Works about DRUG activation

Results: 873

The activation cascade of the broad-spectrum antiviral bemnifosbuvir characterized at atomic resolution.
Published in:
PLoS Biology, 2024, v. 22, n. 8, p. 1, doi. 10.1371/journal.pbio.3002743
By:
- Chazot, Aurélie;
- Zimberger, Claire;
- Feracci, Mikael;
- Moussa, Adel;
- Good, Steven;
- Sommadossi, Jean-Pierre;
- Alvarez, Karine;
- Ferron, François;
- Canard, Bruno
Publication type:
Article
Glutamate Decarboxylase from Lactobacillus brevis: Activation by Ammonium Sulfate.
Published in:
Bioscience, Biotechnology & Biochemistry, 2008, v. 72, n. 5, p. 1299, doi. 10.1271/bbb.70782
By:
- Hiraga, Kazumi;
- Ueno, Yoshie;
- Oda, Kohei
Publication type:
Article
Facile Synthesis of Ladder‐Type Polyacenes with Perylene‐Fused‐Pyrene Structures.
Published in:
Macromolecular Chemistry & Physics, 2018, v. 219, n. 17, p. 1, doi. 10.1002/macp.201800201
By:
- Hu, Chaoying;
- Chen, Weiping;
- Yao, Haicui;
- Ren, Xiaojie;
- Zhang, Hailei;
- Zhao, Hongchi;
- Wu, Yonggang;
- Ba, Xinwu
Publication type:
Article
A Degradable and Antimicrobial Surface‐Attached Polymer Hydrogel.
Published in:
Macromolecular Chemistry & Physics, 2018, v. 219, n. 17, p. 1, doi. 10.1002/macp.201800198
By:
- Erath, Roman;
- Lienkamp, Karen
Publication type:
Article
Computational Design, Synthesis, and Photochemistry of Cy7‐PPG, an Efficient NIR‐Activated Photolabile Protecting Group for Therapeutic Applications.
Published in:
Angewandte Chemie, 2022, v. 134, n. 27, p. 1, doi. 10.1002/ange.202201308
By:
- Alachouzos, Georgios;
- Schulte, Albert M.;
- Mondal, Anirban;
- Szymanski, Wiktor;
- Feringa, Ben L.
Publication type:
Article
New Designs for Phototherapeutic Transition Metal Complexes.
Published in:
Angewandte Chemie, 2020, v. 132, n. 1, p. 61, doi. 10.1002/ange.201905171
By:
- Imberti, Cinzia;
- Zhang, Pingyu;
- Huang, Huaiyi;
- Sadler, Peter J.
Publication type:
Article
Dual‐Targeting Dual‐Action Platinum(IV) Platform for Enhanced Anticancer Activity and Reduced Nephrotoxicity.
Published in:
Angewandte Chemie, 2019, v. 131, n. 24, p. 8193, doi. 10.1002/ange.201903112
By:
- Babak, Maria V.;
- Zhi, Yang;
- Czarny, Bertrand;
- Toh, Tan Boon;
- Hooi, Lissa;
- Chow, Edward Kai‐Hua;
- Ang, Wee Han;
- Gibson, Dan;
- Pastorin, Giorgia
Publication type:
Article
Altered pharmacokinetics of enrofloxacin in experimental models of hepatic and renal impairment.
Published in:
Veterinary Research Communications, 2009, v. 33, n. 5, p. 481
By:
- J. Lim;
- B. Park;
- H. Yun
Publication type:
Article
Pharmacopoeial Quality Requirements for Medicinal Products.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 11, p. 936, doi. 10.1007/s11094-019-01929-w
By:
- Olefir, Yu. V.;
- Sakanyan, E. I.;
- Shishova, L. I.;
- Senchenko, S. P.
Publication type:
Article
Development of a Dosage Form of the New Antitumor Antibiotic Olivamide.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 11, p. 930, doi. 10.1007/s11094-019-01928-x
By:
- Tevyashova, A. N.;
- Bychkova, E. N.;
- Dezhenkova, L. G.;
- Shchekotikhin, A. E.
