Works in Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, Vol 32, Issue 1

Results: 143

Editorial Board.

Published in:: Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. ebi, doi. 10.1080/14756366.2017.1398806
Publication type:: Article

Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1305, doi. 10.1080/14756366.2017.1386660

By:

Akocak, Suleyman;
Lolak, Nabih;
Vullo, Daniela;
Durgun, Mustafa;
Supuran, Claudiu T.

Publication type:

Article

In vitro and in vivo antitumour effects of phenylboronic acid against mouse mammary adenocarcinoma 4T1 and squamous carcinoma SCCVII cells.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1299, doi. 10.1080/14756366.2017.1384823

By:

Marasovic, Maja;
Ivankovic, Sinisa;
Stojkovic, Ranko;
Djermic, Damir;
Galic, Borivoj;
Milos, Mladen

Publication type:

Article

Resveratrol-based cinnamic ester hybrids: synthesis, characterization, and anti-inflammatory activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1282, doi. 10.1080/14756366.2017.1381090

By:

Ruan, Ban-Feng;
Ge, Wei-Wei;
Cheng, Hui-Jie;
Xu, Hua-Jian;
Li, Qing-Shan;
Liu, Xin-Hua

Publication type:

Article

Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1274, doi. 10.1080/14756366.2017.1380638

By:

Ramya, P. V. Sri;
Angapelly, Srinivas;
Angeli, Andrea;
Digwal, Chander Singh;
Arifuddin, Mohammed;
Babu, Bathini Nagendra;
Supuran, Claudiu T.;
Kamal, Ahmed

Publication type:

Article

Dual targeting of cancer-related human matrix metalloproteinases and carbonic anhydrases by chiral N -(biarylsulfonyl)-phosphonic acids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1260, doi. 10.1080/14756366.2017.1378192

By:

Luisi, Grazia;
Angelini, Guido;
Gasbarri, Carla;
Laghezza, Antonio;
Agamennone, Mariangela;
Loiodice, Fulvio;
Supuran, Claudiu T.;
Campestre, Cristina;
Tortorella, Paolo

Publication type:

Article

Neem oil nanoemulsions: characterisation and antioxidant activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1265, doi. 10.1080/14756366.2017.1378190

By:

Rinaldi, Federica;
Hanieh, Patrizia Nadia;
Longhi, Catia;
Carradori, Simone;
Secci, Daniela;
Zengin, Gokhan;
Ammendolia, Maria Grazia;
Mattia, Elena;
Del Favero, Elena;
Marianecci, Carlotta;
Carafa, Maria

Publication type:

Article

Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1253, doi. 10.1080/14756366.2017.1375485

By:

Angeli, Andrea;
Vaiano, Fabio;
Mari, Francesco;
Bertol, Elisabetta;
Supuran, Claudiu T.

Publication type:

Article

Development of terphenyl-2-methyloxazol-5(4 H )-one derivatives as selective reversible MAGL inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1240, doi. 10.1080/14756366.2017.1375484

By:

Granchi, Carlotta;
Caligiuri, Isabella;
Bertelli, Eleonora;
Poli, Giulio;
Rizzolio, Flavio;
Macchia, Marco;
Martinelli, Adriano;
Minutolo, Filippo;
Tuccinardi, Tiziano

Publication type:

Article

Antimycobacterial activity of nitrogen heterocycles derivatives: 7-(pyridine-4-yl)-indolizine derivatives. Part VII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1291, doi. 10.1080/14756366.2017.1375483

By:

Olaru, Anda-Mihaela;
Vasilache, Violeta;
Danac, Ramona;
Mangalagiu, Ionel I.

