Works matching DE "CALCIUM channel inhibition"

Results: 39

The Use of Calcium Channel Blockers in the Treatment of Coronary Spasm and Atrioventricular Block.

Published in:

Cell Biochemistry & Biophysics, 2015, v. 72, n. 2, p. 527, doi. 10.1007/s12013-014-0498-z

By:

Gao, Bo;
Zhang, Zhenjian;
Qian, Jin;
Cao, Chuanbin;
Hua, Xianping;
Chu, Mengting;
HE, Xingwei;
Zeng, Hesong

Publication type:

Article

Serotonin Regulates the Firing of Principal Cells of the Subiculum by Inhibiting a T-type Ca2+ Current.

Published in:

Frontiers in Cellular Neuroscience, 2017, v. 11, p. 1, doi. 10.3389/fncel.2017.00060

By:

Petersen, Anders V.;
Jensen, Camilla S.;
Crépel, Valérie;
Falkerslev, Mathias;
Perrier, Jean-François

Publication type:

Article

Pharmacological effects of purple basil extract on isolated mouse bladder functions and underlying molecular mechanisms.

Published in:

Research Results in Pharmacology, 2024, v. 10, n. 4, p. 113, doi. 10.18413/rrpharmacology.10.507

By:

Arslan, Beyza N.;
Dondas, Naciye Y.

Publication type:

Article

Optimization of TRPV6 Calcium Channel Inhibitors Using a 3D Ligand-Based Virtual Screening Method.

Published in:

Angewandte Chemie International Edition, 2015, v. 54, n. 49, p. 14748, doi. 10.1002/anie.201507320

By:

Simonin, Céline;
Awale, Mahendra;
Brand, Michael;
van Deursen, Ruud;
Schwartz, Julian;
Fine, Michael;
Kovacs, Gergely;
Häfliger, Pascal;
Gyimesi, Gergely;
Sithampari, Abilashan;
Charles, Roch‐Philippe;
Hediger, Matthias A.;
Reymond, Jean‐Louis

Publication type:

Article

Neuroanatomy of pain-deficiency and cross-modal activation in calcium channel subunit (CACN) α2δ3 knockout mice.

Published in:

Brain Structure & Function, 2018, v. 223, n. 1, p. 111, doi. 10.1007/s00429-017-1473-4

By:

Landmann, Julia;
Richter, Franziska;
Oros-Peusquens, Ana-Maria;
Shah, N. Jon;
Classen, Joseph;
Neely, G. Gregory;
Richter, Angelika;
Penninger, Josef M.;
Bechmann, Ingo

Publication type:

Article

Brain-Derived Neurotrophic Factor Inhibits Calcium Channel Activation, Exocytosis, and Endocytosis at a Central Nerve Terminal.

Published in:

Journal of Neuroscience, 2015, v. 35, n. 11, p. 4676, doi. 10.1523/JNEUROSCI.2695-14.2015

By:

Baydyuk, Maryna;
Xin-Sheng Wu;
Liming He;
Ling-Gang Wu

Publication type:

Article

Inhibition of A-Type Potassium Current by the Peptide Toxin SNX-482.

Published in:

Journal of Neuroscience, 2014, v. 34, n. 28, p. 9182, doi. 10.1523/JNEUROSCI.0339-14.2014

By:

Kimm, Tilia;
Bean, Bruce P.

Publication type:

Article

Presynaptic Calcium Channel Inhibition Underlies CB1 Cannabinoid Receptor-Mediated Suppression of GABA Release.

Published in:

Journal of Neuroscience, 2014, v. 34, n. 23, p. 7958, doi. 10.1523/JNEUROSCI.0247-14.2014

By:

Szabó, Gergely G.;
Lenkey, Nora;
Holderith, Noemi;
Andrási, Tibor;
Nusser, Zoltan;
Hájos, Norbert

Publication type:

Article

Heme oxygenase-1 regulates cell proliferation via carbon monoxide-mediated inhibition of T-type Ca channels.

Published in:

Pflügers Archiv: European Journal of Physiology, 2015, v. 467, n. 2, p. 415, doi. 10.1007/s00424-014-1503-5

By:

Duckles, Hayley;
Boycott, Hannah;
Al-Owais, Moza;
Elies, Jacobo;
Johnson, Emily;
Dallas, Mark;
Porter, Karen;
Giuntini, Francesca;
Boyle, John;
Scragg, Jason;
Peers, Chris

Publication type:

Article

Tetrodotoxin blocks L-type Ca channels in canine ventricular cardiomyocytes.

