Works matching DE "DRUG derivatives"

Results: 380

A Metal‐Free and Operationally Simple Radical Trifluoromethylative Borylation of Unactivated Alkenes.

Published in:

Chemistry - A European Journal, 2024, v. 30, n. 6, p. 1, doi. 10.1002/chem.202303468

By:

Keerthika, K.;
Muhammed S, Bazil;
Geetharani, K.

Publication type:

Article

Direct C(3)5−H Polyfluoroarylation of 2‐Amino/alkoxy Pyridines Enabled by a Transient and Electron‐deficient Palladium Intermediate.

Published in:

Chemistry - A European Journal, 2023, v. 29, n. 41, p. 1, doi. 10.1002/chem.202301436

By:

Das, Animesh;
Maji, Biplab

Publication type:

Article

Synthesis of Polysubstituted Enamides by Hydrogen Atom Transfer Alkene Isomerization Using Dual Cobalt/Photoredox Catalysis.

Published in:

Chemistry - A European Journal, 2023, v. 29, n. 37, p. 1, doi. 10.1002/chem.202300804

By:

Seino, Yusuke;
Yamaguchi, Yuto;
Suzuki, Akihiko;
Yamashita, Masaaki;
Kamei, Yuji;
Kamiyama, Futa;
Yoshino, Tatsuhiko;
Kojima, Masahiro;
Matsunaga, Shigeki

Publication type:

Article

Pharmacokinetic and pharmacodynamic comparison of fluoropyrimidine derivatives, capecitabine and 5'-deoxy-5-fluorouridine (5'-DFUR).

Published in:

Cancer Chemotherapy & Pharmacology, 2005, v. 56, n. 2, p. 205, doi. 10.1007/s00280-004-0934-7

By:

Ebi, Hiromichi;
Sigeoka, Yasushi;
Saeki, Toshiaki;
Kawada, Kenji;
Igarashi, Tadahiko;
Usubuchi, Noriko;
Ueda, Ryuzo;
Sasaki, Yasutsuna;
Minami, Hironobu

Publication type:

Article

Unusual reactivity of β-hydroxy-serotonin, a forgotten serotonin derivative.

Published in:

Amino Acids, 2015, v. 47, n. 1, p. 189, doi. 10.1007/s00726-014-1854-4

By:

Kawashima, Takaaki;
Salinger, Jeremy;
Hida, Koichi;
Takai, Katsuji;
Nakamaru-Ogiso, Eiko

Publication type:

Article

Synthesis, Antidiabetic Evaluation and Molecular Docking Studies of Thiazolidine-2,4-Dione Analogues.

Published in:

Indian Journal of Pharmaceutical Education & Research, 2023, v. 57, p. s98, doi. 10.5530/ijper.57.1s.11

By:

Pardeshi, Dolly R.;
Kulkarni, Vithal M.;
Pathare, Sandeep S.

Publication type:

Article

Synthesis, Crystal Structure, Hirshfeld Surface Analyses and Biological Activity of Novel Cinnamide Derivatives as Neuroprotective Drugs.

Published in:

Polycyclic Aromatic Compounds, 2024, v. 44, n. 8, p. 5138, doi. 10.1080/10406638.2023.2261586

By:

Wang, Yuying;
Gao, Mengjie;
Zhong, Yan;
Wu, Bin

Publication type:

Article

Design, Synthesis, Bioactivity Analyses, and Molecular Docking Study of Triazine-Tyrosine Based Derivatives as Drugs like Fingolimod for Treatment of Multiple Sclerosis.

Published in:

Polycyclic Aromatic Compounds, 2024, v. 44, n. 4, p. 2292, doi. 10.1080/10406638.2023.2215375

By:

Asadi, Parvin;
Khodarahmi, Ghadamali;
Rafiee, Amin;
Aliomrani, Mehdi;
Hassanzadeh, Farshid

Publication type:

Article

Microwave Assisted Synthesis and Antimicrobial Activities of Carboxylpyrazoline Derivatives: Molecular Docking and DFT Influence in Bioisosteric Replacement.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 8, p. 5422, doi. 10.1080/10406638.2021.1937236

By:

Farooq, Saba;
Ngaini, Zainab;
Daud, Adibah Izzati;
Khairul, Wan M.

