

Sabuakham, Sahachai;
Nasoontorn, Sutita;
Kongtaworn, Napat;
Rungrotmongkol, Thanyada;
Silsirivanit, Atit;
Pingaew, Ratchanok;
Mahalapbutr, Panupong

Publication type:

Article

Watermelon: setup and validation of an in silico fragment-based approach.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2356179

By:

Di Stefano, Miriana;
Galati, Salvatore;
Piazza, Lisa;
Gado, Francesca;
Granchi, Carlotta;
Macchia, Marco;
Giordano, Antonio;
Tuccinardi, Tiziano;
Poli, Giulio

Publication type:

Article

Identification of novel PD-1/PD-L1 small molecule inhibitors: virtual screening, synthesis and in vitro characterisation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2353711

By:

Wu, Tingting;
Cheng, Hu;
Sima, Lijie;
Wang, Zhongyuan;
Ouyang, Weiwei;
Wang, Jianta;
Hou, Yunlei;
Zhao, Dongsheng;
Liao, Weike;
Hu, Chujiao

Publication type:

Article

Exploring of N-phthalimide-linked 1,2,3-triazole analogues with promising -anti-SARS-CoV-2 activity: synthesis, biological screening, and molecular modelling studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2351861

By:

Aljuhani, Ateyatallah;
Alsehli, Mosa;
Seleem, Mohamed A.;
Alraqa, Shaya Y.;
Ahmed, Hany E. A.;
Rezki, Nadjet;
Aouad, Mohamed R.

Publication type:

Article

Cloning, expression, and purification of an α-carbonic anhydrase from Toxoplasma gondii to unveil its kinetic parameters and anion inhibition profile.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2346523

By:

De Luca, Viviana;
Giovannuzzi, Simone;
Capasso, Clemente;
Supuran, Claudiu T.

Publication type:

Article

The activity of pyrazolo[4,3-e][1,2,4]triazine and pyrazolo[4,3-e]tetrazolo[1,5-b][1,2,4]triazine sulphonamide derivatives in monolayer and spheroid breast cancer cell cultures.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2343352

By:

Szymanowska, Anna;
Radomska, Dominika;
Czarnomysy, Robert;
Mojzych, Mariusz;
Kotwica-Mojzych, Katarzyna;
Bielawski, Krzysztof;
Bielawska, Anna

Publication type:

Article

Discovery of novel FGFR4 inhibitors through a build-up fragment strategy.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2343350

By:

Kim, Jihyung;
Im, Chang Gyun;
Oh, Kyujin;
Lee, Ji Min;
Al-Rubaye, Fatimah;
Min, Kyung Hoon

Publication type:

Article

Effects of thymoquinone and the curcumin analog EF-24 on the activity of the enzyme paraoxonase-1 in human glioblastoma cells U87MG.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2339901

By:

Simsek, Ender;
Sunguroglu, Asuman;
Kilic, Ahmet;
Özgültekin, Nurbanu;
Ozensoy Guler, O.

Publication type:

Article

Evaluation of the anticancer effects exerted by 5-fluorouracil and heme oxygenase-1 inhibitor hybrids in HTC116 colorectal cancer cells.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2337191

By:

Salerno, Loredana;
Notaro, Antonietta;
Consoli, Valeria;
Affranchi, Federica;
Pittalà, Valeria;
Sorrenti, Valeria;
Vanella, Luca;
Giuliano, Michela;
Intagliata, Sebastiano

Publication type:

Article

Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide–hydantoin hybrids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2335927

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Gratteri, Paola;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Targeting bacterial growth in biofilm conditions: rational design of novel inhibitors to mitigate clinical and food contamination using QSAR.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2330907

By:

Galvez-Llompart, Maria;
Hierrezuelo, Jesús;
Blasco, Mariluz;
Zanni, Riccardo;
Galvez, Jorge;
de Vicente, Antonio;
Pérez-García, Alejandro;
Romero, Diego

Publication type:

Article

Elucidation of critical chemical moieties of metallo-β-lactamase inhibitors and prioritisation of target metallo-β-lactamases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2318830

By:

Lee, Jung Hun;
Kim, Sang-Gyu;
Jang, Kyung-Min;
Shin, Kyoungmin;
Jin, Hyeonku;
Kim, Dae-Wi;
Jeong, Byeong Chul;
Lee, Sang Hee

Publication type:

Article

Discovery of novel anaplastic lymphoma kinase (ALK) and histone deacetylase (HDAC) dual inhibitors exhibiting antiproliferative activity against non-small cell lung cancer.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2318645

By:

Wang, Kang-Li;
Yeh, Tsung-Yu;
Hsu, Pei-Chen;
Wong, Tzu-Hsuan;
Liu, Jia-Rong;
Chern, Ji-Wang;
Lin, Miao-Hsia;
Yu, Chao-Wu

Publication type:

Article

Design, synthesis, in vitro and in vivo biological evaluation of pterostilbene derivatives for anti-inflammation therapy.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2315227

By:

Chen, Liuzeng;
Wang, Ke;
Liu, Xiaohan;
Wang, Lifan;
Zou, Hui;
Hu, Shuying;
Zhou, Lingling;
Li, Rong;
Cao, Shiying;
Ruan, Banfeng;
Cui, Quanren

Publication type:

Article

Design, synthesis, and evaluation of cyclic C7-bridged monocarbonyl curcumin analogs containing an o-methoxy phenyl group as potential agents against gastric cancer.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2314233

By:

Gan, Xin;
Wu, Yuna;
Zhu, Min;
Liu, Bo;
Kong, Miaomiao;
Xi, Zixuan;
Li, Ke;
Wang, Haibao;
Su, Tiande;
Yao, Jiali;
Khushafah, Fatehi;
Yi, Baozhu;
Wang, Jiabing;
Li, Wulan;
Wu, Jianzhang

Publication type:

Article