Published in:

Pflügers Archiv: European Journal of Physiology, 2012, v. 464, n. 2, p. 167, doi. 10.1007/s00424-012-1114-y

By:

Hegyi, Bence;
Bárándi, László;
Komáromi, István;
Papp, Ferenc;
Horváth, Balázs;
Magyar, János;
Bányász, Tamás;
Krasznai, Zoltán;
Szentandrássy, Norbert;
Nánási, Péter

Publication type:

Article

Cocaine inhibits store-operated Ca2+ entry in brain microvascular endothelial cells: critical role for sigma-1 receptors.

Published in:

Biochemical Journal, 2016, v. 473, n. 1, p. 1, doi. 10.1042/BJ20150934

By:

Brailoiu, G. Cristina;
Deliu, Elena;
Console-Bram, Linda M.;
Soboloff, Jonathan;
Abood, Mary E.;
Unterwald, Ellen M.;
Brailoiu, Eugen

Publication type:

Article

Pharmacological evaluation and validation for the folkloric use of Oligochaeta ramose in constipation and diarrhea.

Published in:

Bangladesh Journal of Pharmacology, 2014, v. 9, n. 4, p. 617, doi. 10.3329/bjp.v9i4.20566

By:

Hussain, Musaddique;
Raza, Shahid Masood;
Janbaz, Khalid Hussain

Publication type:

Article

Functional nature of the spasmolytic effect, phytochemical composition and acute toxicity studies on Sauromatum guttatum.

Published in:

Bangladesh Journal of Pharmacology, 2014, v. 9, n. 2, p. 203, doi. 10.3329/bjp.v9i2.18602

By:

Shah, Nabi;
Shah, Abdul Jabbar;
Ahmed, Manzoor;
Gilani, Anwarul Hassan

Publication type:

Article

Antimicrobial, antioxidant and calcium channel blocking activities of Amberboa divaricata.

Published in:

Bangladesh Journal of Pharmacology, 2014, v. 9, n. 1, p. 29, doi. 10.3329/bjp.v9i1.16989

By:

Iqbal, Shahid Muhammad;
Mushtaq, Aamir;
Jabeen, Qaiser

Publication type:

Article

N-type calcium channel blockade: a new approach to preventing sudden cardiac death?

Published in:

Cardiovascular Research, 2014, v. 104, n. 1, p. 1, doi. 10.1093/cvr/cvu197

By:

Nattel, Stanley

Publication type:

Article

Regulation of BMP2-induced intracellular calcium increases in osteoblasts.

Published in:

Journal of Orthopaedic Research, 2016, v. 34, n. 10, p. 1725, doi. 10.1002/jor.23196

By:

Xu, Wenfeng;
Liu, Bo;
Liu, Xue;
Chiang, Martin Y. M.;
Li, Bo;
Xu, Zichen;
Liao, Xiaoling

Publication type:

Article

Inhibition of N-Type Calcium Channels by Fluorophenoxyanilide Derivatives.

Published in:

Marine Drugs, 2015, v. 13, n. 4, p. 2030, doi. 10.3390/md13042030

By:

Gleeson, Ellen C.;
Graham, Janease E.;
Spiller, Sandro;
Vetter, Irina;
Lewis, Richard J.;
Duggan, Peter J.;
Tuck, Kellie L.

Publication type:

Article

ω-Conotoxin GVIA Mimetics that Bind and Inhibit Neuronal Cav2.2 Ion Channels.

Published in:

Marine Drugs, 2012, v. 10, n. 10, p. 2349, doi. 10.3390/md10102349

By:

Tranberg, Charlotte Elisabet;
Yang, Aijun;
Vetter, Irina;
McArthur, Jeffrey R.;
Baell, Jonathan B.;
Lewis, Richard J.;
Tuck, Kellie L.;
Duggan, Peter J.

Publication type:

Article

An Automated Electrophysiological Assay for Differentiating CaV2.2 Inhibitors Based on State Dependence and Kinetics.

Published in:

Assay & Drug Development Technologies, 2012, v. 10, n. 6, p. 542, doi. 10.1089/adt.2011.437

By:

Swensen, Andrew M.;
Niforatos, Wende;
Vortherms, Timothy A.;
Perner, Richard J.;
Li, Tao;
Schrimpf, Michael R.;
Scott, Victoria E.;
Lee, Lance;
Jarvis, Michael F.;
McGaraughty, Steve

Publication type:

Article

Calcium channel antagonist and beta-blocker overdose: antidotes and adjunct therapies.

