Works matching IS 00071188 AND DT 2015 AND VI 172 AND IP 5

Results: 22

AQW051, a novel, potent and selective α7 nicotinic ACh receptor partial agonist: pharmacological characterization and phase I evaluation.

Published in:

2015

By:

Feuerbach, Dominik;
Pezous, Nicole;
Weiss, Markus;
Shakeri-Nejad, Kasra;
Lingenhoehl, Kurt;
Hoyer, Daniel;
Hurth, Konstanze;
Bilbe, Graeme;
Pryce, Christopher R;
McAllister, Kevin;
Chaperon, Frederique;
Kucher, Klaus;
Johns, Donald;
Blaettler, Thomas;
Lopez Lopez, Cristina

Publication type:

journal article

Localization of α-adrenoceptors: JR Vane Medal Lecture.

Published in:

2015

By:

McGrath, John C

Publication type:

journal article

Differential activation of human constitutive androstane receptor and its SV23 and SV24 splice variants by rilpivirine and etravirine.

Published in:

2015

By:

Sharma, Devinder;
Lau, Aik Jiang;
Sherman, Matthew A;
Chang, Thomas K H

Publication type:

journal article

Synthesis and SAR studies of novel 6,7,8-substituted 4-substituted benzyloxyquinolin-2(1H)-one derivatives for anticancer activity.

Published in:

2015

By:

Chen, Yi-Fong;
Lin, Yi-Chien;
Morris-Natschke, Susan L;
Wei, Chen-Fang;
Shen, Ting-Chen;
Lin, Hui-Yi;
Hsu, Mei-Hua;
Chou, Li-Chen;
Zhao, Yu;
Kuo, Sheng-Chu;
Lee, Kuo-Hsiung;
Huang, Li-Jiau

Publication type:

journal article

Histamine H₄ receptors in the gastrointestinal tract.

Published in:

2015

By:

Deiteren, A;
De Man, J G;
Pelckmans, P A;
De Winter, B Y

Publication type:

journal article

The activation of supraspinal GPR40/FFA1 receptor signalling regulates the descending pain control system.

Published in:

2015

By:

Nakamoto, K;
Nishinaka, T;
Sato, N;
Aizawa, F;
Yamashita, T;
Mankura, M;
Koyama, Y;
Kasuya, F;
Tokuyama, S

Publication type:

journal article

The phytocannabinoid, Δ9-tetrahydrocannabivarin, can act through 5- HT1A receptors to produce antipsychotic effects.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1305, doi. 10.1111/bph.13000

By:

Cascio, Maria Grazia;
Zamberletti, Erica;
Marini, Pietro;
Parolaro, Daniela;
Pertwee, Roger G

Publication type:

Article

AQW051, a novel, potent and selective α7 nicotinic ACh receptor partial agonist: pharmacological characterization and phase I evaluation.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1292, doi. 10.1111/bph.13001

By:

Feuerbach, Dominik;
Pezous, Nicole;
Weiss, Markus;
Shakeri ‐ Nejad, Kasra;
Lingenhoehl, Kurt;
Hoyer, Daniel;
Hurth, Konstanze;
Bilbe, Graeme;
Pryce, Christopher R;
McAllister, Kevin;
Chaperon, Frederique;
Kucher, Klaus;
Johns, Donald;
Blaettler, Thomas;
Lopez Lopez, Cristina

Publication type:

Article

Inhibition of L-carnitine biosynthesis and transport by methyl-γ-butyrobetaine decreases fatty acid oxidation and protects against myocardial infarction.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1319, doi. 10.1111/bph.13004

By:

Liepinsh, E;
Makrecka ‐ Kuka, M;
Kuka, J;
Vilskersts, R;
Makarova, E;
Cirule, H;
Loza, E;
Lola, D;
Grinberga, S;
Pugovics, O;
Kalvins, I;
Dambrova, M

Publication type:

Article

Interaction between positive allosteric modulators and trapping blockers of the NMDA receptor channel.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1333, doi. 10.1111/bph.13007

By:

Emnett, Christine M;
Eisenman, Lawrence N;
Mohan, Jayaram;
Taylor, Amanda A;
Doherty, James J;
Paul, Steven M;
Zorumski, Charles F;
Mennerick, Steven

Publication type:

Article

Issue Information.

Published in:: British Journal of Pharmacology, 2015, v. 172, n. 5, p. i, doi. 10.1111/bph.12912
Publication type:: Article

The activation of supraspinal GPR40/ FFA1 receptor signalling regulates the descending pain control system.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1250, doi. 10.1111/bph.13003

By:

Nakamoto, K;
Nishinaka, T;
Sato, N;
Aizawa, F;
Yamashita, T;
Mankura, M;
Koyama, Y;
Kasuya, F;
Tokuyama, S

Publication type:

Article

Histamine H4 receptors in the gastrointestinal tract.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1165, doi. 10.1111/bph.12989

By:

Deiteren, A;
De Man, J G;
Pelckmans, P A;
De Winter, B Y

Publication type:

Article

Identification of muscarinic receptor subtypes involved in catecholamine secretion in adrenal medullary chromaffin cells by genetic deletion.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1348, doi. 10.1111/bph.13011

By:

Harada, Keita;
Matsuoka, Hidetada;
Miyata, Hironori;
Matsui, Minoru;
Inoue, Masumi

Publication type:

Article

An analysis of glucocorticoid receptor-mediated gene expression in BEAS-2B human airway epithelial cells identifies distinct, ligand-directed, transcription profiles with implications for asthma therapeutics.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1360, doi. 10.1111/bph.13014

By:

Joshi, T;
Johnson, M;
Newton, R;
Giembycz, M

Publication type:

Article

Clinically used selective oestrogen receptor modulators increase LDL receptor activity in primary human lymphocytes.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1379, doi. 10.1111/bph.13016

By:

Cerrato, F;
Fernández ‐ Suárez, M E;
Alonso, R;
Alonso, M;
Vázquez, C;
Pastor, O;
Mata, P;
Lasunción, M A;
Gómez ‐ Coronado, D

Publication type:

Article

Localization of α-adrenoceptors: JR Vane Medal Lecture.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1179, doi. 10.1111/bph.13008

By:

McGrath, John C

Publication type:

Article

Synthesis and SAR studies of novel 6,7,8-substituted 4-substituted benzyloxyquinolin-2(1 H)-one derivatives for anticancer activity.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1195, doi. 10.1111/bph.12992

By:

Chen, Yi ‐ Fong;
Lin, Yi ‐ Chien;
Morris ‐ Natschke, Susan L;
Wei, Chen ‐ Fang;
Shen, Ting ‐ Chen;
Lin, Hui ‐ Yi;
Hsu, Mei ‐ Hua;
Chou, Li ‐ Chen;
Zhao, Yu;
Kuo, Sheng ‐ Chu;
Lee, Kuo ‐ Hsiung;
Huang, Li ‐ Jiau

Publication type:

Article

FM19 G11 reverses endothelial dysfunction in rat and human arteries through stimulation of the PI3K/Akt/eNOS pathway, independently of mTOR/ HIF-1α activation.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1277, doi. 10.1111/bph.12993

By:

El Assar, M;
Sánchez ‐ Puelles, J M;
Royo, I;
López ‐ Hernández, E;
Sánchez ‐ Ferrer, A;
Aceña, J L;
Rodríguez ‐ Mañas, L;
Angulo, J

Publication type:

Article

Differential activation of human constitutive androstane receptor and its SV23 and SV24 splice variants by rilpivirine and etravirine.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1263, doi. 10.1111/bph.12997

By:

Sharma, Devinder;
Lau, Aik Jiang;
Sherman, Matthew A;
Chang, Thomas K H

Publication type:

Article

MLN4924 sensitizes monocytes and maturing dendritic cells for TNF-dependent and -independent necroptosis.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1222, doi. 10.1111/bph.12998

By:

El ‐ Mesery, Mohamed;
Seher, Axel;
Stühmer, Thorsten;
Siegmund, Daniela;
Wajant, Harald

Publication type:

Article

Novel Nrf2 activators from microbial transformation products inhibit blood-retinal barrier permeability in rabbits.

Published in:

British Journal of Pharmacology, 2015, v. 172, n. 5, p. 1237, doi. 10.1111/bph.12999

By:

Nakagami, Yasuhiro;
Masuda, Kayoko;
Hatano, Emiko;
Inoue, Tatsuya;
Matsuyama, Takuya;
Iizuka, Mayumi;
Ono, Yasunori;
Ohnuki, Takashi;
Murakami, Yoko;
Iwasaki, Masaru;
Yoshida, Kazuhiro;
Kasuya, Yuji;
Komoriya, Satoshi

Publication type:

Article

Works matching IS 00071188 AND DT 2015 AND VI 172 AND IP 5

AQW051, a novel, potent and selective α7 nicotinic ACh receptor partial agonist: pharmacological characterization and phase I evaluation.

Localization of α-adrenoceptors: JR Vane Medal Lecture.

Differential activation of human constitutive androstane receptor and its SV23 and SV24 splice variants by rilpivirine and etravirine.

Synthesis and SAR studies of novel 6,7,8-substituted 4-substituted benzyloxyquinolin-2(1H)-one derivatives for anticancer activity.

Histamine H₄ receptors in the gastrointestinal tract.

The activation of supraspinal GPR40/FFA1 receptor signalling regulates the descending pain control system.

The phytocannabinoid, Δ<sup>9</sup>-tetrahydrocannabivarin, can act through 5- HT<sub>1</sub><sub>A</sub> receptors to produce antipsychotic effects.

AQW051, a novel, potent and selective α7 nicotinic ACh receptor partial agonist: pharmacological characterization and phase I evaluation.

Inhibition of L-carnitine biosynthesis and transport by methyl-γ-butyrobetaine decreases fatty acid oxidation and protects against myocardial infarction.

Interaction between positive allosteric modulators and trapping blockers of the NMDA receptor channel.

Issue Information.

The activation of supraspinal GPR40/ FFA1 receptor signalling regulates the descending pain control system.

Histamine H<sub>4</sub> receptors in the gastrointestinal tract.

Identification of muscarinic receptor subtypes involved in catecholamine secretion in adrenal medullary chromaffin cells by genetic deletion.

An analysis of glucocorticoid receptor-mediated gene expression in BEAS-2B human airway epithelial cells identifies distinct, ligand-directed, transcription profiles with implications for asthma therapeutics.

Clinically used selective oestrogen receptor modulators increase LDL receptor activity in primary human lymphocytes.

Localization of α-adrenoceptors: JR Vane Medal Lecture.

Synthesis and SAR studies of novel 6,7,8-substituted 4-substituted benzyloxyquinolin-2(1 H)-one derivatives for anticancer activity.

FM19 G11 reverses endothelial dysfunction in rat and human arteries through stimulation of the PI3K/Akt/eNOS pathway, independently of mTOR/ HIF-1α activation.

Differential activation of human constitutive androstane receptor and its SV23 and SV24 splice variants by rilpivirine and etravirine.

MLN4924 sensitizes monocytes and maturing dendritic cells for TNF-dependent and -independent necroptosis.

Novel Nrf2 activators from microbial transformation products inhibit blood-retinal barrier permeability in rabbits.