Works matching DE "CARBONIC anhydrase inhibitors"

Results: 682

Topiramate induces acute intracellular acidification in glioblastoma.

Published in:

Journal of Neuro-Oncology, 2016, v. 130, n. 3, p. 465, doi. 10.1007/s11060-016-2258-y

By:

Marathe, Kamini;
McVicar, Nevin;
Li, Alex;
Bellyou, Miranda;
Meakin, Susan;
Bartha, Robert

Publication type:

Article

An Original Aspirin-Containing Carbonic Anhydrase 9 Inhibitor Overcomes Hypoxia-Induced Drug Resistance to Enhance the Efficacy of Myocardial Protection.

Published in:

Cardiovascular Drugs & Therapy, 2022, v. 36, n. 4, p. 605, doi. 10.1007/s10557-021-07182-2

By:

Zhou, Wen;
Zhang, Bin;
Fan, Keyu;
Yin, Xiaojian;
Liu, Jinfeng;
Gou, Shaohua

Publication type:

Article

An Update on Synthesis of Coumarin Sulfonamides as Enzyme Inhibitors and Anticancer Agents.

Published in:

Molecules, 2022, v. 27, n. 5, p. 1604, doi. 10.3390/molecules27051604

By:

Rubab, Laila;
Afroz, Sumbal;
Ahmad, Sajjad;
Hussain, Saddam;
Nawaz, Iram;
Irfan, Ali;
Batool, Fozia;
Kotwica-Mojzych, Katarzyna;
Mojzych, Mariusz

Publication type:

Article

Design, Synthesis and Molecular Docking Study of Novel 3-Phenyl-β-Alanine-Based Oxadiazole Analogues as Potent Carbonic Anhydrase II Inhibitors.

Published in:

Molecules, 2022, v. 27, n. 3, p. 816, doi. 10.3390/molecules27030816

By:

Rafiq, Kashif;
Ur Rehman, Najeeb;
Halim, Sobia Ahsan;
Khan, Majid;
Khan, Ajmal;
Al-Harrasi, Ahmed

Publication type:

Article

Carbonic Anhydrase Inhibitors and Epilepsy: State of the Art and Future Perspectives.

Published in:

Molecules, 2021, v. 26, n. 21, p. 6380, doi. 10.3390/molecules26216380

By:

Ciccone, Lidia;
Cerri, Chiara;
Nencetti, Susanna;
Orlandini, Elisabetta

Publication type:

Article

The Glitazone Class of Drugs as Carbonic Anhydrase Inhibitors—A Spin-Off Discovery from Fragment Screening.

Published in:

Molecules, 2021, v. 26, n. 10, p. 3010, doi. 10.3390/molecules26103010

By:

Mueller, Sarah L.;
Chrysanthopoulos, Panagiotis K.;
Halili, Maria A.;
Hepburn, Caryn;
Nebl, Tom;
Supuran, Claudiu T.;
Nocentini, Alessio;
Peat, Thomas S.;
Poulsen, Sally-Ann;
Alfonso-Prieto, Mercedes

Publication type:

Article

Development and Validation of High-Throughput Bioanalytical Liquid Chromatography-Tandem Mass Spectrometry (LC-MS/MS) Method for the Quantification of Newly Synthesized Antitumor Carbonic Anhydrase Inhibitors in Human Plasma.

Published in:

Molecules, 2020, v. 25, n. 23, p. 5753, doi. 10.3390/molecules25235753

By:

Abdel-Megied, Ahmed M.;
Eldehna, Wagdy M.;
Abdelrahman, Mohamed A.;
Elbarbry, Fawzy A.;
Petruczynik, Anna;
Tuzimski, Tomasz

Publication type:

Article

Hypoxia-Activated Prodrug Derivatives of Carbonic Anhydrase Inhibitors in Benzenesulfonamide Series: Synthesis and Biological Evaluation.

