Works about PYRIMIDINE derivatives
Results: 742
Mechanochemical Regioselective [3+3] Annulation of 6‐Amino Uracil with Propargyl Alcohols Catalyzed by a Brønsted Acid/Hexafluoroisopropanol.
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- Chemistry - A European Journal, 2024, v. 30, n. 48, p. 1, doi. 10.1002/chem.202401480
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- Article
The Boekelheide Rearrangement of Pyrimidine N‐oxides as a Case Study of Closed or Open Shell Reactions ‐ Experimental and Computational Evidence for the Participation of Radical Intermediates.
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- Chemistry - A European Journal, 2023, v. 29, n. 26, p. 1, doi. 10.1002/chem.202204015
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Air‐Stable Oxyallyl Patterns and a Switchable N‐Heterocyclic Carbene.
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- Angewandte Chemie, 2020, v. 132, n. 28, p. 11613, doi. 10.1002/ange.202002669
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- Article
Analgesic Activity and Acute Toxicity of Dihydrotetrazolo[1,5-a]Pyrimidine Derivatives.
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- Pharmaceutical Chemistry Journal, 2021, v. 55, n. 3, p. 228, doi. 10.1007/s11094-021-02403-2
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Development of Fused and Substituted Pyrimidine Derivatives as Potent Anticancer Agents (A Review).
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- Pharmaceutical Chemistry Journal, 2021, v. 54, n. 12, p. 1215, doi. 10.1007/s11094-021-02346-8
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- Article
Synthesis and Neurotropic Activity of Novel Condensed Cyclopentanopyrido[3',2':4,5]-Thieno[3,2-D]Pyrimidine Derivatives.
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- Pharmaceutical Chemistry Journal, 2020, v. 54, n. 7, p. 707, doi. 10.1007/s11094-020-02259-y
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Synthesis of Pyrimidino Derivatives: Potent Antimicrobial Candidates.
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- Pharmaceutical Chemistry Journal, 2017, v. 50, n. 10, p. 678, doi. 10.1007/s11094-017-1511-9
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Synthesis and Anticonvulsant Activity of 7(8)-Amino Derivatives of Condensed Thieno[3,2- d]Pyrimidines.
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- Pharmaceutical Chemistry Journal, 2016, v. 50, n. 5, p. 296, doi. 10.1007/s11094-016-1439-5
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Synthesis and Anticonvulsive Activity of 5-Pyrrolidin-1-Ylpyrano[4″,3″:4′,5′]Pyrido-3′,2′:4,5]Thieno[3,2- D]Pyrimidine Derivatives.
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- Pharmaceutical Chemistry Journal, 2016, v. 50, n. 4, p. 221, doi. 10.1007/s11094-016-1426-x
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- Article
Synthesis and Analgesic Activity of N,6-diaryl-4-methyl-2-thioxo-1,2,3,6-tetrahydropyrimidine-5-carboxamides.
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- Pharmaceutical Chemistry Journal, 2016, v. 50, n. 4, p. 226, doi. 10.1007/s11094-016-1427-9
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- Article
Biological Activity of Adamantane-Containing Mono- and Polycyclic Pyrimidine Derivatives* (A Review).
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- Pharmaceutical Chemistry Journal, 2016, v. 50, n. 2, p. 63, doi. 10.1007/s11094-016-1400-7
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- Article
Synthesis and Antimycobacterial Activity of 5-(Arylmethylene)Hexahydropyrimidine-2,4,6-Triones.
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- Pharmaceutical Chemistry Journal, 2016, v. 49, n. 12, p. 810, doi. 10.1007/s11094-016-1376-3
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Synthesis and Antifungal Activity Against Candida Albicans of 6-Aryl-3,4-Dimethyl- N-Phenyl-2-Oxo-1,2,3,6-Tetrahydropyrimidine-5-Carboxamides.
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- Pharmaceutical Chemistry Journal, 2015, v. 49, n. 8, p. 509, doi. 10.1007/s11094-015-1316-7
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Synthesis and Antimicrobial Activity of N-5-Diaryl-7-Methyl-3-OXO-2,3-Dihydro-5 H-[1,3]Thiazolo[3,2- a]Pyrimidine-6-Carboxamide Hydrochlorides.
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- Pharmaceutical Chemistry Journal, 2015, v. 49, n. 8, p. 512, doi. 10.1007/s11094-015-1317-6
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Synthesis and Antioxidant Activity of Ammonium Salts of 4-(3-Bromophenyl)-5-Methoxycarbonyl-1-( N, N-Dimethylaminopropyl)-3,4-Dihydropyrimidin-2-(1 H)-One.
