Works matching DE "PHOSPHATASE inhibitors"

Results: 183

A Novel Phosphatase Inhibitor May Be a STEP Toward Ameliorating Cognitive Dysfunction.

Published in:

PLoS Biology, 2014, v. 12, n. 8, p. 1, doi. 10.1371/journal.pbio.1001924

By:

Robinson, Richard

Publication type:

Article

A Reappraisal of the Utility of L-012 to Measure Superoxide from Biologically Relevant Sources.

Published in:

Antioxidants, 2023, v. 12, n. 9, p. 1689, doi. 10.3390/antiox12091689

By:

Haigh, Stephen;
Brown, Zach L.;
Shivers, Mitch A.;
Sellers, Hunter G.;
West, Madison A.;
Barman, Scott A.;
Stepp, David W.;
Csanyi, Gabor;
Fulton, David J. R.

Publication type:

Article

Effect of sodium stibogluconate in recruiting and awakening immune cells in the pleural fluid of pancreatic cancer: preparation for immunotherapy.

Published in:

Frontiers in Immunology, 2024, p. 1, doi. 10.3389/fimmu.2023.1315468

By:

Baofa Yu;
Peng Jing;
Feng Gao;
Peicheng Zhang;
Guoqin Zheng;
Xiaomin Zhang

Publication type:

Article

Inhibition of Trypanosoma evansi Protein-Tyrosine Phosphatase by Myristic Acid Analogues Isolated from Khaya senegalensis and Tamarindus indica.

Published in:

Journal of Experimental Pharmacology, 2019, v. 11, p. 135, doi. 10.2147/JEP.S226632

By:

Dingwoke, Emeka John;
Adamude, Fatima Amin;
Chukwuocha, Chimee Ethel;
Ambi, Ahmed Adamu;
Nwobodo, Nwobodo Ndubuisi;
Sallau, Abdullahi Balarabe;
Nzelibe, Humphrey Chukwuemeka

Publication type:

Article

Differentiated proteome pattern of genetic absence epilepsy rats treated with ketogenic diet.

Published in:

Anatomy: International Journal of Experimental & Clinical Anatomy, 2022, v. 16, p. 243, doi. 10.2399/ana.22.003s

By:

Günel, Aslıhan;
Açıkgöz, Nazlı Başak;
Toplu, Aylin;
Güler, Ülkü;
Salih, Bekir;
Türkdoğan, Dilşad;
Onat, Filiz

Publication type:

Article

Nicotinamide mononucleotide attenuates glucocorticoid-induced osteogenic inhibition by regulating the SIRT1/PGC-1α signaling pathway.

Published in:

Molecular Medicine Reports, 2020, v. 22, n. 1, p. 145, doi. 10.3892/mmr.2020.11116

By:

Huang, Rui-Xiong;
Tao, Jun

Publication type:

Article

Fructose-1,6-bisphosphatase-1 decrease may promote carcinogenesis and chemoresistance in cervical cancer.

Published in:

Molecular Medicine Reports, 2017, v. 16, n. 6, p. 8563, doi. 10.3892/mmr.2017.7665

By:

HAORAN LI;
MENGJIAO LI;
YANGYANG PANG;
FEI LIU;
DONG SHENG;
XI CHENG

Publication type:

Article

MicroRNA‑198 contributes to lupus nephritis progression by inhibition of phosphatase and tensin homology deleted on chromosome ten expression.

Published in:

Molecular Medicine Reports, 2017, v. 16, n. 5, p. 7813, doi. 10.3892/mmr.2017.7527

By:

DANYU CUI;
DINGJI ZHU;
HAO REN;
JINGLI LIN;
WEINAN LAI;
QIN HUANG;
JINJUN ZHAO;
MIN YANG

Publication type:

Article

Clinical significance of Wip1 overexpression and its association with the p38MAPK/p53/p16 pathway in NSCLC.

