Works matching DE "RIMONABANT"

Results: 112

One‐Pot Double Oxidation Synthesis of N‐1‐Piperidonyl Amides From N‐1‐Piperidinyl Amides with meta‐Chloroperbenzoic Acid: Rimonabant Analogue as Model Study.

Published in:

Chemistry - A European Journal, 2023, v. 29, n. 45, p. 1, doi. 10.1002/chem.202300702

By:

Chen, Yu‐Chieh;
Zeng, Wei‐Zheng;
Li, Sin‐Min;
Chou, Jia‐Yu;
Tsai, Shuo‐En;
Fuh Wong, Fung

Publication type:

Article

Novel Fubinaca/Rimonabant hybrids as endocannabinoid system modulators.

Published in:

Amino Acids, 2018, v. 50, n. 11, p. 1595, doi. 10.1007/s00726-018-2636-1

By:

Stefanucci, Azzurra;
Macedonio, Giorgia;
Dvorácskó, Szabolcs;
Tömböly, Csaba;
Mollica, Adriano

Publication type:

Article

Possible Therapeutic Doses of Cannabinoid Type 1 Receptor Antagonist Reverses Key Alterations in Fragile X Syndrome Mouse Model.

Published in:

Genes, 2016, v. 7, n. 9, p. 56, doi. 10.3390/genes7090056

By:

Gomis-González, Maria;
Busquets-Garcia, Arnau;
Matute, Carlos;
Maldonado, Rafael;
Mato, Susana;
Ozaita, Andrés

Publication type:

Article

Patients' experiences of prescribed anti-obesity drugs and perceptions of support from primary care: a qualitative study.

Published in:

Primary Health Care Research & Development, 2010, v. 11, n. 3, p. 250, doi. 10.1017/S1463423610000083

By:

Psarou, Aikaterini;
Brown, Ian

Publication type:

Article

CB1 receptor blockade ameliorates hepatic fat infiltration and inflammation and increases Nrf2-AMPK pathway in a rat model of severely uncontrolled diabetes.

Published in:

PLoS ONE, 2018, v. 13, n. 10, p. 1, doi. 10.1371/journal.pone.0206152

By:

Chang, Eugene;
Kim, Dae-Hee;
Yang, Hyekyung;
Lee, Da Hyun;
Bae, Soo Han;
Park, Cheol-Young

Publication type:

Article

Nonopioid placebo analgesia is mediated by CB1 cannabinoid receptors.

Published in:

Nature Medicine, 2011, v. 17, n. 10, p. 1228, doi. 10.1038/nm.2435

By:

Benedetti, Fabrizio;
Amanzio, Martina;
Rosato, Rosalba;
Blanchard, Catherine

Publication type:

Article

Efficacy and Safety of Ezetimibe Plus Orlistat or Rimonabant in Statin-Intolerant Nondiabetic Overweight/Obese Patients With Dyslipidemia.

Published in:

Journal of Cardiovascular Pharmacology & Therapeutics, 2009, v. 14, n. 4, p. 274, doi. 10.1177/1074248409343935

By:

Florentin, Matilda;
Kostapanos, Michael S.;
Nakou, Eleni S.;
Elisaf, Moses;
Liberopoulos, Evangelos N.

Publication type:

Article

Interfering with reconsolidation by rimonabant results in blockade of heroin-associated memory.

Published in:

Frontiers in Pharmacology, 2024, p. 01, doi. 10.3389/fphar.2024.1361838

By:

Jiang Lin;
Yilin Peng;
Jinlong Zhang;
Junzhe Cheng;
Qianqian Chen;
Binbin Wang;
Yuhang Liu;
Shuliang Niu;
Jie Yan

Publication type:

Article

The Gastric CB1 Receptor Modulates Ghrelin Production through the mTOR Pathway to Regulate Food Intake.

Published in:

PLoS ONE, 2013, v. 8, n. 11, p. 1, doi. 10.1371/journal.pone.0080339

By:

Senin, Lucia L.;
Al-Massadi, Omar;
Folgueira, Cintia;
Castelao, Cecilia;
Pardo, Maria;
Barja-Fernandez, Silvia;
Roca-Rivada, Arturo;
Amil, Maria;
Crujeiras, Ana B.;
Garcia-Caballero, Tomas;
Gabellieri, Enrico;
Leis, Rosaura;
Dieguez, Carlos;
Pagotto, Uberto;
Casanueva, Felipe F.;
Seoane, Luisa M.

Publication type:

Article

Obesity, the Endocannabinoid System, and Bias Arising from Pharmaceutical Sponsorship.