Published in:

Molecules, 2020, v. 25, n. 10, p. 2347, doi. 10.3390/molecules25102347

By:

Anduran, Emilie;
Aspatwar, Ashok;
Parvathaneni, Nanda-Kumar;
Suylen, Dennis;
Bua, Silvia;
Nocentini, Alessio;
Parkkila, Seppo;
Supuran, Claudiu T.;
Dubois, Ludwig;
Lambin, Philippe;
Winum, Jean-Yves;
Carta, Fabrizio;
Angeli, Andrea

Publication type:

Article

Dual P-Glycoprotein and CA XII Inhibitors: A New Strategy to Reverse the P-gp Mediated Multidrug Resistance (MDR) in Cancer Cells †.

Published in:

Molecules, 2020, v. 25, n. 7, p. 1748, doi. 10.3390/molecules25071748

By:

Teodori, Elisabetta;
Braconi, Laura;
Bua, Silvia;
Lapucci, Andrea;
Bartolucci, Gianluca;
Manetti, Dina;
Romanelli, Maria Novella;
Dei, Silvia;
Supuran, Claudiu T.;
Coronnello, Marcella;
Ferreira, Maria José Umbelino

Publication type:

Article

Cloning, Characterization and Anion Inhibition Studies of a β-Carbonic Anhydrase from the Pathogenic Protozoan Entamoeba histolytica.

Published in:

Molecules, 2018, v. 23, n. 12, p. 3112, doi. 10.3390/molecules23123112

By:

Haapanen, Susanna;
Bua, Silvia;
Kuuslahti, Marianne;
Parkkila, Seppo;
Supuran, Claudiu T.

Publication type:

Article

Potent and Selective Carboxylic Acid Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII.

Published in:

Molecules, 2018, v. 23, n. 1, p. 17, doi. 10.3390/molecules23010017

By:

Cau, Ylenia;
Vullo, Daniela;
Mori, Mattia;
Dreassi, Elena;
Supuran, Claudiu T.;
Botta, Maurizio

Publication type:

Article

Novel Sulfamide-Containing Compounds as Selective Carbonic Anhydrase I Inhibitors.

Published in:

Molecules, 2017, v. 22, n. 7, p. 1049, doi. 10.3390/molecules22071049

By:

Berrino, Emanuela;
Bua, Silvia;
Mori, Mattia;
Botta, Maurizio;
Murthy, Vallabhaneni S.;
Vijayakumar, Vijayaparthasarathi;
Tamboli, Yasinalli;
Bartolucci, Gianluca;
Mugelli, Alessandro;
Cerbai, Elisabetta;
Supuran, Claudiu T.;
Carta, Fabrizio

Publication type:

Article

Phenols and Polyphenols as Carbonic Anhydrase Inhibitors.

Published in:

Molecules, 2016, v. 21, n. 12, p. 1649, doi. 10.3390/molecules21121649

By:

Karioti, Anastasia;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Nitric Oxide Donors and Selective Carbonic Anhydrase Inhibitors: A Dual Pharmacological Approach for the Treatment of Glaucoma, Cancer and Osteoporosis.

Published in:

Molecules, 2015, v. 20, n. 4, p. 5667, doi. 10.3390/molecules20045667

By:

Carradori, Simone;
Mollica, Adriano;
De Monte, Celeste;
Granese, Arianna;
Supuran, Claudiu T.

Publication type:

Article

4-Amino-substituted Benzenesulfonamides as Inhibitors of Human Carbonic Anhydrases.

Published in:

Molecules, 2014, v. 19, n. 11, p. 17356, doi. 10.3390/molecules191117356

By:

Rutkauskas, Kęstutis;
Zubrienė, Asta;
Tumosienė, Ingrida;
Kantminienė, Kristina;
Kažemėkaitė, Marytė;
Smirnov, Alexey;
Kazokaitė, Justina;
Morkūnaitė, Vaida;
Čapkauskaitė, Edita;
Manakova, Elena;
Gražulis, Saulius;
Beresnevičius, Zigmuntas J.;
Matulis, Daumantas

Publication type:

Article

Utilization of Physiologically based Biopharmaceutical Modelling and Simulations for Proposed Dissolution Specifications of Acetazolamide ER Capsules 500 mg.

