Works matching IS 00071188 AND DT 2012 AND VI 165 AND IP 5

Results: 42

Effects of atorvastatin metabolites on induction of drug-metabolizing enzymes and membrane transporters through human pregnane X receptor.

Published in:

2012

By:

Hoffart E;
Ghebreghiorghis L;
Nussler AK;
Thasler WE;
Weiss TS;
Schwab M;
Burk O;
Hoffart, E;
Ghebreghiorghis, L;
Nussler, A K;
Thasler, W E;
Weiss, T S;
Schwab, M;
Burk, O

Publication type:

journal article

The evolving science of detection of 'blood doping'.

Published in:

2012

By:

Lundby C;
Robach P;
Saltin B;
Lundby, Carsten;
Robach, Paul;
Saltin, Bengt

Publication type:

journal article

Tau-targeted treatment strategies in Alzheimer's disease.

Published in:

2012

By:

Götz J;
Ittner A;
Ittner LM;
Götz, Jürgen;
Ittner, Arne;
Ittner, Lars M

Publication type:

journal article

Cyclic nucleotide phosphodiesterase (PDE) isozymes as targets of the intracellular signalling network: benefits of PDE inhibitors in various diseases and perspectives for future therapeutic developments.

Published in:

2012

By:

Keravis T;
Lugnier C;
Keravis, Thérèse;
Lugnier, Claire

Publication type:

journal article

What makes the α(1A)-adrenoceptor gene express the α(1L)-adrenoceptor functional phenotype?

Published in:

2012

By:

Ventura S;
Ventura, Sabatino

Publication type:

journal article

β(2)-Adrenoceptors increase translocation of GLUT4 via GPCR kinase sites in the receptor C-terminal tail.

Published in:

2012

By:

Dehvari N;
Hutchinson DS;
Nevzorova J;
Dallner OS;
Sato M;
Kocan M;
Merlin J;
Evans BA;
Summers RJ;
Bengtsson T;
Dehvari, Nodi;
Hutchinson, Dana S;
Nevzorova, Julia;
Dallner, Olof S;
Sato, Masaaki;
Kocan, Martina;
Merlin, Jon;
Evans, Bronwyn A;
Summers, Roger J;
Bengtsson, Tore

Publication type:

journal article

A β-amyloid oligomer directly modulates P/Q-type calcium currents in Xenopus oocytes.

Published in:

2012

By:

Mezler M;
Barghorn S;
Schoemaker H;
Gross G;
Nimmrich V;
Mezler, M;
Barghorn, S;
Schoemaker, H;
Gross, G;
Nimmrich, V

Publication type:

journal article

TASK1 (K(2P)3.1) K(+) channel inhibition by endothelin-1 is mediated through Rho kinase-dependent phosphorylation.

Published in:

2012

By:

Seyler C;
Duthil-Straub E;
Zitron E;
Gierten J;
Scholz EP;
Fink RH;
Karle CA;
Becker R;
Katus HA;
Thomas D;
Seyler, C;
Duthil-Straub, E;
Zitron, E;
Gierten, J;
Scholz, E P;
Fink, R H A;
Karle, C A;
Becker, R;
Katus, H A;
Thomas, D

Publication type:

journal article

Phenotype pharmacology of lower urinary tract α(1)-adrenoceptors.

Published in:

2012

By:

Nishimune A;
Yoshiki H;
Uwada J;
Anisuzzaman AS;
Umada H;
Muramatsu I;
Nishimune, A;
Yoshiki, H;
Uwada, J;
Anisuzzaman, A S M;
Umada, H;
Muramatsu, I

Publication type:

journal article

Modulating human proteinase activated receptor 2 with a novel antagonist (GB88) and agonist (GB110).

Published in:

2012

By:

Suen JY;
Barry GD;
Lohman RJ;
Halili MA;
Cotterell AJ;
Le GT;
Fairlie DP;
Suen, J Y;
Barry, G D;
Lohman, R J;
Halili, M A;
Cotterell, A J;
Le, G T;
Fairlie, D P

Publication type:

journal article

Different tests for a difference: how do we do research?