Published in:

Molecular Medicine Reports, 2017, v. 15, n. 2, p. 719, doi. 10.3892/mmr.2016.6032

By:

Shize Yang;
Siyuan Dong;
Xiaohan Qu;
Xinwen Zhong;
Qigang Zhang

Publication type:

Article

Gαq Sensitizes TRPM8 to Inhibition by PI(4,5)P2 Depletion upon Receptor Activation.

Published in:

Journal of Neuroscience, 2019, v. 39, n. 31, p. 6067, doi. 10.1523/JNEUROSCI.2304-18.2019

By:

Luyu Liu;
Yevgen Yudin;
Nagwekar, Janhavi;
Chifei Kang;
Shirokova, Natalia;
Rohacs, Tibor

Publication type:

Article

Phosphatase inhibition prevents the activity-dependent trafficking of GABAA receptors during status epilepticus in the young animal.

Published in:

Epilepsia (Series 4), 2015, v. 56, n. 9, p. 1355, doi. 10.1111/epi.13098

By:

Joshi, Suchitra;
Rajasekaran, Karthik;
Hawk, Kyle M.;
Brar, Jasmit;
Ross, Brittany M.;
Tran, Christine A.;
Chester, Stephen J.;
Goodkin, Howard P.

Publication type:

Article

Protein tyrosine phosphatase 1B inhibitors from a marine-derived fungal strain aspergillus sp. SF-5929.

Published in:

Natural Product Research, 2020, v. 34, n. 5, p. 675, doi. 10.1080/14786419.2018.1499629

By:

Kim, Dong-Cheol;
Minh Ha, Tran;
Sohn, Jae Hak;
Yim, Joung Han;
Oh, Hyuncheol

Publication type:

Article

Improved immunohistochemical detection of phosphorylated mitogen-activated protein kinases in the injured rat optic nerve head.

Published in:

Histochemistry & Cell Biology, 2019, v. 151, n. 5, p. 435, doi. 10.1007/s00418-019-01771-x

By:

Mammone, Teresa;
Chidlow, Glyn;
Casson, Robert J.;
Wood, John P. M.

Publication type:

Article

Effects of Midazolam on Antioxidant Levels, Biochemical and Metabolic Parameters in Eurygaster integriceps Puton (Hemiptera: Scutelleridae) Eggs Parasitized by Trissolcus semistriatus Nees (Hymenoptera: Scelionidae).

Published in:

Bulletin of Environmental Contamination & Toxicology, 2023, v. 110, n. 1, p. 1, doi. 10.1007/s00128-022-03648-7

By:

Sugeçti, Serkan;
Kepekçi, Ali Bestemi;
Büyükgüzel, Kemal

Publication type:

Article

Pyrin–PSTPIP1 colocalises at the leading edge during cell migration.

Published in:

Cell Biology International, 2015, v. 39, n. 12, p. 1384, doi. 10.1002/cbin.10514

By:

Akkaya‐Ulum, Yeliz Z.;
Balci‐Peynircioglu, Banu;
Purali, Nuhan;
Yilmaz, Engin

Publication type:

Article

Design of an Electrochemical Device for the Detection of Alkaline Phosphatase Inhibitors in Seawater.

Published in:

ChemElectroChem, 2024, v. 11, n. 16, p. 1, doi. 10.1002/celc.202400271

By:

Sáenz‐Espinar, María J.;
Hafed‐Khatiri, Salma;
Salinas‐Torres, David;
Montilla, Francisco;
Huerta, Francisco

Publication type:

Article

The Role of Hypoxia on the Trimethylation of H3K27 in Podocytes.

Published in:

Biomedicines, 2023, v. 11, n. 9, p. 2475, doi. 10.3390/biomedicines11092475

By:

Barth, Johanna;
Loeffler, Ivonne;
Bondeva, Tzvetanka;
Liebisch, Marita;
Wolf, Gunter

Publication type:

Article

Determination of rate of inorganic phosphorus consumption in natural waters using alkaline phosphatase inhibitors.

