Works in Journal of Labelled Compounds & Radiopharmaceuticals, 2013, Vol 56, Issue 9/10

Results: 24

A perspective on tritium versus carbon-14: ensuring optimal label selection in pharmaceutical research and development.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 441, doi. 10.1002/jlcr.3085

By:

Krauser, Joel A.

Publication type:

Article

Syntheses of C-13 and C-14-labeled versions of the investigational proteasome inhibitor MLN9708.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 464, doi. 10.1002/jlcr.3079

By:

Plesescu, Mihaela;
Elliott, Eric L.;
Li, Yuexian;
Prakash, Shimoga R.

Publication type:

Article

Biodistribution (as determined by the radiolabelled equivalent) of a gold(III) bis(pyrrolide-imine) Schiff base complex: a potential chemotherapeutic.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 530, doi. 10.1002/jlcr.3068

By:

Akerman, Matthew P.;
Munro, Orde Q.;
Mongane, Modisenyane;
Staden, Johan A.;
Rae, William I. D.;
Bester, Cornelius J.;
Marjanovic Painter, Biljana;
Szucs, Zoltan;
Zeevaart, Jan Rijn

Publication type:

Article

11th International Isotope Symposium on the Synthesis and Applications of Isotopes and Isotopically Labelled Compounds (IIS2012).

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 397, doi. 10.1002/jlcr.3101

By:

Atzrodt, Jens;
Derdau, Volker;
Allen, John

Publication type:

Article

Kinetic deuterium isotope effects in cytochrome P450 oxidation reactions.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 428, doi. 10.1002/jlcr.3031

By:

Guengerich, F. Peter

Publication type:

Article

18F-labeled folic acid derivatives for imaging of the folate receptor via positron emission tomography.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 432, doi. 10.1002/jlcr.3104

By:

Schieferstein, Hanno;
Ross, Tobias L.

Publication type:

Article

Imaging agent of a TRPA1 inhibitor.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 536, doi. 10.1002/jlcr.3030

By:

Malmquist, Jonas;
Bernlind, Alexandra;
Lindberg, Sandra

Publication type:

Article

Scientific Program IIS2012, Heidelberg.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 399, doi. 10.1002/jlcr.3100

By:

Atzrodt, Jens;
Derdau, Volker;
Allen, John

Publication type:

Article

Selected Scientific Topics of the 11th International Isotope Symposium on the Synthesis and Applications of Isotopes and Isotopically Labeled Compounds.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 408, doi. 10.1002/jlcr.3096

By:

Atzrodt, Jens;
Derdau, Volker

Publication type:

Article

Preparation of [3H]fluoroethyl tosylate and its use in the labelling of the dopamine transporter radioligand [3H]FE-PE2I.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 447, doi. 10.1002/jlcr.3012

By:

Cochrane, Alison R;
Kerr, William John;
Sandell, Johan

Publication type:

Article

Carbon-14 labelled Tribendimidine, a broad-spectrum anthelmintic drug.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 471, doi. 10.1002/jlcr.3070

By:

Fontana, Erminia;
Pignatti, Alberto;
Ghiglieri, Alberto;
Battaglia, Rosangela;
Cinato, Flavio;
Wang, Chong;
Hostos, Eugenio

Publication type:

Article

Melvin Calvin award lecture, Isotopic chemistry: the most varied of careers...with tritium and deuterium the most versatile of the isotopes.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 417, doi. 10.1002/jlcr.3045

By:

Lockley, William J. S.

Publication type:

Article

Synthesis of isotopically labeled versions of L-MTP-PE (mifamurtide) and MDP.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 475, doi. 10.1002/jlcr.3078

By:

Li, Yuexian;
Plesescu, Mihaela;
Prakash, Shimoga R.

Publication type:

Article

Radiolabelling of steroids: the synthesis of 17 α-[4-14C]trenbolone.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 455, doi. 10.1002/jlcr.3089

By:

Hendry, David;
Knagg, Eric;
Smith, Neil A.;
Woolley, Geoffrey T.

Publication type:

Article

Preparation of labeled human drug metabolites and drug-drug interaction-probes with fungal peroxygenases.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 513, doi. 10.1002/jlcr.3103

By:

Poraj Kobielska, Marzena;
Atzrodt, Jens;
Holla, Wolfgang;
Sandvoss, Martin;
Gröbe, Glenn;
Scheibner, Katrin;
Hofrichter, Martin

Publication type:

Article

Editorial Board.

Published in:: Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. i, doi. 10.1002/jlcr.3132
Publication type:: Article

Production of high specific activity 195mPt-cisplatinum at South African Nuclear Energy Corporation for Phase 0 clinical trials in healthy individual subjects.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 495, doi. 10.1002/jlcr.3091

By:

Zeevaart, Jan Rijn;
Wagener, Judith;
Marjanovic Painter, Biljana;
Sathekge, Mike;
Soni, Nischal;
Zinn, Christa;
Perkins, Gary;
Smith, Suzanne V.

