Works matching DE "PHOSPHATASE inhibitors"
Results: 180
LB-100 Enhances Drugs Efficacy Through Inhibition of P-Glycoprotein Expression in Multidrug-Resistant Glioblastoma and Non-Small Cell Lung Carcinoma Cellular Models.
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- Pharmaceutics, 2025, v. 17, n. 2, p. 189, doi. 10.3390/pharmaceutics17020189
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- Article
Improved immunohistochemical detection of phosphorylated mitogen-activated protein kinases in the injured rat optic nerve head.
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- Histochemistry & Cell Biology, 2019, v. 151, n. 5, p. 435, doi. 10.1007/s00418-019-01771-x
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- Article
Off-target effects of protein tyrosine phosphatase inhibitors on oncostatin M-treated human epidermal keratinocytes: the phosphatase targeting STAT1 remains unknown.
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- PeerJ, 2020, p. 1, doi. 10.7717/peerj.9504
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- Article
Synthesis, kinetic studies and in-silico investigations of novel quinolinyl-iminothiazolines as alkaline phosphatase inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2163394
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- Article
Design, synthesis and biological evaluation of novel triazoloquinazolinone and imidazoquinazolinone derivatives as allosteric inhibitors of SHP2 phosphatase.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1495, doi. 10.1080/14756366.2022.2078968
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- Article
Inhibition mechanism of naphthylphenylamine derivatives acting on the CDC25B dual phosphatase and analysis of the molecular processes involved in the high cytotoxicity exerted by one selected derivative in melanoma cells.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1866, doi. 10.1080/14756366.2020.1819257
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- Article
Identification of flavonolignans from Silybum marianum seeds as allosteric protein tyrosine phosphatase 1B inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1283, doi. 10.1080/14756366.2018.1497020
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- Article
Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 25, doi. 10.1080/14756366.2016.1201480
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- Article
Screening of indeno[1,2- b ]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 25, doi. 10.1080/14756366.2016.1201480
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- Article
Protein tyrosine phosphatase 1B inhibitors isolated from Artemisia roxburghiana.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 4, p. 563, doi. 10.3109/14756366.2015.1047358
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- Article
Development of Specific Inhibitors for Oncogenic Phosphatase PPM1D by Using Ion-Responsive DNA Aptamer Library.
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- Catalysts (2073-4344), 2020, v. 10, n. 10, p. 1153, doi. 10.3390/catal10101153
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- Article
Role of Protein Tyrosine Phosphatase 1B Inhibitor in Early Brain Injury of Subarachnoid Hemorrhage in Mice.
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- Brain Sciences (2076-3425), 2023, v. 13, n. 5, p. 816, doi. 10.3390/brainsci13050816
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- Article
Neuronal-Specific Inhibition of Endoplasmic Reticulum Mg2+/Ca2+ ATPase Ca2+ Uptake in a Mixed Primary Hippocampal Culture Model of Status Epilepticus.
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- Brain Sciences (2076-3425), 2020, v. 10, n. 7, p. 438, doi. 10.3390/brainsci10070438
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- Article
Attenuation of STAT3 Signaling Cascade by Daidzin Can Enhance the Apoptotic Potential of Bortezomib against Multiple Myeloma.
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- Biomolecules (2218-273X), 2020, v. 10, n. 1, p. 1, doi. 10.3390/biom10010023
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- Article
Infection by the Protozoan Parasite Toxoplasma gondii Inhibits Host MNK1/2-eIF4E Axis to Promote Its Survival.
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- Frontiers in Cellular & Infection Microbiology, 2020, v. 10, p. N.PAG, doi. 10.3389/fcimb.2020.00488
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- Article
Analysis of Phosphatase Activity in a Droplet-Based Microfluidic Chip.
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- Biosensors (2079-6374), 2022, v. 12, n. 9, p. 740, doi. 10.3390/bios12090740
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- Article
Optimalisation of the Activation Medium and Effect of Inhibiting Activities of Acid Phosphatase, Lactate Dehydrogenase and β-N-Acetylglucosaminidase on the Fertilisation Success of Eurasian Perch (Perca fluviatilis L.).
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- Animals (2076-2615), 2022, v. 12, n. 3, p. 307, doi. 10.3390/ani12030307
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- Article
In silico identification and analysis of potential inhibitors for acid phosphatase, HppA from Helicobacter pylori.
