Works about DRUG derivatives

Results: 388

Synthesis of Salidroside Derivatives at C4 Position of Benzene Ring and Its Effect on Hep3B Cell Viability.

Published in:

Chemical Biology & Drug Design, 2025, v. 105, n. 6, p. 1, doi. 10.1111/cbdd.70131

By:

Wang, Juntao;
Yang, Zhaoqi;
Feng, Zili;
Zhao, Hongbo;
Duan, Congxue;
Sheng, Yunzhi;
Du, Pengfei;
Chen, Wang;
Chen, Qingjuan;
Xiao, Dong

Publication type:

Article

Investigation on the chiral recognition mechanism between verteporfin and cholate salts by capillary electrophoresis.

Published in:

Journal of Separation Science, 2020, v. 43, n. 14, p. 2905, doi. 10.1002/jssc.202000026

By:

Xu, Zhongqi;
Xue, Tianfeng;
He, Tao

Publication type:

Article

Colchicine derivative as a potential anti-glioma compound.

Published in:

Journal of Neuro-Oncology, 2015, v. 124, n. 3, p. 403, doi. 10.1007/s11060-015-1874-2

By:

Fang, Kuan-Min;
Liu, Jun-Jen;
Li, Chun-Chun;
Cheng, Chih-Chi;
Hsieh, Yun-Ti;
Chai, Kit;
Lien, Yu-An;
Tzeng, Shun-Fen

Publication type:

Article

Piperazine derivatives with potent drug moiety as efficient acetylcholinesterase, butyrylcholinesterase, and glutathione S‐transferase inhibitors.

Published in:

2023

By:

Karaytuğ, Mahmut Onur;
Balcı, Neslihan;
Türkan, Fikret;
Gürbüz, Mahmut;
Demirkol, Mehmet Emin;
Namlı, Zeynep;
Tamam, Lut;
Gülçin, İlhami

Publication type:

Editorial

Synthesis, molecular docking, and cytotoxicity of quinazolinone and dihydroquinazolinone derivatives as cytotoxic agents.

Published in:

BMC Chemistry, 2022, v. 16, n. 1, p. 1, doi. 10.1186/s13065-022-00825-x

By:

Taayoshi, Fahimeh;
Iraji, Aida;
Moazzam, Ali;
Soleimani, Meysam;
Asadi, Mehdi;
Pedrood, Keyvan;
Akbari, Mosayeb;
Salehabadi, Hafezeh;
Larijani, Bagher;
Adibpour, Neda;
Mahdavi, Mohammad

Publication type:

Article

Proteolysis targeting chimera (PROTAC)-driven antibody internalization of oncogenic cell surface receptors.

Published in:

Communications Biology, 2024, v. 7, n. 1, p. 1, doi. 10.1038/s42003-024-07439-0

By:

Tolosa, Ezequiel J.;
Yang, Lin;
Ayers-Ringler, Jennifer;
Suzuki, Shinichiro;
Mallareddy, Jayapal Reddy;
Schaefer-Klein, Janet;
Borad, Mitesh;
Kosari, Farhad;
Natarajan, Amarnath;
Mansfield, Aaron S.

Publication type:

Article

The Presence of New Psychoactive Substances in a Tor Network Marketplace Environment.

Published in:

2016

By:

Dolliver, Diana S.;
Kuhns, Joseph B.

Publication type:

journal article

Comparison of LC-MS and LC-DAD Methods of Detecting Abused Piperazine Designer Drugs.

Published in:

Journal of Clinical Medicine, 2022, v. 11, n. 7, p. 1758, doi. 10.3390/jcm11071758

By:

Welz, Anna;
Koba, Marcin;
Kośliński, Piotr;
Siódmiak, Joanna

Publication type:

Article

Taurine and Its Derivatives: Analysis of the Inhibitory Effect on Platelet Function and Their Antithrombotic Potential.

Published in:

Journal of Clinical Medicine, 2022, v. 11, n. 3, p. 666, doi. 10.3390/jcm11030666

By:

Roşca, Adrian Eugen;
Vlădăreanu, Ana-Maria;
Mirica, Radu;
Anghel-Timaru, Cristina-Mihaela;
Mititelu, Alina;
Popescu, Bogdan Ovidiu;
Căruntu, Constantin;
Voiculescu, Suzana Elena;
Gologan, Şerban;
Onisâi, Minodora;
Iordan, Iuliana;
Zăgrean, Leon

Publication type:

Article

In vitro and in silico biological evaluation of phthalimide derivatives as antiproliferative agents.