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1217, doi. 10.1111/j.1476-5381.2011.01809.x

By:

Drummond, Gordon B;
Vowler, Sarah L

Publication type:

Article

Non-bronchodilating mechanisms of tiotropium prevent airway hyperreactivity in a guinea-pig model of allergic asthma.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1501, doi. 10.1111/j.1476-5381.2011.01632.x

By:

Buels, KS;
Jacoby, DB;
Fryer, AD

Publication type:

Article

Pentoxifylline aggravates fatty liver in obese and diabetic ob/ob mice by increasing intestinal glucose absorption and activating hepatic lipogenesis.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1361, doi. 10.1111/j.1476-5381.2011.01580.x

By:

Massart, J;
Robin, MA;
Noury, F;
Fautrel, A;
Lettéron, P;
Bado, A;
Eliat, PA;
Fromenty, B

Publication type:

Article

Effects of atorvastatin metabolites on induction of drug-metabolizing enzymes and membrane transporters through human pregnane X receptor.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1595, doi. 10.1111/j.1476-5381.2011.01665.x

By:

Hoffart, E;
Ghebreghiorghis, L;
Nussler, AK;
Thasler, WE;
Weiss, TS;
Schwab, M;
Burk, O

Publication type:

Article

Phenotype pharmacology of lower urinary tract α1-adrenoceptors.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1226, doi. 10.1111/j.1476-5381.2011.01591.x

By:

Nishimune, A;
Yoshiki, H;
Uwada, J;
Anisuzzaman, ASM;
Umada, H;
Muramatsu, I

Publication type:

Article

Endothelin and bradykinin: 'brothers-in-arms' in Chagas vasculopathies?

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1330, doi. 10.1111/j.1476-5381.2011.01636.x

By:

D'Orléans-Juste, Pedro;
Bkaily, Ghassan;
Rae, Giles Alexander

Publication type:

Article

β2-Adrenoceptors increase translocation of GLUT4 via GPCR kinase sites in the receptor C-terminal tail.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1442, doi. 10.1111/j.1476-5381.2011.01647.x

By:

Dehvari, Nodi;
Hutchinson, Dana S;
Nevzorova, Julia;
Dallner, Olof S;
Sato, Masaaki;
Kocan, Martina;
Merlin, Jon;
Evans, Bronwyn A;
Summers, Roger J;
Bengtsson, Tore

Publication type:

Article

The evolving science of detection of 'blood doping'.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1306, doi. 10.1111/j.1476-5381.2011.01822.x

By:

Lundby, Carsten;
Robach, Paul;
Saltin, Bengt

Publication type:

Article

Angiotensin-(1-7) inhibits epidermal growth factor receptor transactivation via a Mas receptor-dependent pathway.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1390, doi. 10.1111/j.1476-5381.2011.01613.x

By:

Akhtar, Saghir;
Yousif, Mariam HM;
Dhaunsi, Gursev S;
Chandrasekhar, Bindu;
Al-Farsi, Omama;
Benter, Ibrahim F

Publication type:

Article

TM-25659 enhances osteogenic differentiation and suppresses adipogenic differentiation by modulating the transcriptional co-activator TAZ.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1584, doi. 10.1111/j.1476-5381.2011.01664.x

By:

Jang, EJ;
Jeong, H;
Kang, JO;
Kim, NJ;
Kim, MS;
Choi, SH;
Yoo, SE;
Hong, JH;
Bae, MA;
Hwang, ES

Publication type:

Article

A β-amyloid oligomer directly modulates P/Q-type calcium currents in Xenopus oocytes.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1572, doi. 10.1111/j.1476-5381.2011.01646.x

By:

Mezler, M;
Barghorn, S;
Schoemaker, H;
Gross, G;
Nimmrich, V

Publication type:

Article

Inhibiting the TLR4-MyD88 signalling cascade by genetic or pharmacological strategies reduces acute alcohol-induced sedation and motor impairment in mice.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1319, doi. 10.1111/j.1476-5381.2011.01572.x

By:

Wu, Yue;
Lousberg, Erin L;
Moldenhauer, Lachlan M;
Hayball, John D;
Coller, Janet K;
Rice, Kenner C;
Watkins, Linda R;
Somogyi, Andrew A;
Hutchinson, Mark R