Publication type:

Article

Characterization of human S-adenosyl-homocysteine hydrolase in vitro and identification of its potential inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1209, doi. 10.1080/14756366.2017.1370584

By:

Hao, Weiwei;
Li, Yanhua;
Shan, Qiuli;
Han, Tian;
Li, Wencheng;
He, Sheng;
Zhu, Kongkai;
Li, Yumei;
Tan, Xiaojun;
Gu, Jinsong

Publication type:

Article

Reactive oxygen species inhibit catalytic activity of peptidylarginine deiminase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1203, doi. 10.1080/14756366.2017.1368505

By:

Damgaard, Dres;
Bjørn, Mads Emil;
Jensen, Peter Østrup;
Nielsen, Claus Henrik

Publication type:

Article

Synthesis, in vitro antitumour activity, and molecular docking study of novel 2-substituted mercapto-3-(3,4,5-trimethoxybenzyl)-4(3H)-quinazolinone analogues.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1229, doi. 10.1080/14756366.2017.1368504

By:

El-Azab, Adel S.;
Abdel-Aziz, Alaa A.-M.;
Ghabbour, Hazem A.;
Al-Gendy, Manal A.

Publication type:

Article

α-Glucosidase inhibition by flavonoids: an in vitro and in silico structure–activity relationship study.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1216, doi. 10.1080/14756366.2017.1368503

By:

Proença, Carina;
Freitas, Marisa;
Ribeiro, Daniela;
Oliveira, Eduardo F. T.;
Sousa, Joana L. C.;
Tomé, Sara M.;
Ramos, Maria J.;
Silva, Artur M. S.;
Fernandes, Pedro A.;
Fernandes, Eduarda

Publication type:

Article

Inhibition of protein tyrosine phosphatase (PTP1B) and α-glucosidase by geranylated flavonoids from Paulownia tomentosa.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1195, doi. 10.1080/14756366.2017.1368502

By:

Song, Yeong Hun;
Uddin, Zia;
Jin, Young Min;
Li, Zuopeng;
Curtis-Long, Marcus John;
Kim, Kwang Dong;
Cho, Jung Keun;
Park, Ki Hun

Publication type:

Article

Synthesis and biological evaluation of aminomethyl and alkoxymethyl derivatives as carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1174, doi. 10.1080/14756366.2017.1368019

By:

Gulçin, İlhami;
Abbasova, Malahat;
Taslimi, Parham;
Huyut, Zübeyir;
Safarova, Leyla;
Sujayev, Afsun;
Farzaliyev, Vagif;
Beydemir, Şükrü;
Alwasel, Saleh H.;
Supuran, Claudiu T.

Publication type:

Article

Synthesis and biological evaluation of benzenesulphonamide-bearing 1,4,5-trisubstituted-1,2,3-triazoles possessing human carbonic anhydrase I, II, IV, and IX inhibitory activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1187, doi. 10.1080/14756366.2017.1367775

By:

Kumar, Rajiv;
Sharma, Vikas;
Bua, Silvia;
Supuran, Claudiu T.;
Sharma, Pawan K.

Publication type:

Article

Design, synthesis and biological activity of pyrazinamide derivatives for anti- Mycobacterium tuberculosis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1183, doi. 10.1080/14756366.2017.1367774

By:

Zhou, Shiyang;
Yang, Shanbin;
Huang, Gangliang

Publication type:

Article

The use of dimethylsulfoxide as a solvent in enzyme inhibition studies: the case of aldose reductase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1152, doi. 10.1080/14756366.2017.1363744

By:

Misuri, Livia;
Cappiello, Mario;
Balestri, Francesco;
Moschini, Roberta;
Barracco, Vito;
Mura, Umberto;
Del-Corso, Antonella

Publication type:

Article

New quinoxalinone inhibitors targeting secreted phospholipase A2 and α-glucosidase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1143, doi. 10.1080/14756366.2017.1363743

By:

Alasmary, Fatmah A. S.;
Alnahdi, Fatima S.;
Ben Bacha, Abir;
El-Araby, Amr M.;
Moubayed, Nadine;
Alafeefy, Ahmed M.;
El-Araby, Moustafa E.

