Works matching DE "PROTEASE inhibitors synthesis"

Results: 13

Drug-1,3,4-Thiadiazole Conjugates as Novel Mixed-Type Inhibitors of Acetylcholinesterase: Synthesis, Molecular Docking, Pharmacokinetics, and ADMET Evaluation.

Published in:

Molecules, 2019, v. 24, n. 5, p. 860, doi. 10.3390/molecules24050860

By:

Ujan, Rabail;
Saeed, Aamer;
Channar, Pervaiz Ali;
Larik, Fayaz Ali;
Abbas, Qamar;
Alajmi, Mohamed F.;
El-Seedi, Hesham R.;
Rind, Mahboob Ali;
Hassan, Mubashir;
Raza, Hussain;
Seo, Sung-Yum

Publication type:

Article

Optimization, purification and characterization of novel thermostable, haloalkaline, solvent stable protease from Bacillus halodurans CAS6 using marine shellfish wastes: a potential additive for detergent and antioxidant synthesis.

Published in:

Bioprocess & Biosystems Engineering, 2013, v. 36, n. 7, p. 873, doi. 10.1007/s00449-012-0820-3

By:

Annamalai, Neelamegam;
Rajeswari, Mayavan;
Thavasi, Rengathavasi;
Vijayalakshmi, Shanmugam;
Balasubramanian, Thangavel

Publication type:

Article

Site-2 protease responds to oxidative stress and regulates oxidative injury in mammalian cells.

Published in:

Scientific Reports, 2014, p. 1, doi. 10.1038/srep06268

By:

Yong Gu;
Waisin Lee;
Jiangang Shen

Publication type:

Article

Granzyme B-inhibitor serpina3n induces neuroprotection in vitro and in vivo.

Published in:

Journal of Neuroinflammation, 2015, v. 12, n. 1, p. 1, doi. 10.1186/s12974-015-0376-7

By:

Haile, Yohannes;
Carmine-Simmen, Katia;
Olechowski, Camille;
Kerr, Bradley;
Bleackley, R. Chris;
Giuliani, Fabrizio

Publication type:

Article

Loss of CD26 protease activity in recipient mice during hematopoietic stem cell transplantation results in improved transplant efficiency.

Published in:

Transfusion, 2013, v. 53, n. 4, p. 878, doi. 10.1111/j.1537-2995.2012.03826.x

By:

Yoo, Eunsun;
Paganessi, Laura A.;
Alikhan, Wasfia A.;
Paganessi, Elizabeth A.;
Hughes, Frank;
Fung, Henry C.;
Rich, Elizabeth;
Seong, Chu Myong;
Christopherson 2nd, Kent W.

Publication type:

Article

Improving fold resistance prediction of HIV-1 against protease and reverse transcriptase inhibitors using artificial neural networks.

Published in:

BMC Bioinformatics, 2017, v. 18, p. 1, doi. 10.1186/s12859-017-1782-x

By:

Amamuddy, Olivier Sheik;
Bishop, Nigel T.;
Bishop, Özlem Tastan

Publication type:

Article

One-pot Synthesis of 1-Amidoalkyl-2-naphthols under Solvent-free Conditions.

Published in:

Organic Preparations & Procedures International, 2014, v. 46, n. 3, p. 252, doi. 10.1080/00304948.2014.903143

By:

Maleki, Behrooz;
Taimazi, Fereshteh

Publication type:

Article

Reverse Zymography Alone does not Confirm Presence of a Protease Inhibitor.

Published in:

Protein Journal, 2013, v. 32, n. 3, p. 155, doi. 10.1007/s10930-013-9470-9

By:

Dutta, Sangita;
Bhattacharyya, Debasish

Publication type:

Article

Protease-activated receptor-1 activation by granzyme B causes neurotoxicity that is augmented by interleukin-1β.

Published in:

2017

By:

Lee, Paul R.;
Johnson, Tory P.;
Gnanapavan, Sharmilee;
Giovannoni, Gavin;
Tongguang Wang;
Steiner, Joseph P.;
Medynets, Marie;
Vaal, Mark J.;
Gartner, Valerie;
Nath, Avindra;
Wang, Tongguang

Publication type:

journal article

Screening and characterization of protease producing actinomycetes from marine saltern.

Published in:

Journal of Basic Microbiology, 2014, v. 54, n. 10, p. 1098, doi. 10.1002/jobm.201300563

By:

Suthindhiran, Krish;
Jayasri, Mangalam Achuthananda;
Dipali, Dipa;
Prasar, Apurva

Publication type:

Article

Synthesis of carbon-14 and stable isotope labeled Avagacestat: a novel gamma secretase inhibitor for the treatment of Alzheimer's disease.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2014, v. 57, n. 10, p. 600, doi. 10.1002/jlcr.3224

By:

Burrell, Richard C.;
Easter, John A.;
Cassidy, Michael P.;
Gillman, Kevin W.;
Olson, Richard E.;
Bonacorsi, Samuel J.

Publication type:

Article

Statistical medium optimization for the production of collagenolytic protease by Pseudomonas sp. SUK using response surface methodology.

Published in:

Microbiology (00262617), 2015, v. 84, n. 4, p. 520, doi. 10.1134/S0026261715040037

By:

Bhagwat, Prashant;
Jhample, Sowmya;
Dandge, Padma

Publication type:

Article

Structural and biochemical analysis of a thermostable membrane-bound stomatin-specific protease.

Published in:

Journal of Synchrotron Radiation, 2013, v. 20, n. 6, p. 933, doi. 10.1107/S0909049513021328

By:

Yokoyama, Hideshi;
Kobayashi, Daisuke;
Takizawa, Naoto;
Fujii, Satoshi;
Matsui, Ikuo

Publication type:

Article