Published in:

TIP Revista Especializada en Ciencias Químico-Biológicas, 2021, v. 24, p. 1, doi. 10.22201/fesz.23958723e.2021.314

By:

Sierra-Rivera, Crystel A.;
Kashif, Muhammad;
Vázquez-Jiménez, Lenci K.;
Zugasti-Cruz, Alejandro;
Juárez-Saldivar, Alfredo;
Paz-González, Alma D.;
Rivera, Gildardo

Publication type:

Article

3D QSAR investigations on locomotor activity of 5--cyano--N1,6--disubstituted 2--thiouracil derivatives.

Published in:

Humanity & Society, 2010, v. 34, n. 2, p. 168

By:

Kuchekar, Bhanudas S.;
Pore, Yogesh V.

Publication type:

Article

Natural Compounds and Derivatives as New Drug Candidates for Endocrine and Metabolic Disorders: Over One and a Half Decades.

Published in:

Malaysian Journal of Medicine & Health Sciences, 2024, v. 20, p. 4

By:

Manikkam, Rajalakshmi

Publication type:

Article

Ethno-Medicine Survey of Medicinal Plants Used by Villagers in Kudat, Sabah, Malaysia.

Published in:

Malaysian Journal of Medicine & Health Sciences, 2019, v. 15, p. 65

By:

Shimmi, Sadia Choudhury;
Kabir, Shaila;
Parash, M. Tanveer Hossain;
Hossain, A. B. M. Tofazzal;
Khaing, Mya Sanda;
Yunus, Razlan Bin Muhd

Publication type:

Article

Organogels based on amino acid derivatives and their optimization for drug release using response surface methodology.

Published in:

Artificial Cells, Nanomedicine & Biotechnology, 2020, v. 48, n. 1, p. 266, doi. 10.1080/21691401.2019.1699833

By:

Hu, Beibei;
Yan, Haipeng;
Sun, Yanping;
Chen, Xi;
Sun, Yujuan;
Li, Sanming;
Jing, Yongshuai;
Li, Heran

Publication type:

Article

Cover Feature: Synthesis and Antitumor Evaluation of Novel Hybrids of Phenylsulfonylfuroxan and Estradiol Derivatives (ChemistryOpen 2/2020).

Published in:

ChemistryOpen, 2020, v. 9, n. 2, p. 98, doi. 10.1002/open.202000011

By:

Wan, Qi;
Deng, Yan;
Huang, Yaoqing;
Yu, Zhihui;
Wang, Chunli;
Wang, Ke;
Dong, Jibin;
Chen, Ying

Publication type:

Article

SYNTHESES AND ANTIOXIDANT ACTIVITIES OF SOME HYDROXY DIMETHOXY CHALCONE DERIVATIVES.

Published in:

Indonesian Journal of Pharmacy / Majalah Farmasi Indonesia, 2014, v. 25, n. 1, p. 17, doi. 10.14499/indonesianjpharm25iss1pp17

By:

Elfi Susanti, V. H.;
Matsjeh, Sabirin;
Mustofa;
Redjeki, Tri;
Wahyuningsih, Tutik Dwi

Publication type:

Article

The synthesis and antitubercular activity of substituted hydrazone,2-pyrazoline-5-one and 2-isoxazoline-5-one derivatives possessing 1,3,4-thiadiazole moiety.

Published in:

Marmara Pharmaceutical Journal, 2012, v. 16, n. 3, p. 222

By:

Oral, Başak;
Rollas, Sevim

Publication type:

Article

Formononetin: a review of its source, pharmacology, drug combination, toxicity, derivatives, and drug delivery systems.

Published in:

2025

By:

Jin, Min;
Wei, Linfang;
Wang, Jianhua;
Shen, Yuehong;
Gao, Lei;
Zhao, Fan;
Gao, Qianying;
Ma, Yifei;
Sun, Yongyan;
Lin, Ying;
Ji, Guanjie;
Cai, Pingping;
Yan, Rugen

Publication type:

Literature Review

A quantitative structure–activity relationship study on CXL017 derivatives as effective drugs for cancer treatment.

