Works matching DE "PYRIDONE derivatives"

Results: 43

Protective Effect of A<sub>2B</sub> Receptor Antagonist (TRP 1) on Acetic Acid Induced Ulcerative Colitis in Rats: in vitro, in vivo and in silico Methods.

Published in:

Indian Journal of Pharmaceutical Education & Research, 2018, v. 52, n. 1, p. 101, doi. 10.5530/ijper.52.1.12

By:

Pasala, Praveen Kumar;
Alluri, Ramesh;
Mavulati, Sri Chandana;
Mailavaram, Raghu Prasad;
Shaik, Khasim;
Konduri, Prasad

Publication type:

Article

Similar pyridinone compounds with different activities of anti -HIV-1 reverse transcriptase.

Published in:

Journal of Chinese Pharmaceutical Sciences, 2018, v. 27, n. 7, p. 469, doi. 10.5246/jcps.2018.07.048

By:

Yunqi Liu;
Xixi Li;
Xiaodong Dou;
Chao Tian;
Zhili Zhang;
Junyi Liu;
Xiaowei Wang

Publication type:

Article

Microwave-assisted synthesis of 2-pyridone 2-pyridone-based compounds.

Published in:

Chemical Industry / Hemijska Industrija, 2014, v. 68, n. 1, p. 1, doi. 10.2298/HEMIND121204021M

By:

Mijin, Dušan Ž.;
Marković, Jelena M.;
Brković, Danijela V.;
Marinković, Aleksandar D.

Publication type:

Article

Four-component reaction between cyanoacetamide, aryl aldehydes, and ethyl acetoacetate with ammonium carbonate.

Published in:

Research on Chemical Intermediates, 2015, v. 41, n. 2, p. 1001, doi. 10.1007/s11164-013-1250-9

By:

Dehghan, Alimohammad;
Singh, Sonia;
Anary-Abbasinejad, Mohammad;
Hassanabadi, Alireza

Publication type:

Article

Synthesis, preliminary biological evaluation and 3D-QSAR study of novel 1,5-disubstituted-2(1H)-pyridone derivatives as potential anti-lung cancer agents.

Published in:

Arabian Journal of Chemistry, 2016, v. 9, n. 5, p. 721, doi. 10.1016/j.arabjc.2015.08.001

By:

Xu, Qifei;
Jiang, Xiaoding;
Zhu, Weixing;
Chen, Chuo;
Hu, Gaoyun;
Li, Qianbin

Publication type:

Article

Efficient One-Pot Four-Component Synthesis and X-ray Crystallographic Structure of 2-Pyridone Derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2013, v. 50, n. 6, p. 1272, doi. 10.1002/jhet.1632

By:

Balalaie, Saeed;
Hashemi, Mohammed M.;
Khezri, S. Hadi;
Rominger, Frank;
Ghabraie, Elmira;
Oeser, Thomas

Publication type:

Article

Simultaneous measurement of nicotinamide and its catabolites, nicotinamide N-oxide, N¹-methyl-2-pyridone-5-carboxamide, and N¹-methyl-4-pyridone-3-carboxamide, in mice urine.

Published in:

Bioscience, Biotechnology & Biochemistry, 2014, v. 78, n. 8, p. 1306, doi. 10.1080/09168451.2014.918495

By:

Akihiro Maeta;
Mitsue Sano;
Tsutomu Fukuwatari;
Katsumi Shibata

Publication type:

Article

Classical QSAR and Docking Simulation of 4-Pyridone Derivatives for Their Antimalarial Activity.

Published in:

Molecules, 2018, v. 23, n. 12, p. 3166, doi. 10.3390/molecules23123166

By:

Flores-Sumoza, Máryury;
Alcázar, Jackson J.;
Márquez, Edgar;
Mora, José R.;
Lezama, Jesús;
Puello, Esneyder;
Brogi, Simone

Publication type:

Article

Rhodium(I)-Complexes Catalyzed 1,4-Conjugate Addition of Arylzinc Chlorides to N-Boc-4-pyridone.