Published in:

PLoS ONE, 2009, v. 4, n. 3, p. 1, doi. 10.1371/journal.pone.0005092

By:

McPartland, John M.

Publication type:

Article

Different Transcriptional Control of Metabolism and Extracellular Matrix in Visceral and Subcutaneous Fat of Obese and Rimonabant Treated Mice.

Published in:

PLoS ONE, 2008, v. 3, n. 10, p. 1, doi. 10.1371/journal.pone.0003385

By:

Poussin, Carine;
Hall, Diana;
Minehira, Kaori;
Galzin, Anne-Marie;
Tarussio, David;
Thorens, Bernard

Publication type:

Article

The Orexigenic Effect of Ghrelin Is Mediated through Central Activation of the Endogenous Cannabinoid System.

Published in:

PLoS ONE, 2008, v. 3, n. 3, p. 1, doi. 10.1371/journal.pone.0001797

By:

Kola, Blerina;
Farkas, Imre;
Christ-Crain, Mirjam;
Wittmann, Gábor;
Lolli, Francesca;
Amin, Faisal;
Harvey-White, Judith;
Liposits, Zsolt;
Kunos, George;
Grossman, Ashley B.;
Fekete, Csaba;
Korbonits, Márta

Publication type:

Article

CB1 cannabinoid receptors promote oxidative stress and cell death in murine models of doxorubicin-induced cardiomyopathy and in human cardiomyocytes.

Published in:

Cardiovascular Research, 2010, v. 85, n. 4, p. 773, doi. 10.1093/cvr/cvp369

By:

Mukhopadhyay, Partha;
Rajesh, Mohanraj;
Bátkai, Sándor;
Patel, Vivek;
Kashiwaya, Yoshihiro;
Liaudet, Lucas;
Evgenov, Oleg V.;
Mackie, Ken;
Haskó, György;
Pacher, Pál

Publication type:

Article

Computational investigation on the binding modes of Rimonabant analogs with CB1 and CB2.

Published in:

Chemical Biology & Drug Design, 2018, v. 92, n. 3, p. 1699, doi. 10.1111/cbdd.13337

By:

Liu, Cheng;
Yuan, Congmin;
Wu, Pinwen;
Zhu, Chen;
Fang, Hao;
Wang, Lili;
Fu, Wei

Publication type:

Article

CB1 receptor antagonist rimonabant protects against chronic intermittent hypoxia-induced renal injury in rats.

Published in:

2021

By:

Zhao, Li;
Liu, Tao;
Dou, Zhan-jun;
Wang, Mei-ting;
Hu, Zi-xuan;
Wang, Bei

Publication type:

journal article

A dual inhibitor of FAAH and TRPV1 channels shows dose-dependent effect on depression-like behaviour in rats.

Published in:

Acta Neuropsychiatrica, 2017, v. 29, n. 6, p. 324, doi. 10.1017/neu.2016.68

By:

Kirkedal, Christian;
Wegener, Gregers;
Moreira, Fabricio;
Joca, Sâmia Regiane Lourenco;
Liebenberg, Nico

Publication type:

Article

Rimonabant improves obesity but not the overall cardiovascular risk and quality of life; results from CARDIO-REDUSE (CArdiometabolic Risk reDuctIOn by Rimonabant: the Effectiveness in Daily practice and its USE).

Published in:

Family Practice, 2012, v. 29, n. 5, p. 521, doi. 10.1093/fampra/cms013

By:

Boesten, Jolien E J;
Kaper, Janneke;
Stoffers, Henri E J H;
Kroon, Abraham A;
van Schayck, Onno C P

Publication type:

Article

Effect of rimonabant and metformin on glucose-dependent insulinotropic polypeptide and glucagon-like peptide-1 in obese women with polycystic ovary syndrome.

Published in:

2010

By:

Sathyapalan, Thozhukat;
Cho, LiWei;
Kilpatrick, Eric S.;
Le Roux, Carel W.;
Coady, Anne-Marie;
Atkin, Stephen L.

Publication type:

Letter

Effect of rimonabant on oesophageal motor function in man.

Published in:

Alimentary Pharmacology & Therapeutics, 2011, v. 33, n. 6, p. 730, doi. 10.1111/j.1365-2036.2011.04576.x

By:

Scarpellini, E.;
Blondeau, K.;
Boecxstaens, V.;
Vos, R.;
Gasbarrini, A.;
Farré, R.;
Tack, J.

Publication type:

Article

Endocannabinoid control of gastric sensorimotor function in man.