Published in:

Russian Journal of General Chemistry, 2016, v. 86, n. 13, p. 3015, doi. 10.1134/S1070363216130156

By:

Ryzhakov, A.;
Stepanova, I.

Publication type:

Article

Constitutive Cell Proliferation Regulating Inhibitor of Protein Phosphatase 2A (CIP2A) Mediates Drug Resistance to Erlotinib in an EGFR Activating Mutated NSCLC Cell Line.

Published in:

Cells (2073-4409), 2021, v. 10, n. 4, p. 716, doi. 10.3390/cells10040716

By:

Saafan, Hisham;
Alahdab, Ahmad;
Michelet, Robin;
Gohlke, Linus;
Ziemann, Janine;
Holdenrieder, Stefan;
McLaughlin, Katie-May;
Wass, Mark N.;
Cinatl Jr., Jindrich;
Michaelis, Martin;
Kloft, Charlotte;
Ritter, Christoph A;
Gray, Steven G.

Publication type:

Article

Development of Specific Inhibitors for Oncogenic Phosphatase PPM1D by Using Ion-Responsive DNA Aptamer Library.

Published in:

Catalysts (2073-4344), 2020, v. 10, n. 10, p. 1153, doi. 10.3390/catal10101153

By:

Kaneko, Atsushi;
Watari, Miyuu;
Mizunuma, Masataka;
Saito, Hikaru;
Furukawa, Kazuhiro;
Chuman, Yoshiro

Publication type:

Article

Influence of acid phosphatase and arylsulfatase inhibitor additions on fertility rate of Siberian sturgeon ( Acipenser baerii Brandt, 1869).

Published in:

Journal of Applied Ichthyology, 2015, v. 31, p. 154, doi. 10.1111/jai.12729

By:

Sarosiek, B.;
Dryl, K.;
Judycka, S.;
Szczepkowski, M.;
Kowalski, R. K.

Publication type:

Article

LB-100 Enhances Drugs Efficacy Through Inhibition of P-Glycoprotein Expression in Multidrug-Resistant Glioblastoma and Non-Small Cell Lung Carcinoma Cellular Models.

Published in:

Pharmaceutics, 2025, v. 17, n. 2, p. 189, doi. 10.3390/pharmaceutics17020189

By:

Podolski-Renić, Ana;
Chigriai, Margarita;
Jovanović Stojanov, Sofija;
Grozdanić, Marija;
Lupšić, Ema;
Nikolić, Igor;
Dragoj, Miodrag;
Dinić, Jelena;
Pešić, Milica

Publication type:

Article

Facile Synthesis of N -(4-Bromo-3-methylphenyl)pyrazine-2-carboxamide Derivatives, Their Antibacterial Activities against Clinically Isolated XDR S. Typhi , Alkaline Phosphatase Inhibitor Activities, and Docking Studies.

Published in:

Pharmaceuticals (14248247), 2024, v. 17, n. 9, p. 1241, doi. 10.3390/ph17091241

By:

Khan, Abdul Hannan;
Bilal, Muhammad;
Mahmood, Abid;
Rasool, Nasir;
Qamar, Muhammad Usman;
Imran, Muhammad;
Toma, Sebastian Ionut;
Andreescu, Oana

Publication type:

Article

CX08005, a Protein Tyrosine Phosphatase 1B Inhibitor, Attenuated Hepatic Lipid Accumulation and Microcirculation Dysfunction Associated with Nonalcoholic Fatty Liver Disease.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 1, p. 106, doi. 10.3390/ph16010106

By:

Li, Jiang;
Zhang, Xiaolin;
Tian, Jinying;
Li, Juan;
Li, Xuechen;
Wu, Song;
Liu, Yuying;
Han, Jingyan;
Ye, Fei

Publication type:

Article

The Potential Use of Ebselen in Treatment-Resistant Depression.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 4, p. N.PAG, doi. 10.3390/ph15040485

By:

Ramli, Fitri Fareez;
Cowen, Philip J.;
Godlewska, Beata R.