Published in:

Journal of the Chinese Chemical Society, 2021, v. 68, n. 10, p. 1972, doi. 10.1002/jccs.202100050

By:

Nekoei, Mehdi;
Mohammadhosseini, Majid;
Pourbasheer, Eslam

Publication type:

Article

Photo-induced hydroxypentafluorosulfanylation of alkenes with SF5Cl and oxygen gas and their further derivatization.

Published in:

Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-54015-5

By:

Jiang, Yuanyang;
Meng, Xiaoli;
Zhang, Jiangshan;
Wu, Gang;
Lin, Xinjing;
Guo, Shuo

Publication type:

Article

Sulfonamide-directed site-selective functionalization of unactivated C(sp3)−H enabled by photocatalytic sequential electron/proton transfer.

Published in:

Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-49337-3

By:

Wang, Chaodong;
Chen, Zhi;
Sun, Jie;
Tong, Luwei;
Wang, Wenjian;
Song, Shengjie;
Li, Jianjun

Publication type:

Article

Experimental and Theoretical Studies of 1, 3-diaminopropylene Derivatives as Poten- tial Antioxidative Agents for Copper Nano-particles in Hydrothermal System.

Published in:

Nano Biomedicine & Engineering, 2011, v. 3, n. 2, p. 130, doi. 10.5101/nbe.v3i2.p130-136

By:

Guo Gao;
Xueqing Zhang;
Kan Wang;
Lili Feng;
Peng Huang;
Yixia Zhang;
Chunlei Zhang;
Meng He;
Xiao Zhi

Publication type:

Article

Distribution and effect of steroidal saponin derivative WRC3 in B16 melanoma cells.

Published in:

Molecular Medicine Reports, 2015, v. 12, n. 4, p. 6019, doi. 10.3892/mmr.2015.4225

By:

ZELIANG WEI;
YUYAN LIANG;
LIMEI MA;
KE LI;
HAI NIU;
WEN HUANG

Publication type:

Article

A Transcriptomics-Based Bioinformatics Approach for Identification and In Vitro Screening of FDA-Approved Drugs for Repurposing against Dengue Virus-2.

Published in:

Viruses (1999-4915), 2022, v. 14, n. 10, p. N.PAG, doi. 10.3390/v14102150

By:

Punekar, Madhura;
Kasabe, Bhagyashri;
Patil, Poonam;
Kakade, Mahadeo B.;
Parashar, Deepti;
Alagarasu, Kalichamy;
Cherian, Sarah

Publication type:

Article

Tetracyclic triterpenoids as inhibitors of cytochrome P450 3A4 and their quantitative structure activity relationship analysis.

Published in:

Arabian Journal of Chemistry, 2023, v. 16, n. 10, p. N.PAG, doi. 10.1016/j.arabjc.2023.105156

By:

Pan, Wei;
Feng, Lei;
Sun, Cheng-Peng;
Tian, Xiang-Ge;
Shi, Chao;
Wang, Chao;
Lv, Xia;
Wang, Yan;
Huang, Shan-Shan;
Zhang, Bao-Jing;
Ning, Jing;
Ma, Xiao-Chi

Publication type:

Article

Synthesis of Salicylate and Salicylamide Alcohols for the Preparation of Phosphorodiamidates and Ifosfamide Prodrugs.

Published in:

Oriental Journal of Chemistry, 2021, v. 37, n. 2, p. 295, doi. 10.13005/ojc/370205

By:

PAL, ASHUTOSH

Publication type:

Article

Eyelash drug launched in national event.

Published in:

Optometry Times, 2009, v. 1, n. 3, p. 8

By:

Charters, Lynda

Publication type:

Article

Enantiospecific sp2-sp3 coupling of secondary and tertiary boronic esters.

Published in:

Nature Chemistry, 2014, v. 6, n. 7, p. 584, doi. 10.1038/nchem.1971

By:

Bonet, Amadeu;
Odachowski, Marcin;
Leonori, Daniele;
Essafi, Stephanie;
Aggarwal, Varinder K.

Publication type:

Article

Partial Purification of Dipeptidyl Peptidase-4 From Human Blood Serum and Study the Inhibitory Effect of Some Nitrile Derivatives on it.

Published in:

Indian Journal of Forensic Medicine & Toxicology, 2021, v. 15, n. 3, p. 2969, doi. 10.37506/ijfmt.v15i3.15755

By:

Algburi, Firas Shawqi;
Al-Tikrity, Nadia Y.;
Ulusal, Hasan;
Taskin-Tok, Tugba;
Ali, Omeed Akbar

Publication type:

Article

Development and Preparation of ciprofloxacin Drug Derivatives for Treatment of Microbial Contamination in Hospitals and Environment.