Published in:

British Journal of Clinical Pharmacology, 2016, v. 81, n. 3, p. 453, doi. 10.1111/bcp.12763

By:

Graudins, Andis;
Lee, Hwee Min;
Druda, Dino

Publication type:

Article

Preparation and preclinical evaluation of 68Ga‑DOTA‑amlodipine for L‑type calcium channel imaging.

Published in:

Indian Journal of Nuclear Medicine, 2016, v. 31, n. 4, p. 267, doi. 10.4103/0972-3919.190797

By:

Firuzyar, Tahereh;
Shafiee‑Ardestani, Mahdi;
Khalaj, Ali;
Jalilian, Amir Reza;
Aboudzadeh, Mohammad Reza;
Sadeghpour, Hossein

Publication type:

Article

Prolonged mydriasis after inadvertent topical administration of the calcium channel antagonist amlodipine: implications for glaucoma drug development.

Published in:

Cutaneous & Ocular Toxicology, 2015, v. 34, n. 1, p. 84, doi. 10.3109/15569527.2014.896016

By:

Roos, Jonathan C. P.;
Haridas, Anjana S.

Publication type:

Article

The effect of intrathecal administration of the neuronal N-type calcium channels antagonist, ω -conotoxin MVIIA, on attenuating the spontaneous and naloxone-precipitated morphine withdrawal in rats.

Published in:

Toxin Reviews, 2016, v. 35, n. 1/2, p. 33, doi. 10.1080/15569543.2016.1181657

By:

Bozorgi, Hooman;
Jahanian-Najafabadi, Ali;
Rabbani, Mohammed

Publication type:

Article

Genetic risk between the CACNA1I gene and schizophrenia in Chinese Uygur population.

Published in:

Hereditas, 2017, p. 1, doi. 10.1186/s41065-017-0037-1

By:

Wei Xu;
Lin He;
Yongyong Shi;
Yahui Liu;
Qingli Guo;
Ke Liu;
Zujia Wen;
Zhaowei Zhou;
Zhijian Song;
Juan Zhou;
Jianhua Chen;
Qizhong Yi

Publication type:

Article

Sigma1 receptors inhibit store-operated Ca2+ entry by attenuating coupling of STIM1 to Orai1.

Published in:

Journal of Cell Biology, 2016, v. 213, n. 1, p. 65, doi. 10.1083/jcb.201506022

By:

Srivats, Shyam;
Balasuriya, Dilshan;
Pasche, Mathias;
Vistal, Gerard;
Edwardson, J. Michael;
Taylor, Colin W.;
Murrell-Lagnado, Ruth D.

Publication type:

Article

Natural regulatory T cells are resistant to calcium release-activated calcium (CRAC/ORAI) channel inhibition.

Published in:

International Immunology, 2013, v. 25, n. 9, p. 497, doi. 10.1093/intimm/dxt013

By:

Jin, Shu;
Chin, Jayne;
Kitson, Christopher;
Woods, John;
Majmudar, Rupal;
Carvajal, Valerie;
Allard, John;
DeMartino, Julie;
Narula, Satwant;
Thomas-Karyat, Dori A.

Publication type:

Article

Plant Calcium-Permeable Channels.

Published in:

Plant Physiology, 2013, v. 163, n. 2, p. 514, doi. 10.1104/pp.113.220855

By:

Swarbreck, Stéphanie M.;
Colaço, Renato;
Davies, Julia M.

Publication type:

Article

Bufalin, a bufanolide steroid from the parotoid glands of the Chinese toad, inhibits L-type Ca2+ channels and contractility in rat ventricular myocytes.

Published in:

Fundamental & Clinical Pharmacology, 2017, v. 31, n. 3, p. 340, doi. 10.1111/fcp.12265

By:

Song, Tao;
Chu, Xi;
Zhang, Xuan;
Song, Qiongtao;
Zhang, Ying;
Zhang, Yuanyuan;
Han, Xue;
Zhang, Jianping;
Chu, Li

Publication type:

Article

Successful catheter ablation of symptomatic premature ventricular contractions originating from mitral annulus.

Published in:

2012

By:

Uz, Ömer;
Kiliçaslan, Fethi;
Tezcan, Mehmet

Publication type:

Case Study

Erratum for "Protective effect of quercetin on bupivacaine-induced neurotoxicity via T-type calcium channel inhibition".

Published in:: 2017
Publication type:: Correction Notice

Inhibition of Voltage-Gated Calcium Channels as Common Mode of Action for (Mixtures of) Distinct Classes of Insecticides.

