Works matching DE "CYCLOPROPYL compounds"

Results: 100

Synthesis and biological evaluation of novel cyclopropyl derivatives as subtype‐selective ligands for estrogen receptor.

Published in:

Journal of Pharmacy & Pharmacology, 2018, v. 70, n. 7, p. 910, doi. 10.1111/jphp.12908

By:

Wang, Zunyuan;
Yang, Yewei;
Zheng, Xiaoliang;
Zhang, Tao;
Huang, Wenhai;
Yan, Dongmei;
Zhang, Wenjun;
Wang, Xiaoju;
Shen, Zhengrong

Publication type:

Article

Chemodivergent assembly of ortho-functionalized phenols with tunable selectivity via rhodium(III)-catalyzed and solvent-controlled C-H activation.

Published in:

Communications Chemistry, 2021, v. 4, n. 1, p. 1, doi. 10.1038/s42004-021-00518-x

By:

Zhang, Haiman;
Lin, Shuang;
Gao, Hui;
Zhang, Kaixin;
Wang, Yi;
Zhou, Zhi;
Yi, Wei

Publication type:

Article

Crystal Structure, DFT Theoretical Study and Herbicidal Activity of Novel 1,2,4-Triazole Compound Containing Cyclopropyl Group.

Published in:

Journal of the Chemical Society of Pakistan, 2015, v. 37, n. 3, p. 567

By:

Guo-Xiang Sun;
Ming-Yan Yang;
Wen Zhao;
Zhao-Hui Sun;
Hong-Ke Wu

Publication type:

Article

Correction to: Pharmacological characterization of the LSD analog N-ethyl-N-cyclopropyl lysergamide (ECPLA).

Published in:

2019

By:

Halberstadt, Adam L.;
Klein, Landon M.;
Chatha, Muhammad;
Valenzuela, Laura B.;
Stratford, Alexander;
Wallach, Jason;
Nichols, David E.;
Brandt, Simon D.

Publication type:

Correction Notice

Pharmacological characterization of the LSD analog N-ethyl-N-cyclopropyl lysergamide (ECPLA).

Published in:

Psychopharmacology, 2019, v. 236, n. 2, p. 799, doi. 10.1007/s00213-018-5055-9

By:

Halberstadt, Adam L.;
Klein, Landon M.;
Chatha, Muhammad;
Valenzuela, Laura B.;
Stratford, Alexander;
Wallach, Jason;
Nichols, David E.;
Brandt, Simon D.

Publication type:

Article

In vitro and in vivo antiviral activity of a fluoronucleoside analog, NCC, against Coxsackie virus B3.

Published in:

Acta Virologica, 2021, v. 65, n. 1, p. 58, doi. 10.4149/av_2021_106

By:

Yafeng Wang;
Xiaokai Zhuan;
Youmei Peng;
Qing Li;
Chenzheng Huang;
He Huang;
Zongxian Liang;
Qingduan Wang;
Junbiao Chang

Publication type:

Article

Synthesis of (±)-terpendole E.

Published in:

Bioscience, Biotechnology & Biochemistry, 2015, v. 79, n. 1, p. 11, doi. 10.1080/09168451.2014.955455

By:

Takaaki Teranishi;
Tetsuro Murokawa;
Masaru Enomoto;
Shigefumi Kuwahara

Publication type:

Article

Targeting HIV-1 Reverse Transcriptase Using a Fragment-Based Approach.

Published in:

Molecules, 2023, v. 28, n. 7, p. 3103, doi. 10.3390/molecules28073103

By:

Mansouri, Mahta;
Rumrill, Shawn;
Dawson, Shane;
Johnson, Adam;
Pinson, Jo-Anne;
Gunzburg, Menachem J.;
Latham, Catherine F.;
Barlow, Nicholas;
Mbogo, George W.;
Ellenberg, Paula;
Headey, Stephen J.;
Sluis-Cremer, Nicolas;
Tyssen, David;
Bauman, Joseph D.;
Ruiz, Francesc X.;
Arnold, Eddy;
Chalmers, David K.;
Tachedjian, Gilda

Publication type:

Article

Sugar-Annulated Oxazoline Ligands: A Novel Pd(II) Complex and Its Application in Allylic Substitution.

