Works in Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, Vol 33, Issue 1

Results: 164
    1
    2
    3
    4
    5
    6
    7
    8
    9

    Target-based drug discovery through inversion of quantitative structure-drug-property relationships and molecular simulation: CA IX-sulphonamide complexes.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1430, doi. 10.1080/14756366.2018.1511551
    By:
    • Žuvela, Petar;
    • Liu, J. Jay;
    • Yi, Myunggi;
    • Pomastowski, Paweł P.;
    • Sagandykova, Gulyaim;
    • Belka, Mariusz;
    • David, Jonathan;
    • Bączek, Tomasz;
    • Szafrański, Krzysztof;
    • Żołnowska, Beata;
    • Sławiński, Jarosław;
    • Supuran, Claudiu T.;
    • Wong, Ming Wah;
    • Buszewski, Bogusław
    Publication type:
    Article
    10
    11
    12
    13
    14
    15
    16
    17
    18
    19
    20
    21
    22
    23
    24
    25

    Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3′,4′,5′-trimethoxyphenyl)-3-(2′-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1225, doi. 10.1080/14756366.2018.1493473
    By:
    • Preti, Delia;
    • Romagnoli, Romeo;
    • Rondanin, Riccardo;
    • Cacciari, Barbara;
    • Hamel, Ernest;
    • Balzarini, Jan;
    • Liekens, Sandra;
    • Schols, Dominique;
    • Estévez-Sarmiento, Francisco;
    • Quintana, José;
    • Estévez, Francisco
    Publication type:
    Article
    26
    27
    28
    29
    30
    31
    32
    33

    Synthesis and pharmacological evaluation of novel isoquinoline N-sulphonylhydrazones designed as ROCK inhibitors.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1181, doi. 10.1080/14756366.2018.1490732
    By:
    • Oliveira, Ramon Guerra de;
    • Guerra, Fabiana Sélos;
    • Mermelstein, Cláudia dos Santos;
    • Fernandes, Patrícia Dias;
    • Bastos, Isadora Tairinne de Sena;
    • Costa, Fanny Nascimento;
    • Barroso, Regina Cely Rodrigues;
    • Ferreira, Fabio Furlan;
    • Fraga, Carlos Alberto Manssour
    Publication type:
    Article
    34

    Synthesis and structure-activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1271, doi. 10.1080/14756366.2018.1490731
    By:
    • Bacsa, Ildikó;
    • Herman, Bianka Edina;
    • Jójárt, Rebeka;
    • Herman, Kevin Stefán;
    • Wölfling, János;
    • Schneider, Gyula;
    • Varga, Mónika;
    • Tömböly, Csaba;
    • Rižner, Tea Lanišnik;
    • Szécsi, Mihály;
    • Mernyák, Erzsébet
    Publication type:
    Article
    35
    36
    37
    38
    39
    40

    Nitroimidazole-based inhibitors DTP338 and DTP348 are safe for zebrafish embryos and efficiently inhibit the activity of human CA IX in Xenopus oocytes.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1064, doi. 10.1080/14756366.2018.1482285
    By:
    • Aspatwar, Ashok;
    • Becker, Holger M.;
    • Parvathaneni, Nanda Kumar;
    • Hammaren, Milka;
    • Svorjova, Aleksandra;
    • Barker, Harlan;
    • Supuran, Claudiu T.;
    • Dubois, Ludwig;
    • Lambin, Philippe;
    • Parikka, Mataleena;
    • Parkkila, Seppo;
    • Winum, Jean-Yves
    Publication type:
    Article
    41
    42
    43
    44
    45
    46
    47
    48
    49
    50

    Dioxygen, an unexpected carbonic anhydrase ligand.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 999, doi. 10.1080/14756366.2018.1475371
    By:
    • Ferraroni, Marta;
    • Gaspari, Roberto;
    • Scozzafava, Andrea;
    • Cavalli, Andrea;
    • Supuran, Claudiu T.
    Publication type:
    Article