Published in:

Frontiers in Health Informatics, 2024, v. 13, n. 8, p. 5453

By:

Kadam, Pramod V.;
Lakshmi, K.

Publication type:

Article

Closure of Full-Thickness Macular Holes Associated with Macular Edema with Medical Therapy.

Published in:

Ophthalmologica, 2022, v. 245, n. 2, p. 179, doi. 10.1159/000516018

By:

Kokame, Gregg T.;
Johnson, Mark W.;
Lim, Jennifer;
Flynn, Harry W.;
de Carlo, Talisa;
Yannuzzi, Nicolas;
Ryan, Edwin H.;
Omizo, Jase N.;
Sridhar, Jayanth;
Staropoli, Patrick;
Goldhagen, Brian;
Lian, Rebecca

Publication type:

Article

Dilatation of Retinal Arterioles Induced by Topical Dorzolamide for One Week Is Impaired in Patients with Type 1 Diabetes and Mild Retinopathy.

Published in:

Ophthalmologica, 2020, v. 243, n. 3, p. 236, doi. 10.1159/000504178

By:

Tilma, Kathrine Kleis;
Bek, Toke

Publication type:

Article

Facile synthesis of aminobiphenyl sulfonamides via Chan–Lam coupling and their biological evaluation as potent carbonic anhydrase inhibitors.

Published in:

Scientific Reports, 2025, v. 15, n. 1, p. 1, doi. 10.1038/s41598-025-10048-4

By:

Sharif, Moniba;
Mahmood, Abid;
Kanwal, Aqsa;
Ahmad, Matloob;
Rasool, Nasir;
Qamar, Muhammad Usman;
Mughram, Mohammed H. AL;
Al-Harethi, Amira Ali Mohammed;
Shah, Tawaf Ali;
Shaikh, Imran Ibrahim

Publication type:

Article

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 10, p. 412, doi. 10.3390/metabo10100412

By:

Angeli, Andrea;
Carta, Fabrizio;
Nocentini, Alessio;
Winum, Jean-Yves;
Zalubovskis, Raivis;
Akdemir, Atilla;
Onnis, Valentina;
Eldehna, Wagdy M.;
Capasso, Clemente;
Simone, Giuseppina De;
Monti, Simona Maria;
Carradori, Simone;
Donald, William A.;
Dedhar, Shoukat;
Supuran, Claudiu T.

Publication type:

Article

Design, Synthesis, and Biological Evaluation of 1,2,3-Triazole-linked triazino[5,6-b]indole-benzene sulfonamide Conjugates as Potent Carbonic Anhydrase I, II, IX, and XIII Inhibitors.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 5, p. 200, doi. 10.3390/metabo10050200

By:

Chinchilli, Krishna Kartheek;
Angeli, Andrea;
Thacker, Pavitra S.;
Korra, Laxman Naik;
Biswas, Rashmita;
Arifuddin, Mohammed;
Supuran, Claudiu T.

Publication type:

Article

Synthesis and Biological Evaluation of Imidazo[2,1-b]Thiazole based Sulfonyl Piperazines as Novel Carbonic Anhydrase II Inhibitors.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 4, p. 136, doi. 10.3390/metabo10040136

By:

Manasa, Kesari Lakshmi;
Pujitha, Sravya;
Sethi, Aaftaab;
Arifuddin, Mohammed;
Alvala, Mallika;
Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors.

Published in:

Metabolites (2218-1989), 2018, v. 8, n. 2, p. 37, doi. 10.3390/metabo8020037

By:

Abdoli, Morteza;
Bozdag, Murat;
Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Amino Acids as Building Blocks for Carbonic Anhydrase Inhibitors.

Published in:

Metabolites (2218-1989), 2018, v. 8, n. 2, p. 36, doi. 10.3390/metabo8020036

By:

Chiaramonte, Niccolò;
Romanelli, Maria Novella;
Teodori, Elisabetta;
Supuran, Claudiu T.

Publication type:

Article

Carbonic Anhydrases: Role in pH Control and Cancer.