Publication type:

Article

Yy1 regulates Senp1 contributing to AMPA receptor GluR1 expression following neuronal depolarization.

Published in:

Journal of Biomedical Science, 2019, v. 26, p. 1, doi. 10.1186/s12929-019-0582-1

By:

Tao Wu;
Donohoe, Mary E.

Publication type:

Article

The mode of action of the Protein tyrosine phosphatase 1B inhibitor Ertiprotafib.

Published in:

PLoS ONE, 2020, v. 15, n. 10, p. 1, doi. 10.1371/journal.pone.0240044

By:

Kumar, Ganesan Senthil;
Page, Rebecca;
Peti, Wolfgang

Publication type:

Article

Novel indolotacrine hybrids as acetylcholinesterase inhibitors: design, synthesis, biological evaluation, and molecular docking studies.

Published in:

Journal of the Iranian Chemical Society, 2023, v. 20, n. 5, p. 1049, doi. 10.1007/s13738-022-02726-1

By:

Babaee, Saeed;
Zolfigol, Mohammad Ali;
Chehardoli, Gholamabbas;
Faramarzi, Mohammad Ali;
Mojtabavi, Somayeh;
Akbarzadeh, Tahmineh;
Hariri, Roshanak;
Rastegari, Arezoo;
Homayouni Moghadam, Farshad;
Mahdavi, Mohammad;
Najafi, Zahra

Publication type:

Article

A freeze-and-thaw-induced fragment of the microtubule-associated protein tau in rat brain extracts: implications for the biochemical assessment of neurotoxicity.

Published in:

Bioscience Reports, 2021, v. 41, n. 3, p. 1, doi. 10.1042/BSR20203980

By:

Vasconcelos, Israel C.;
Campos, Raquel M.;
Schwaemmle, Hanna K.;
Masson, Ana P.;
Ferrari, Gustavo D.;
Alberici, Luciane C.;
Faça, Vitor M.;
Garcia-Cairasco, Norberto;
Sebollela, Adriano

Publication type:

Article

The in vivo disposition of subcutaneous injected 14C-razuprotafib (14C-AKB-9778), a sulphamic acid phosphatase inhibitor, in nonclinical species and human.

Published in:

Xenobiotica, 2021, v. 51, n. 10, p. 1132, doi. 10.1080/00498254.2021.1972358

By:

Soldo, Brandi Lynn;
Camilleri, Patrick;
Buch, Akshay;
Janusz, John

Publication type:

Article

Oxidative metabolism of razuprotafib (AKB-9778), a sulfamic acid phosphatase inhibitor, in human microsomes and recombinant human CYP2C8 enzyme.

Published in:

Xenobiotica, 2021, v. 51, n. 10, p. 1110, doi. 10.1080/00498254.2021.1969482

By:

Camilleri, Patrick;
Soldo, Brandi;
Buch, Akshay;
Janusz, John

Publication type:

Article

Relationship between uterine smooth muscular CPI-17-signal pathway-mediated Ca2+ sensitivity changes and uterine atony-induced postpartum haemorrhage.

Published in:

2019

By:

Liao, Qiuping;
Yan, Jianying;
Luo, Jinying;
Han, Qing;
Zhang, Qinjian;
Chen, Rongxin;
Zhou, Zhimei

Publication type:

journal article

Synthesis, kinetic studies and in-silico investigations of novel quinolinyl-iminothiazolines as alkaline phosphatase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2163394

By:

Mustafa, Muhammad Naeem;
Channar, Pervaiz Ali;
Sarfraz, Muhammad;
Saeed, Aamer;
Ejaz, Syeda Abida;
Aziz, Mubashir;
Alasmary, Fatmah Ali;
Alsoqair, Hanadi Yaqob;
Raza, Hussain;
Kim, Song Ja;
Hamad, Asad

Publication type:

Article

Design, synthesis and biological evaluation of novel triazoloquinazolinone and imidazoquinazolinone derivatives as allosteric inhibitors of SHP2 phosphatase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1495, doi. 10.1080/14756366.2022.2078968

By:

Wenjun Ye;
Ye Liu;
Qian Ren;
Tianhui Liao;
Yumei Chen;
Dongmei Chen;
Sisi Wang;
Lihong Yao;
Yihe Jia;
Chunshen Zhao;
Zhixu Zhou

Publication type:

Article

Inhibition mechanism of naphthylphenylamine derivatives acting on the CDC25B dual phosphatase and analysis of the molecular processes involved in the high cytotoxicity exerted by one selected derivative in melanoma cells.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1866, doi. 10.1080/14756366.2020.1819257

By:

Aliotta, Federica;
Nasso, Rosarita;
Rullo, Rosario;
Arcucci, Alessandro;
Avagliano, Angelica;
Simonetti, Martina;
Sanità, Gennaro;
Masullo, Mariorosario;
Lavecchia, Antonio;
Ruocco, Maria Rosaria;
Vendittis, Emmanuele De

Publication type:

Article

Identification of flavonolignans from Silybum marianum seeds as allosteric protein tyrosine phosphatase 1B inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1283, doi. 10.1080/14756366.2018.1497020

By:

Qin, Ningbo;
Sasaki, Tatsunori;
Li, Wei;
Wang, Jian;
Zhang, Xiangyu;
Li, Dahong;
Li, Zhanlin;
Cheng, Maosheng;
Hua, Huiming;
Koike, Kazuo

Publication type:

Article

Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 25, doi. 10.1080/14756366.2016.1201480

By:

Alchab, Faten;
Sibille, Estelle;
Ettouati, Laurent;
Bana, Emilie;
Bouaziz, Zouhair;
Mularoni, Angélique;
Monniot, Elodie;
Bagrel, Denyse;
Jose, Joachim;
Le Borgne, Marc;
Chaimbault, Patrick

Publication type:

Article

Screening of indeno[1,2- b ]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 25, doi. 10.1080/14756366.2016.1201480

By:

Alchab, Faten;
Sibille, Estelle;
Ettouati, Laurent;
Bana, Emilie;
Bouaziz, Zouhair;
Mularoni, Angélique;
Monniot, Elodie;
Bagrel, Denyse;
Jose, Joachim;
Le Borgne, Marc;
Chaimbault, Patrick

Publication type:

Article

Protein tyrosine phosphatase 1B inhibitors isolated from Artemisia roxburghiana.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 4, p. 563, doi. 10.3109/14756366.2015.1047358

By:

Shah, Muhammad Raza;
Ishtiaq;
Hizbullah, Syed Muhammad;
Habtemariam, Solomon;
Zarrelli, Armando;
Muhammad, Akhtar;
Collina, Simona;
Khan, Inamulllah

Publication type:

Article

The Anti-Fungal Activity of Nitropropenyl Benzodioxole (NPBD), a Redox-Thiol Oxidant and Tyrosine Phosphatase Inhibitor.

Published in:

Antibiotics (2079-6382), 2022, v. 11, n. 9, p. 1188, doi. 10.3390/antibiotics11091188

By:

Nicoletti, Gina;
White, Kylie

Publication type:

Article

Broad Spectrum Anti-Bacterial Activity of a Recombinant Phosphatase-Like Protein (rPLP), Isolated from the Shrimp Penaeus monodon.

Published in:

Israeli Journal of Aquaculture-Bamidgeh, 2015, v. 67, p. 1, doi. 10.46989/001c.20721

By:

Banerjee, Debashis;
Maiti, Biswajit;
Girisha, S. K.;
Venugopal, M. N.;
Karunasagar, Indrani

Publication type:

Article

Imide cantharidin derivatives: Synthesis and HBV-DNA inhibitory properties.

