Works matching IS 00071188 AND DT 2014 AND VI 171 AND IP 23

Results: 31

In vivo properties of KNT-127, a novel δ opioid receptor agonist: receptor internalization, antihyperalgesia and antidepressant effects in mice.

Published in:

2014

By:

Nozaki, C;
Nagase, H;
Nemoto, T;
Matifas, A;
Kieffer, B L;
Gaveriaux-Ruff, C

Publication type:

journal article

Modulation of K2P 2.1 and K2P 10.1 K(+) channel sensitivity to carvedilol by alternative mRNA translation initiation.

Published in:

2014

By:

Kisselbach, J;
Seyler, C;
Schweizer, P A;
Gerstberger, R;
Becker, R;
Katus, H A;
Thomas, D

Publication type:

journal article

The neurosteroid 5β-pregnan-3α-ol-20-one enhances actions of etomidate as a positive allosteric modulator of α1β2γ2L GABAA receptors.

Published in:

2014

By:

Li, P;
Bracamontes, J R;
Manion, B D;
Mennerick, S;
Steinbach, J H;
Evers, A S;
Akk, G

Publication type:

journal article

Detection of the secondary, low-affinity β1 -adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR-CGP.

Published in:

2014

By:

Gherbi, K;
Briddon, S J;
Hill, S J

Publication type:

journal article

δ-Opioid receptors up-regulate excitatory amino acid transporters in mouse astrocytes.

Published in:

2014

By:

Liang, Jianfeng;
Chao, Dongman;
Sandhu, Harleen K;
Yu, Yanbing;
Zhang, Li;
Balboni, Gianfranco;
Kim, Dong H;
Xia, Ying

Publication type:

journal article

Modulation of K2P2.1 and K2P10.1 K+ channel sensitivity to carvedilol by alternative mRNA translation initiation.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5182, doi. 10.1111/bph.12596

By:

Kisselbach, J;
Seyler, C;
Schweizer, P A;
Gerstberger, R;
Becker, R;
Katus, H A;
Thomas, D

Publication type:

Article

Analgesic tolerance to morphine is regulated by PPARγ.

Published in:

2014

By:

de Guglielmo, Giordano;
Kallupi, Marsida;
Scuppa, Giulia;
Stopponi, Serena;
Demopulos, Gregory;
Gaitanaris, George;
Ciccocioppo, Roberto

Publication type:

journal article

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptor.

Published in:

2014

By:

Guo, Dong;
Venhorst, Suzanne N;
Massink, Arnault;
van Veldhoven, Jacobus P D;
Vauquelin, Georges;
IJzerman, Adriaan P;
Heitman, Laura H

Publication type:

journal article

Identification of novel insulin mimetic drugs by quantitative total internal reflection fluorescence (TIRF) microscopy.

Published in:

2014

By:

Lanzerstorfer, Peter;
Stadlbauer, Verena;
Chtcheglova, Lilia A;
Haselgrübler, Renate;
Borgmann, Daniela;
Wruss, Jürgen;
Hinterdorfer, Peter;
Schröder, Klaus;
Winkler, Stephan M;
Höglinger, Otmar;
Weghuber, Julian

Publication type:

journal article

UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations.

Published in:

2014

By:

Hassan-Mohamed, I;
Giorgio, C;
Incerti, M;
Russo, S;
Pala, D;
Pasquale, E B;
Zanotti, I;
Vicini, P;
Barocelli, E;
Rivara, S;
Mor, M;
Lodola, A;
Tognolini, M

Publication type:

journal article

Heteromerization of GPR55 and cannabinoid CB2 receptors modulates signalling.

Published in:

2014

By:

Balenga, N A;
Martínez-Pinilla, E;
Kargl, J;
Schröder, R;
Peinhaupt, M;
Platzer, W;
Bálint, Z;
Zamarbide, M;
Dopeso-Reyes, I G;
Ricobaraza, A;
Pérez-Ortiz, J M;
Kostenis, E;
Waldhoer, M;
Heinemann, A;
Franco, R

Publication type:

journal article

Uni PR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5195, doi. 10.1111/bph.12669

By:

Hassan ‐ Mohamed, I;
Giorgio, C;
Incerti, M;
Russo, S;
Pala, D;
Pasquale, E B;
Zanotti, I;
Vicini, P;
Barocelli, E;
Rivara, S;
Mor, M;
Lodola, A;
Tognolini, M

Publication type:

Article

Heteromerization of GPR55 and cannabinoid CB2 receptors modulates signalling.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5387, doi. 10.1111/bph.12850

By:

Balenga, N A;
Martínez ‐ Pinilla, E;
Kargl, J;
Schröder, R;
Peinhaupt, M;
Platzer, W;
Bálint, Z;
Zamarbide, M;
Dopeso ‐ Reyes, I G;
Ricobaraza, A;
Pérez ‐ Ortiz, J M;
Kostenis, E;
Waldhoer, M;
Heinemann, A;
Franco, R