Published in:

Alimentary Pharmacology & Therapeutics, 2010, v. 31, n. 10, p. 1123, doi. 10.1111/j.1365-2036.2010.04259.x

By:

AMELOOT, K.;
JANSSEN, P.;
SCARPELLINI, E.;
VOS, R.;
BOESMANS, W.;
DEPOORTERE, I.;
VANDEN BERGHE, P.;
TACK, J.

Publication type:

Article

Comparative effects of cannabinoid CB1 receptor agonist and antagonist on timing impulsivity induced by d-amphetamine in a differential reinforcement of low-rate response task in male rats.

Published in:

Psychopharmacology, 2022, v. 239, n. 5, p. 1459, doi. 10.1007/s00213-021-06018-z

By:

Chen, Shuo-Fu;
Hsu, Wei-Chung;
Lu, Xi-Yun;
Chuang, Chuen-Yu;
Liao, Ruey-Ming

Publication type:

Article

Cannabinoid receptor-1 signaling contributions to sign-tracking and conditioned reinforcement in rats.

Published in:

Psychopharmacology, 2018, v. 235, n. 10, p. 3031, doi. 10.1007/s00213-018-4993-6

By:

Bacharach, Sam Z.;
Nasser, Helen M.;
Zlebnik, Natalie E.;
Dantrassy, Hannah M.;
Kochli, Daniel E.;
Gyawali, Utsav;
Cheer, Joseph F.;
Calu, Donna J.

Publication type:

Article

Δ9 -Tetrahydrocannabinol-like discriminative stimulus effects of five novel synthetic cannabinoids in rats.

Published in:

Psychopharmacology, 2018, v. 235, n. 3, p. 673, doi. 10.1007/s00213-017-4783-6

By:

Gatch, Michael B.;
Forster, Michael J.

Publication type:

Article

Cannabinoid withdrawal in mice: inverse agonist vs neutral antagonist.

Published in:

Psychopharmacology, 2015, v. 232, n. 15, p. 2751, doi. 10.1007/s00213-015-3907-0

By:

Tai, Sherrica;
Nikas, Spyros;
Shukla, Vidyanand;
Vemuri, Kiran;
Makriyannis, Alexandros;
Järbe, Torbjörn

Publication type:

Article

Rimonabant's reductive effects on high densities of food reinforcement, but not palatability, in lean and obese Zucker rats.

Published in:

Psychopharmacology, 2014, v. 231, n. 10, p. 2159, doi. 10.1007/s00213-013-3366-4

By:

Buckley, Jessica;
Rasmussen, Erin

Publication type:

Article

Differentiation between low- and high-efficacy CB receptor agonists using a drug discrimination protocol for rats.

Published in:

Psychopharmacology, 2014, v. 231, n. 3, p. 489, doi. 10.1007/s00213-013-3257-8

By:

Järbe, Torbjörn;
LeMay, Brian;
Halikhedkar, Aneetha;
Wood, JodiAnne;
Vadivel, Subramanian;
Zvonok, Alexander;
Makriyannis, Alexandros

Publication type:

Article

Tethered agonist activated ADGRF1 structure and signalling analysis reveal basis for G protein coupling.

Published in:

Nature Communications, 2023, v. 14, n. 1, p. 1, doi. 10.1038/s41467-023-38083-7

By:

Jones, Daniel T. D.;
Dates, Andrew N.;
Rawson, Shaun D.;
Burruss, Maggie M.;
Lipper, Colin H.;
Blacklow, Stephen C.

Publication type:

Article

Oral Communication 12, Tuesday Sept. 25th 5.00 pm–6.00 pm; Room: Lecture Hall 3.

Published in:: Alcohol & Alcoholism. Supplement, 2007, v. 42, p. i46, doi. 10.1093/alcalc/agm124
Publication type:: Article

Symposium 17 Monday Sept. 24th 6.30 pm–8.00 pm; Room: Lecture Hall 1.

Published in:: 2007
Publication type:: Proceeding

A systematic review of the effectiveness of smoking relapse prevention interventions for abstinent smokers.

Published in:

Addiction, 2010, v. 105, n. 8, p. 1362, doi. 10.1111/j.1360-0443.2010.02996.x

By:

Agboola, Shade;
McNeill, Ann;
Coleman, Tim;
Leonardi Bee, Jo

Publication type:

Article

Potential antipsychotic properties of central cannabinoid (CB1) receptor antagonists.

Published in:

World Journal of Biological Psychiatry, 2010, v. 11, n. 2_2, p. 208, doi. 10.3109/15622970801908047

By:

Roser, Patrik;
Vollenweider, Franz X.;
Kawohl, Wolfram

Publication type:

Article

Compensatory Activation of Cannabinoid CB2 Receptor Inhibition of GABA Release in the Rostral Ventromedial Medulla in Inflammatory Pain.