Publication type:

Article

Azithromycin distinctively modulates classical activation of human monocytes in vitro.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1348, doi. 10.1111/j.1476-5381.2011.01576.x

By:

Vrančić, M;
Banjanac, M;
Nujić, K;
Bosnar, M;
Murati, T;
Munić, V;
Stupin Polančec, D;
Belamarić, D;
Parnham, MJ;
Eraković Haber, V

Publication type:

Article

Cyclosporin A and cardioprotection: from investigative tool to therapeutic agent.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1235, doi. 10.1111/j.1476-5381.2011.01700.x

By:

Hausenloy, DJ;
Boston-Griffiths, EA;
Yellon, DM

Publication type:

Article

5-HT receptors as novel targets for optimizing pigmentary responses in dorsal skin melanophores of frog, Hoplobatrachus tigerinus.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1515, doi. 10.1111/j.1476-5381.2011.01630.x

By:

Ali, Sharique A;
Salim, Saima;
Sahni, Tarandeep;
Peter, Jaya;
Ali, Ayesha S

Publication type:

Article

Pharmacokinetics and in vivo potency of soluble epoxide hydrolase inhibitors in cynomolgus monkeys.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1401, doi. 10.1111/j.1476-5381.2011.01641.x

By:

Ulu, A;
Appt, SE;
Morisseau, C;
Hwang, SH;
Jones, PD;
Rose, TE;
Dong, H;
Lango, J;
Yang, J;
Tsai, HJ;
Miyabe, C;
Fortenbach, C;
Adams, MR;
Hammock, BD

Publication type:

Article

Dynamic monitoring of beating periodicity of stem cell-derived cardiomyocytes as a predictive tool for preclinical safety assessment.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1424, doi. 10.1111/j.1476-5381.2011.01623.x

By:

Abassi, Yama A;
Xi, Biao;
Li, Nan;
Ouyang, Wei;
Seiler, Alexander;
Watzele, Manfred;
Kettenhofen, Ralf;
Bohlen, Heribert;
Ehlich, Andreas;
Kolossov, Eugen;
Wang, Xiaobo;
Xu, Xiao

Publication type:

Article

What makes the α1A-adrenoceptor gene express the α1L-adrenoceptor functional phenotype?

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1223, doi. 10.1111/j.1476-5381.2011.01663.x

By:

Ventura, S

Publication type:

Article

Activation of transient receptor potential A1 by a non-pungent capsaicin-like compound, capsiate.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1476, doi. 10.1111/j.1476-5381.2011.01634.x

By:

Shintaku, Kenji;
Uchida, Kunitoshi;
Suzuki, Yoshiro;
Zhou, Yiming;
Fushiki, Tohru;
Watanabe, Tatsuo;
Yazawa, Susumu;
Tominaga, Makoto

Publication type:

Article

Long-term treatment with ivabradine in post-myocardial infarcted rats counteracts f-channel overexpression.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1457, doi. 10.1111/j.1476-5381.2011.01627.x

By:

Suffredini, S;
Stillitano, F;
Comini, L;
Bouly, M;
Brogioni, S;
Ceconi, C;
Ferrari, R;
Mugelli, A;
Cerbai, E

Publication type:

Article

Clozapine, but not haloperidol, enhances glial d-serine and L-glutamate release in rat frontal cortex and primary cultured astrocytes.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1543, doi. 10.1111/j.1476-5381.2011.01638.x

By:

Tanahashi, Shunske;
Yamamura, Satoshi;
Nakagawa, Masanori;
Motomura, Eishi;
Okada, Motohiro

Publication type:

Article

Trypanosoma cruzi invades host cells through the activation of endothelin and bradykinin receptors: a converging pathway leading to chagasic vasculopathy.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1333, doi. 10.1111/j.1476-5381.2011.01609.x

By:

Andrade, Daniele;
Serra, Rafaela;
Svensjö, Erik;
Lima, Ana Paula C;
Ramos Junior, Erivan S;
Fortes, Fabio S;
Morandini, Ana Carolina F;
Morandi, Verônica;
Soeiro, Maria de N;
Tanowitz, Herbert B;
Scharfstein, Julio