Publication type:

Article

Analgesic tolerance to morphine is regulated by PPARγ.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5407, doi. 10.1111/bph.12851

By:

Guglielmo, Giordano;
Kallupi, Marsida;
Scuppa, Giulia;
Stopponi, Serena;
Demopulos, Gregory;
Gaitanaris, George;
Ciccocioppo, Roberto

Publication type:

Article

In vivo properties of KNT-127, a novel δ opioid receptor agonist: receptor internalization, antihyperalgesia and antidepressant effects in mice.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5376, doi. 10.1111/bph.12852

By:

Nozaki, C;
Nagase, H;
Nemoto, T;
Matifas, A;
Kieffer, B L;
Gaveriaux ‐ Ruff, C

Publication type:

Article

Alteration of vascular reactivity in heart failure: role of phosphodiesterases 3 and 4.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5361, doi. 10.1111/bph.12853

By:

Hubert, F;
Belacel ‐ Ouari, M;
Manoury, B;
Zhai, K;
Domergue ‐ Dupont, V;
Mateo, P;
Joubert, F;
Fischmeister, R;
Leblais, V

Publication type:

Article

δ-Opioid receptors up-regulate excitatory amino acid transporters in mouse astrocytes.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5417, doi. 10.1111/bph.12857

By:

Liang, Jianfeng;
Chao, Dongman;
Sandhu, Harleen K;
Yu, Yanbing;
Zhang, Li;
Balboni, Gianfranco;
Kim, Dong H;
Xia, Ying

Publication type:

Article

Detection of the secondary, low-affinity β1-adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR- CGP.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5431, doi. 10.1111/bph.12858

By:

Gherbi, K;
Briddon, S J;
Hill, S J

Publication type:

Article

Issue Information.

Published in:: British Journal of Pharmacology, 2014, v. 171, n. 23, p. i, doi. 10.1111/bph.12392
Publication type:: Article

TRPC6 regulates cell cycle progression by modulating membrane potential in bone marrow stromal cells.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5280, doi. 10.1111/bph.12840

By:

Ichikawa, Jun;
Inoue, Ryuji

Publication type:

Article

Nicotinic acetylcholine receptors control acetylcholine and noradrenaline release in the rodent habenulo-interpeduncular complex.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5209, doi. 10.1111/bph.12841

By:

Beiranvand, F;
Zlabinger, C;
Orr ‐ Urtreger, A;
Ristl, R;
Huck, S;
Scholze, P

Publication type:

Article

Determination of the binding mode for the cyclopentapeptide CXCR4 antagonist FC131 using a dual approach of ligand modifications and receptor mutagenesis.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5313, doi. 10.1111/bph.12842

By:

Thiele, S;
Mungalpara, J;
Steen, A;
Rosenkilde, M M;
Våbenø, J

Publication type:

Article

Novel coumarin modified GLP-1 derivatives with enhanced plasma stability and prolonged in vivo glucose-lowering ability.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5252, doi. 10.1111/bph.12843

By:

Han, Jing;
Sun, Lidan;
Huang, Xun;
Li, Zheng;
Zhang, Chenyu;
Qian, Hai;
Huang, Wenlong

Publication type:

Article

Identification of novel insulin mimetic drugs by quantitative total internal reflection fluorescence ( TIRF) microscopy.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5237, doi. 10.1111/bph.12845

By:

Lanzerstorfer, Peter;
Stadlbauer, Verena;
Chtcheglova, Lilia A;
Haselgrübler, Renate;
Borgmann, Daniela;
Wruss, Jürgen;
Hinterdorfer, Peter;
Schröder, Klaus;
Winkler, Stephan M;
Höglinger, Otmar;
Weghuber, Julian

Publication type:

Article

Metabolic characteristics of 13-cis-retinoic acid (isotretinoin) and anti-tumour activity of the 13-cis-retinoic acid metabolite 4-oxo-13-cis-retinoic acid in neuroblastoma.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5330, doi. 10.1111/bph.12846

By:

Sonawane, Poonam;
Cho, Hwang Eui;
Tagde, Ashujit;
Verlekar, Dattesh;
Yu, Alice L;
Reynolds, C Patrick;
Kang, Min H

Publication type:

Article

Glutathione administration reduces mitochondrial damage and shifts cell death from necrosis to apoptosis in ageing diabetic mice hearts during exercise.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5345, doi. 10.1111/bph.12847

By:

Golbidi, S;
Botta, A;
Gottfred, S;
Nusrat, A;
Laher, I;
Ghosh, S

Publication type:

Article

The neurosteroid 5β-pregnan-3α-ol-20-one enhances actions of etomidate as a positive allosteric modulator of α1β2γ2 L GABAA receptors.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5446, doi. 10.1111/bph.12861

By:

Li, P;
Bracamontes, J R;
Manion, B D;
Mennerick, S;
Steinbach, J H;
Evers, A S;
Akk, G

Publication type:

Article

Inhibition of phosphodiesterase-3 by levosimendan is sufficient to account for its inotropic effect in failing human heart.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5169, doi. 10.1111/bph.12647

By:

Ørstavik, Ø;
Ata, S H;
Riise, J;
Dahl, C P;
Andersen, G Ø;
Levy, F O;
Skomedal, T;
Osnes, J ‐ B;
Qvigstad, E

Publication type:

Article

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptor.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5295, doi. 10.1111/bph.12836

By:

Guo, Dong;
Venhorst, Suzanne N;
Massink, Arnault;
Veldhoven, Jacobus P D;
Vauquelin, Georges;
IJzerman, Adriaan P;
Heitman, Laura H

Publication type:

Article

Celastrol protects ischaemic myocardium through a heat shock response with up-regulation of haeme oxygenase-1.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5265, doi. 10.1111/bph.12838

By:

Der Sarkissian, S;
Cailhier, J ‐ F;
Borie, M;
Stevens, L ‐ M;
Gaboury, L;
Mansour, S;
Hamet, P;
Noiseux, N

Publication type:

Article

Endocannabinoid modulation by FAAH and monoacylglycerol lipase within the analgesic circuitry of the periaqueductal grey.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 23, p. 5225, doi. 10.1111/bph.12839

By:

Lau, Benjamin K;
Drew, Geoffrey M;
Mitchell, Vanessa A;
Vaughan, Christopher W

Publication type:

Article

Works matching IS 00071188 AND DT 2014 AND VI 171 AND IP 23

In vivo properties of KNT-127, a novel δ opioid receptor agonist: receptor internalization, antihyperalgesia and antidepressant effects in mice.

Modulation of K2P 2.1 and K2P 10.1 K(+) channel sensitivity to carvedilol by alternative mRNA translation initiation.

The neurosteroid 5β-pregnan-3α-ol-20-one enhances actions of etomidate as a positive allosteric modulator of α1β2γ2L GABAA receptors.

Detection of the secondary, low-affinity β1 -adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR-CGP.

δ-Opioid receptors up-regulate excitatory amino acid transporters in mouse astrocytes.

Modulation of K<sub>2P</sub>2.1 and K<sub>2P</sub>10.1 K<sup>+</sup> channel sensitivity to carvedilol by alternative mRNA translation initiation.

Analgesic tolerance to morphine is regulated by PPARγ.

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptor.

Identification of novel insulin mimetic drugs by quantitative total internal reflection fluorescence (TIRF) microscopy.

UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations.

Heteromerization of GPR55 and cannabinoid CB2 receptors modulates signalling.

Uni PR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations.

Heteromerization of GPR55 and cannabinoid CB<sub>2</sub> receptors modulates signalling.

Analgesic tolerance to morphine is regulated by PPARγ.

In vivo properties of KNT-127, a novel δ opioid receptor agonist: receptor internalization, antihyperalgesia and antidepressant effects in mice.

Alteration of vascular reactivity in heart failure: role of phosphodiesterases 3 and 4.

δ-Opioid receptors up-regulate excitatory amino acid transporters in mouse astrocytes.

Detection of the secondary, low-affinity β<sub>1</sub>-adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR- CGP.

Issue Information.

TRPC6 regulates cell cycle progression by modulating membrane potential in bone marrow stromal cells.

Nicotinic acetylcholine receptors control acetylcholine and noradrenaline release in the rodent habenulo-interpeduncular complex.

Determination of the binding mode for the cyclopentapeptide CXCR4 antagonist FC131 using a dual approach of ligand modifications and receptor mutagenesis.

Novel coumarin modified GLP-1 derivatives with enhanced plasma stability and prolonged in vivo glucose-lowering ability.

Identification of novel insulin mimetic drugs by quantitative total internal reflection fluorescence ( TIRF) microscopy.

Metabolic characteristics of 13-cis-retinoic acid (isotretinoin) and anti-tumour activity of the 13-cis-retinoic acid metabolite 4-oxo-13-cis-retinoic acid in neuroblastoma.

Glutathione administration reduces mitochondrial damage and shifts cell death from necrosis to apoptosis in ageing diabetic mice hearts during exercise.

The neurosteroid 5β-pregnan-3α-ol-20-one enhances actions of etomidate as a positive allosteric modulator of α1β2γ2 L GABA<sub>A</sub> receptors.

Inhibition of phosphodiesterase-3 by levosimendan is sufficient to account for its inotropic effect in failing human heart.

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A<sub>1</sub> adenosine receptor.

Celastrol protects ischaemic myocardium through a heat shock response with up-regulation of haeme oxygenase-1.

Endocannabinoid modulation by FAAH and monoacylglycerol lipase within the analgesic circuitry of the periaqueductal grey.