Published in:

Journal of Neuroscience, 2017, v. 37, n. 3, p. 626, doi. 10.1523/JNEUROSCI.1310-16.2017

By:

Ming-Hua Li;
Suchland, Katherine L.;
Ingram, Susan L.

Publication type:

Article

Effect of CB1 Receptor Blockade on Food-Reinforced Responding and Associated Nucleus Accumbens Neuronal Activity in Rats.

Published in:

Journal of Neuroscience, 2012, v. 32, n. 33, p. 11467, doi. 10.1523/JNEUROSCI.1833-12.2012

By:

Hernandez, Giovanni;
Cheer, Joseph F.

Publication type:

Article

Reduced Food Intake is the Major Contributor to the Protective Effect of Rimonabant on Islet in Established Obesity-Associated Type 2 Diabetes.

Published in:

Yonsei Medical Journal, 2013, v. 54, n. 5, p. 1127, doi. 10.3349/ymj.2013.54.5.1127

By:

Sang-Man Jin;
Bae Jun Oh;
Suel Lee;
Jung Mook Choi;
Soo Jin Yang;
Sung Woo Park;
Kwang-Won Kim;
Jae Hyeon Kim;
Cheol-Young Park

Publication type:

Article

Uso terapêutico dos canabinoides em psiquiatria.

Published in:

Brazilian Journal of Psychiatry / Revista Brasileira de Psiquiatria, 2010, v. 32, p. S56

By:

Crippa, José Alexandre S.;
Zuardi, Antonio Waldo;
Hallak, Jaime E. C.

Publication type:

Article

Targeting the Endocannabinoid/CB1 Receptor System For Treating Major Depression Through Antidepressant Activities of Curcumin and Dexanabinol-Loaded Solid Lipid Nanoparticles.

Published in:

Cellular Physiology & Biochemistry (Karger AG), 2017, v. 42, n. 6, p. 2281, doi. 10.1159/000480001

By:

He, Xiaolie;
Yang, Li;
Wang, Mei;
Zhuang, Xizhen;
Huang, Ruiqi;
Zhu, Rongrong;
Wang, Shilong

Publication type:

Article

Exploring the first Rimonabant analog-opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 444, doi. 10.1080/14756366.2016.1260565

By:

Mollica, Adriano;
Pelliccia, Sveva;
Famiglini, Valeria;
Stefanucci, Azzurra;
Macedonio, Giorgia;
Chiavaroli, Annalisa;
Orlando, Giustino;
Brunetti, Luigi;
Ferrante, Claudio;
Pieretti, Stefano;
Novellino, Ettore;
Benyhe, Sandor;
Zador, Ferenc;
Erdei, Anna;
Szucs, Edina;
Samavati, Reza;
Dvorácskó, Szabolcs;
Tomboly, Csaba;
Ragno, Rino;
Patsilinakos, Alexandros

Publication type:

Article

The CB1 Neutral Antagonist AM4113 Retains the Therapeutic Efficacy of the Inverse Agonist Rimonabant for Nicotine Dependence and Weight Loss with Better Psychiatric Tolerability.

Published in:

International Journal of Neuropsychopharmacology, 2016, v. 19, n. 12, p. 1, doi. 10.1093/ijnp/pyw068

By:

Gueye, Aliou B.;
Pryslawsky, Yaroslaw;
Trigo, Jose M.;
Poulia, Nafsika;
Delis, Foteini;
Antoniou, Katerina;
Loureiro, Michael;
Laviolette, Steve R.;
Vemuri, Kiran;
Makriyannis, Alexandros;
Le Foll, Bernard

Publication type:

Article

The CB1 Neutral Antagonist Tetrahydrocannabivarin Reduces Default Mode Network and Increases Executive Control Network Resting State Functional Connectivity in Healthy Volunteers.

Published in:

International Journal of Neuropsychopharmacology, 2016, v. 19, n. 2, p. 1, doi. 10.1093/ijnp/pyv092

By:

Rzepa, Ewelina;
Tudge, Luke;
McCabe, Ciara

Publication type:

Article

Neural Effects of Cannabinoid CB1 Neutral Antagonist Tetrahydrocannabivarin on Food Reward and Aversion in Healthy Volunteers.

Published in:

International Journal of Neuropsychopharmacology, 2015, v. 18, n. 6, p. 1, doi. 10.1093/ijnp/pyu094

By:

Tudge, Luke;
Williams, Clare;
Cowen, Philip J.;
McCabe, Ciara

Publication type:

Article

Reduced neural response to reward following 7 days treatment with the cannabinoid CB1 antagonist rimonabant in healthy volunteers.