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- Pharmaceutical Chemistry Journal, 2015, v. 49, n. 8, p. 515, doi. 10.1007/s11094-015-1318-5
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Synthesis and Evaluation of Thiazole - Pyrimidine Derivatives as New Anticandidal and Cytotoxic Agents.
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- Pharmaceutical Chemistry Journal, 2014, v. 48, n. 7, p. 452, doi. 10.1007/s11094-014-1130-7
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- Article
Synthesis and Neurotropic Activity of 8-Amino Derivatives of Condensed Thieno[3,2- d]- and Furo[3,2- d]Pyrimidines.
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- Pharmaceutical Chemistry Journal, 2014, v. 47, n. 12, p. 655, doi. 10.1007/s11094-014-1026-6
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- Article
Synthesis and Neurotropic Activity of New Condensed Pyrido[3′,2′:4,5]furo[3,2- d]-pyrimidine Derivatives.
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- Pharmaceutical Chemistry Journal, 2013, v. 47, n. 3, p. 135, doi. 10.1007/s11094-013-0911-8
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- Article
Antagonists of serotonin 5-HT receptors. III. Pyridine-substituted 3-(phenylsulfonyl)pyrazolo[1,5- a]pyrimidines: synthesis and structure - activity relationship.
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- Pharmaceutical Chemistry Journal, 2012, v. 46, n. 7, p. 406, doi. 10.1007/s11094-012-0810-4
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- Article
Synthesis and neurotropic activity of new condensed pyrido[3',2':4,5]thieno[3,2- d]pyrimidine derivatives.
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- Pharmaceutical Chemistry Journal, 2012, v. 46, n. 5, p. 271, doi. 10.1007/s11094-012-0778-0
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- Article
Synthesis and neurotropic activity of condensed thieno[2,3 e][1,2,4]triazolo[4,3-c]pyrimidine derivatives.
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- Pharmaceutical Chemistry Journal, 2012, v. 46, n. 3, p. 154, doi. 10.1007/s11094-012-0750-z
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Thiopyrimidine derivatives: synthesis and antibacterial activity.
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- Pharmaceutical Chemistry Journal, 2012, v. 46, n. 2, p. 117, doi. 10.1007/s11094-012-0744-x
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- Article
Structure of new derivatives of perhydropyrimidine-2-ones and intermolecular interactions in their crystals.
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- Journal of Structural Chemistry, 2017, v. 58, n. 2, p. 283, doi. 10.1134/S0022476617020093
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- Article
An unusual conformational change in the folded trimethylene/leonard linker pyrazolo[3,4- d]pyrimidine analogue of the theophylline compound due to structural changes.
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- Journal of Structural Chemistry, 2015, v. 56, n. 7, p. 1437, doi. 10.1134/S0022476615070306
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Synthesis and crystal structure analysis of two thiazolo[3,2- a]pyrimidine derivatives.
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- Journal of Structural Chemistry, 2014, v. 55, n. 8, p. 1521, doi. 10.1134/S0022476614080204
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Synthesis and crystal structure analysis of two thiazolo[3,2- a]pyrimidine derivatives.
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- Journal of Structural Chemistry, 2014, v. 55, n. 7, p. 1521, doi. 10.1134/S0022476614080204
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1SYNTHESIS AND ANTIOXIDANT ACTIVITY OF NEW 2-(2-OXOINDOLINE-3-YLYDENE) SUBSTITUTED 5,6-DIHYDROIMIDAZO[2,1-b]THIAZOLONES AND 6,7-DIHYDRO-THIAZOLO[3,2-a]PYRIMIDINONES.
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- Issues of Chemistry & Chemical Technology / Voprosy Khimii & Khimicheskoi Tekhnologii, 2025, n. 1, p. 71, doi. 10.32434/0321-4095-2025-158-1-71-79
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SYNTHESIS OF PYRAZOLO[1,5-a][1,3,5]TRIAZINE AND OXAZOLO[4,5-d]PYRIMIDINE DERIVATIVES AND STUDY OF THEIR VASODILATOR ACTIVITY.
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- Issues of Chemistry & Chemical Technology / Voprosy Khimii & Khimicheskoi Tekhnologii, 2023, n. 2, p. 51, doi. 10.32434/0321-4095-2023-147-2-51-60
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Synthesis of new imine-/amine-bearing imidazo[1,2-a]pyrimidine derivatives and screening of their cytotoxic activity.
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- Turkish Journal of Chemistry, 2023, v. 47, n. 5, p. 1064, doi. 10.55730/1300-0527.3594
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Recent synthetic methodologies for pyrimidine and its derivatives.
