Works matching IS 1475-6366 AND VI 35 AND IP 1 AND DT 2020

Results: 185
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    Scaffold hopping and optimisation of 3',4'-dihydroxyphenyl- containing thienopyrimidinones: synthesis of quinazolinone derivatives as novel allosteric inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1953, doi. 10.1080/14756366.2020.1835884
    By:
    • Tocco, Graziella;
    • Esposito, Francesca;
    • Caboni, Pierluigi;
    • Laus, Antonio;
    • Beutler, John A.;
    • Wilson, Jennifer A.;
    • Corona, Angela;
    • Le Grice, Stuart F. J.;
    • Tramontano, Enzo
    Publication type:
    Article
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    Multidirectional in vitro and in cellulo studies as a tool for identification of multi-target-directed ligands aiming at symptoms and causes of Alzheimer's disease.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1944, doi. 10.1080/14756366.2020.1835882
    By:
    • Szałaj, Natalia;
    • Godyń, Justyna;
    • Jończyk, Jakub;
    • Pasieka, Anna;
    • Panek, Dawid;
    • Wichur, Tomasz;
    • Więckowski, Krzysztof;
    • Zaręba, Paula;
    • Bajda, Marek;
    • Pislar, Anja;
    • Malawska, Barbara;
    • Sabate, Raimon;
    • Więckowska, Anna
    Publication type:
    Article
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    Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1840, doi. 10.1080/14756366.2020.1825408
    By:
    • Elie, Jonathan;
    • Feizbakhsh, Omid;
    • Desban, Nathalie;
    • Josselin, Béatrice;
    • Baratte, Blandine;
    • Bescond, Amandine;
    • Duez, Julien;
    • Fant, Xavier;
    • Bach, Stéphane;
    • Marie, Dominique;
    • Place, Matthieu;
    • Ben Salah, Sami;
    • Chartier, Agnes;
    • Berteina-Raboin, Sabine;
    • Chaikuad, Apirat;
    • Knapp, Stefan;
    • Carles, Fabrice;
    • Bonnet, Pascal;
    • Buron, Frédéric;
    • Routier, Sylvain
    Publication type:
    Article
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    Inhibition mechanism of naphthylphenylamine derivatives acting on the CDC25B dual phosphatase and analysis of the molecular processes involved in the high cytotoxicity exerted by one selected derivative in melanoma cells.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1866, doi. 10.1080/14756366.2020.1819257
    By:
    • Aliotta, Federica;
    • Nasso, Rosarita;
    • Rullo, Rosario;
    • Arcucci, Alessandro;
    • Avagliano, Angelica;
    • Simonetti, Martina;
    • Sanità, Gennaro;
    • Masullo, Mariorosario;
    • Lavecchia, Antonio;
    • Ruocco, Maria Rosaria;
    • Vendittis, Emmanuele De
    Publication type:
    Article
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    The intensification of anticancer activity of LFM-A13 by erythropoietin as a possible option for inhibition of breast cancer.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1697, doi. 10.1080/14756366.2020.1818738
    By:
    • Rozkiewicz, Dariusz;
    • Hermanowicz, Justyna Magdalena;
    • Tankiewicz-Kwedlo, Anna;
    • Sieklucka, Beata;
    • Pawlak, Krystyna;
    • Czarnomysy, Robert;
    • Bielawski, Krzysztof;
    • Surazynski, Arkadiusz;
    • Kalafut, Joanna;
    • Przybyszewska, Alicja;
    • Koda, Mariusz;
    • Jakubowska, Katarzyna;
    • Rivero-Muller, Adolfo;
    • Pawlak, Dariusz
    Publication type:
    Article
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    New classes of potent heparanase inhibitors from ligand-based virtual screening.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1685, doi. 10.1080/14756366.2020.1811701
    By:
    • Pala, Daniele;
    • Scalvini, Laura;
    • Elisi, Gian Marco;
    • Lodola, Alessio;
    • Mor, Marco;
    • Spadoni, Gilberto;
    • Ferrara, Fabiana F.;
    • Pavoni, Emiliano;
    • Roscilli, Giuseppe;
    • Milazzo, Ferdinando M.;
    • Battistuzzi, Gianfranco;
    • Rivara, Silvia;
    • Giannini, Giuseppe
    Publication type:
    Article
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    Cytotoxic substituted indolizines as new colchicine site tubulin polymerisation inhibitors.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1581, doi. 10.1080/14756366.2020.1801671
    By:
    • Sardaru, Monica-Cornelia;
    • Craciun, Anda Mihaela;
    • Al Matarneh, Cristina-Maria;
    • Sandu, Isabela Andreea;
    • Amarandi, Roxana Maria;
    • Popovici, Lacramioara;
    • Ciobanu, Catalina Ionica;
    • Peptanariu, Dragos;
    • Pinteala, Mariana;
    • Mangalagiu, Ionel I.;
    • Danac, Ramona
    Publication type:
    Article
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    Synthesis and evaluation of 2,4,5-trisubstitutedthiazoles as carbonic anhydrase-III inhibitors.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1483, doi. 10.1080/14756366.2020.1786820
    By:
    • Al-Jaidi, Bilal A.;
    • Deb, Pran Kishore;
    • Telfah, Soha Taher;
    • Dakkah, Abdel Naser;
    • Bataineh, Yazan A.;
    • Khames Aga, Qutaiba Ahmed Al;
    • Al-dhoun, Mohammad A.;
    • Ahmad Al-Subeihi, Ala' Ali;
    • Odetallah, Haifa'a Marouf;
    • Bardaweel, Sanaa K.;
    • Mailavaram, Raghuprasad;
    • Venugopala, Katharigatta N.;
    • Nair, Anroop B.
    Publication type:
    Article
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