Published in:

Molecules, 2016, v. 21, n. 12, p. 1704, doi. 10.3390/molecules21121704

By:

Kraft, Jochen;
Mill, Katharina;
Ziegler, Thomas

Publication type:

Article

Correlations between metabolism and structural elements of the alicyclic fentanyl analogs cyclopropyl fentanyl, cyclobutyl fentanyl, cyclopentyl fentanyl, cyclohexyl fentanyl and 2,2,3,3-tetramethylcyclopropyl fentanyl studied by human hepatocytes and LC-QTOF-MS

Published in:

Archives of Toxicology, 2019, v. 93, n. 1, p. 95, doi. 10.1007/s00204-018-2330-9

By:

Åstrand, Anna;
Töreskog, Amanda;
Watanabe, Shimpei;
Kronstrand, Robert;
Gréen, Henrik;
Vikingsson, Svante

Publication type:

Article

Formal synthesis of laurencione via MgBr-catalyzed rearrangement of α,ß-epoxy ketones to 1,2-diketones.

Published in:

Chemistry of Heterocyclic Compounds, 2013, v. 49, n. 5, p. 676, doi. 10.1007/s10593-013-1297-y

By:

Astashko, D.;
Habrus, Y.;
Yurevich, S.;
Tyvorskii, V.

Publication type:

Article

Synthesis of (2S)-4-Methyl- and (2S)-4-Methyl-6-oxo-3,6-dihydro-2H-pyran-2-carbaldehydes as Precursors to C22-C27 Fragments of Fijianolides and Their Synthetic Analogs.

Published in:

Russian Journal of Organic Chemistry, 2018, v. 54, n. 9, p. 1341, doi. 10.1134/S1070428018090130

By:

Mineeva, I. V.

Publication type:

Article

Reductive Heterocyclization of 2-Cyanobenzophenones by the Action of NaBH4. New Efficient Synthesis of 3-Arylphthalides.

Published in:

Russian Journal of Organic Chemistry, 2018, v. 54, n. 4, p. 568, doi. 10.1134/S1070428018040085

By:

Mochalov, S. S.;
Fedotov, A. N.;
Trofimova, E. V.;
Zefirov, N. S.

Publication type:

Article

Methyl (5 R)-5-hydroxy-3-methylidenedecanoate as a promising building block in asymmetric syntheses of bioactive natural compounds.

Published in:

Russian Journal of Organic Chemistry, 2013, v. 49, n. 7, p. 979, doi. 10.1134/S107042801307004X

By:

Mineeva, I.

Publication type:

Article

Efficient regioselective synthesis of 3-substituted 6,7-dihydro-5 H-pyrrolo[1,2- c][1,3]thiazol-4-ium bromides.

Published in:

Russian Journal of Organic Chemistry, 2012, v. 48, n. 1, p. 143, doi. 10.1134/S1070428012010241

By:

Dyachenko, V.

Publication type:

Article

Single atom changes in newly synthesized HIV protease inhibitors reveal structural basis for extreme affinity, high genetic barrier, and adaptation to the HIV protease plasticity.

Published in:

Scientific Reports, 2020, v. 10, n. 1, p. 1, doi. 10.1038/s41598-020-65993-z

By:

Bulut, Haydar;
Hattori, Shin-ichiro;
Aoki-Ogata, Hiromi;
Hayashi, Hironori;
Das, Debananda;
Aoki, Manabu;
Davis, David A.;
Rao, Kalapala Venkateswara;
Nyalapatla, Prasanth R.;
Ghosh, Arun K.;
Mitsuya, Hiroaki

Publication type:

Article

An Expedient Stereoselective Synthesis of Spirocyclopropyl Oxindoles from Indolin-2-One/ N-Protected Indolin-2-Ones and Bromonitroalkenes.

Published in:

Journal of the Chinese Chemical Society, 2013, v. 60, n. 6, p. 597, doi. 10.1002/jccs.201200557

By:

Roy, Suparna;
Chen, Kwunmin

Publication type:

Article

Metal-Porphyrin Orbital Interactions in Paramagnetic Iron Complexes Having Planar and Deformed Porphyrin Ring.

Published in:

Journal of the Chinese Chemical Society, 2013, v. 60, n. 1, p. 9, doi. 10.1002/jccs.201200474

By:

Nakamura, Mikio;
Ikezaki, Akira;
Takahashi, Masashi

Publication type:

Article

Trace Level Quantification of the ( — )2-(2-amino-5- chlorophenyl)-4-cyclopropyl-1,1,1-trifluoro-3-butyn- 2-ol Genotoxic Impurity in Efavirenz Drug Substance and Drug Product Using LC–MS/MS.