Publication type:

Article

Diethyl (2-Amino-3-Cyano-4H-Chromen-4-yl)Phosphonate and Its Halogenated Derivatives as Effective Drug: A Theoretical and an Experimental Spectroscopic Study.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 5, p. 2305, doi. 10.1080/10406638.2020.1832126

By:

Yadav, Krishna Kant;
Kumar, Abhishek;
Kumar, Amarendra;
Brahmachari, Goutam;
Misra, Neeraj

Publication type:

Article

Synthesis of Thiazole Linked Imidazo[2,1-b]Thiazoles as Anticancer Agents.

Published in:

Polycyclic Aromatic Compounds, 2021, v. 41, n. 8, p. 1608, doi. 10.1080/10406638.2019.1689514

By:

Mahmoud, Huda K.;
Gomha, Sobhi M.;
Farghaly, Thoraya A.;
Awad, Hanem M.

Publication type:

Article

Oral isotretinoin and sacroiliitis: causal link or coincidence? Discussion points emerging from a case-based review.

Published in:

Rheumatology / Reumatologia, 2022, v. 60, n. 5, p. 357, doi. 10.5114/reum.2022.120761

By:

Sargin, Betül;
Manzo, Ciro

Publication type:

Article

Cover Feature: Synthesis and in vivo Evaluation of Fluorobenzyl Metformin Derivatives as Potential Drugs in The Diabetes Treatment (Asian J. Org. Chem. 7/2023).

Published in:

Asian Journal of Organic Chemistry, 2023, v. 12, n. 7, p. 1, doi. 10.1002/ajoc.202300276

By:

Hernández‐Velázquez, Edson D.;
Herrera, Mayra D.;
Alba‐Betancourt, Clara;
Navarro‐Santos, Pedro;
Ortíz‐Alvarado, Rafael;
Solorio‐Alvarado, César R.

Publication type:

Article

Synthesis and in vivo Evaluation of Fluorobenzyl Metformin Derivatives as Potential Drugs in The Diabetes Treatment.

Published in:

Asian Journal of Organic Chemistry, 2023, v. 12, n. 7, p. 1, doi. 10.1002/ajoc.202300200

By:

Hernández‐Velázquez, Edson D.;
Herrera, Mayra D.;
Alba‐Betancourt, Clara;
Navarro‐Santos, Pedro;
Ortíz‐Alvarado, Rafael;
Solorio‐Alvarado, César R.

Publication type:

Article

Synergistic interaction and activation of the opioid receptor-NO-cGMP-K+ channel pathway on peripheral antinociception induced by the α-Bisabolol-diclofenac combination.

Published in:

Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1158236

By:

Ortiz, Mario I.

Publication type:

Article

Corrigendum: Anti-viral drug discovery against monkeypox and smallpox infection by natural curcumin derivatives: a computational drug design approach.

Published in:: Frontiers in Cellular & Infection Microbiology, 2023, p. 1, doi. 10.3389/fcimb.2023.1217334
Publication type:: Article

POM analyses of Raltegravir derivatives: a new reflection enlightening the mechanism of HIV-integrase inhibition.

Published in:

Research on Chemical Intermediates, 2015, v. 41, n. 8, p. 5121, doi. 10.1007/s11164-014-1616-7

By:

Lahsasni, Siham;
Ben Hadda, Taibi;
Masand, Vijay;
Pathan, Naziyanaz;
Parvez, Ali;
Warad, Ismail;
Shaheen, Usama;
Bader, Ammar;
Aljofan, Mohamad

Publication type:

Article

Pharmacological evaluation of isochromen-1-ones and their thioanalogues derived from anti-inflammatory drug ketoprofen.