Publication type:

Article

Novel series of 1,2,4-trioxane derivatives as antimalarial agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1159, doi. 10.1080/14756366.2017.1363742

By:

Rudrapal, Mithun;
Chetia, Dipak;
Singh, Vineeta

Publication type:

Article

Inhibition of human cytochromes P450 2A6 and 2A13 by flavonoids, acetylenic thiophenes and sesquiterpene lactones from Pluchea indica and Vernonia cinerea.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1136, doi. 10.1080/14756366.2017.1363741

By:

Boonruang, Supattra;
Prakobsri, Khanistha;
Pouyfung, Phisit;
Srisook, Ekaruth;
Prasopthum, Aruna;
Rongnoparut, Pornpimol;
Sarapusit, Songklod

Publication type:

Article

Multicomponent synthesis of some new (1 S ,4 S )-2,5-diazabicyclo[2.2.1]heptane-dithiocarbamates and their in vitro anti-proliferative activity against CaSki, MDA-MB-231 and SK-Lu-1 tumour cells as apoptosis inducing agents without necrosis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1129, doi. 10.1080/14756366.2017.1363197

By:

Laskar, Sujay;
Sánchez-Sánchez, Luis;
López-Ortiz, Manuel;
López-Muñoz, Hugo;
Escobar-Sánchez, María L.;
Sánchez, Arturo T.;
Regla, Ignacio

Publication type:

Article

Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1071, doi. 10.1080/14756366.2017.1356295

By:

Abdoli, Morteza;
Angeli, Andrea;
Bozdag, Murat;
Carta, Fabrizio;
Kakanejadifard, Ali;
Saeidian, Hamid;
Supuran, Claudiu T.

Publication type:

Article

A one-step procedure for immobilising the thermostable carbonic anhydrase (SspCA) on the surface membrane of Escherichia coli.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1120, doi. 10.1080/14756366.2017.1355794

By:

Del Prete, Sonia;
Perfetto, Rosa;
Rossi, Mosè;
Alasmary, Fatmah A. S.;
Osman, Sameh M.;
AlOthman, Zeid;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Allosteric inhibition of carnosinase (CN1) by inducing a conformational shift.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1102, doi. 10.1080/14756366.2017.1355793

By:

Peters, Verena;
Schmitt, Claus P.;
Weigand, Tim;
Klingbeil, Kristina;
Thiel, Christian;
van den Berg, Antje;
Calabrese, Vittorio;
Nawroth, Peter;
Fleming, Thomas;
Forsberg, Elisabete;
Wagner, Andreas H.;
Hecker, Markus;
Vistoli, Giulio

Publication type:

Article

Inhibition of dengue virus replication by novel inhibitors of RNA-dependent RNA polymerase and protease activities.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1091, doi. 10.1080/14756366.2017.1355791

By:

Pelliccia, Sveva;
Wu, Yu-Hsuan;
Coluccia, Antonio;
La Regina, Giuseppe;
Tseng, Chin-Kai;
Famiglini, Valeria;
Masci, Domiziana;
Hiscott, John;
Lee, Jin-Ching;
Silvestri, Romano

Publication type:

Article

Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1064, doi. 10.1080/14756366.2017.1355307

By:

Nocentini, Alessio;
Vullo, Daniela;
Del Prete, Sonia;
Osman, Sameh M.;
Alasmary, Fatmah A.S.;
AlOthman, Zeid;
Capasso, Clemente;
Carta, Fabrizio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Quantitative assessment of specific carbonic anhydrase inhibitors effect on hypoxic cells using electrical impedance assays.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1079, doi. 10.1080/14756366.2017.1355306

By:

Stanica, Luciana;
Gheorghiu, Mihaela;
Stan, Miruna;
Polonschii, Cristina;
David, Sorin;
Bratu, Dumitru;
Dinischiotu, Anca;
Supuran, Claudiu T.;
Gheorghiu, Eugen

Publication type:

Article

Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1053, doi. 10.1080/14756366.2017.1354858

By:

Campestre, Cristina;
Locatelli, Marcello;
Guglielmi, Paolo;
De Luca, Elisa;
Bellagamba, Giuseppe;
Menta, Sergio;
Zengin, Gokhan;
Celia, Christian;
Di Marzio, Luisa;
Carradori, Simone

Publication type:

Article

Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1042, doi. 10.1080/14756366.2017.1354857

By:

Zengin Kurt, Belma;
Sonmez, Fatih;
Durdagi, Serdar;
Aksoydan, Busecan;
Ekhteiari Salmas, Ramin;
Angeli, Andrea;
Kucukislamoglu, Mustafa;
Supuran, Claudiu T.

