Works matching IS 1475-6366 AND VI 32 AND IP 1 AND DT 2017
Results: 143
Editorial Board.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. ebi, doi. 10.1080/14756366.2017.1398806
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Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1305, doi. 10.1080/14756366.2017.1386660
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In vitro and in vivo antitumour effects of phenylboronic acid against mouse mammary adenocarcinoma 4T1 and squamous carcinoma SCCVII cells.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1299, doi. 10.1080/14756366.2017.1384823
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Resveratrol-based cinnamic ester hybrids: synthesis, characterization, and anti-inflammatory activity.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1282, doi. 10.1080/14756366.2017.1381090
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Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1274, doi. 10.1080/14756366.2017.1380638
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Dual targeting of cancer-related human matrix metalloproteinases and carbonic anhydrases by chiral N -(biarylsulfonyl)-phosphonic acids.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1260, doi. 10.1080/14756366.2017.1378192
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Neem oil nanoemulsions: characterisation and antioxidant activity.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1265, doi. 10.1080/14756366.2017.1378190
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Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1253, doi. 10.1080/14756366.2017.1375485
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Development of terphenyl-2-methyloxazol-5(4 H )-one derivatives as selective reversible MAGL inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1240, doi. 10.1080/14756366.2017.1375484
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Antimycobacterial activity of nitrogen heterocycles derivatives: 7-(pyridine-4-yl)-indolizine derivatives. Part VII.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1291, doi. 10.1080/14756366.2017.1375483
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Characterization of human S-adenosyl-homocysteine hydrolase in vitro and identification of its potential inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1209, doi. 10.1080/14756366.2017.1370584
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Reactive oxygen species inhibit catalytic activity of peptidylarginine deiminase.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1203, doi. 10.1080/14756366.2017.1368505
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Synthesis, in vitro antitumour activity, and molecular docking study of novel 2-substituted mercapto-3-(3,4,5-trimethoxybenzyl)-4(3H)-quinazolinone analogues.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1229, doi. 10.1080/14756366.2017.1368504
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α-Glucosidase inhibition by flavonoids: an in vitro and in silico structure–activity relationship study.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1216, doi. 10.1080/14756366.2017.1368503
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Inhibition of protein tyrosine phosphatase (PTP1B) and α-glucosidase by geranylated flavonoids from Paulownia tomentosa.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1195, doi. 10.1080/14756366.2017.1368502
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Novel series of 1,2,4-trioxane derivatives as antimalarial agents.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1159, doi. 10.1080/14756366.2017.1363742
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Inhibition of human cytochromes P450 2A6 and 2A13 by flavonoids, acetylenic thiophenes and sesquiterpene lactones from Pluchea indica and Vernonia cinerea.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1136, doi. 10.1080/14756366.2017.1363741
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Design, synthesis and biological activity of pyrazinamide derivatives for anti- Mycobacterium tuberculosis.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1183, doi. 10.1080/14756366.2017.1367774
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The use of dimethylsulfoxide as a solvent in enzyme inhibition studies: the case of aldose reductase.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1152, doi. 10.1080/14756366.2017.1363744
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New quinoxalinone inhibitors targeting secreted phospholipase A2 and α-glucosidase.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1143, doi. 10.1080/14756366.2017.1363743
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Synthesis and biological evaluation of aminomethyl and alkoxymethyl derivatives as carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1174, doi. 10.1080/14756366.2017.1368019
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Synthesis and biological evaluation of benzenesulphonamide-bearing 1,4,5-trisubstituted-1,2,3-triazoles possessing human carbonic anhydrase I, II, IV, and IX inhibitory activity.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1187, doi. 10.1080/14756366.2017.1367775
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Multicomponent synthesis of some new (1 S ,4 S )-2,5-diazabicyclo[2.2.1]heptane-dithiocarbamates and their in vitro anti-proliferative activity against CaSki, MDA-MB-231 and SK-Lu-1 tumour cells as apoptosis inducing agents without necrosis.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1129, doi. 10.1080/14756366.2017.1363197
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Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1071, doi. 10.1080/14756366.2017.1356295
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A one-step procedure for immobilising the thermostable carbonic anhydrase (SspCA) on the surface membrane of Escherichia coli.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1120, doi. 10.1080/14756366.2017.1355794