Published in:

Research on Chemical Intermediates, 2013, v. 39, n. 3, p. 1343, doi. 10.1007/s11164-012-0690-y

By:

Napoleon, A.;
Bhagwat, Swati;
Khan, Fazlur-Rahman

Publication type:

Article

Tetracyclic triterpenoids as inhibitors of cytochrome P450 3A4 and their quantitative structure activity relationship analysis.

Published in:

Arabian Journal of Chemistry, 2023, v. 16, n. 10, p. N.PAG, doi. 10.1016/j.arabjc.2023.105156

By:

Pan, Wei;
Feng, Lei;
Sun, Cheng-Peng;
Tian, Xiang-Ge;
Shi, Chao;
Wang, Chao;
Lv, Xia;
Wang, Yan;
Huang, Shan-Shan;
Zhang, Bao-Jing;
Ning, Jing;
Ma, Xiao-Chi

Publication type:

Article

Review on recent development of quinoline for anticancer activities.

Published in:

Arabian Journal of Chemistry, 2022, v. 15, n. 11, p. N.PAG, doi. 10.1016/j.arabjc.2022.104168

By:

Ilakiyalakshmi, Mohan;
Arumugam Napoleon, Ayyakannu

Publication type:

Article

Greener pastures in evaluating antidiabetic drug for a quinoxaline Derivative: Synthesis, Characterization, Molecular Docking, in vitro and HSA/DFT/XRD studies.

Published in:

Arabian Journal of Chemistry, 2022, v. 15, n. 6, p. N.PAG, doi. 10.1016/j.arabjc.2022.103851

By:

Missioui, Mohcine;
Mortada, Salma;
Guerrab, Walid;
Demirtaş, Güneş;
Mague, Joel T.;
Ansar, M'hammed;
El Abbes Faouzi, My;
Essassi, E.M.;
Mehdar, Yassin T.H.;
Aljohani, Faizah S.;
Said, Musa A.;
Ramli, Youssef

Publication type:

Article

Eyelash drug launched in national event.

Published in:

Optometry Times, 2009, v. 1, n. 3, p. 8

By:

Charters, Lynda

Publication type:

Article

Study on the Activation of the Opioid Receptors by a Set of Morphine Derivatives in a Well-Defined Assay System.

Published in:

Neurochemical Research, 2012, v. 37, n. 2, p. 410, doi. 10.1007/s11064-011-0627-7

By:

Zhang, Yan;
Wang, Zhiwei;
Cox, D.;
Civelli, Olivier

Publication type:

Article

Investigating the potential of monocyclic B9N9 and C18 rings for the electrochemical sensing, and adsorption of carbazole-based anti-cancer drug derivatives: DFT-based first-principle study.

Published in:

Journal of Molecular Modeling, 2024, v. 30, n. 8, p. 1, doi. 10.1007/s00894-024-06049-1

By:

Niamat, Yumna;
Yaqoob, Junaid;
Khan, Muhammad Usman;
Hussain, Riaz;
Gilani, Mazhar Amjad;
Hassan, Abrar Ul;
Ahamad, Tansir

Publication type:

Article

Identification of novel C-15 fluoro isosteviol derivatives for GABA-AT inhibition by in silico investigations.

Published in:

Journal of Molecular Modeling, 2023, v. 29, n. 3, p. 1, doi. 10.1007/s00894-023-05479-7

By:

Salaria, Punam;
Akshinthala, Parameswari;
Kapavarapu, Ravikumar;
M, Amarendar Reddy

Publication type:

Article

Drugs of Abuse 2012 Update.

Published in:

Pediatric Emergency Medicine Reports, 2012, v. 17, n. 12, p. 145

By:

Felter, Robert A.

Publication type:

Article

The potential use of bacteria and bacterial derivatives as drug delivery systems for viral infection.

Published in:

Virology Journal, 2023, v. 20, n. 1, p. 1, doi. 10.1186/s12985-023-02183-z

By:

Faghihkhorasani, Amirhosein;
Ahmed, Hanan Hassan;
Mashool, Noor Muhammad;
Alwan, Mariem;
Assefi, Marjan;
Adab, Aya Hussein;
Yasamineh, Saman;
Gholizadeh, Omid;
Baghani, Moein

Publication type:

Article

Synthesis and in vitro anti-breast cancer activity of some novel 1,5-benzothiazepine derivatives.