Publication type:

Article

Cloning, expression and purification of the α-carbonic anhydrase from the mantle of the Mediterranean mussel, Mytilus galloprovincialis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1029, doi. 10.1080/14756366.2017.1353502

By:

Perfetto, Rosa;
Del Prete, Sonia;
Vullo, Daniela;
Carginale, Vincenzo;
Sansone, Giovanni;
Barone, Carmela M. A.;
Rossi, Mosè;
Alasmary, Fatmah A. S.;
Osman, Sameh M.;
AlOthman, Zeid;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

New sulfurated derivatives of cinnamic acids and rosmaricine as inhibitors of STAT3 and NF-κB transcription factors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1012, doi. 10.1080/14756366.2017.1350658

By:

Gabriele, Elena;
Brambilla, Dario;
Ricci, Chiara;
Regazzoni, Luca;
Taguchi, Kyoko;
Ferri, Nicola;
Asai, Akira;
Sparatore, Anna

Publication type:

Article

Insights into the binding mode of sulphamates and sulphamides to hCA II: crystallographic studies and binding free energy calculations.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1002, doi. 10.1080/14756366.2017.1349764

By:

De Simone, Giuseppina;
Langella, Emma;
Esposito, Davide;
Supuran, Claudiu T.;
Monti, Simona Maria;
Winum, Jean-Yves;
Alterio, Vincenzo

Publication type:

Article

Design and synthesis of benzopyran-based inhibitors of the hypoxia-inducible factor-1 pathway with improved water solubility.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 992, doi. 10.1080/14756366.2017.1347784

By:

Ferguson, Jalisa H.;
De Los Santos, Zeus;
Devi, Saroja N.;
Kaluz, Stefan;
Van Meir, Erwin G.;
Zingales, Sarah K.;
Wang, Binghe

Publication type:

Article

Rosmarinic acid prevents fibrillization and diminishes vibrational modes associated to β sheet in tau protein linked to Alzheimer’s disease.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 945, doi. 10.1080/14756366.2017.1347783

By:

Cornejo, Alberto;
Aguilar Sandoval, Felipe;
Caballero, Leonardo;
Machuca, Luis;
Muñoz, Patricio;
Caballero, Julio;
Perry, George;
Ardiles, Alejandro;
Areche, Carlos;
Melo, Francisco

Publication type:

Article

Water permeability is a measure of severity in acute appendicitis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1036, doi. 10.1080/14756366.2017.1347167

By:

Pini, Nicola;
Pfeifle, Viktoria A.;
Kym, Urs;
Keck, Simone;
Galati, Virginie;
Holland-Cunz, Stefan;
Gros, Stephanie J.

Publication type:

Article

Cancer stem cells CD133 inhibition and cytotoxicity of certain 3-phenylthiazolo[3,2- a ]benzimidazoles: design, direct synthesis, crystal study and in vitro biological evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 986, doi. 10.1080/14756366.2017.1347166

By:

Al-Ansary, Ghada H.;
Eldehna, Wagdy M.;
Ghabbour, Hazem A.;
Al-Rashood, Sara T. A.;
Al-Rashood, Khalid A.;
Eladwy, Radwa A.;
Al-Dhfyan, Abdullah;
Kabil, Maha M.;
Abdel-Aziz, Hatem A.