Published in:

Molecules, 2017, v. 22, n. 5, p. 723, doi. 10.3390/molecules22050723

By:

Fenghai Guo;
McGilvary, Matthew A.;
Jeffries, Malcolm C.;
Graves, Briana N.;
Graham, Shekinah A.;
Yuelin Wu

Publication type:

Article

Synthesis of Substituted α-Trifluoromethyl Piperidinic Derivatives.

Published in:

Molecules, 2017, v. 22, n. 3, p. 483, doi. 10.3390/molecules22030483

By:

Rioton, Sarah;
Pardo, Domingo Gomez;
Cossy, Janine

Publication type:

Article

Synthesis of Substituted 2-Pyridones Using Arylamidoesters of Malonic Acid.

Published in:

Chemistry of Heterocyclic Compounds, 2014, v. 50, n. 8, p. 1126, doi. 10.1007/s10593-014-1572-6

By:

Hayotsyan, S.;
Hasratyan, A.;
Kon'kova, S.;
Khachatryan, A.;
Ayvazyan, A.;
Panosyan, G.;
Sargsyan, M.

Publication type:

Article

Synthesis of new tetrahydrobenzo[ b]pyrimido- [5,4- g][1,8]naphthyridine-2,4-diones from 6-aminouracils.

Published in:

Russian Journal of Organic Chemistry, 2017, v. 53, n. 10, p. 1609, doi. 10.1134/S1070428017100232

By:

Karakhanyan, G.

Publication type:

Article

Synthesis of pyrido[2,3- d]pyrimidines from 6-amino-1,3-dimethyluracil and aldehydes.

Published in:

Russian Journal of Organic Chemistry, 2015, v. 51, n. 12, p. 1784, doi. 10.1134/S1070428015120210

By:

Azev, Yu.;
Ermakova, O.;
Gibor, A.;
Bakulev, V.;
Ezhikova, M.;
Kodess, M.

Publication type:

Article

Indium-promoted Conversion of Allylic Bromide to Alcohol Moiety and Synthesis of Pipermethystine Skeletons.

Published in:

Journal of the Chinese Chemical Society, 2016, v. 63, n. 9, p. 818, doi. 10.1002/jccs.201600239

By:

Liou, Bo ‐ Sian;
Chou, Shang ‐ Shing Peter

Publication type:

Article

Dual targeting of MDM2 with a novel small-molecule inhibitor overcomes TRAIL resistance in cancer.

Published in:

Carcinogenesis, 2016, v. 37, n. 11, p. 1027, doi. 10.1093/carcin/bgw088

By:

Singh, Anup Kumar;
Chauhan, Shikha S.;
Singh, Sudhir Kumar;
Verma, Ved Vrat;
Singh, Akhilesh;
Arya, Rakesh Kumar;
Maheshwari, Shrankhla;
Akhtar, Md. Sohail;
Sarkar, Jayanta;
Rangnekar, Vivek M.;
Chauhan, Prem M. S.;
Datta, Dipak

Publication type:

Article

Synthesis of Pyridone Derivatives from 7-Hydroxy-7-polyfluoroalkylhexahydroimidazo[1,2-a]pyridin-5-ones.

Published in:

European Journal of Organic Chemistry, 2017, v. 2017, n. 27, p. 3986, doi. 10.1002/ejoc.201700683

By:

Goryaeva, Marina V.;
Burgart, Yanina V.;
Kudyakova, Yulia S.;
Ezhikova, Marina A.;
Kodess, Mikhail I.;
Saloutin, Victor I.

Publication type:

Article

Pyridone Functionalization: Regioselective Deprotonation of 6-Methylpyridin-2(1 H)- and -4(1 H)-one Derivatives.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 31, p. 5238, doi. 10.1002/ejoc.201601156

By:

Diaz Ropero, Beatriz P. Fernandez;
Elsegood, Mark R. J.;
Fairley, Gary;
Pritchard, Gareth J.;
Weaver, George W.

