Works about MICROSOMES
Results: 1145
Characterization of Coumarin-Specific Prenyltransferase Activities in Citrus limon Peel.
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- Bioscience, Biotechnology & Biochemistry, 2012, v. 76, n. 7, p. 1389, doi. 10.1271/bbb.120192
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- Article
The Formation of g = 2.49-Species of Cytochrome P450 in the Rat Liver by PCB126 Oral Administration: Identification of Heme Axial Ligands by EPR Spectroscopy.
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- Bioscience, Biotechnology & Biochemistry, 2006, v. 70, n. 12, p. 2974, doi. 10.1271/bbb.60367
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- Article
Biotransformation of (—)-Menthone by Human Liver Microsomes.
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- Bioscience, Biotechnology & Biochemistry, 2006, v. 70, n. 5, p. 1259, doi. 10.1271/bbb.70.1259
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- Article
Catalytic Reaction of Basiodiomycete Lentinula edodes Cytochrome P450, Le.CYP1 Enzyme Produced in Yeast.
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- Bioscience, Biotechnology & Biochemistry, 2004, v. 68, n. 1, p. 79, doi. 10.1271/bbb.68.79
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- Article
Reaction phenotyping of vinblastine metabolism in dogs.
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- Veterinary & Comparative Oncology, 2016, v. 14, n. 2, p. 161, doi. 10.1111/vco.12084
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- Article
Dasotraline as a selective cytochrome 2B6 inhibitor for reaction phenotyping.
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- Biopharmaceutics & Drug Disposition, 2019, v. 40, n. 9, p. 358, doi. 10.1002/bdd.2207
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- Article
Pharmacokinetic interference of doxorubicin with tolbutamide due to reduced metabolic clearance with increased serum unbound fraction in rats.
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- Biopharmaceutics & Drug Disposition, 2019, v. 40, n. 7, p. 225, doi. 10.1002/bdd.2195
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- Article
In vitro investigation on the impact of the surface-active excipients Cremophor EL, Tween 80 and Solutol HS 15 on the metabolism of midazolam.
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- Biopharmaceutics & Drug Disposition, 2004, v. 25, n. 1, p. 37, doi. 10.1002/bdd.383
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- Article
Isolated Cardiac Ryanodine Receptor Function Varies Between Mammals.
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- Journal of Membrane Biology, 2024, v. 257, n. 1/2, p. 25, doi. 10.1007/s00232-023-00301-0
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- Article
Evaluation of cytochrome P450 activity in vitro, using dermal and hepatic microsomes from four species and two keratinocyte cell lines in culture.
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- Archives of Dermatological Research, 2008, v. 300, n. 1, p. 11, doi. 10.1007/s00403-007-0811-4
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- Article
Effect of pyridine and quinoline N-oxides on microsomal Na,K-ATPase activity.
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- Pharmaceutical Chemistry Journal, 2006, v. 40, n. 7, p. 347, doi. 10.1007/s11094-006-0124-5
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- Article
Comparative 1-Substituted Imidazole Inhibition of Cytochrome P450 Isozyme-Selective Activities in Human and Mouse Hepatic Microsomes.
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- Drug Metabolism Reviews, 2007, v. 39, n. 2/3, p. 309, doi. 10.1080/03602530701498570
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- Article
Ronald W. Estabrook, Ph.D., M.D. (Hon.): Boss, Mentor, Colleague, and Friend.
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- Drug Metabolism Reviews, 2007, v. 39, n. 2/3, p. 271, doi. 10.1080/03602530701498117
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- Article
Relevance of Cytochrome P450s in Plants: Also One of Ron Estabrook's Research Interests.
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- Drug Metabolism Reviews, 2007, v. 39, n. 2/3, p. 273, doi. 10.1080/03602530701468268
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- Article
Application of Chimeric Mice with Humanized Liver for Predictive ADME.
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- Drug Metabolism Reviews, 2007, v. 39, n. 1, p. 145, doi. 10.1080/03602530601021340
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- Article
Organophosphorus Chemicals: Potent Inhibitors of the Human Metabolism of Steroid Hormones and Xenobiotics.