Publication type:

Article

Kinetic study on the inhibition of xanthine oxidase by acylated derivatives of flavonoids synthesised enzymatically.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 978, doi. 10.1080/14756366.2017.1347165

By:

de Araújo, Maria Elisa Melo Branco;
Franco, Yollanda Edwirges Moreira;
Alberto, Thiago Grando;
Messias, Marcia Cristina Fernandes;
Leme, Camila Wielewski;
Sawaya, Alexandra Christine Helena Frankland;
Carvalho, Patricia de Oliveira

Publication type:

Article

Discovery of novel isoflavone derivatives as AChE/BuChE dual-targeted inhibitors: synthesis, biological evaluation and molecular modelling.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 968, doi. 10.1080/14756366.2017.1347163

By:

Feng, Bo;
Li, Xinpeng;
Xia, Jie;
Wu, Song

Publication type:

Article

Synthesis and biological evaluation of novel 7-hydroxy-4-phenylchromen-2-one–linked to triazole moieties as potent cytotoxic agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1111, doi. 10.1080/14756366.2017.1344982

By:

Liu, Chuan-Feng;
Shen, Qing-Kun;
Li, Jia-Jun;
Tian, Yu-Shun;
Quan, Zheshan

Publication type:

Article

Synthesis, anticancer and apoptosis-inducing activities of quinazoline–isatin conjugates: epidermal growth factor receptor-tyrosine kinase assay and molecular docking studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 935, doi. 10.1080/14756366.2017.1344981

By:

El-Azab, Adel S.;
Al-Dhfyan, Abdullah;
Abdel-Aziz, Alaa A.-M.;
Abou-Zeid, Laila A.;
Alkahtani, Hamad M.;
Al-Obaid, Abdulrahman M.;
Al-Gendy, Manal A.

Publication type:

Article

Subnanomolar indazole-5-carboxamide inhibitors of monoamine oxidase B (MAO-B) continued: indications of iron binding, experimental evidence for optimised solubility and brain penetration.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 960, doi. 10.1080/14756366.2017.1344980

By:

Tzvetkov, Nikolay T.;
Antonov, Liudmil

Publication type:

Article

Design and synthesis of a novel photoaffinity probe for labelling EGF receptor tyrosine kinases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 954, doi. 10.1080/14756366.2017.1344979

By:

Zheng, You-Guang;
Wu, Xiao-Qing;
Su, Jun;
Jiang, Ping;
Xu, Liang;
Gao, Jian;
Cai, Bin;
Ji, Min

Publication type:

Article

Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 920, doi. 10.1080/14756366.2017.1344236

By:

Krasavin, Mikhail;
Korsakov, Mikhail;
Ronzhina, Oksana;
Tuccinardi, Tiziano;
Kalinin, Stanislav;
Tanç, Muhammet;
Supuran, Claudiu T.

Publication type:

Article

Beta-lactamase database (BLDB) – structure and function.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 917, doi. 10.1080/14756366.2017.1344235

By:

Naas, Thierry;
Oueslati, Saoussen;
Bonnin, Rémy A.;
Dabos, Maria Laura;
Zavala, Agustin;
Dortet, Laurent;
Retailleau, Pascal;
Iorga, Bogdan I.

Publication type:

Article

Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 885, doi. 10.1080/14756366.2017.1337759

By:

Bozdag, Murat;
Bua, Silvia;
Osman, Sameh M.;
AlOthman, Zeid;
Supuran, Claudiu T.

Publication type:

Article

Syntheses and evaluation of multicaulin and miltirone-like compounds as antituberculosis agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 878, doi. 10.1080/14756366.2017.1337758

By:

Burmaoğlu, Serdar;
Seçinti, Hatice;
Mozioğlu, Erkan;
Gören, Ahmet C.;
Altundaş, Ramazan;
Seçen, Hasan

Publication type:

Article

Natural extracellular nanovesicles and photodynamic molecules: is there a future for drug delivery?

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 908, doi. 10.1080/14756366.2017.1335310

By:

Kusuzaki, Katsuyuki;
Matsubara, Takao;
Murata, Hiroaki;
Logozzi, Mariantonia;
Iessi, Elisabetta;
Di Raimo, Rossella;
Carta, Fabrizio;
Supuran, Claudiu T.;
Fais, Stefano

Publication type:

Article

VEGFR-2 inhibitors and apoptosis inducers: synthesis and molecular design of new benzo [g] quinazolin bearing benzenesulfonamide moiety.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 893, doi. 10.1080/14756366.2017.1334650

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Soliman, Aiten M.;
Ragab, Fatma A.

Publication type:

Article