Publication type:

Article

Time-Efficient Synthesis of Pyrido[2,3- d]pyrimidinones via α-Oxoketenes.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 11, p. 1994, doi. 10.1002/ejoc.201600171

By:

Castillo, Juan‐Carlos;
Quiroga, Jairo;
Rodriguez, Jean;
Coquerel, Yoann

Publication type:

Article

Pirfenidone for the treatment of idiopathic pulmonary fibrosis.

Published in:

Expert Review of Clinical Pharmacology, 2017, v. 10, n. 5, p. 483, doi. 10.1080/17512433.2017.1295846

By:

George, Peter M;
Wells, Athol U

Publication type:

Article

N-Heterocyclic Carbene Catalyzed Cyclocondensation of a,b- Unsaturated Carboxylic Acids: Enantioselective Synthesis of Pyrrolidinone and Dihydropyridinone Derivatives.

Published in:

Angewandte Chemie International Edition, 2014, v. 53, n. 43, p. 11611, doi. 10.1002/anie.201407469

By:

Chen, Xiang‐Yu;
Gao, Zhong‐Hua;
Song, Chun‐Yu;
Zhang, Chun‐Lin;
Wang, Zhi‐Xiang;
Ye, Song

Publication type:

Article

Fluorofenidone attenuates vascular remodeling in hypoxia-induced pulmonary hypertension of rats.

Published in:

Canadian Journal of Physiology & Pharmacology, 2014, v. 92, n. 1, p. 58, doi. 10.1139/cjpp-2013-0056

By:

Li, Xian-Wei;
Du, Jie;
Hu, Gao-Yun;
Hu, Chang-Ping;
Li, Dai;
Li, Yuan-Jian;
Li, Xiao-Hui

Publication type:

Article

RP-HPLC and UV Spectrophotometric Methods for Estimation of Pirfenidone in Pharmaceutical Formulations.

Published in:

Indian Journal of Pharmaceutical Sciences, 2014, v. 76, n. 3, p. 225

By:

PARMAR, V. K.;
DESAI, S. B.;
VAJA, T.

Publication type:

Article

Modification of microcrystalline cellulose with pyridone derivatives for removal of cationic dyes from aqueous solutions.

Published in:

Cellulose, 2016, v. 23, n. 5, p. 2917, doi. 10.1007/s10570-016-1024-9

By:

Sun, Chang;
Huang, Zhiyong;
Wang, Jiaxin;
Rao, Liming;
Zhang, Jingjing;
Yu, Jiao;
Du, Jinmei;
Xu, Changhai

Publication type:

Article

Anti-mycobacterial activities of copper(II) complexes. Part II. Lipophilic hydroxypyridinones derived from maltol.

Published in:

Canadian Journal of Chemistry, 2015, v. 93, n. 3, p. 334, doi. 10.1139/cjc-2014-0426

By:

Salsbury, Lauren E.;
Robertson, Katherine N.;
Flewelling, Andrew J.;
Li, Hoaxin;
Geier, Stephen J.;
Vogels, Christopher M.;
Gray, Christopher A.;
Westcott, Stephen A.

Publication type:

Article

Enantioselective Pd-Catalyzed Allylic Alkylation Reactions of Dihydropyrido[1,2- a]indolone Substrates: Efficient Syntheses of (−)-Goniomitine, (+)-Aspidospermidine, and (−)-Quebrachamine.

Published in:

Angewandte Chemie, 2016, v. 128, n. 43, p. 13727, doi. 10.1002/ange.201608138

By:

Pritchett, Beau P.;
Kikuchi, Jun;
Numajiri, Yoshitaka;
Stoltz, Brian M.

Publication type:

Article

N-Heterocyclic Carbene Catalyzed Cyclocondensation of α,β- Unsaturated Carboxylic Acids: Enantioselective Synthesis of Pyrrolidinone and Dihydropyridinone Derivatives.