Published in:

Indian Journal of Forensic Medicine & Toxicology, 2020, v. 14, n. 2, p. 1188, doi. 10.37506/ijfmt.v14i2.3067

By:

Jawad, Aseel Mahmood;
Aljamali, Nagham Mahmood;
Jwad, Saher Mahmood

Publication type:

Article

Study on the Analysis and Synthesis of Designer Drugs, Piperazine.

Published in:

Indian Journal of Forensic Medicine & Toxicology, 2019, v. 13, n. 2, p. 125, doi. 10.5958/0973-9130.2019.00098.7

By:

Gandhi, Rhythm;
Chauhan, Amit;
Shukla, S. K.

Publication type:

Article

Characterization of the designer drug bk-2C-B (2-amino-1-(bromodimethoxyphenyl) ethan-1-one) by gas chromatography/mass spectrometry without and with derivatization with 2,2,2-trichloroethyl chloroformate, liquid chromatography/high-resolution mass spectrometry, and nuclear magnetic resonance

Published in:

Rapid Communications in Mass Spectrometry: RCM, 2015, v. 29, n. 13, p. 1196, doi. 10.1002/rcm.7211

By:

Frison, Giampietro;
Odoardi, Sara;
Frasson, Samuela;
Sciarrone, Rocco;
Ortar, Giorgio;
Romolo, Francesco Saverio;
Strano Rossi, Sabina

Publication type:

Article

Delineation of a Novel Non-Steroidal Anti-Inflammatory Drugs Derivative Using Molecular Docking and Pharmacological Assessment.

Published in:

Indian Journal of Pharmaceutical Sciences, 2022, v. 84, n. 3, p. 642

By:

SHAH, K.;
MUJWAR, S.

Publication type:

Article

Application of Chitosan and Its Derivatives in Transdermal Drug Delivery.

Published in:

Advances in Polymer Science, 2021, v. 288, p. 411, doi. 10.1007/12_2021_102

By:

Panonnummal, Rajitha;
Kumar, Vrinda S.;
Jayakumar, R.;
Sabitha, M.

Publication type:

Article

A Metal‐Free and Operationally Simple Radical Trifluoromethylative Borylation of Unactivated Alkenes.

Published in:

Chemistry - A European Journal, 2024, v. 30, n. 6, p. 1, doi. 10.1002/chem.202303468

By:

Keerthika, K.;
Muhammed S, Bazil;
Geetharani, K.

Publication type:

Article

Direct C(3)5−H Polyfluoroarylation of 2‐Amino/alkoxy Pyridines Enabled by a Transient and Electron‐deficient Palladium Intermediate.

Published in:

Chemistry - A European Journal, 2023, v. 29, n. 41, p. 1, doi. 10.1002/chem.202301436

By:

Das, Animesh;
Maji, Biplab

Publication type:

Article

Synthesis of Polysubstituted Enamides by Hydrogen Atom Transfer Alkene Isomerization Using Dual Cobalt/Photoredox Catalysis.

Published in:

Chemistry - A European Journal, 2023, v. 29, n. 37, p. 1, doi. 10.1002/chem.202300804

By:

Seino, Yusuke;
Yamaguchi, Yuto;
Suzuki, Akihiko;
Yamashita, Masaaki;
Kamei, Yuji;
Kamiyama, Futa;
Yoshino, Tatsuhiko;
Kojima, Masahiro;
Matsunaga, Shigeki

Publication type:

Article

Remote Radical Desaturation of Unactivated C−H Bonds in Amides.

Published in:

Chemistry - A European Journal, 2021, v. 27, n. 67, p. 16621, doi. 10.1002/chem.202103509

By:

Xia, Yong;
Jana, Kalipada;
Studer, Armido

Publication type:

Article

Electrochemical NiH‐Catalyzed C(sp3)−C(sp3) Coupling of Alkyl Halides and Alkyl Alkenes.

Published in:

Angewandte Chemie, 2023, v. 135, n. 44, p. 1, doi. 10.1002/ange.202311941

By:

Li, Pengfei;
Kou, Guangsheng;
Feng, Tian;
Wang, Minyan;
Qiu, Youai

Publication type:

Article

A General and Practical Route to Functionalized Bicyclo[1.1.1]Pentane‐Heteroaryls Enabled by Photocatalytic Multicomponent Heteroarylation of [1.1.1]Propellane.

