Works in Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, Vol 30, Issue 6

Results: 25

Editorial Board.

Published in:: Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. ebi, doi. 10.3109/14756366.2015.1113026
Publication type:: Article

The impact of hydroquinone on acetylcholine esterase and certain human carbonic anhydrase isoenzymes (hCA I, II, IX, and XII).

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 941, doi. 10.3109/14756366.2014.999236

By:

Scozzafava, Andrea;
Kalın, Pınar;
Supuran, Claudiu T.;
Gülçin, İlhami;
Alwasel, Saleh H.

Publication type:

Article

Chemical constituents of Hericium erinaceum associated with the inhibitory activity against cellular senescence in human umbilical vascular endothelial cells.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 934, doi. 10.3109/14756366.2014.995181

By:

Noh, Hyung Jun;
Yang, Hyo Hyun;
Kim, Geum Soog;
Lee, Seung Eun;
Lee, Dae Young;
Choi, Je Hun;
Kim, Seung Yu;
Lee, Eun Suk;
Ji, Seung Heon;
Kang, Ki Sung;
Park, Hye-Jin;
Kim, Jae-Ryong;
Kim, Ki Hyun

Publication type:

Article

Studies on the antiplatelet and antithrombotic profile of anti-inflammatory coumarin derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 925, doi. 10.3109/14756366.2014.995180

By:

Kontogiorgis, Christos;
Nicolotti, Orazio;
Mangiatordi, Giuseppe Felice;
Tognolini, Massimiliano;
Karalaki, Foteini;
Giorgio, Carmine;
Patsilinakos, Alexandros;
Carotti, Angelo;
Hadjipavlou-Litina, Dimitra;
Barocelli, Elisabetta

Publication type:

Article

Search for human DNA topoisomerase II poisons in the group of 2,5-disubstituted-1,3,4-thiadiazoles.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 1021, doi. 10.3109/14756366.2014.995179

By:

Plech, Tomasz;
Kaproń, Barbara;
Paneth, Agata;
Wujec, Monika;
Czarnomysy, Robert;
Bielawska, Anna;
Bielawski, Krzysztof;
Trotsko, Nazar;
Kuśmierz, Edyta;
Paneth, Piotr

Publication type:

Article

Protonography, a technique applicable for the analysis of η -carbonic anhydrase activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 920, doi. 10.3109/14756366.2014.990963

By:

Del Prete, Sonia;
De Luca, Viviana;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 908, doi. 10.3109/14756366.2014.987138

By:

D'Ascenzio, Melissa;
Chimenti, Paola;
Gidaro, Maria Concetta;
De Monte, Celeste;
De Vita, Daniela;
Granese, Arianna;
Scipione, Luigi;
Di Santo, Roberto;
Costa, Giosuè;
Alcaro, Stefano;
Yáñez, Matilde;
Carradori, Simone

Publication type:

Article

High-efficient synthesis and biological activities of allosamidins.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 863, doi. 10.3109/14756366.2014.987137

By:

Huang, Gangliang;
Peng, Daquan;
Mei, Xinya;
Chen, Xin;
Xiao, Feng;
Tang, Qilin

Publication type:

Article

Inhibition of β -carbonic anhydrases from Brucella suis with C -cinnamoyl glycosides incorporating the phenol moiety.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 1017, doi. 10.3109/14756366.2014.986120

By:

Riafrecha, Leonardo E.;
Vullo, Daniela;
Ouahrani-Bettache, Safia;
Köhler, Stephan;
Dumy, Pascal;
Winum, Jean-Yves;
Supuran, Claudiu T.;
Colinas, Pedro A.

Publication type:

Article

N-glycosyl-N-hydroxysulfamides as potent inhibitors of Brucella suis carbonic anhydrases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 1010, doi. 10.3109/14756366.2014.986119

By:

Ombouma, Joanna;
Vullo, Daniela;
Köhler, Stephan;
Dumy, Pascal;
Supuran, Claudiu T.;
Winum, Jean-Yves

Publication type:

Article

Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 901, doi. 10.3109/14756366.2014.986118

By:

Singasane, Namrata;
Kharkar, Prashant S.;
Ceruso, Mariangela;
Supuran, Claudiu T.;
Toraskar, Mrunmayee P.

Publication type:

Article

Synthesis of 3,4-dihydroxypyrrolidine-2,5-dione and 3,5-dihydroxybenzoic acid derivatives and evaluation of the carbonic anhydrase I and II inhibition.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 896, doi. 10.3109/14756366.2014.983917

By:

Arslan, Mehmet;
Şentürk, Murat;
Fidan, İsmail;
Talaz, Oktay;
Ekinci, Deniz;
Coşgun, Sedat;
Supuran, Claudiu T.

Publication type:

Article

Design and synthesis of resveratrol–salicylate hybrid derivatives as CYP1A1 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 884, doi. 10.3109/14756366.2014.979347

By:

Aldawsari, Fahad S.;
Elshenawy, Osama H.;
El Gendy, Mohamed A. M.;
Aguayo-Ortiz, Rodrigo;
Baksh, Shairaz;
El-Kadi, Ayman O. S.;
Velázquez-Martínez, Carlos A.