Published in:

Metabolites (2218-1989), 2018, v. 8, n. 1, p. 19, doi. 10.3390/metabo8010019

By:

Mboge, Mam Y.;
Mahon, Brian P.;
McKenna, Robert;
Frost, Susan C.

Publication type:

Article

Carbonic Anhydrase Inhibition and the Management of Hypoxic Tumors.

Published in:

Metabolites (2218-1989), 2017, v. 7, n. 3, p. 48, doi. 10.3390/metabo7030048

By:

Supuran, Claudiu T.

Publication type:

Article

Bilateral Choroidal Detachment Following Pseudophakic Cystoid Macular Edema Treatment with Oral Acetazolamide.

Published in:

2025

By:

Kudasiewicz-Kardaszewska, Agnieszka;
Ozimek, Małgorzata;
Urbański, Tomasz;
Cisiecki, Sławomir

Publication type:

Case Study

Comparative efficacy of selenoureido carbonic anhydrase inhibitors and azole antifungal drugs against clinical isolates of Malassezia pachydermatis.

Published in:

Veterinary Dermatology, 2025, v. 36, n. 3, p. 302, doi. 10.1111/vde.13336

By:

Spadini, Costanza;
Mezzasalma, Nicolò;
Odigie, Amienwanlen Eugene;
Angeli, Andrea;
Carta, Fabrizio;
Selleri, Silvia;
Gandolfo, Emanuele;
Taddei, Simone;
Franceschi, Valentina;
Minesso, Sergio;
Supuran, Claudiu T.;
Cabassi, Clotilde Silvia

Publication type:

Article

Intrinsic thermodynamics of high affinity inhibitor binding to recombinant human carbonic anhydrase IV.

Published in:

European Biophysics Journal, 2018, v. 47, n. 3, p. 271, doi. 10.1007/s00249-017-1256-0

By:

Mickevičiūtė, Aurelija;
Timm, David D.;
Gedgaudas, Marius;
Linkuvienė, Vaida;
Chen, Zhiwei;
Waheed, Abdul;
Michailovienė, Vilma;
Zubrienė, Asta;
Smirnov, Alexey;
Čapkauskaitė, Edita;
Baranauskienė, Lina;
Jachno, Jelena;
Revuckienė, Jurgita;
Manakova, Elena;
Gražulis, Saulius;
Matulienė, Jurgita;
Di Cera, Enrico;
Sly, William S.;
Matulis, Daumantas

Publication type:

Article

Severe Vaso-Occlusive and Ocular Decompression Retinopathy Revealing a Sickle Cell Trait in a Patient with Herpetic Uveitis.

Published in:

2024

By:

Toutain, Jonathan;
Fares, Selim;
Cochereau, Isabelle;
Gargouri, Mohamed Ali;
Titah, Chérif

Publication type:

Case Study

The Effectiveness of Pharmacological Agents for the Treatment of Uveitic Macular Edema (UMO): A Systematic Review.

Published in:

2019

By:

Tallouzi, Mohammad O.;
Moore, David J.;
Barry, Robert J.;
Calvert, Melanie;
Mathers, Jonathan;
Murray, Philip I.;
Denniston, Alastair K.

Publication type:

journal article

A Retrospective Study of Transcleral Cyclophotocoagulation Using the Slow Coagulation Technique for the Treatment of Refractory Glaucoma.

Published in:

2019

By:

Fong, Yoly Yeuk Ying;
Wong, Billy Kwok Tung;
Li, Felix Chi Hong;
Young, Alvin Lerrmann

Publication type:

journal article

Management of Cystoid Macular Edema in Retinitis Pigmentosa.

Published in:

2017

By:

Huckfeldt, Rachel M.;
Comander, Jason

Publication type:

journal article

Carbonic anhydrase 2 inhibits epithelial-mesenchymal transition and metastasis in hepatocellular carcinoma.

Published in:

Carcinogenesis, 2018, v. 39, n. 4, p. 562, doi. 10.1093/carcin/bgx148

By:

Chenyue Zhang;
Haiyong Wang;
Zhiao Chen;
Liping Zhuang;
Litao Xu;
Zhouyu Ning;
Zhenfeng Zhu;
Peng Wang;
Zhiqiang Meng

Publication type:

Article

Rho-Associated Kinase Inhibitors: Evolving Strategies in Glaucoma Treatment.