Publication type:
Article
Antiproliferative Evaluation of (E)-3-(3-(Allyloxy)-2-Methoxyphenyl)-1-(2,4,6-Trimethoxyphenyl)Prop-2-En-1-One as a Novel Apoptosis Inducer Against Prostate Cancer PC-3 Cells.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 11, p. 917, doi. 10.1007/s11094-019-01926-z
By:
- Fu, Dong-Jun;
- Li, Ping;
- Kuang, Yi-Rui;
- Jiang, Li-Le;
- Zhu, Ming-Chao;
- Li, Si-Chen;
- Zheng, Guo;
- Zhang, Rui;
- Zhang, Sai-Yang;
- Li, Jiang-Feng
Publication type:
Article
Synthesis, Antimicrobial Properties, and Toxicity of a Nanobiocomposite Based on Ag(0) Particles and Poly(1-Vinyl-1,2,4-Triazole).
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 11, p. 912, doi. 10.1007/s11094-019-01925-0
By:
- Sosedova, L. M.;
- Novikov, M. A.;
- Titov, E. A.;
- Pozdnyakov, A. S.;
- Korzhova, S. A.;
- Ermakova, T. G.;
- Prozorova, G. F.
Publication type:
Article
Synthesis and Anti-Inflammatory Activity of Tyrosol and Its Structural Analogs.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 11, p. 907, doi. 10.1007/s11094-019-01924-1
By:
- Krysin, A. P.;
- Tolstikova, T. G.;
- Dolgikh, M. P.;
- Shul'ts, E. E.;
- Pokrovskii, L. M.
Publication type:
Article
Antitumor Activity and Toxicity of Olivamide Dosage Form, a New Semi-Synthetic Olivomycin a Derivative.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 11, p. 902, doi. 10.1007/s11094-019-01923-2
By:
- Treshchalin, I. D.;
- Treshchalin, M. I.;
- Tevyashova, A. N.;
- Pereverzeva, E. R.
Publication type:
Article
Quantitative Determination of Total Flavonoids in Blood-Red Hawthorn Leaves.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 10, p. 850, doi. 10.1007/s11094-019-1913-y
By:
- Kurkin, V. A.;
- Morozova, T. V.;
- Pravdivtseva, O. E.;
- Kurkina, A. V.
Publication type:
Article
Synthesis and Neurotropic Activity of New Condensed Pyrano[4,3-b]-Pyridines Derivatives.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 10, p. 844, doi. 10.1007/s11094-019-1912-z
By:
- Dabaeva, V. V.;
- Bagdasaryan, M. R.;
- Dashyan, Sh. Sh.;
- Dzhagatspanyan, I. A.;
- Nazaryan, I. M.;
- Akopyan, A. G.;
- Paronikyan, R. G.
Publication type:
Article
Synthesis and Neurotropic Activity of 4-Phenylpyridine-3-Carboxylic Acid and 3-Hydroxy-4-Phenylthieno[2,3-b]-Pyridine Derivatives.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 10, p. 839, doi. 10.1007/s11094-019-1911-0
By:
- Paronikyan, E. G.;
- Ogannisyan, A. V.;
- Paronikyan, R. G.;
- Dzhagatspanyan, I. A.;
- Nazaryan, I. M.;
- Akopyan, A. G.;
- Minasyan, N. S.
Publication type:
Article
Modification of the Benzene Moiety in the Quinolone Nucleus of 4-Hydroxy-6,7-Dimethoxy-2-Oxo-N-(Pyridin-3-Ylmethyl)-1,2-Dihydroquinoline-3-Carboxamide as an Attempt to Enhance its Analgesic Activity.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 10, p. 825, doi. 10.1007/s11094-019-1908-8
By:
- Ukrainets, I. V.;
- Mospanova, E. V.;
- Bereznyakova, N. L.;
- Davidenko, A. A.
Publication type:
Article
Synthesis and Antiviral Activity of Polycyclic N-Amidoimides Based on 4-Oxatetracyclo-[5.3.2.02, 6.08, 10]Dodec-11-Ene-3,5-Dione.
Published in:
Pharmaceutical Chemistry Journal, 2019, v. 52, n. 10, p. 820, doi. 10.1007/s11094-019-1907-9
By:
- Selivanov, B. A.;
- Bormotov, N. I.;
- Shishkina, L. N.;
- Belanov, E. F.;
- Serova, O. A.;
- Kabanov, A. S.;
- Mazurkov, O. Yu.;
- Tikhonov, A. Ya.
Publication type:
Article
Synthesis, Spectroscopic Studies, Antibacterial Activity, and Colorimetric Evaluation of the Time-Killing Assay for Newly Synthesized Chalcones Using Resazurin.