Published in:

International Journal of Neuropsychopharmacology, 2010, v. 13, n. 8, p. 1103, doi. 10.1017/S1461145710000453

By:

Horder, Jamie;
Harmer, Catherine J.;
Cowen, Philip J.;
McCabe, Ciara

Publication type:

Article

Mitochondrial ADP/ATP exchange inhibition: a novel off-target mechanism underlying ibipinabant-induced myotoxicity.

Published in:

Scientific Reports, 2015, p. 14533, doi. 10.1038/srep14533

By:

Schirris, Tom J. J.;
Ritschel, Tina;
Herma Renkema, G.;
Willems, Peter H. G. M.;
Smeitink, Jan A. M.;
Russel, Frans G. M.

Publication type:

Article

The Endocannabinoid System and Cannabidiol's Promise for the Treatment of Substance Use Disorder.

Published in:

Frontiers in Psychiatry, 2019, p. N.PAG, doi. 10.3389/fpsyt.2019.00063

By:

Chye, Yann;
Christensen, Erynn;
Solowij, Nadia;
Yücel, Murat

Publication type:

Article

INVENTIVE MEDICINES - COSTLY MIRACLES OR MAYH EM OF THE MODERN SCIENCE.

Published in:

Review of Economic Studies & Research Virgil Madgearu, 2012, v. 5, n. 2, p. 139

By:

KESIČ, Dragan;
BERTONCELJ, Andrej

Publication type:

Article

Rimonabant assoziiert mit gravierenden neuropsychiatrischen Nebenwirkungen.

Published in:

Praxis (16618157), 2010, v. 99, n. 23, p. 1439, doi. 10.1024/1661-8157/a000314

By:

Steurer, Johann

Publication type:

Article

Effects of 7 days of treatment with the cannabinoid type 1 receptor antagonist, rimonabant, on emotional processing.

Published in:

Journal of Psychopharmacology, 2012, v. 26, n. 1, p. 125, doi. 10.1177/0269881111400649

By:

Horder, Jamie;
Browning, Michael;
Di Simplicio, Martina;
Cowen, Philip J;
Harmer, Catherine J

Publication type:

Article

Effects of Cannabinoid Exposure during Adolescence on the Conditioned Rewarding Effects of WIN 55212-2 and Cocaine in Mice: Influence of the Novelty-Seeking Trait.

Published in:

Neural Plasticity, 2015, v. 2015, p. 1, doi. 10.1155/2016/6481862

By:

Rodríguez-Arias, M.;
Roger-Sánchez, C.;
Vilanova, I.;
Revert, N.;
Manzanedo, C.;
Miñarro, J.;
Aguilar, M. A.

Publication type:

Article

Rimonabant Precipitates Anxiety in Rats Withdrawn from Palatable Food: Role of the Central Amygdala.

Published in:

Neuropsychopharmacology, 2013, v. 38, n. 12, p. 2498, doi. 10.1038/npp.2013.153

By:

Blasio, Angelo;
Iemolo, Attilio;
Sabino, Valentina;
Petrosino, Stefania;
Steardo, Luca;
Rice, Kenner C;
Orlando, Pierangelo;
Iannotti, Fabio Arturo;
Di Marzo, Vincenzo;
Zorrilla, Eric P;
Cottone, Pietro

Publication type:

Article

Genetic Deletion of Fatty Acid Amide Hydrolase Alters Emotional Behavior and Serotonergic Transmission in the Dorsal Raphe, Prefrontal Cortex, and Hippocampus.

Published in:

Neuropsychopharmacology, 2010, v. 35, n. 10, p. 2083, doi. 10.1038/npp.2010.80

By:

Bambico, Francis Rodriguez;
Cassano, Tommaso;
Dominguez-Lopez, Sergio;
Katz, Noam;
Walker, Claire Dominique;
Piomelli, Daniele;
Gobbi, Gabriella

Publication type:

Article

A Common Polymorphism in the Cannabinoid Receptor 1 (CNR1) Gene is Associated with Antipsychotic-Induced Weight Gain in Schizophrenia.

Published in:

Neuropsychopharmacology, 2010, v. 35, n. 6, p. 1315, doi. 10.1038/npp.2009.235

By:

Tiwari, Arun K.;
Zai, Clement C.;
Likhodi, Olga;
Lisker, Annika;
Singh, Deepika;
Souza, Renan P.;
Batra, Poonam;
Zaidi, Syed H. E.;
Sheng Chen;
Fang Liu;
Puls, Imke;
Meltzer, Herbert Y.;
Lieberman, Jeffrey A.;
Kennedy, James L.;
Müller, Daniel J

Publication type:

Article