Published in:

Toxicological Sciences, 2014, v. 141, n. 1, p. 103, doi. 10.1093/toxsci/kfu110

By:

Meijer, Marieke;
Dingemans, Milou M.L.;
van den Berg, Martin;
Westerink, Remco H.S.

Publication type:

Article

Synthesis and biological evaluation of pyrrolidine-based T-type calcium channel inhibitors for the treatment of neuropathic pain.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1460, doi. 10.1080/14756366.2018.1513926

By:

Yang, Hak Kyun;
Son, Woo Seung;
Lim, Keon Seung;
Kim, Gun Hee;
Lim, Eun Jeong;
Gadhe, Changdev G.;
Lee, Jae Yeol;
Jeong, Kyu-Sung;
Lim, Sang Min;
Pae, Ae Nim

Publication type:

Article

Synthesis and evaluation of 5,6-disubstituted thiopyrimidine aryl aminothiazoles as inhibitors of the calcium-activated chloride channel TMEM16A/Ano1.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1362, doi. 10.3109/14756366.2015.1135912

By:

Piechowicz, Katarzyna A.;
Truong, Eric C.;
Javed, Kashif M.;
Chaney, Rachelle R.;
Wu, Johnny Y.;
Phuan, Puay W.;
Verkman, Alan S.;
Anderson, Marc O.

Publication type:

Article

Arterial hypertension, a tricky side of Parkinson's disease: physiopathology and therapeutic features.

Published in:

Neurological Sciences, 2013, v. 34, n. 5, p. 621, doi. 10.1007/s10072-012-1251-2

By:

Mazza, Alberto;
Ravenni, Roberta;
Antonini, Angelo;
Casiglia, Edoardo;
Rubello, Domenico;
Pauletto, Paolo

Publication type:

Article

Angiotensin II signalling kicks out p27Kip1: casein kinase 2 augmentation of Cav1.2 L-type Ca2+ channel activity in immature ventricular cardiomyocytes.

Published in:

Journal of Physiology, 2017, v. 595, n. 13, p. 4131, doi. 10.1113/JP274260

By:

Horne, Mary C.;
Hell, Johannes W.

Publication type:

Article

Diltiazem prevents stress-induced contractile deficits in cardiomyocytes, but does not reverse the cardiomyopathy phenotype in Mybpc3-knock-in mice.

Published in:

Journal of Physiology, 2017, v. 595, n. 12, p. 3987, doi. 10.1113/JP273769

By:

Flenner, Frederik;
Geertz, Birgit;
Reischmann‐Düsener, Silke;
Weinberger, Florian;
Eschenhagen, Thomas;
Carrier, Lucie;
Friedrich, Felix W.

Publication type:

Article

The Effects of Amlodipine Administration and In Vitro Addition of Pentoxifylline on Sperm Parameters in Mice.

Published in:

Medical Journal of Tabriz University of Medical Sciences & Health Services, 2012, v. 33, n. 6, p. 16

By:

Oskouei, Behnaz Sadeghzadeh;
Ghanbar, Ahmad Ali;
Roshangar, Leila;
Khaki, Amir Afshin;
Rad, Jafar Soleimani

Publication type:

Article

Protein kinase D regulates the human cardiac L-type voltage-gated calcium channel through serine 1884

Published in:

FEBS Letters, 2011, v. 585, n. 24, p. 3903, doi. 10.1016/j.febslet.2011.11.011

By:

Aita, Yusuke;
Kurebayashi, Nagomi;
Hirose, Shigehisa;
Maturana, Andrés D.

Publication type:

Article

Resolving the Reversed Rate Effect of Calcium Channel Blockers on Human-Induced Pluripotent Stem Cell-Derived Cardiomyocytes and the Impact on In Vitro Cardiac Safety Evaluation.

Published in:

Toxicological Sciences, 2019, v. 167, n. 2, p. 573, doi. 10.1093/toxsci/kfy264

By:

Zeng, Haoyu;
Wang, Jixin;
Clouse, Holly;
Lagrutta, Armando;
Sannajust, Frederick

Publication type:

Article

Works matching DE "CALCIUM channel inhibition"

The Use of Calcium Channel Blockers in the Treatment of Coronary Spasm and Atrioventricular Block.

Serotonin Regulates the Firing of Principal Cells of the Subiculum by Inhibiting a T-type Ca<sup>2+</sup> Current.

Pharmacological effects of purple basil extract on isolated mouse bladder functions and underlying molecular mechanisms.