Published in:

Journal of the Serbian Chemical Society, 2012, v. 77, n. 6, p. 725, doi. 10.2298/JSC110715219A

By:

Ameta, K. L.;
Rathore, Nitu S.;
Kumar, Biresh

Publication type:

Article

Antithyroid activity of some 6-(alkylsulfanyl)-9H-purines.

Published in:

Journal of the Serbian Chemical Society, 2011, v. 76, n. 10, p. 1355, doi. 10.2298/JSC101209041I

By:

Fatima, Ismat;
Munawar, Munawar A.;
Tasneem, Affia;
Jahan, Sarwat;
Khan, Misbahul A.;
Ahmed, Shakeel

Publication type:

Article

Synthesis and antimicrobial activity of a new series of 1,4-dihydropyridine derivatives.

Published in:

Journal of the Serbian Chemical Society, 2011, v. 76, n. 1, p. 1, doi. 10.2298/JSC091127003K

By:

KUMAR, RADHAKRISHNAN SURENDRA;
IDHAYADHULLA, AKBAR;
NASSER, ABDUL JAMAL ABDUL;
SELVIN, JOSEPH

Publication type:

Article

Synthesis and properties of some new 4-succinamoyl piperazine-2,6-dione derivatives.

Published in:

Chemija, 2007, v. 18, n. 1, p. 50

By:

Švedaitė, Irena

Publication type:

Article

Synthesis and growth regulatory activity of pyrazolesulfanyl- and isoxazolesulfanyl-1 H-[1,2,4]triazoles and their azinyl derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2011, v. 48, n. 1, p. 188, doi. 10.1002/jhet.514

By:

Eliazyan, Karine A.;
Shahbazyan, Lusya V.;
Pivazyan, Vergush A.;
Yengoyan, Aleksandr P.

Publication type:

Article

XQ2, a Novel TPZ Derivative, Induced G2/M Phase Arrest and Apoptosis under Hypoxia in Non-Small Cell Lung Cancer. Cells.

Published in:

Bioscience, Biotechnology & Biochemistry, 2010, v. 74, n. 6, p. 1181, doi. 10.1271/bbb.90889

By:

Jianshu Lou;
XingLu Zhou;
Qinjie Weng;
Duo-duo Wang;
Qing Xia;
Yongzhou Hu;
Qiaojun He;
Bo Yang;
Peihua Lou

Publication type:

Article

New vanadyl complexes with metformin derivatives as potential insulin mimetic agents.

Published in:

Journal of Thermal Analysis & Calorimetry, 2012, v. 110, n. 1, p. 257, doi. 10.1007/s10973-012-2274-x

By:

Olar, Rodica;
Dogaru, Andreea;
Marinescu, Dana;
Badea, Mihaela

Publication type:

Article

Colchicine derivative as a potential anti-glioma compound.

Published in:

Journal of Neuro-Oncology, 2015, v. 124, n. 3, p. 403, doi. 10.1007/s11060-015-1874-2

By:

Fang, Kuan-Min;
Liu, Jun-Jen;
Li, Chun-Chun;
Cheng, Chih-Chi;
Hsieh, Yun-Ti;
Chai, Kit;
Lien, Yu-An;
Tzeng, Shun-Fen

Publication type:

Article

K-80003 Inhibition of Macrophage Apoptosis and Necrotic Core Development in Atherosclerotic Vulnerable Plaques.

Published in:

Cardiovascular Drugs & Therapy, 2022, v. 36, n. 6, p. 1061, doi. 10.1007/s10557-021-07237-4

By:

Wang, Xiaolei;
Sun, Zhe;
Yuan, Ruosen;
Zhang, Weifeng;
Shen, Yejiao;
Yin, Anwen;
Li, Yanjie;
Ji, Qingqi;
Wang, Xia;
Li, Yi;
Zhang, Min;
Pan, Xin;
Shen, Linghong;
He, Ben

Publication type:

Article

Synthesis and Pharmacological Evaluation of 6-Arylpyridazinones as Potent Vasorelaxants.