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Allosteric inhibition of carnosinase (CN1) by inducing a conformational shift.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1102, doi. 10.1080/14756366.2017.1355793
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Inhibition of dengue virus replication by novel inhibitors of RNA-dependent RNA polymerase and protease activities.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1091, doi. 10.1080/14756366.2017.1355791
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Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1064, doi. 10.1080/14756366.2017.1355307
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Quantitative assessment of specific carbonic anhydrase inhibitors effect on hypoxic cells using electrical impedance assays.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1079, doi. 10.1080/14756366.2017.1355306
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Design and synthesis of benzopyran-based inhibitors of the hypoxia-inducible factor-1 pathway with improved water solubility.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 992, doi. 10.1080/14756366.2017.1347784
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Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1042, doi. 10.1080/14756366.2017.1354857
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Cloning, expression and purification of the α-carbonic anhydrase from the mantle of the Mediterranean mussel, Mytilus galloprovincialis.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1029, doi. 10.1080/14756366.2017.1353502
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New sulfurated derivatives of cinnamic acids and rosmaricine as inhibitors of STAT3 and NF-κB transcription factors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1012, doi. 10.1080/14756366.2017.1350658
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Insights into the binding mode of sulphamates and sulphamides to hCA II: crystallographic studies and binding free energy calculations.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1002, doi. 10.1080/14756366.2017.1349764
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Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1053, doi. 10.1080/14756366.2017.1354858
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Rosmarinic acid prevents fibrillization and diminishes vibrational modes associated to β sheet in tau protein linked to Alzheimer’s disease.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 945, doi. 10.1080/14756366.2017.1347783
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Water permeability is a measure of severity in acute appendicitis.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1036, doi. 10.1080/14756366.2017.1347167
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Cancer stem cells CD133 inhibition and cytotoxicity of certain 3-phenylthiazolo[3,2- a ]benzimidazoles: design, direct synthesis, crystal study and in vitro biological evaluation.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 986, doi. 10.1080/14756366.2017.1347166
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Discovery of novel isoflavone derivatives as AChE/BuChE dual-targeted inhibitors: synthesis, biological evaluation and molecular modelling.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 968, doi. 10.1080/14756366.2017.1347163
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Kinetic study on the inhibition of xanthine oxidase by acylated derivatives of flavonoids synthesised enzymatically.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 978, doi. 10.1080/14756366.2017.1347165
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Synthesis and biological evaluation of novel 7-hydroxy-4-phenylchromen-2-one–linked to triazole moieties as potent cytotoxic agents.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1111, doi. 10.1080/14756366.2017.1344982
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Synthesis, anticancer and apoptosis-inducing activities of quinazoline–isatin conjugates: epidermal growth factor receptor-tyrosine kinase assay and molecular docking studies.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 935, doi. 10.1080/14756366.2017.1344981
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Subnanomolar indazole-5-carboxamide inhibitors of monoamine oxidase B (MAO-B) continued: indications of iron binding, experimental evidence for optimised solubility and brain penetration.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 960, doi. 10.1080/14756366.2017.1344980
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Design and synthesis of a novel photoaffinity probe for labelling EGF receptor tyrosine kinases.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 954, doi. 10.1080/14756366.2017.1344979
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Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 920, doi. 10.1080/14756366.2017.1344236
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Beta-lactamase database (BLDB) – structure and function.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 917, doi. 10.1080/14756366.2017.1344235
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Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 885, doi. 10.1080/14756366.2017.1337759
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Syntheses and evaluation of multicaulin and miltirone-like compounds as antituberculosis agents.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 878, doi. 10.1080/14756366.2017.1337758
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Natural extracellular nanovesicles and photodynamic molecules: is there a future for drug delivery?
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 908, doi. 10.1080/14756366.2017.1335310
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VEGFR-2 inhibitors and apoptosis inducers: synthesis and molecular design of new benzo [g] quinazolin bearing benzenesulfonamide moiety.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 893, doi. 10.1080/14756366.2017.1334650
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