Published in:

Angewandte Chemie, 2014, v. 126, n. 43, p. 11795, doi. 10.1002/ange.201407469

By:

Chen, Xiang ‐ Yu;
Gao, Zhong ‐ Hua;
Song, Chun ‐ Yu;
Zhang, Chun ‐ Lin;
Wang, Zhi ‐ Xiang;
Ye, Song

Publication type:

Article

A Facile Synthesis of Pyrido[2,3 :3,4]pyrazolo[1,5-a]pyrimidine and Pyrido[2',3':3,4]pyrazolo[5,1-c][1,2,4]triazine Bearing a Thiophene Moiety.

Published in:

Journal of Chemistry, 2013, p. 1, doi. 10.1155/2013/463515

By:

Elsaman, Tilal;
Fares, Mohamed;
Abdel-Aziz, Hatem A.;
Attia, Mohamed I.;
Ghabbour, Hazem A.;
Dawood, Kamal M.

Publication type:

Article

Focused microwave-assisted efficient and convenient synthesis of new pyrido[2,3- d]pyrimidinone derivatives.

Published in:

Heterocyclic Communications, 2012, v. 18, n. 5/6, p. 257, doi. 10.1515/hc-2012-0131

By:

Quan, Zheng-Jun;
Liang, Jun-Ling;
Bai, Lin;
Zhang, Zhang;
Da, Yu-Xia;
Wang, Xi-Cun

Publication type:

Article

Synthesis of ester functionalized 2-pyridone derivatives using KF/Alumina as a catalyst.

Published in:

Organic Communications, 2016, v. 9, n. 1, p. 15

By:

Mahesh, Bellam;
Reddy, Kandula Madhu Kumar;
Reddy, Gajjala Raghavendra;
Reddy, Nadiveedhi Maheshwara;
Reddy, Cirandur Suresh

Publication type:

Article

Preparation, Characterization, Redox, and Photoinduced Electron-Transfer Properties of the NIR-Absorbing N-Ferrocenyl-2-pyridone BODIPYs.

Published in:

European Journal of Inorganic Chemistry, 2017, v. 2017, n. 2, p. 318, doi. 10.1002/ejic.201600855

By:

Zatsikha, Yuriy V.;
Didukh, Natalia O.;
Blesener, Tanner;
Kayser, Mathew P.;
Kovtun, Yuriy P.;
Blank, David A.;
Nemykin, Victor N.

Publication type:

Article

Effects of 4-Pyridone-3-carboxamide-1β-D-ribonucleoside on adenine nucleotide catabolism in the aortic wall; Implications for atherosclerosis in ApoE-/-LDLR-/- mice.

Published in:

Nucleosides, Nucleotides & Nucleic Acids, 2016, v. 35, n. 10-12, p. 720, doi. 10.1080/15257770.2016.1154970

By:

Zabielska, Magdalena;
Kutryb-Zajac, Barbara;
Żukowska, Paulina;
Slominska, Ewa;
Smoleński, Ryszard

Publication type:

Article

3D-QSAR studies on a diverse set of heterocyclic MMP inhibitors.

Published in:

International Journal of Pharmacy & Life Sciences, 2012, v. 3, n. 7, p. 1819

By:

Gade, Swetha;
Mahmood, Shaik

Publication type:

Article

Pirfenidone Induces G1 Arrest in Human Tenon's Fibroblasts In Vitro Involving AKT and MAPK Signaling Pathways.

Published in:

2017

By:

Guo, Xiujuan;
Yang, Yangfan;
Liu, Liling;
Liu, Xiaoan;
Xu, Jiangang;
Wu, Kaili;
Yu, Minbin

Publication type:

journal article

The discovery of S/GSK1265744: a carbamoyl pyridone HIV-1 integrase inhibitor.

Published in:

Journal of the International AIDS Society, 2012, v. 15, p. 1, doi. 10.7448/IAS.15.6.18267

By:

Taoda, Y;
Johns, B;
Weatherhead, J;
Temelkoff, D;
Kawasuji, T;
Yoshida, H;
Taishi, T;
Kiyama, R;
Fuji, M;
Murai, H;
Yoshinaga, T;
Sato, A;
Fujiwara, T

Publication type:

Article

Wide‐Range Columnar and Lamellar Photoluminescent Liquid‐Crystalline Lanthanide Complexes with Mesogenic 4‐Pyridone Derivatives.