Published in:

Angewandte Chemie, 2023, v. 135, n. 24, p. 1, doi. 10.1002/ange.202302223

By:

Huang, Weichen;
Keess, Sebastian;
Molander, Gary A.

Publication type:

Article

Transition‐Metal‐Free Difunctionalization of Sulfur Nucleophiles**.

Published in:

Angewandte Chemie, 2023, v. 135, n. 8, p. 1, doi. 10.1002/ange.202216296

By:

Mondal, Shobhan;
Di Tommaso, Ester Maria;
Olofsson, Berit

Publication type:

Article

Metal‐Free Electrochemical Carboxylation of Organic Halides in the Presence of Catalytic Amounts of an Organomediator.

Published in:

Angewandte Chemie, 2022, v. 134, n. 41, p. 1, doi. 10.1002/ange.202210201

By:

Wang, Yanwei;
Zhao, Zhiwei;
Pan, Deng;
Wang, Siyi;
Jia, Kangping;
Ma, Dengke;
Yang, Guoqing;
Xue, Xiao‐Song;
Qiu, Youai

Publication type:

Article

Electrocarboxylation of Aryl Epoxides with CO2 for the Facile and Selective Synthesis of β‐Hydroxy Acids.

Published in:

Angewandte Chemie, 2022, v. 134, n. 38, p. 1, doi. 10.1002/ange.202207746

By:

Wang, Yanwei;
Tang, Shunyao;
Yang, Guoqing;
Wang, Siyi;
Ma, Dengke;
Qiu, Youai

Publication type:

Article

Nickel‐Catalyzed Thermal Redox Functionalization of C(sp3)−H Bonds with Carbon Electrophiles**.

Published in:

Angewandte Chemie, 2022, v. 134, n. 22, p. 1, doi. 10.1002/ange.202201662

By:

Gong, Yuxin;
Su, Lei;
Zhu, Zhaodong;
Ye, Yang;
Gong, Hegui

Publication type:

Article

Remote Site‐Selective Radical C(sp3)−H Monodeuteration of Amides using D2O.

Published in:

Angewandte Chemie, 2021, v. 133, n. 34, p. 18793, doi. 10.1002/ange.202104254

By:

Wang, Lin;
Xia, Yong;
Derdau, Volker;
Studer, Armido

Publication type:

Article

Generation and Reactivity of Amidyl Radicals: Manganese‐Mediated Atom‐Transfer Reaction.

Published in:

Angewandte Chemie, 2020, v. 132, n. 11, p. 4458, doi. 10.1002/ange.201913042

By:

Liu, Run‐Zhou;
Li, Jinxia;
Sun, Jun;
Liu, Xian‐Guan;
Qu, Shuanglin;
Li, Ping;
Zhang, Bo

Publication type:

Article

Radical Monofluoroalkylative Alkynylation of Olefins by a Docking–Migration Strategy.

Published in:

Angewandte Chemie, 2019, v. 131, n. 49, p. 17810, doi. 10.1002/ange.201910514

By:

Wang, Min;
Zhang, Huihui;
Liu, Jige;
Wu, Xinxin;
Zhu, Chen

Publication type:

Article

CJX1, an amlodipine derivative, interacts with ATPase of human P-glycoprotein

Published in:

Cell Biology International, 2009, v. 33, n. 10, p. 1073, doi. 10.1016/j.cellbi.2009.06.023

By:

Ji, Bian-Sheng;
He, Ling

Publication type:

Article

Synthesis of tetrazol-1-yl analogs of L-lysine and L-ornithine.

Published in:

Russian Journal of Organic Chemistry, 2015, v. 51, n. 11, p. 1671, doi. 10.1134/S1070428015110287

By:

Chuprun, S.;
Popova, E.;
Mukhametshina, A.;
Trifonov, R.

Publication type:

Article

Synthesis of tetrazol-5-ylethyl derivatives of dipterocarpol.

Published in:

Russian Journal of Organic Chemistry, 2015, v. 51, n. 11, p. 1674, doi. 10.1134/S1070428015110299

By:

Kaledina, A.;
Zorina, A.;
Anokhina, V.;
Trifonov, R.

Publication type:

Article