Optimization of TRPV6 Calcium Channel Inhibitors Using a 3D Ligand-Based Virtual Screening Method.

Neuroanatomy of pain-deficiency and cross-modal activation in calcium channel subunit (CACN) α2δ3 knockout mice.

Brain-Derived Neurotrophic Factor Inhibits Calcium Channel Activation, Exocytosis, and Endocytosis at a Central Nerve Terminal.

Inhibition of A-Type Potassium Current by the Peptide Toxin SNX-482.

Presynaptic Calcium Channel Inhibition Underlies CB<sub>1</sub> Cannabinoid Receptor-Mediated Suppression of GABA Release.

Heme oxygenase-1 regulates cell proliferation via carbon monoxide-mediated inhibition of T-type Ca channels.

Tetrodotoxin blocks L-type Ca channels in canine ventricular cardiomyocytes.

Cocaine inhibits store-operated Ca<sup>2+</sup> entry in brain microvascular endothelial cells: critical role for sigma-1 receptors.

Pharmacological evaluation and validation for the folkloric use of Oligochaeta ramose in constipation and diarrhea.

Functional nature of the spasmolytic effect, phytochemical composition and acute toxicity studies on Sauromatum guttatum.

Antimicrobial, antioxidant and calcium channel blocking activities of Amberboa divaricata.

N-type calcium channel blockade: a new approach to preventing sudden cardiac death?

Regulation of BMP2-induced intracellular calcium increases in osteoblasts.

Inhibition of N-Type Calcium Channels by Fluorophenoxyanilide Derivatives.

ω-Conotoxin GVIA Mimetics that Bind and Inhibit Neuronal Cav2.2 Ion Channels.

An Automated Electrophysiological Assay for Differentiating Ca<sub>V</sub>2.2 Inhibitors Based on State Dependence and Kinetics.

Calcium channel antagonist and beta-blocker overdose: antidotes and adjunct therapies.

Preparation and preclinical evaluation of <sup>68</sup>Ga‑DOTA‑amlodipine for L‑type calcium channel imaging.

Prolonged mydriasis after inadvertent topical administration of the calcium channel antagonist amlodipine: implications for glaucoma drug development.

The effect of intrathecal administration of the neuronal N-type calcium channels antagonist, ω -conotoxin MVIIA, on attenuating the spontaneous and naloxone-precipitated morphine withdrawal in rats.

Genetic risk between the CACNA1I gene and schizophrenia in Chinese Uygur population.

Sigma1 receptors inhibit store-operated Ca<sup>2+</sup> entry by attenuating coupling of STIM1 to Orai1.

Natural regulatory T cells are resistant to calcium release-activated calcium (CRAC/ORAI) channel inhibition.

Plant Calcium-Permeable Channels.

Bufalin, a bufanolide steroid from the parotoid glands of the Chinese toad, inhibits L-type Ca<sup>2+</sup> channels and contractility in rat ventricular myocytes.

Successful catheter ablation of symptomatic premature ventricular contractions originating from mitral annulus.

Erratum for "Protective effect of quercetin on bupivacaine-induced neurotoxicity via T-type calcium channel inhibition".

Inhibition of Voltage-Gated Calcium Channels as Common Mode of Action for (Mixtures of) Distinct Classes of Insecticides.

Synthesis and biological evaluation of pyrrolidine-based T-type calcium channel inhibitors for the treatment of neuropathic pain.

Synthesis and evaluation of 5,6-disubstituted thiopyrimidine aryl aminothiazoles as inhibitors of the calcium-activated chloride channel TMEM16A/Ano1.

Arterial hypertension, a tricky side of Parkinson's disease: physiopathology and therapeutic features.

Angiotensin II signalling kicks out p27<sup>Kip1</sup>: casein kinase 2 augmentation of Ca<sub>v</sub>1.2 L-type Ca<sup>2+</sup> channel activity in immature ventricular cardiomyocytes.

Diltiazem prevents stress-induced contractile deficits in cardiomyocytes, but does not reverse the cardiomyopathy phenotype in Mybpc3-knock-in mice.

The Effects of Amlodipine Administration and In Vitro Addition of Pentoxifylline on Sperm Parameters in Mice.

Protein kinase D regulates the human cardiac L-type voltage-gated calcium channel through serine 1884

Resolving the Reversed Rate Effect of Calcium Channel Blockers on Human-Induced Pluripotent Stem Cell-Derived Cardiomyocytes and the Impact on In Vitro Cardiac Safety Evaluation.