Published in:

Chemistry - A European Journal, 2018, v. 24, n. 51, p. 13512, doi. 10.1002/chem.201801781

By:

Chiriac, Laura F.;
Pasuk, Iuliana;
Secu, Mihail;
Micutz, Marin;
Cîrcu, Viorel

Publication type:

Article

Anticancer evaluation and molecular modeling of multi-targeted kinase inhibitors based pyrido[2,3-d]pyrimidine scaffold.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 546, doi. 10.1080/14756366.2018.1437729

By:

Elzahabi, Heba S. A.;
Nossier, Eman S.;
Khalifa, Nagy M.;
Alasfoury, Rania A.;
El-Manawaty, May A.

Publication type:

Article

Pirfenidone attenuates bladder fibrosis and mitigates deterioration of bladder function in a rat model of partial bladder outlet obstruction.

Published in:

Molecular Medicine Reports, 2015, v. 12, n. 3, p. 3639, doi. 10.3892/mmr.2015.3814

By:

LIU JIAN DUAN;
JUN QI;
TAO HUANG;
XIN GU;
DING XU;
XIANG JIE KONG;
XIAO QIANG QIAN

Publication type:

Article

Clinical detection and categorization of uncommon and concomitant mutations involving BRAF.

Published in:

2015

By:

Gang Zheng;
Li-Hui Tseng;
Guoli Chen;
Haley, Lisa;
Illei, Peter;
Gocke, Christopher D.;
Eshleman, James R.;
Ming-Tseh Lin;
Zheng, Gang;
Tseng, Li-Hui;
Chen, Guoli;
Lin, Ming-Tseh

Publication type:

journal article

Synthesis of 1,3,4-Oxa(Thia)Diazole Derivatives of Amidomethylcytisine.

Published in:

Chemistry of Natural Compounds, 2018, v. 54, n. 4, p. 826, doi. 10.1007/s10600-018-2489-6

By:

Ismailova, D. S.;
Ziyaev, A. A.;
Levkovich, M. G.;
Toshmurodov, T. T.

Publication type:

Article

Search for compounds with antiviral activity among synthetic (-)-cytisine derivatives.

Published in:

Chemistry of Natural Compounds, 2013, v. 48, n. 6, p. 1042, doi. 10.1007/s10600-013-0460-0

By:

Tsypysheva, I.;
Koval'skaya, A.;
Lobov, A.;
Zarubaev, V.;
Karpinskaya, L.;
Petrenko, I.;
Nikolaeva, E.;
Shtro, A.;
Yunusov, M.

Publication type:

Article

The structure of products of phenacylation and subsequent (re)cyclizations of 3-acetyl-4,6-dimethylpyridin-2(1 H)-one according to X-ray structural analysis.

Published in:

Chemistry of Heterocyclic Compounds, 2017, v. 53, n. 9, p. 997, doi. 10.1007/s10593-017-2161-2

By:

Okul', Ekaterina;
Rybakov, Victor;
Babaev, Eugene

Publication type:

Article

Synthesis of 10-alkylsulfanyl-substituted pyrido-[4',3':4,5]thieno[3,2- d]pyrimidines annulated with pyran, cyclohexane, and cyclopentane rings.

Published in:

Chemistry of Heterocyclic Compounds, 2016, v. 52, n. 5, p. 337, doi. 10.1007/s10593-016-1887-6

By:

Paronikyan, Ervand;
Dashyan, Shushanik;
Minasyan, Nune;
Stepanyan, Grachya;
Babaev, Evgene

Publication type:

Article

Recent syntheses of ellipticine and its derivatives.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2018, v. 2018, p. 216, doi. 10.24820/ark.5550190.p010.445

By:

Ibrahim-Ouali, Malika;
Dumur, Frédéric

Publication type:

Article