Published in:

ScienceAsia, 2023, v. 49, n. 1, p. 38, doi. 10.2306/scienceasia1513-1874.2022.117

By:

Chun Bin Tan;
Ya Jing Xing;
Xing Fang Qiao;
Bao Min Fan;
Xiao-Ling Liu;
Yao Bo Zeng

Publication type:

Article

Small molecule. Big biology. Dual phosphatase inhibitor enters the immunotherapy fray.

Published in:

Immunology & Cell Biology, 2024, v. 102, n. 1, p. 8, doi. 10.1111/imcb.12711

By:

Wilson, Nicholas S;
Huntington, Nicholas D

Publication type:

Article

Natural regulatory T cells are resistant to calcium release-activated calcium (CRAC/ORAI) channel inhibition.

Published in:

International Immunology, 2013, v. 25, n. 9, p. 497, doi. 10.1093/intimm/dxt013

By:

Jin, Shu;
Chin, Jayne;
Kitson, Christopher;
Woods, John;
Majmudar, Rupal;
Carvajal, Valerie;
Allard, John;
DeMartino, Julie;
Narula, Satwant;
Thomas-Karyat, Dori A.

Publication type:

Article

Inhibition of Phosphatase Activity Follows Decline in Sulfatase Activity and Leads to Transcriptional Effects through Sustained Phosphorylation of Transcription Factor MITF.

Published in:

PLoS ONE, 2016, v. 11, n. 4, p. 1, doi. 10.1371/journal.pone.0153463

By:

Bhattacharyya, Sumit;
Feferman, Leo;
Tobacman, Joanne K.

Publication type:

Article

Trigonal Bipyramidal or Square Pyramidal Coordination Geometry? Investigating the Most Potent Geometry for Vanadium Phosphatase Inhibitors.

Published in:

European Journal of Inorganic Chemistry, 2014, v. 2014, n. 27, p. 4450, doi. 10.1002/ejic.201402306

By:

Crans, Debbie C.;
Tarlton, Michael L.;
McLauchlan, Craig C.

Publication type:

Article

Partial endothelial-to-mesenchymal transition mediated by HIF-induced CD45 in neointima formation upon carotid artery ligation.

Published in:

Cardiovascular Research, 2023, v. 119, n. 7, p. 1606, doi. 10.1093/cvr/cvac190

By:

Yamashiro, Yoshito;
Ramirez, Karina;
Nagayama, Kazuaki;
Hattori, Naoko;
Liu, Yu-Yu;
Matsunaga, Shinji;
Tomita, Shuhei;
Kubota, Yoshiaki;
Yanagisawa, Hiromi

Publication type:

Article

Phosphatase-1 inhibitor-1 in physiological and pathological β-adrenoceptor signalling.

Published in:

Cardiovascular Research, 2011, v. 91, n. 3, p. 392, doi. 10.1093/cvr/cvr058

By:

Wittköpper, Katrin;
Dobrev, Dobromir;
Eschenhagen, Thomas;
El-Armouche, Ali

Publication type:

Article

Tumor necrosis factor α stimulates expression and secretion of urokinase plasminogen activator in human dental pulp cells.

Published in:

2012

By:

Narita, Takanori;
Muromachi, Koichiro;
Kamio, Naoto;
Nakao, Sumi;
Matsushima, Kiyoshi;
Hashizume, Hideki

Publication type:

journal article

STS1 and STS2 Phosphatase Inhibitor Baicalein Enhances the Expansion of Hematopoietic and Progenitor Stem Cells and Alleviates 5-Fluorouracil-Induced Myelosuppression.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 3, p. 2987, doi. 10.3390/ijms24032987

By:

Li, Na;
Wang, Yanhong;
Wang, Anqing;
Zhang, Jing;
Jia, Chaoran;
Yu, Chunlei;
Song, Zhenbo;
Wang, Shuyue;
Liu, Lei;
Yi, Jingwen;
Bao, Yongli;
Huang, Yanxin;
Sun, Luguo

Publication type:

Article