Published in:

Scientia Pharmaceutica, 2016, v. 84, n. 3, p. 456, doi. 10.3390/scipharm84030456

By:

Jaishetty, Nagadeep;
Palanisamy, Kamaraj;
Maruthapillai, Arthanareeswari;
Jaishetty, Rajamanohar

Publication type:

Article

Gold(III)‐Catalysed cis‐to‐trans Cyclopropyl Isomerization.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 25, p. 3317, doi. 10.1002/ejoc.201800419

By:

Reiersølmoen, Ann Christin;
Østrem, Elise;
Fiksdahl, Anne

Publication type:

Article

Potent Analogues of Abscisic Acid - Identifying Cyano-Cyclopropyl Moieties as Promising Replacements for the Cyclohexenone Headgroup.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 12, p. 1, doi. 10.1002/ejoc.201701769

By:

Frackenpohl, Jens;
Bojack, Guido;
Baltz, Rachel;
Bickers, Udo;
Busch, Marco;
Dittgen, Jan;
Franke, Jana;
Freigang, Jörg;
Grill, Erwin;
Gonzalez, Susana;
Helmke, Hendrik;
Hills, Martin J.;
Hohmann, Sabine;
von Koskull‐Döring, Pascal;
Kleemann, Jochen;
Lange, Gudrun;
Lehr, Stefan;
Schmutzler, Dirk;
Schulz, Arno;
Walther, Kerstin

Publication type:

Article

Direct Oxidation of Cyclopropanated Cyclooctanes as a Synthetic Approach to Polycyclic Cyclopropyl Ketones.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 7, p. 879, doi. 10.1002/ejoc.201701671

By:

Sedenkova, Kseniya N.;
Andriasov, Kristian S.;
Stepanova, Svetlana A.;
Gloriozov, Igor P.;
Grishin, Yuri K.;
Kuznetsova, Tamara S.;
Averina, Elena B.

Publication type:

Article

Stereoselective Synthesis of Stannylated Dehydropiperidines and Dehydroazepanes.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 30, p. 5146, doi. 10.1002/ejoc.201600903

By:

Lumbroso, Alexandre;
Coeffard, Vincent;
Gatineau, David;
Stecko, Sebastian;
Beaudet, Isabelle;
Quintard, Jean‐Paul;
Le Grognec, Erwan

Publication type:

Article

Total Synthesis of the Resveratrol Oligomers (±)-Ampelopsin B and (±)-ϵ-Viniferin.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 3, p. 426, doi. 10.1002/ejoc.201501486

By:

Lindgren, Anders E. G.;
Öberg, Christopher T.;
Hillgren, J. Mikael;
Elofsson, Mikael

Publication type:

Article

Total Synthesis of Solandelactones A and B.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 25, p. 5620, doi. 10.1002/ejoc.201500700

By:

Eichenauer, Nils C.;
Nordschild, Anja C. M.;
Bischop, Martina;
Schumacher, Dominik;
Mackwitz, Marcel K. W.;
Tschersich, Roxanne;
Wilhelm, Thorsten;
Pietruszka, Jörg

Publication type:

Article

A Unified Strategy for Kainoid Synthesis.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 22, p. 4823, doi. 10.1002/ejoc.201402452

By:

Fujii, Masaya;
Yokoshima, Satoshi;
Fukuyama, Tohru

Publication type:

Article

Male-Produced Sex Pheromone of the Stink Bug Edessa meditabunda.

Published in:

Journal of Chemical Ecology, 2012, v. 38, n. 7, p. 825, doi. 10.1007/s10886-012-0144-4

By:

Zarbin, Paulo;
Fávaro, Carla;
Vidal, Diogo;
Rodrigues, Mauro

Publication type:

Article

High Diastereoselectivity in the Yang Photocyclization via Remote Hydrogen Abstraction Reaction.

Published in:

Bulletin of the Korean Chemical Society, 2016, v. 37, n. 9, p. 1509, doi. 10.1002/bkcs.10900

By:

Jang, Mi;
Park, Bong Ser

Publication type:

Article

A DFT Study on the Reaction Mechanism of the Pd( II)-catalyzed Cycloisomerization of 4-Aza-1-cyclopropyl-1,6-enyne: A Solvent Effect.