Publication type:

Article

Inhibiting fatty acid amide hydrolase normalizes endotoxin-induced enhanced gastrointestinal motility in mice.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1556, doi. 10.1111/j.1476-5381.2011.01644.x

By:

Bashashati, M;
Storr, MA;
Nikas, SP;
Wood, JT;
Godlewski, G;
Liu, J;
Ho, W;
Keenan, CM;
Zhang, H;
Alapafuja, SO;
Cravatt, BF;
Lutz, B;
Mackie, K;
Kunos, G;
Patel, KD;
Makriyannis, A;
Davison, JS;
Sharkey, KA

Publication type:

Article

Cyclic nucleotide phosphodiesterase (PDE) isozymes as targets of the intracellular signalling network: benefits of PDE inhibitors in various diseases and perspectives for future therapeutic developments.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1288, doi. 10.1111/j.1476-5381.2011.01729.x

By:

Keravis, Thérèse;
Lugnier, Claire

Publication type:

Article

TLR4-MyD88 signalling: a molecular target for alcohol actions.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1316, doi. 10.1111/j.1476-5381.2011.01695.x

By:

Pandey, Subhash C

Publication type:

Article

TASK1 (K2P3.1) K+ channel inhibition by endothelin-1 is mediated through Rho kinase-dependent phosphorylation.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1467, doi. 10.1111/j.1476-5381.2011.01626.x

By:

Seyler, C;
Duthil-Straub, E;
Zitron, E;
Gierten, J;
Scholz, EP;
Fink, RHA;
Karle, CA;
Becker, R;
Katus, HA;
Thomas, D

Publication type:

Article

Long-lasting neuroprotection and neurological improvement in stroke models with new, potent and brain permeable inhibitors of poly(ADP-ribose) polymerase.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1487, doi. 10.1111/j.1476-5381.2011.01666.x

By:

Moroni, F;
Cozzi, A;
Chiarugi, A;
Formentini, L;
Camaioni, E;
Pellegrini-Giampietro, DE;
Chen, Y;
Liang, S;
Zaleska, MM;
Gonzales, C;
Wood, A;
Pellicciari, R

Publication type:

Article

A naturally occurring naringenin derivative exerts potent bone anabolic effects by mimicking oestrogen action on osteoblasts.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1526, doi. 10.1111/j.1476-5381.2011.01637.x

By:

Swarnkar, Gaurav;
Sharan, Kunal;
Siddiqui, Jawed A;
Mishra, Jay Sharan;
Khan, Kainat;
Khan, Mohd Parvez;
Gupta, Varsha;
Rawat, Preeti;
Maurya, Rakesh;
Dwivedi, Anil K;
Sanyal, Sabyasachi;
Chattopadhyay, Naibedya

Publication type:

Article

Treatment of depressive-like behaviour in Huntington's disease mice by chronic sertraline and exercise.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1375, doi. 10.1111/j.1476-5381.2011.01567.x

By:

Renoir, Thibault;
Pang, Terence YC;
Zajac, Michelle S;
Chan, Grace;
Du, Xin;
Leang, Leah;
Chevarin, Caroline;
Lanfumey, Laurence;
Hannan, Anthony J

Publication type:

Article

Tau-targeted treatment strategies in Alzheimer's disease.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1246, doi. 10.1111/j.1476-5381.2011.01713.x

By:

Götz, Jürgen;
Ittner, Arne;
Ittner, Lars M

Publication type:

Article

Modulating human proteinase activated receptor 2 with a novel antagonist (GB88) and agonist (GB110).

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1413, doi. 10.1111/j.1476-5381.2011.01610.x

By:

Suen, JY;
Barry, GD;
Lohman, RJ;
Halili, MA;
Cotterell, AJ;
Le, GT;
Fairlie, DP

Publication type:

Article

OATPs, OATs and OCTs: the organic anion and cation transporters of the SLCO and SLC22A gene superfamilies.

Published in:

British Journal of Pharmacology, 2012, v. 165, n. 5, p. 1260, doi. 10.1111/j.1476-5381.2011.01724.x

By:

Roth, Megan;
Obaidat, Amanda;
Hagenbuch, Bruno

Publication type:

Article