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- Drug Metabolism Reviews, 2006, v. 38, n. 1/2, p. 149, doi. 10.1080/03602530600569984
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- Article
Cytochromes P450—A Family of Proteins and Scientists–Understanding their Relationships.
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- Drug Metabolism Reviews, 2006, v. 38, n. 1/2, p. 209, doi. 10.1080/03602530600570065
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- Article
HUMAN METABOLISM AND METABOLIC INTERACTIONS OF DEPLOYMENT-RELATED CHEMICALS.
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- Drug Metabolism Reviews, 2005, v. 37, n. 1, p. 1, doi. 10.1081/DMR-46955
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- Article
257. ROLE OF POLYPHORPHIC HUMAN CYP2B6 IN CYCLOPHOSPHAMIDE BIOACTIVATION.
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- 2003
- Publication type:
- Abstract
251. CYP3A4 ACTIVITY IN RAT LIVER MICROSOMES USING 7-BENZYLOXYQUINOLINE AND HPLC DETERMINATION.
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- 2003
- Publication type:
- Abstract
241. IN VITRO METABOLISM OF CLOMETHIAZOLE BY HUMAN LIVER MICROSOMES AND HUMAN CYTOCHROME P450 ISOFORMS.
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- 2003
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- Abstract
160. FISH MICROSOMAL CYP450 ACTIVITIES AND ENDOCRINE DISRUPTION SCREENING.
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- 2003
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- Abstract
137. IN VITRO METABOLISM OF CRUDE PETROLEUM FROM "ERIKA" OIL SPILL BY FISH (SOLEA SOLEA) AND MUSSELS (MYTILUS EDULIS) MICROSOMES.
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- 2003
- Publication type:
- Abstract
125. QUANTITATIVE PREDICTION OF DRUG-DRUG INTERACTIONS: A COMPARISON BETWEEN MICROSOMES AND HEPATOCYTES FOR AZOLE-TOLBUTAMIDE INTERACTIONS.
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- 2003
- Publication type:
- Abstract
120. INVESTIGATION OF GLUCURONIDATION OF 5'-DFCR, THE FIRST INTERMEDIARY METABOLITE OF CAPECITABINE, IN MICROSOMES FROM RAT AND HUMAN LIVERS.
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- 2003
- Publication type:
- Abstract
114. REDOX REGULATION OF ACTIVITY OF TWO UGT ISOFORMS, 1A6 AND 2B1, IN TRANSFECTED V79 CELLS AND RAT BRAIN ASTROCYTES.
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- 2003
- Publication type:
- Abstract
113. O-GLUCURONIDATION OF THE PHOSPHODIESTERASE 4 INHIBITOR AWD 12-281 IN HUMAN LIVER MICROSOMES AND RECOMBINANT UDP-GLUCURONOSYLTRANSFERASES.
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- 2003
- Publication type:
- Abstract
112. HETERO-OLIGOMERIC INTERACTION BETWEEN UDP-GLUCURONOSYL-TRANSFERASE (UGT) ISOZYMES IN HEPATIC MICROSOMES.
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- 2003
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- Abstract
110. MIDAZOLAM IS METABOLIZED BY UGT1A4 IN HUMAN HEPATOCYTES AND HEPATIC MICROSOMES.
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- 2003
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- Abstract
108. AS IN HUMANS A GENETIC POLYMORPHISM OF FMO2 EXISTS IN RATS.
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- 2003
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- Abstract
105. CO-EXPRESSION OF CYP AND FMO ISOFORMS BASED ON ENZYMATIC ACTIVITY IN RAT AND IN HUMAN LIVER MICROSOMES.
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- 2003
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- Abstract
59. STEREOSELECTIVITY OF CETIRIZINE METABOLISM.
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- 2003
- Publication type:
- Abstract
411. IN VITRO BIOTRANSFORMATION OF RO3300074-000 IN HUMANS: IDENTIFICATION OF ISOFORMS OF CYTOCHROME P-450 RESPONSIBLE FOR METABOLISM AND INHIBITION KINETICS OF KETOCONAZOLE, MIDAZOLAM, AND ERYTHROMYCIN IN HUMAN HEPATIC MICROSOMES.
