Works matching DE "GUANIDINE derivatives"


Results: 166
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    A Review of the Biological Activity of Amidrazone Derivatives.

    Published in:
    Pharmaceuticals (14248247), 2022, v. 15, n. 10, p. 1219, doi. 10.3390/ph15101219
    By:
    • Paprocka, Renata;
    • Wiese-Szadkowska, Małgorzata;
    • Kosmalski, Tomasz;
    • Frisch, Daria;
    • Ratajczak, Magdalena;
    • Modzelewska-Banachiewicz, Bożena;
    • Studzińska, Renata
    Publication type:
    Article
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    Synthesis and pharmacological evaluation of guanidinederivatives with potential hypoglycemic activity.

    Published in:
    2014
    By:
    • de Albuquerque Sarmento, Patrícia;
    • Cavalcante-Araújo, Polliane Maria;
    • de Melo, Igor Santana;
    • Barcellos França, Paulo Henrique;
    • de Medeiros, Návylla Candeia;
    • de Oliveira, Tales Lyra;
    • Lins, Thaís Honório;
    • Santos Veríssimo, Regina Célia Sales;
    • de Assis Bastos, Maria Lysete;
    • Nogueira Ribeiro, Êurica Adélia;
    • Sabino-Silva, Robinson;
    • de Araújo-Júnior, João Xavier
    Publication type:
    Abstract
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    A novel synthetic derivative of biaryl guanidine as a potential BACE1 inhibitor, to treat Alzheimer's disease: In-silico, in-vitro and in-vivo evaluation.

    Published in:
    Pakistan Journal of Pharmaceutical Sciences, 2022, v. 35, n. 5, p. 1339, doi. 10.36721/PJPS.2022.35.5.REG.1339-1345.1
    By:
    • Ali, Sayyad;
    • Hassan Bin Asad, Muhammad Hassham;
    • Javed, Muhammad Arslan;
    • Javed, Tariq;
    • Al-Kharaman, Yasser MSA;
    • Latif, Muhammad;
    • Mohsin, Sabeeh;
    • Nawaz, Taufiq;
    • Farid Hasan, Syed Muhammad;
    • Iqbal, Jamshed;
    • Babak, Borhan;
    • Hussain, Izhar
    Publication type:
    Article
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    Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivity.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201403
    By:
    • Allam, Heba Abdelrasheed;
    • Albakry, Mohamed E.;
    • Mahmoud, Walaa R.;
    • Bonardi, Alessandro;
    • Moussa, Shaimaa A.;
    • Mohamady, Samy;
    • Abdel-Aziz, Hatem A.;
    • Supuran, Claudiu T.;
    • Ibrahim, Hany S.
    Publication type:
    Article
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    Guanidine Derivatives of Quinazoline-2,4(1 H ,3 H)-Dione as NHE-1 Inhibitors and Anti-Inflammatory Agents.

    Published in:
    Life (2075-1729), 2022, v. 12, n. 10, p. 1647, doi. 10.3390/life12101647
    By:
    • Spasov, Alexander;
    • Ozerov, Alexander;
    • Kosolapov, Vadim;
    • Gurova, Natalia;
    • Kucheryavenko, Aida;
    • Naumenko, Ludmila;
    • Babkov, Denis;
    • Sirotenko, Viktor;
    • Taran, Alena;
    • Borisov, Alexander;
    • Sokolova, Elena;
    • Klochkov, Vladlen;
    • Merezhkina, Darya;
    • Miroshnikov, Mikhail;
    • Ovsyankina, Nadezhda;
    • Smirnov, Alexey;
    • Velikorodnaya, Yulia
    Publication type:
    Article
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    Implications of Guanidine Substitution on Copper Complexes as Entatic-State Models.

    Published in:
    European Journal of Inorganic Chemistry, 2016, v. 2016, n. 29, p. 4731, doi. 10.1002/ejic.201600655
    By:
    • Hoffmann, Alexander;
    • Stanek, Julia;
    • Dicke, Benjamin;
    • Peters, Laurens;
    • Grimm‐Lebsanft, Benjamin;
    • Wetzel, Alina;
    • Jesser, Anton;
    • Bauer, Matthias;
    • Gnida, Manuel;
    • Meyer‐Klaucke, Wolfram;
    • Rübhausen, Michael;
    • Herres‐Pawlis, Sonja
    Publication type:
    Article
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