Published in:
Pharmaceutical Chemistry Journal, 2018, v. 52, n. 6, p. 518, doi. 10.1007/s11094-018-1852-z
By:
- Prasad, Sunnapu;
- Francis Saleshier, M.;
- Krishnan, S.;
- Bharathi, P.
Publication type:
Article
Structure and Analgesic Activity of 13-(N-Aryl(N,N-Diethyl)Aminocarbonyl)-9-Methyl-11-Thioxo-8-Oxa-10,12-Diazatricyclo [7.3.1.02,7]Trideca-2,4,6-Trienes and Their 10-N-Phenyl Derivatives.
Published in:
Pharmaceutical Chemistry Journal, 2018, v. 52, n. 6, p. 515, doi. 10.1007/s11094-018-1851-0
By:
- Gein, V. L.;
- Zamaraeva, T. M.;
- Buzmakova, N. A.;
- Rudakova, I. P.;
- Dmitriev, M. V.
Publication type:
Article
Synthesis and Biological Activity of 6-(1,3-Benzoxazol-2-Yl)-5-Methylthieno-[2,3-d]Pyrimidines.
Published in:
Pharmaceutical Chemistry Journal, 2018, v. 52, n. 6, p. 510, doi. 10.1007/s11094-018-1850-1
By:
- Vlasov, S. V.;
- Kovalenko, S. N.;
- Osolodchenko, T. P.;
- Lenitskaya, E. B.;
- Chernykh, V. P.
Publication type:
Article
Synthesis and Antimicrobial Activity of 5-(Arylmethylidene)-2,4,6-Pyrimidine-2,4,6(1H,3H,5H)-Triones.
Published in:
Pharmaceutical Chemistry Journal, 2018, v. 52, n. 6, p. 506, doi. 10.1007/s11094-018-1849-7
By:
- Luzhnova, S. A.;
- Tyrkov, A. G.;
- Gabitova, N. M.;
- Yurtaeva, E. A.
Publication type:
Article
Structure-Activity (Antihypoxic) Relationship in a Series of Substituted Glyprolines.
Published in:
Pharmaceutical Chemistry Journal, 2018, v. 52, n. 6, p. 501, doi. 10.1007/s11094-018-1848-8
By:
- Kolyasnikova, K. N.;
- Kuznetsova, E. A.;
- Nikolaev, S. V.;
- Antipova, T. A.;
- Gudasheva, T. A.;
- Seredenin, S. B.
Publication type:
Article
Polymeric Complexes of Ofloxacin and Their Activity Against Tuberculosis Mycobacteria.
Published in:
Pharmaceutical Chemistry Journal, 2017, v. 51, n. 4, p. 250, doi. 10.1007/s11094-017-1592-5
By:
- Solovskii, M.;
- Borisenko, M.;
- Vlasova, E.;
- Tarabukina, E.;
- Zakharova, N.;
- Prazdnikova, T.
Publication type:
Article
Some Physicochemical Properties and Antifungal Activity of Cetylpyridinium Peroxodisulfate.
Published in:
Pharmaceutical Chemistry Journal, 2017, v. 51, n. 4, p. 254, doi. 10.1007/s11094-017-1593-4
By:
- Dovlatyan, A.;
- Kazaryan, P.;
- Arutyunyan, R.
Publication type:
Article
Synthesis, Immunomodulating and Antitumor Activities of Copolymers of Dialkylaminoethyl Methacrylates and Vinylsaccharides.
Published in:
Pharmaceutical Chemistry Journal, 2017, v. 51, n. 4, p. 245, doi. 10.1007/s11094-017-1591-6
By:
- Nazarova, O.;
- Potapenkova, L.;
- Stukov, A.;
- Zolotova, Yu.;
- Zhuravskaya, O.;
- Nekrasova, T.;
- Panarin, E.
Publication type:
Article
Synthesis, Hydrolysis, and Analgesic Activity of 3-[3-(1-arylethylcarbamoyl)-4-hydroxy-2-oxo-1,2-dihydroquinolin-1-yl]propanenitriles and Their Derivatives.
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 431, doi. 10.1007/s11094-016-1464-4
By:
- Ukrainets, I.;
- Taran, E.;
- Andreeva, K.
Publication type:
Article
Synthesis and Antimicrobial Activity of 5-(Heterylmethylene)Hexahydropyrimidin-2,4,6-Triones.
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 436, doi. 10.1007/s11094-016-1465-3
By:
- Tyrkov, A.;
- Sukhenko, L.;
- Yurtaeva, E.