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- 2002
- Publication type:
- Abstract
408. OPTIMIZING LCQ DYNAMIC EXCLUSION ANALYSIS FOR HIGHER THROUGHPUT METABOLITE STRUCTURE ELUCIDATION IN DRUG DISCOVERY.
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- 2002
- Publication type:
- Abstract
403. DISCOVERY P450 INHIBITION SCREENING: HOW DOES A 5-IN-1 LC-MS/MS ASSAY COMPARE TO COMMONLY USED FLUOROMETRIC ASSAYS?
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- 2002
- Publication type:
- Abstract
397. METABOLIC CHARACTERIZATION OF A SET OF TWENTY-THREE COMPOUNDS IN LIVER MICROSOMES OBTAINED FROM NUDE AND CD-1 MICE AND FROM WISTAR AND SPRAGUE DAWLEY RATS.
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- 2002
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- Abstract
370. EFFECT OF COMMOM ORGANIC SOLVENTS ON HUMAN UGT ENZYME ACTIVITIES.
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- 2002
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- Abstract
352. INHIBITOR POTENCY OF TWO FUROCOUMARINS TOWARD CYP3A4 ACTIVITY IS SUBSTRATE DEPENDENT IN A WHOLE CELL SYSTEM.
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- 2002
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- Abstract
345. STEREOSELECTIVE METABOLISM OF OXAZOLIDINONE ALPHA-1A ADRENERGIC RECEPTOR ANTAGONISTS BY CYP3A AND RESULTING MECHANISM-BASED ENZYME INHIBITION.
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- 2002
- Publication type:
- Abstract
215. SIMULTANEOUS QUANTITATION OF CYP3A4 AND 3A7 IN HUMAN LIVER MICROSOMES USING DEHYDROEPIANDROSTERONE (DHEA).
- Published in:
- 2002
- Publication type:
- Abstract
210. A COMPARISON OF CYTOCHROME P450 ACTIVITIES IN BACTOSOMES, SUPERSOMES, AND HUMAN LIVER MICROSOMES.
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- 2002
- Publication type:
- Abstract
153. MATRIX INHIBITION METHOD A NEW METHOD FOR SIMULTANEOUS ESTIMATION OF PROTEIN BINDING AND INTRINSIC CLEARANCE.
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- 2002
- Publication type:
- Abstract
143. IN VITRO ASSESSMENT OF METABOLIC STABILITY, PERMEABILITY AND EFFICACY OF TRYPTANTHRINS: A NOVEL CLASS OF PROPHYLACTIC ANTIMALARIAL DRUG CANDIDATES.
- Published in:
- 2002
- Publication type:
- Abstract
137. IN VITRO METABOLISM OF A NEW NEUROPROTECTIVE AGENT KR-31543 IN HUMAN LIVER MICROSOMES.
- Published in:
- 2002
- Publication type:
- Abstract
136. METABOLISM OF A NEW ERECTOGENIC DA-8159 IN HUMAN LIVER MICROSOMES AND CHARACTERIZATION OF CYTOCHROME P450.
- Published in:
- 2002
- Publication type:
- Abstract
131. IDENTIFICATION OF AN OXIDATION METABOLIC PATHWAY OF ITRIGLUMIDE IN HUMAN LIVER MICROSOMES.
- Published in:
- 2002
- Publication type:
- Abstract
130. BIOTRANSFORMATION OF [<sup>14</sup>C]BMS-275183 IN BILE-DUCT CANNULATED (BDC) RATS.
- Published in:
- 2002
- Publication type:
- Abstract
129. METABOLISM OF [<sup>14</sup>C]BMS-275183 IN MOUSE, RAT, DOG, MONKEY AND HUMAN LIVER MICROSOMES.
- Published in:
- 2002
- Publication type:
- Abstract
127. EXPERIMENTAL SET-UP FOR THE COMPARISON OF THE METABOLISM OF XENOBIOTICS IN VIVO AND IN VITRO.
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- 2002
- Publication type:
- Abstract
126. THE METABOLIC PROFILING OF STEREO ISOMERS IN970, IN971 IN RAT, DOG AND HUMAN LIVER MICROSOME.
- Published in:
- 2002
- Publication type:
- Abstract