Published in:

Drugs, 2019, v. 79, n. 10, p. 1031, doi. 10.1007/s40265-019-01130-z

By:

Schehlein, Emily M.;
Robin, Alan L.

Publication type:

Article

DEVELOPMENT AND VALIDATION OF ANALYTICAL METHOD FOR SIMULTANEOUS ESTIMATION OF BRINZOLAMIDE AND TIMOLOL BY HPLC FROM OPHTHALMIC PREPARATION.

Published in:

International Journal of Pharmacy & Life Sciences, 2014, v. 5, n. 3, p. 1001, doi. 10.13040/IJPSR.0975-8232.5(3).1001-07

By:

Khatun, Rahima;
Islam, S. M. Ashraful

Publication type:

Article

Management of obesity and cardiometabolic risk - role of phentermine/extended release topiramate.

Published in:

Diabetes, Metabolic Syndrome & Obesity: Targets & Therapy, 2014, v. 7, p. 35, doi. 10.2147/DMSO.S38979

By:

Sweeting, Arianne N.;
Tabet, Eddy;
Caterson, Ian D.;
Markovic, Tania P.

Publication type:

Article

Novel pyrazole-3,4-dicarboxamides bearing biologically active sulfonamide moiety as potential carbonic anhydrase inhibitors.

Published in:

Arabian Journal of Chemistry, 2019, v. 12, n. 8, p. 2740, doi. 10.1016/j.arabjc.2015.05.020

By:

Mert, Samet;
Alım, Zuhal;
İşgör, Mehmet Mustafa;
Anıl, Barış;
Kasımoğulları, Rahmi;
Beydemir, Şükrü

Publication type:

Article

Prescribing trends of glaucoma drugs in six major cities of China from 2013 to 2017.

Published in:

PLoS ONE, 2020, v. 15, n. 1, p. 1, doi. 10.1371/journal.pone.0227595

By:

Yu, Lingyan;
Ding, Kai;
Luo, Lifang;
Yu, Zhenwei

Publication type:

Article

Oculohypotensive effects of various acetozolamide nanopreparations for topical treatment of animal model-induced glaucoma and their impact on optic nerve.

Published in:

PLoS ONE, 2019, v. 14, n. 2, p. 1, doi. 10.1371/journal.pone.0212588

By:

Mahmoud, Sherif S.;
ElAbrak, Eman S.;
Aly, Mervat A.;
Ali, Eman M.

Publication type:

Article

Reverse-phase LC method development and validation for the quantification of acetazolamide and its specified and unspecified degradation products in hard gelatin capsule formulations.

Published in:

Journal of the Iranian Chemical Society, 2022, v. 19, n. 3, p. 775, doi. 10.1007/s13738-021-02341-6

By:

Chinta, Srinivasa Reddy;
Paidikondala, Kalyani;
Katari, Naresh Kumar;
Dongala, Thirupathi;
Ediga, Sasikiran Goud;
Marisetti, Vishnu Murthy

Publication type:

Article

Carbonic Anhydrase Inhibitors Featuring a Porphyrin Scaffold: Synthesis, Optical and Biological Properties.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 21, p. 1, doi. 10.1002/ejoc.202101538

By:

Merabti, Amina;
Roger, Maxime;
Nguyen, Christophe;
Nocentini, Alessio;
Gerbier, Philippe;
Richeter, Sébastien;
Gary‐Bobo, Magali;
Supuran, Claudiu T.;
Clément, Sébastien;
Winum, Jean‐Yves

Publication type:

Article

Adipocyte proteome and secretome influence inflammatory and hormone pathways in glioma.