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- Turkish Journal of Chemistry, 2018, v. 42, n. 6, p. 1421, doi. 10.3906/kim-1806-8
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Synthesis, reaction, and evaluation of the anticancer activity of 6,7,8,9-tetrahydro-5H-cyclohepta[4,5]selenopheno[2,3-d]pyrimidine derivatives.
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- Turkish Journal of Chemistry, 2016, v. 40, n. 4, p. 631, doi. 10.3906/kim-1508-69
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- Article
Synthesis of new pyrazole and antibacterial pyrazolopyrimidine derivatives.
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- Turkish Journal of Chemistry, 2014, v. 38, n. 2, p. 210, doi. 10.3906/kim-1303-20
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Design, synthesis, docking, MD simulations, and anti-proliferative evaluation of thieno[2,3-d]pyrimidine derivatives as new EGFR inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2220579
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Design, synthesis, and biological evaluation of pyrido[2,3-d]pyrimidine and thieno[2,3-d]pyrimidine derivatives as novel EGFR<sup>L858R/T790M</sup> inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2205605
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Synthesis, DFT calculations, and anti-proliferative evaluation of pyrimidine and selenadiazolopyrimidine derivatives as dual Topoisomerase II and HSP90 inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2198163
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Correction.
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- 2023
- Publication type:
- Correction Notice
Design, synthesis and biological evaluation of 2-((4-sulfamoylphenyl)amino)-pyrrolo[2,3-d]pyrimidine derivatives as CDK inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2169282
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Biological evaluation, docking studies, and in silico ADME prediction of some pyrimidine and pyridine derivatives as potential EGFR<sup>WT</sup> and EGFR<sup>T790M</sup> inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 176, doi. 10.1080/14756366.2022.2135512
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Targeting p21-activated kinase 4 (PAK4) with pyrazolo[3,4-d]pyrimidine derivative SPA7012 attenuates hepatic ischaemia-reperfusion injury in mice.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 2133, doi. 10.1080/14756366.2022.2106478
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Discovery of new 1H-pyrazolo[3,4-d]pyrimidine derivatives as anticancer agents targeting EGFR<sup>WT</sup> and EGFR<sup>T790M</sup>.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 2283, doi. 10.1080/14756366.2022.2112575
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Design, synthesis, and biological evaluation of new thieno[2,3-d] pyrimidine derivatives as targeted therapy for PI3K with molecular modelling study.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 315, doi. 10.1080/14756366.2021.2010729
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Synthesis and biological evaluation of novel thienopyrimidine derivatives as diacylglycerol acyltransferase 1 (DGAT-1) inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 227, doi. 10.1080/14756366.2019.1693555
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Design, synthesis, molecular modelling, and biological evaluation of novel substituted pyrimidine derivatives as potential anticancer agents for hepatocellular carcinoma.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1110, doi. 10.1080/14756366.2019.1612889
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Novel thienopyrimidine derivatives as dual EGFR and VEGFR-2 inhibitors: design, synthesis, anticancer activity and effect on cell cycle profile.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 838, doi. 10.1080/14756366.2019.1593160
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- Article
Synthesis and in vivo anti-ulcer evaluation of some novel piperidine linked dihydropyrimidinone derivatives.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 978, doi. 10.1080/14756366.2018.1474212
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Synthesis and evaluation of novel spiro derivatives for pyrrolopyrimidines as anti-hyperglycemia promising compounds.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 809, doi. 10.1080/14756366.2018.1461854
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Synthesis of new pyridothienopyrimidinone and pyridothienotriazolopyrimidine derivatives as pim-1 inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 58, doi. 10.1080/14756366.2017.1389921
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Design, synthesis and biological activity of N<sup>4</sup>-phenylsubstituted-7H-pyrrolo[2,3-d]pyrimidin-4-amines as dual inhibitors of aurora kinase A and epidermal growth factor receptor kinase.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 74, doi. 10.1080/14756366.2017.1376666
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The role of 5-arylalkylamino- and 5-piperazino- moieties on the 7-aminopyrazolo[4,3- d ]pyrimidine core in affecting adenosine A 1 and A 2A receptor affinity and selectivity profiles.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 248, doi. 10.1080/14756366.2016.1247060
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Synthesis, cyclooxygenase inhibition, anti-inflammatory evaluation and ulcerogenic liability of new 1-phenylpyrazolo[3,4- d ]pyrimidine derivatives.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 6, doi. 10.1080/14756366.2016.1186018
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- Article