Publication type:

Article

Design, synthesis and bioevaluation of novel umbelliferone analogues as potential mushroom tyrosinase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 874, doi. 10.3109/14756366.2014.979346

By:

Ashraf, Zaman;
Rafiq, Muhammad;
Seo, Sung-Yum;
Babar, Mustafeez Mujtaba;
Zaidi, Najam-us-Sahar Sadaf

Publication type:

Article

Perturbation response scanning specifies key regions in subtilisin serine protease for both function and stability.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 867, doi. 10.3109/14756366.2014.979345

By:

Abdizadeh, Haleh;
Guven, Gokce;
Atilgan, Ali Rana;
Atilgan, Canan

Publication type:

Article

Production of collagen micro- and nanofibers for potential drug-carrier systems.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 1013, doi. 10.3109/14756366.2014.976567

By:

Aras, Onur;
Kazanci, Murat

Publication type:

Article

Synthesis of some novel heterocylic compounds derived from 2-[3-(4-chlorophenyl)-5-(4-methoxybenzyl)-4H-1,2,4-triazol-4-yl]acetohydrazide and investigation of their lipase and α -glucosidase inhibition.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 1002, doi. 10.3109/14756366.2014.1003213

By:

Bekircan, Olcay;
Ülker, Serdar;
Menteşe, Emre

Publication type:

Article

Tacrine–propargylamine derivatives with improved acetylcholinesterase inhibitory activity and lower hepatotoxicity as a potential lead compound for the treatment of Alzheimer’s disease.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 995, doi. 10.3109/14756366.2014.1003212

By:

Mao, Fei;
Li, Jianheng;
Wei, Hui;
Huang, Ling;
Li, Xingshu

Publication type:

Article

A failed tentative to design a super carbonic anhydrase having the biochemical properties of the most thermostable CA (SspCA) and the fastest (SazCA) enzymes.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 989, doi. 10.3109/14756366.2014.1002403

By:

De Luca, Viviana;
Del Prete, Sonia;
Carginale, Vincenzo;
Vullo, Daniela;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Anagliptin, a potent dipeptidyl peptidase IV inhibitor: its single-crystal structure and enzyme interactions.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 981, doi. 10.3109/14756366.2014.1002402

By:

Watanabe, Yukihisa S.;
Yasuda, Yoshika;
Kojima, Yuko;
Okada, Shino;
Motoyama, Tomoko;
Takahashi, Ryo;
Oka, Mitsuru

Publication type:

Article

Synthesis and evaluation of biological and antitumor activities of 5,7-dimethyl- oxazolo[5,4- d ]pyrimidine-4,6(5 H ,7 H )-dione derivatives as novel inhibitors of FGFR1.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 961, doi. 10.3109/14756366.2014.1002401

By:

Ye, Faqing;
Wang, Yuewu;
Nian, Siyun;
Wang, Yu;
Chen, Di;
Yu, Shufang;
Wang, Sicen

Publication type:

Article

Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti- Helicobacter pylori , anti-malarial and anti-leishmanial agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 1027, doi. 10.3109/14756366.2014.1001755

By:

De Monte, Celeste;
Bizzarri, Bruna;
Gidaro, Maria Concetta;
Carradori, Simone;
Mollica, Adriano;
Luisi, Grazia;
Granese, Arianna;
Alcaro, Stefano;
Costa, Giosuè;
Basilico, Nicoletta;
Parapini, Silvia;
Scaltrito, Maria Maddalena;
Masia, Carla;
Sisto, Francesca

Publication type:

Article

Esterase activity of carbonic anhydrases serves as surrogate for selecting antibodies blocking hydratase activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 955, doi. 10.3109/14756366.2014.1001754

By:

Uda, Narasimha Rao;
Seibert, Volker;
Stenner-Liewen, Frank;
Müller, Philipp;
Herzig, Petra;
Gondi, Gabor;
Zeidler, Reinhard;
van Dijk, Marc;
Zippelius, Alfred;
Renner, Christoph

Publication type:

Article

Kinetic characterization of 4,4′-biphenylsulfonamides as selective non-zinc binding MMP inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 947, doi. 10.3109/14756366.2014.1000889

By:

Santamaria, Salvatore;
Nuti, Elisa;
Cercignani, Giovanni;
La Regina, Giuseppe;
Silvestri, Romano;
Supuran, Claudiu T.;
Rossello, Armando

Publication type:

Article

Synthesis of pro-apoptotic indapamide derivatives as anticancer agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 967, doi. 10.3109/14756366.2014.1001756

By:

Yılmaz, Özgür;
Özbaş Turan, Suna;
Akbuğa, Jülide;
Tiber, Pınar Mega;
Orun, Oya;
Supuran, Claudiu T.;
Küçükgüzel, Ş. Güniz

Publication type:

Article