Published in:

Bulletin of the Korean Chemical Society, 2016, v. 37, n. 6, p. 898, doi. 10.1002/bkcs.10799

By:

Park, Ji Eun;
Kang, Youn Kyung

Publication type:

Article

(R)-7-(Azepan-3-ylamino)-8-chloro-1-cyclopropyl-6-fluoro-4- oxo-1,4-dihydroquinoline-3-carboxylic Acid Hydrochloride.

Published in:

Molbank, 2013, v. 13, n. 2, p. 1, doi. 10.3390/M801

By:

Zhengjun Xia;
Zaixin Chen;
Shuitao Yu

Publication type:

Article

A Dft Investigation of the Interaction of B- And Al-Doped C60 Fullerenes with Cyclopropylpipezarine.

Published in:

Journal of Structural Chemistry, 2018, v. 59, n. 6, p. 1271, doi. 10.1134/S0022476618060045

By:

Bilge, M.

Publication type:

Article

DFT Mechanistic Investigation of the Gold(I)-Catalyzed Synthesis of Azepino[1,2- a]indoles.

Published in:

ChemCatChem, 2015, v. 7, n. 16, p. 2480, doi. 10.1002/cctc.201500429

By:

Giacinto, Pietro;
Cera, Gianpiero;
Bottoni, Andrea;
Bandini, Marco;
Miscione, Gian Pietro

Publication type:

Article

Iron-Catalyzed Synthesis of Cyclopropyl Halides.

Published in:

ChemCatChem, 2013, v. 5, n. 3, p. 706, doi. 10.1002/cctc.201200740

By:

Grupe, Sabine;
Jacobi von Wangelin, Axel

Publication type:

Article

The (+)- cis- and (+)- trans-Olibanic Acids: Key Odorants of Frankincense.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 44, p. 13719, doi. 10.1002/anie.201605242

By:

Cerutti-Delasalle, Céline;
Mehiri, Mohamed;
Cagliero, Cecilia;
Rubiolo, Patrizia;
Bicchi, Carlo;
Meierhenrich, Uwe J.;
Baldovini, Nicolas

Publication type:

Article

Asymmetric Ring Opening/Cyclization/Retro-Mannich Reaction of Cyclopropyl Ketones with Aryl 1,2-Diamines for the Synthesis of Benzimidazole Derivatives.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 40, p. 12228, doi. 10.1002/anie.201604735

By:

Xia, Yong;
Lin, Lili;
Chang, Fenzhen;
Liao, Yuting;
Liu, Xiaohua;
Feng, Xiaoming

Publication type:

Article

Rhodium-Catalyzed Enantioselective Silylation of Cyclopropyl C−H Bonds.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 30, p. 8723, doi. 10.1002/anie.201603153

By:

Lee, Taegyo;
Hartwig, John F.

Publication type:

Article

Temporary Generation of a Cyclopropyl Oxocarbenium Ion Enables Highly Diastereoselective Donor-Acceptor Cyclopropane Cycloaddition.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 23, p. 6780, doi. 10.1002/anie.201601340

By:

Sabbatani, Juliette;
Maulide, Nuno

Publication type:

Article

Tandem Allylboration-Prins Reaction for the Rapid Construction of Substituted Tetrahydropyrans: Application to the Total Synthesis of (−)-Clavosolide A.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 7, p. 2498, doi. 10.1002/anie.201511140

By:

Millán, Alba;
Smith, James R.;
Chen, Jack L.-Y.;
Aggarwal, Varinder K.

Publication type:

Article

Brook Rearrangement as a Trigger for the Ring Opening of Strained Carbocycles.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 2, p. 714, doi. 10.1002/anie.201510094

By:

Zhang, Fa‐Guang;
Eppe, Guillaume;
Marek, Ilan

Publication type:

Article

Asymmetric Ring-Opening of Cyclopropyl Ketones with Thiol, Alcohol, and Carboxylic Acid Nucleophiles Catalyzed by a Chiral N, N′-Dioxide-Scandium(III) Complex.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 46, p. 13748, doi. 10.1002/anie.201506909

By:

Xia, Yong;
Lin, Lili;
Chang, Fenzhen;
Fu, Xuan;
Liu, Xiaohua;
Feng, Xiaoming

Publication type:

Article

Palladium-Catalyzed Direct Cyclopropylation of Heterocycles.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 33, p. 9601, doi. 10.1002/anie.201504735

By:

Wu, Xiaojin;
Lei, Chuanhu;
Yue, Guizhou;
Zhou, Jianrong (Steve)

Publication type:

Article

Synthesis and Characterization of a Gold Vinylidene Complex Lacking π-Conjugated Heteroatoms.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 23, p. 6867, doi. 10.1002/anie.201501474

By:

Harris, Robert J.;
Widenhoefer, Ross A.