Published in:

Metabolic Brain Disease, 2019, v. 34, n. 1, p. 141, doi. 10.1007/s11011-018-0327-y

By:

Almeida, J.;
Costa, J.;
Coelho, P.;
Cea, V.;
Galesio, M.;
Noronha, J. P.;
Diniz, M. S.;
Prudêncio, C.;
Soares, R.;
Sala, C.;
Fernandes, Rúben

Publication type:

Article

Potential Anti-carcinogenic Effect of Acetazolamide, a Carbonic Anhydrase Enzyme Inhibitor, in Diethylnitrosamine - Induced Hepatocarcinogenesis in Rats.

Published in:

QJM: An International Journal of Medicine, 2021, v. 114, p. i210, doi. 10.1093/qjmed/hcab100.141

By:

Sayed, Moataz Mohamed;
Soliman, Mohamed Lotfy;
Tamim, Yomna Mohamed;
Osman, Ahmed H.;
Abdul-Rasheed Hussain, Muhammad Saleh

Publication type:

Article

Evidence for Bicarbonate Secretion by Ameloblasts in a Novel Cellular Model.

Published in:

2016

By:

Bori, E.;
Guo, J.;
Rácz, R.;
Burghardt, B.;
Földes, A.;
Kerémi, B.;
Harada, H.;
Steward, M. C.;
Den Besten, P.;
Bronckers, A. L. J. J.;
Varga, G.

Publication type:

journal article

A family of amphiphilic dioxidovanadium(V) hydrazone complexes as potent carbonic anhydrase inhibitors along with anti-diabetic and cytotoxic activities.

Published in:

BioMetals, 2022, v. 35, n. 3, p. 499, doi. 10.1007/s10534-022-00384-7

By:

Ghosh, Chiranjit;
Patra, Debashis;
Bala, Niranjan;
Majumder, Indira;
Sepay, Nayim;
Mukhopadhyay, Prabuddha;
Das, Sukhen;
Kundu, Rita;
Drew, Michael G. B.;
León, Armando Rafael;
Ghosh, Tapas;
Pradhan, Manik

Publication type:

Article

Synthesis of new series of thiazol‐(2(3H)‐ylideneamino)benzenesulfonamide derivatives as carbonic anhydrase inhibitors.

Published in:

Journal of Biochemical & Molecular Toxicology, 2020, v. 34, n. 12, p. 1, doi. 10.1002/jbt.22596

By:

Berber, Nurcan;
Arslan, Mustafa;
Vural, Fırat;
Ergun, Adem;
Gençer, Nahit;
Arslan, Oktay

Publication type:

Article

Native mass spectrometry of human carbonic anhydrase I and its inhibitor complexes.

Published in:

Journal of Biological Inorganic Chemistry (JBIC), 2020, v. 25, n. 7, p. 979, doi. 10.1007/s00775-020-01818-8

By:

Zoppi, Carlotta;
Nocentini, Alessio;
Supuran, Claudiu T.;
Pratesi, Alessandro;
Messori, Luigi

Publication type:

Article

In Vitro CO-Releasing and Antioxidant Properties of Sulfonamide-Based CAI-CORMs in a H 2 O 2 -Stimulated Human Achilles Tendon-Derived Cell Model.

Published in:

Molecules, 2025, v. 30, n. 3, p. 593, doi. 10.3390/molecules30030593

By:

Berrino, Emanuela;
Guglielmi, Paolo;
Carta, Fabrizio;
Carradori, Simone;
Campestre, Cristina;
Angeli, Andrea;
Arrighi, Francesca;
Pontecorvi, Virginia;
Chimenti, Paola;
Secci, Daniela;
Supuran, Claudiu T.;
Gallorini, Marialucia

Publication type:

Article

Privileged Scaffold Hybridization in the Design of Carbonic Anhydrase Inhibitors.

Published in:

Molecules, 2024, v. 29, n. 18, p. 4444, doi. 10.3390/molecules29184444

By:

Secci, Daniela;
Sanna, Erica;
Distinto, Simona;
Onali, Alessia;
Lupia, Antonio;
Demuru, Laura;
Atzeni, Giulia;
Meleddu, Rita;
Cottiglia, Filippo;
Angeli, Andrea;
Supuran, Claudiu T.;
Maccioni, Elias

Publication type:

Article