Publication type:
Article
Synthesis and Hypotensive Activity of Novel Styryl Derivatives Based on Ethyl-4-(4-Methoxyphenyl)-2-Thioxo-1,2,3,4-Tetrahydropyrimidine-5-Carboxylate.
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 440, doi. 10.1007/s11094-016-1466-2
By:
- Fazylov, S.;
- Nurkenov, O.;
- Zhivotova, T.;
- Arinova, A.;
- Tolepbek, I.;
- Zhakupova, A.;
- Bakirova, R.;
- Muravleva, L.
Publication type:
Article
Synthesis, Antimicrobial and In Silico EGFR Inhibitory Activity Evaluation of Sulfonylamino Pyrrolidine Derivatives.
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 443, doi. 10.1007/s11094-016-1467-1
By:
- Kumar, B.;
- Prasad, A.;
- Reddy, P.;
- Ravindranath, L.
Publication type:
Article
Antimicrobial Activity of Dioxidine Against Strains of Potential Pathogens of Otorhinolarygological Infections.
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 465, doi. 10.1007/s11094-016-1470-6
By:
- Gus'kova, T.;
- Durnev, A.;
- Reikhart, D.;
- Chernyavtseva, A.
Publication type:
Article
Antiproliferative Activity of Niclosamide Against Melanoma and Colorectal Cancer Cells.
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 471, doi. 10.1007/s11094-016-1471-5
By:
- Zhirnik, A.;
- Semochkina, Yu.;
- Moskaleva, E.;
- Perevozchikova, V.;
- Rodina, A.;
- Severin, S.
Publication type:
Article
Use of Impedance Biotesting to Assess the Actions of Pharmaceutical Compounds on the Growth of Microorganisms.
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 481, doi. 10.1007/s11094-016-1473-3
By:
- Sibirtsev, V.;
- Naumov, I.;
- Kuprina, E.;
- Olekhnovich, R.
Publication type:
Article
Olivomycin A - an Antitumor Antibiotic of the Aureolic Acid Group (Review).
Published in:
Pharmaceutical Chemistry Journal, 2016, v. 50, n. 7, p. 425, doi. 10.1007/s11094-016-1463-5
By:
- Tevyashova, A.
Publication type:
Article
Interspecies Pharmacokinetics. 2. Analysis of the Structure of Interspecies Relationships Between Parameters of Drug Pharmacokinetics.
Published in:
Pharmaceutical Chemistry Journal, 2015, v. 48, n. 10, p. 635, doi. 10.1007/s11094-015-1162-7
By:
- Polekhina, O.;
- Obraztsov, N.;
- Petrunin, V.;
- Vysotskaya, T.
Publication type:
Article
Synthesis And Analgesic Activity Of 4-Aryl-2-Arylamino-4-OXO-2-Butenoic Acid Hetarylamides.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 11, doi. 10.1007/s11094-014-1034-6
By:
- Pulina, N.;
- Sobin, F.;
- Kozhukhar', V.;
- Makhmudov, R.;
- Rubtsov, A.;
- Naugol'nykh, E.
Publication type:
Article
Chemical Constituents, Antimicrobial Activity, Antioxidant and Total Phenolic Content in the Leaves of Thecocarpus Meifolious Boiss. Umbelliferae Herbs Growing Wild in Iran.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 44, doi. 10.1007/s11094-014-1043-5
By:
- Taherkhani, M.;
- Rustaiyan, A.;
- Rasouli, I.;
- Taherkhani, T.
Publication type:
Article
Synthesis and Antimicrobial Activity of Phenylthioand Benzylsulfonylacetic Acids Based on 2-amino-5-alkyl(arylalkyl)-1,3,4-thiadiazoles.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 20, doi. 10.1007/s11094-014-1037-3
By:
- Serkov, S.;
- Sigai, N.;
- Kostikova, N.;
- Bulatov, P.;
- Epishina, M.
Publication type:
Article
Synthesis, Toxicity, and Antituberculosis Activity of Isoniazid Derivatives Containing Sterically Hindered Phenols.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 5, doi. 10.1007/s11094-014-1032-8
By:
- Oludina, Yu.;
- Voloshina, A.;
- Kulik, M.;
- Zobov, V.;
- Bukharov, S.;
- Tagasheva, R.;
- Nugumanova, G.;
- Burilov, A.;
- Kravchenko, M.;
- Skornyakov, S.;
- Rusinov, G.