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- Journal of Molecular Recognition, 2023, v. 36, n. 9, p. 1, doi. 10.1002/jmr.3049
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- Article
Differentiated proteome pattern of genetic absence epilepsy rats treated with ketogenic diet.
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- Anatomy: International Journal of Experimental & Clinical Anatomy, 2022, v. 16, p. 243, doi. 10.2399/ana.22.003s
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- Article
Inhibition of PI3K/p70 S6K and p38 MAPK cascades increases osteoblastic differentiation induced by BMP-2.
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- FEBS Letters, 2002, v. 510, n. 1-2, p. 99, doi. 10.1016/S0014-5793(01)03236-7
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- Article
Protein Tyrosine Phosphatase α in the Dorsomedial Striatum Promotes Excessive Ethanol-Drinking Behaviors.
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- Journal of Neuroscience, 2013, v. 33, n. 36, p. 14369, doi. 10.1523/JNEUROSCI.1954-13.2013
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- Article
Cytoplasmic SET induces tau hyperphosphorylation through a decrease of methylated phosphatase 2A.
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- BMC Neuroscience, 2014, v. 15, n. 1, p. 1, doi. 10.1186/1471-2202-15-82
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- Article
Identification of inhibitors that target dual-specificity phosphatase 5 provide new insights into the binding requirements for the two phosphate pockets.
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- BMC Biochemistry, 2015, v. 16, n. 1, p. 1, doi. 10.1186/s12858-015-0048-3
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- Article
MAP4K4 expression in cardiomyocytes: multiple isoforms, multiple phosphorylations and interactions with striatins.
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- Biochemical Journal, 2021, v. 478, n. 11, p. 2121, doi. 10.1042/BCJ20210003
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- Article
Cancerous inhibitor of protein phosphatase 2A (CIP2A) modifies energy metabolism via 5' AMP-activated protein kinase signalling in malignant cells.
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- Biochemical Journal, 2019, v. 476, n. 15, p. 2255, doi. 10.1042/BCJ20190121
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- Article
Some Plant Enzymes Are Highly Sensitive to Inhibition by Zinc Ions.
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- Russian Journal of Plant Physiology, 2019, v. 66, n. 4, p. 591, doi. 10.1134/S1021443719040198
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- Article
The Role of Hypoxia on the Trimethylation of H3K27 in Podocytes.
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- Biomedicines, 2023, v. 11, n. 9, p. 2475, doi. 10.3390/biomedicines11092475
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- Article
A Plasmodium falciparum protein tyrosine phosphatase inhibitor identified from the ChEMBL‐NTD database blocks parasite growth.
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- FEBS Open Bio, 2021, v. 11, n. 7, p. 1921, doi. 10.1002/2211-5463.13171
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- Article
Protein Tyrosine Phosphatase 1B Inhibitors from the Root Bark of Pseudolarix amabilis (Nelson) Rehd. (Pinaceae).
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- Records of Natural Products, 2019, v. 13, n. 6, p. 475, doi. 10.25135/rnp.125.18.12.1132
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- Article
Novel indolotacrine hybrids as acetylcholinesterase inhibitors: design, synthesis, biological evaluation, and molecular docking studies.
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- Journal of the Iranian Chemical Society, 2023, v. 20, n. 5, p. 1049, doi. 10.1007/s13738-022-02726-1
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- Article
A freeze-and-thaw-induced fragment of the microtubule-associated protein tau in rat brain extracts: implications for the biochemical assessment of neurotoxicity.
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- Bioscience Reports, 2021, v. 41, n. 3, p. 1, doi. 10.1042/BSR20203980
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- Article
Partial endothelial-to-mesenchymal transition mediated by HIF-induced CD45 in neointima formation upon carotid artery ligation.
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- Cardiovascular Research, 2023, v. 119, n. 7, p. 1606, doi. 10.1093/cvr/cvac190
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- Article
Novel fluorochromes label tonoplast in living plant cells and reveal changes in vacuolar organization after treatment with protein phosphatase inhibitors.
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- Protoplasma, 2018, v. 255, n. 3, p. 829, doi. 10.1007/s00709-017-1190-0
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- Article
Molecular basis for the selective and ABA-independent inhibition of PP2CA by PYL13.
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- Cell Research, 2013, v. 23, n. 12, p. 1369, doi. 10.1038/cr.2013.143
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- Article
A Kinetic Process to Determine the Interaction Type Between Two Compounds, One of Which Is a Reaction Product, Using Alkaline Phosphatase Inhibition as a Case Study.