Publication type:

Article

Syntheses of 3H-labeled, 14C-labeled, and 2H4-labeled SCH 444877, phosphodiesterase type 5 inhibitors.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 480, doi. 10.1002/jlcr.3080

By:

Ren, Sumei;
Hesk, David;
McNamara, Paul;
Koharski, David;
Hendershot, Sharon

Publication type:

Article

Application of neutral iridium(I) N-heterocyclic carbene complexes in ortho-directed hydrogen isotope exchange.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 451, doi. 10.1002/jlcr.3084

By:

Cochrane, Alison R.;
Irvine, Stephanie;
Kerr, William J.;
Reid, Marc;
Andersson, Shalini;
Nilsson, Göran N.

Publication type:

Article

Carbon-14 labeling of K777•HCl, a therapeutic agent for Chagas disease.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 461, doi. 10.1002/jlcr.3107

By:

Rhee, Sung Whi;
Bradford, Wallace W.;
Malerich, Jeremiah P.;
Tanga, Mary J.

Publication type:

Article

The synthesis of a carbon-14 labeled pegylated Adnectin™ for placental transfer studies in guinea pigs.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 492, doi. 10.1002/jlcr.3077

By:

Maxwell, Brad D.;
Cao, Kai;
Bonacorsi, Samuel;
Sivaraman, Lakshmi;
Wang, Bonnie;
McNerney, MaryEllen;
Wang, Lifei;
Christopher, Lisa J.;
Fung, Nga Kit Eliza;
Wang, Jian;
Arnold, Mark E.

Publication type:

Article

Synthesis of deuterated [D32]oleic acid and its phospholipid derivative [D64]dioleoyl- sn-glycero-3-phosphocholine.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 520, doi. 10.1002/jlcr.3088

By:

Darwish, Tamim A.;
Luks, Emily;
Moraes, Greta;
Yepuri, Nageshwar R.;
Holden, Peter J.;
James, Michael

Publication type:

Article

A convergent stereocontrolled synthesis of [3-14C]solanesol.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 485, doi. 10.1002/jlcr.3083

By:

Roe, Stephen J.;
Oldfield, Mark F.;
Geach, Neil;
Baxter, Andrew

Publication type:

Article

Effect of deuteration on the metabolism and clearance of some pharmacologically active compounds-synthesis and in vitro metabolism of deuterated derivatives of dronedadrone.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2013, v. 56, n. 9/10, p. 504, doi. 10.1002/jlcr.3090

By:

Schofield, Joseph;
Brasseur, Denis;
Bruin, Béatrice;
Vassal, Thierry;
Klieber, Sylvie;
Arabeyre, Catherine;
Bourrié, Martine;
Sadoun, Freddy;
Fabre, Gérard

Publication type:

Article

Works in Journal of Labelled Compounds & Radiopharmaceuticals, 2013, Vol 56, Issue 9/10

A perspective on tritium versus carbon-14: ensuring optimal label selection in pharmaceutical research and development.

Syntheses of C-13 and C-14-labeled versions of the investigational proteasome inhibitor MLN9708.

Biodistribution (as determined by the radiolabelled equivalent) of a gold(III) bis(pyrrolide-imine) Schiff base complex: a potential chemotherapeutic.

11th International Isotope Symposium on the Synthesis and Applications of Isotopes and Isotopically Labelled Compounds (IIS2012).

Kinetic deuterium isotope effects in cytochrome P450 oxidation reactions.

<sup>18</sup>F-labeled folic acid derivatives for imaging of the folate receptor via positron emission tomography.

Imaging agent of a TRPA1 inhibitor.

Scientific Program IIS2012, Heidelberg.

Selected Scientific Topics of the 11th International Isotope Symposium on the Synthesis and Applications of Isotopes and Isotopically Labeled Compounds.

Preparation of [<sup>3</sup>H]fluoroethyl tosylate and its use in the labelling of the dopamine transporter radioligand [<sup>3</sup>H]FE-PE2I.

Carbon-14 labelled Tribendimidine, a broad-spectrum anthelmintic drug.

Melvin Calvin award lecture, Isotopic chemistry: the most varied of careers...with tritium and deuterium the most versatile of the isotopes.

Synthesis of isotopically labeled versions of L-MTP-PE (mifamurtide) and MDP.

Radiolabelling of steroids: the synthesis of 17 α-[4-<sup>14</sup>C]trenbolone.

Preparation of labeled human drug metabolites and drug-drug interaction-probes with fungal peroxygenases.

Editorial Board.

Production of high specific activity <sup>195m</sup>Pt-cisplatinum at South African Nuclear Energy Corporation for Phase 0 clinical trials in healthy individual subjects.

Syntheses of <sup>3</sup>H-labeled, <sup>14</sup>C-labeled, and <sup>2</sup>H<sub>4</sub>-labeled SCH 444877, phosphodiesterase type 5 inhibitors.

Application of neutral iridium(I) N-heterocyclic carbene complexes in ortho-directed hydrogen isotope exchange.

Carbon-14 labeling of K777•HCl, a therapeutic agent for Chagas disease.

The synthesis of a carbon-14 labeled pegylated Adnectin™ for placental transfer studies in guinea pigs.

Synthesis of deuterated [D<sub>32</sub>]oleic acid and its phospholipid derivative [D<sub>64</sub>]dioleoyl- sn-glycero-3-phosphocholine.

A convergent stereocontrolled synthesis of [3-<sup>14</sup>C]solanesol.

Effect of deuteration on the metabolism and clearance of some pharmacologically active compounds-synthesis and in vitro metabolism of deuterated derivatives of dronedadrone.