Published in:

Drug Development Research, 2013, v. 74, n. 5, p. 296, doi. 10.1002/ddr.21079

By:

Bansal, Ranju;
Kumar, Dinesh;
Sharma, Deepika;
Calle, Carmen;
Carron, Rosalia

Publication type:

Article

Interaction of Doxorubicin Embedded into Phospholipid Nanoparticles and Targeted Peptide-Modified Phospholipid Nanoparticles with DNA.

Published in:

Molecules, 2023, v. 28, n. 14, p. 5317, doi. 10.3390/molecules28145317

By:

Pronina, Veronica V.;
Kostryukova, Lyubov V.;
Bulko, Tatiana V.;
Shumyantseva, Victoria V.

Publication type:

Article

Pyridyl Methylsulfinyl Benzimidazole Derivatives as Promising Agents against Giardia lamblia and Trichomonas vaginalis.

Published in:

Molecules, 2022, v. 27, n. 24, p. 8902, doi. 10.3390/molecules27248902

By:

Hernández-Ochoa, Beatriz;
Martínez-Rosas, Víctor;
Morales-Luna, Laura;
Calderón-Jaimes, Ernesto;
Rocha-Ramírez, Luz María;
Ortega-Cuellar, Daniel;
Rufino-González, Yadira;
González-Valdez, Abigail;
Arreguin-Espinosa, Roberto;
Enríquez-Flores, Sergio;
Castillo-Rodríguez, Rosa Angélica;
Cárdenas-Rodríguez, Noemí;
Wong-Baeza, Carlos;
Baeza-Ramírez, Isabel;
Gómez-Manzo, Saúl

Publication type:

Article

Histone Deacetylase Inhibitory Activity and Antiproliferative Potential of New [6]-Shogaol Derivatives.

Published in:

Molecules, 2022, v. 27, n. 10, p. 3332, doi. 10.3390/molecules27103332

By:

Phaosiri, Chanokbhorn;
Yenjai, Chavi;
Senawong, Thanaset;
Senawong, Gulsiri;
Saenglee, Somprasong;
Somsakeesit, La-or;
Kumboonma, Pakit

Publication type:

Article

Albatrellus confluens (Alb. & Schwein.) Kotl. & Pouz.: Natural Fungal Compounds and Synthetic Derivatives with In Vitro Anthelmintic Activities and Antiproliferative Effects against Two Human Cancer Cell Lines.

Published in:

Molecules, 2022, v. 27, n. 9, p. 2950, doi. 10.3390/molecules27092950

By:

Dube, Mthandazo;
Llanes, Dayma;
Saoud, Mohamad;
Rennert, Robert;
Imming, Peter;
Häberli, Cécile;
Keiser, Jennifer;
Arnold, Norbert

Publication type:

Article

Research Progress in the Field of Gambogic Acid and Its Derivatives as Antineoplastic Drugs.

Published in:

Molecules, 2022, v. 27, n. 9, p. 2937, doi. 10.3390/molecules27092937

By:

Li, Meng;
Su, Fali;
Zhu, Mingtao;
Zhang, Huan;
Wei, Yuxin;
Zhao, Yang;
Li, Jianmin;
Lv, Shaowa

Publication type:

Article

Distinct Mechanisms of Cytotoxicity in Novel Nitrogenous Heterocycles: Future Directions for a New Anti-Cancer Agent.

Published in:

Molecules, 2022, v. 27, n. 8, p. N.PAG, doi. 10.3390/molecules27082409

By:

Suliman, Rasha Saad;
Alghamdi, Sahar Saleh;
Ali, Rizwan;
Rahman, Ishrat;
Alqahtani, Tariq;
Frah, Ibrahim K.;
Aljatli, Dimah A.;
Huwaizi, Sarah;
Algheribe, Shatha;
Alehaideb, Zeyad;
Islam, Imadul

Publication type:

Article

Novel 1,2,3-Triazole-Coumarin Hybrid Glycosides and Their Tetrazolyl Analogues: Design, Anticancer Evaluation and Molecular Docking Targeting EGFR, VEGFR-2 and CDK-2.