Publication type:
Article
Synthesis and Antimicrobial Activity of Anilines with 1,3,5-Cycloheptatriene and 5H-Dibenzo[ a, d]Annulene Fragments.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 22, doi. 10.1007/s11094-014-1038-2
By:
- Yunnikova, L.;
- Akent'eva, T.;
- Aleksandrova, G.;
- Mikhailova, L.;
- Eliseev, S.
Publication type:
Article
Antinociceptive Activity of Dimethyl 7-aryl-2-(2-rimino)-8-[(3-aryl)quinoxalin-2-yl]-9-oxo-1,6-dioxaspiro[4.4]non-3,7-diene-3,4-dicarboxylates.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 18, doi. 10.1007/s11094-014-1036-4
By:
- Lisovenko, N.;
- Dryakhlov, A.;
- Makhmudov, R.
Publication type:
Article
Synthesis of a New Class of Strongly Antibacterial Heterocyclic Compounds: 8-Bromo-6-alkyl-1-aryl-6 H-isoxazolo[4,3- E]indoles.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 34, doi. 10.1007/s11094-014-1041-7
By:
- Jajarmi, Maryam;
- Pordel, Mehdi;
- Allameh, Sadegh
Publication type:
Article
Synthesis and Local-Anesthetic Activity of New Arylpyruvic Acid Derivatives.
Published in:
Pharmaceutical Chemistry Journal, 2014, v. 48, n. 1, p. 8, doi. 10.1007/s11094-014-1033-7
By:
- Chernov, I.;
- Chashchina, S.;
- Igidov, N.;
- Syropyatov, B.
Publication type:
Article
Synthesis and Antimicrobial Activity of 2-Chloro(bromo)-(2-methyl)-3-arylpropionamides.
Published in:
Pharmaceutical Chemistry Journal, 2013, v. 47, n. 6, p. 307, doi. 10.1007/s11094-013-0949-7
By:
- Grishchuk, B.;
- Symchak, R.;
- Baranovskii, V.;
- Klimnyuk, S.;
- Pokryshko, E.
Publication type:
Article
Erratum to: Synthesis and characterization of polysulfanilamide and its copolymers: bioactivity and drug release.
Published in:
2012
By:
- Alsughayer, Abdulhakeem;
- Elassar, Abdel-Zaher;
- Sagheer, Fakhreia;
- Mustafa, Seham
Publication type:
Correction Notice
Synthesis and antimicrobial activity of 3-aryl-4,5,6,7-tetrahydroindazoles.
Published in:
Pharmaceutical Chemistry Journal, 2012, v. 46, n. 8, p. 470, doi. 10.1007/s11094-012-0827-8
By:
- Pantyukhin, A.;
- Mikhailovskii, A.;
- Aleksandrova, G.;
- Makhmudov, R.;
- Pershina, N.;
- Vakhrin, M.
Publication type:
Article
Anxiolytic activity of biologically active compounds from Filipendula vulgaris.
Published in:
Pharmaceutical Chemistry Journal, 2012, v. 46, n. 8, p. 492, doi. 10.1007/s11094-012-0832-y
By:
- Udut, V.;
- Vengerovskii, A.;
- Suslov, N.;
- Shilova, I.;
- Kaigorodtsev, A.;
- Polomeeva, N.;
- Dygai, A.
Publication type:
Article
Synthesis of Betulin Derivatives: N'{N-[3-OXO-20(29)-Lupen-28-OYL]-9-Aminononanoyl}3-Amino-3-Phenylpropionic Acid.
Published in:
Pharmaceutical Chemistry Journal, 2012, v. 46, n. 8, p. 473, doi. 10.1007/s11094-012-0828-7
By:
- Sysolyatin, S.;
- Surmachev, V.;
- Malykhin, V.;
- Kalashnikov, A.;
- Surmacheva, I.;
- Sonina, E.;
- Dubkov, A.;
- Tolstikov, G.;
- Shul'ts, E.;
- Salakhutdinov, N.;
- Dzhemilev, U.
Publication type:
Article
Antioxidant activity of polyphenols and polyphenol complex from the far-eastern tree Maackia amurensis.
Published in:
Pharmaceutical Chemistry Journal, 2012, v. 46, n. 8, p. 488, doi. 10.1007/s11094-012-0831-z
By:
- Utkina, N.;
- Kulesh, N.
Publication type:
Article