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- Applied Biochemistry & Biotechnology, 2020, v. 191, n. 2, p. 657, doi. 10.1007/s12010-019-03213-9
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- Article
Protein tyrosine phosphatase 1B inhibitors from a marine-derived fungal strain aspergillus sp. SF-5929.
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- Natural Product Research, 2020, v. 34, n. 5, p. 675, doi. 10.1080/14786419.2018.1499629
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- Article
Exploration of newly synthesized azo-thiohydantoins as the potential alkaline phosphatase inhibitors via advanced biochemical characterization and molecular modeling approaches.
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- BMC Chemistry, 2024, v. 18, n. 1, p. 1, doi. 10.1186/s13065-024-01149-8
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- Article
[1, 8]-Naphthyridine derivatives as dual inhibitor of alkaline phosphatase and carbonic anhydrase.
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- BMC Chemistry, 2023, v. 17, n. 1, p. 1, doi. 10.1186/s13065-023-01052-8
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- Article
In situ visualization of opioid and cannabinoid drug effects using phosphosite-specific GPCR antibodies.
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- Communications Biology, 2023, v. 6, n. 1, p. 1, doi. 10.1038/s42003-023-04786-2
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- Article
Constitutive Cell Proliferation Regulating Inhibitor of Protein Phosphatase 2A (CIP2A) Mediates Drug Resistance to Erlotinib in an EGFR Activating Mutated NSCLC Cell Line.
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- Cells (2073-4409), 2021, v. 10, n. 4, p. 716, doi. 10.3390/cells10040716
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- Article
Zoledronic acid in combination with serine/threonine phosphatase inhibitors induces enhanced cytotoxicity and apoptosis in hormone-refractory prostate cancer cell lines by decreasing the activities of PP1 and PP2A.
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- BJU International, 2012, v. 110, n. 11c, p. E1147, doi. 10.1111/j.1464-410X.2012.11392.x
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- Article
Cracking the ANP32 whips: Important functions, unequal requirement, and hints at disease implications.
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- BioEssays, 2014, v. 36, n. 11, p. 1062, doi. 10.1002/bies.201400058
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- Article
Stabilities and Biological Activities of Vanadium Drugs: What is the Nature of the Active Species?
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- Chemistry - An Asian Journal, 2017, v. 12, n. 14, p. 1692, doi. 10.1002/asia.201700463
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- Article
The role of phosphorylation in the elasticity of the tethers that connect telomeres of separating anaphase chromosomes.
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- Nucleus (1949-1034), 2020, v. 11, n. 1, p. 19, doi. 10.1080/19491034.2019.1710329
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- Article
The induction of HAD-like phosphatases by multiple signaling pathways confers resistance to the metabolic inhibitor 2-deoxyglucose.
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- Science Signaling, 2019, v. 12, n. 597, p. 1, doi. 10.1126/scisignal.aaw8000
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- Article
Design and rationale of the ATHENA study--A 12-month, multicentre, prospective study evaluating the outcomes of a de novo everolimus-based regimen in combination with reduced cyclosporine or tacrolimus versus a standard regimen in kidney transplant patients: study protocol for a randomised controlled trial.
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- 2016
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- Publication type:
- journal article
In Vitro and In Vivo Pharmacological Profiles of DS‐1211, a Novel Potent, Selective, and Orally Bioavailable Tissue‐Nonspecific Alkaline Phosphatase Inhibitor.
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- Journal of Bone & Mineral Research, 2022, v. 37, n. 10, p. 2033, doi. 10.1002/jbmr.4680
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- Article
The in vivo disposition of subcutaneous injected <sup>14</sup>C-razuprotafib (<sup>14</sup>C-AKB-9778), a sulphamic acid phosphatase inhibitor, in nonclinical species and human.
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- Xenobiotica, 2021, v. 51, n. 10, p. 1132, doi. 10.1080/00498254.2021.1972358
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- Article
Oxidative metabolism of razuprotafib (AKB-9778), a sulfamic acid phosphatase inhibitor, in human microsomes and recombinant human CYP2C8 enzyme.
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- Xenobiotica, 2021, v. 51, n. 10, p. 1110, doi. 10.1080/00498254.2021.1969482
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- Article
A Novel Phosphatase Inhibitor May Be a STEP Toward Ameliorating Cognitive Dysfunction.
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- PLoS Biology, 2014, v. 12, n. 8, p. 1, doi. 10.1371/journal.pbio.1001924
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- Article