Publication type:

Article

Synthesis of Cyclopropyl-Substituted Furans by Brønsted Acid Promoted Cascade Reactions.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 19, p. 5744, doi. 10.1002/anie.201500625

By:

Clark, J. Stephen;
Romiti, Filippo;
Hogg, Kirsten F.;
Hamid, Malai Haniti S. A.;
Richter, Sven C.;
Boyer, Alistair;
Redman, Joanna C.;
Farrugia, Louis J.

Publication type:

Article

Discovery and Reconstitution of the Cycloclavine Biosynthetic Pathway-Enzymatic Formation of a Cyclopropyl Group.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 17, p. 5117, doi. 10.1002/anie.201410002

By:

Jakubczyk, Dorota;
Caputi, Lorenzo;
Hatsch, Anaëlle;
Nielsen, Curt A. F.;
Diefenbacher, Melanie;
Klein, Jens;
Molt, Andrea;
Schröder, Hartwig;
Cheng, Johnathan Z.;
Naesby, Michael;
O'Connor, Sarah E.

Publication type:

Article

Total Synthesis of (−)-Lundurine A and Determination of its Absolute Configuration.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 7, p. 2228, doi. 10.1002/anie.201409963

By:

Jin, Shuaijiang;
Gong, Jing;
Qin, Yong

Publication type:

Article

Stereodivergent Synthesis of Arylcyclopropylamines by Sequential CH Borylation and Suzuki-Miyaura Coupling.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 3, p. 846, doi. 10.1002/anie.201409186

By:

Miyamura, Shin;
Araki, Misaho;
Suzuki, Takayoshi;
Yamaguchi, Junichiro;
Itami, Kenichiro

Publication type:

Article

Gold-Catalyzed C(sp3)H/C(sp)H Coupling/Cyclization/Oxidative Alkynylation Sequence: A Powerful Strategy for the Synthesis of 3-Alkynyl Polysubstituted Furans.

Published in:

Angewandte Chemie International Edition, 2014, v. 53, n. 30, p. 7870, doi. 10.1002/anie.201402475

By:

Ma, Yuanhong;
Zhang, Shuai;
Yang, Shiping;
Song, Feijie;
You, Jingsong

Publication type:

Article

4-Cyclopropyl-1-(1-methyl-4-nitro-1 H-imidazol-5-yl)-1 H-1,2,3-triazole and Ethyl 1-(1-methyl-4-nitro-1 H-imidazol-5-yl)-1 H-1,2,3-triazole-4-carboxylate.

Published in:

Journal of Chemical Crystallography, 2016, v. 46, n. 6/7, p. 296, doi. 10.1007/s10870-016-0659-6

By:

Boechat, Núbia;
Carvalho, Alcione;
Quaresma, Bruna;
Wardell, James;
Wardell, Solange

Publication type:

Article

Crystal structure of catena-poly-[(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-ium-1-yl)-1,4-dihydroquinoline-3-carboxylate- κ2 O, O′)-(μ2-4,4′-sulfonyldibenzoato- κ4 O, O′: O′′, O′′′)zinc(II)] hemihydrate, C31H27ZnFN3O9.5S

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 4, p. 1203, doi. 10.1515/ncrs-2016-0132

By:

Fan, Zhuo-Wen;
Wang, Liang-Liang;
Meng, Ying;
Cui, Kuo;
Liu, Ji-Zhi

Publication type:

Article

Design, Synthesis, Biological Evaluation, and Docking Studies of ( S)-Phenylalanine Derivatives with a 2-Cyanopyrrolidine Moiety as Potent Dipeptidyl Peptidase 4 Inhibitors.

Published in:

Chemical Biology & Drug Design, 2013, v. 82, n. 2, p. 140, doi. 10.1111/cbdd.12139

By:

Liu, Yang;
Wu, Yizhe;
Wu, Haoshu;
Tang, Li;
Wu, Peng;
Liu, Tao;
Hu, Yongzhou

Publication type:

Article