Published in:

Molecules, 2022, v. 27, n. 7, p. 2047, doi. 10.3390/molecules27072047

By:

El-Sayed, Wael A.;
Alminderej, Fahad M.;
Mounier, Marwa M.;
Nossier, Eman S.;
Saleh, Sayed M.;
Kassem, Asmaa F.

Publication type:

Article

Exploring the Synergistic Anticancer Potential of Benzofuran–Oxadiazoles and Triazoles: Improved Ultrasound- and Microwave-Assisted Synthesis, Molecular Docking, Hemolytic, Thrombolytic and Anticancer Evaluation of Furan-Based Molecules.

Published in:

Molecules, 2022, v. 27, n. 3, p. 1023, doi. 10.3390/molecules27031023

By:

Irfan, Ali;
Faiz, Sadia;
Rasul, Azhar;
Zafar, Rehman;
Zahoor, Ameer Fawad;
Kotwica-Mojzych, Katarzyna;
Mojzych, Mariusz

Publication type:

Article

Evaluation of Anticancer and Antibacterial Activity of Four 4-Thiazolidinone-Based Derivatives.

Published in:

Molecules, 2022, v. 27, n. 3, p. 894, doi. 10.3390/molecules27030894

By:

Skóra, Bartosz;
Lewińska, Anna;
Kryshchyshyn-Dylevych, Anna;
Kaminskyy, Danylo;
Lesyk, Roman;
Szychowski, Konrad A.

Publication type:

Article

Aurones: A Golden Resource for Active Compounds.

Published in:

Molecules, 2022, v. 27, n. 1, p. 2, doi. 10.3390/molecules27010002

By:

Mazziotti, Ilaria;
Petrarolo, Giovanni;
La Motta, Concettina

Publication type:

Article

The Molecular Structure and Self-Assembly Behavior of Reductive Amination of Oxidized Alginate Derivative for Hydrophobic Drug Delivery.

Published in:

Molecules, 2021, v. 26, n. 19, p. 5821, doi. 10.3390/molecules26195821

By:

Chen, Xiuqiong;
Zhu, Qingmei;
Li, Zhengyue;
Yan, Huiqiong;
Lin, Qiang

Publication type:

Article

Rosin Derivatives as a Platform for the Antiviral Drug Design.

Published in:

Molecules, 2021, v. 26, n. 13, p. 3836, doi. 10.3390/molecules26133836

By:

Popova, Larisa;
Ivanchenko, Olga;
Pochkaeva, Evgeniia;
Klotchenko, Sergey;
Plotnikova, Marina;
Tsyrulnikova, Angelica;
Aronova, Ekaterina

Publication type:

Article

Investigation of Antifungal Properties of Synthetic Dimethyl-4-Bromo-1-(Substituted Benzoyl) Pyrrolo[1,2-a] Quinoline-2,3-Dicarboxylates Analogues: Molecular Docking Studies and Conceptual DFT-Based Chemical Reactivity Descriptors and Pharmacokinetics Evaluation

Published in:

Molecules, 2021, v. 26, n. 9, p. 2722, doi. 10.3390/molecules26092722

By:

Uppar, Vijayakumar;
Chandrashekharappa, Sandeep;
Shivamallu, Chandan;
P, Sushma;
Kollur, Shiva Prasad;
Ortega-Castro, Joaquín;
Frau, Juan;
Flores-Holguín, Norma;
Basarikatti, Atiyaparveen I.;
Chougala, Mallikarjun;
Mohan M, Mrudula;
Banuprakash, Govindappa;
Jayadev;
Venugopala, Katharigatta N.;
Nandeshwarappa, Belakatte P.;
Veerapur, Ravindra;
Al-Kheraif, Abdulaziz A.;
Elgorban, Abdallah M.;
Syed, Asad;
Mudnakudu-Nagaraju, Kiran K.

Publication type:

Article