Works matching DE "BROMODOMAIN-containing proteins"


Results: 268
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    Unveiling New Triazoloquinoxaline‐Based PROTACs Designed for the Selective Degradation of the ncBAF Chromatin Remodeling Subunit BRD9.

    Published in:
    Chemistry - A European Journal, 2025, v. 31, n. 34, p. 1, doi. 10.1002/chem.202404218
    By:
    • Pierri, Martina;
    • Bove, Guglielmo;
    • Gazzillo, Erica;
    • Colarusso, Ester;
    • Scala, Francesca;
    • Pepe, Giacomo;
    • Terracciano, Stefania;
    • Chini, Maria Giovanna;
    • Simonelli, Nicla;
    • Bruno, Ines;
    • Nebbioso, Angela;
    • Campiglia, Pietro;
    • Bifulco, Giuseppe;
    • Altucci, Lucia;
    • Del Gaudio, Nunzio;
    • Lauro, Gianluigi
    Publication type:
    Article
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    Development of novel cellular histone-binding and chromatin-displacement assays for bromodomain drug discovery.

    Published in:
    Epigenetics & Chromatin, 2015, v. 8, n. 1, p. 1, doi. 10.1186/s13072-015-0026-4
    By:
    • Zhan, Yanai;
    • Kost-Alimova, Maria;
    • Xi Shi;
    • Leo, Elisabetta;
    • Bardenhagen, Jennifer P.;
    • Shepard, Hannah E.;
    • Appikonda, Srikanth;
    • Vangamudi, Bhavatarini;
    • Zhao, Shuping;
    • Tieu, Trang N.;
    • Jiang, Shiming;
    • Heffernan, Timothy P.;
    • Marszalek, Joseph R.;
    • Toniatti, Carlo;
    • Draetta, Giulio;
    • Tyler, Jessica;
    • Barton, Michelle;
    • Jones, Philip;
    • Palmer, Wylie S.;
    • Geck Do, Mary K.
    Publication type:
    Article
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    Development of novel cellular histone-binding and chromatin-displacement assays for bromodomain drug discovery.

    Published in:
    Epigenetics & Chromatin, 2015, v. 8, n. 1, p. 1, doi. 10.1186/s13072-015-0026-4
    By:
    • Zhan, Yanai;
    • Kost-Alimova, Maria;
    • Xi Shi;
    • Leo, Elisabetta;
    • Bardenhagen, Jennifer P.;
    • Shepard, Hannah E.;
    • Appikonda, Srikanth;
    • Vangamudi, Bhavatarini;
    • Shuping Zhao;
    • Tieu, Trang N.;
    • Shiming Jiang;
    • Heffernan, Timothy P.;
    • Marszalek, Joseph R.;
    • Toniatti, Carlo;
    • Draetta, Giulio;
    • Tyler, Jessica;
    • Barton, Michelle;
    • Jones, Philip;
    • Palmer, Wylie S.;
    • Geck Do, Mary K.
    Publication type:
    Article
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    Inhibition of bromodomain and extra-terminal (BET) proteins increases NKG2D ligand MICA expression and sensitivity to NK cell-mediated cytotoxicity in multiple myeloma cells: role of cMYC-IRF4-miR-125b interplay.

    Published in:
    Journal of Hematology & Oncology, 2016, v. 9, p. 1, doi. 10.1186/s13045-016-0362-2
    By:
    • Abruzzese, Maria Pia;
    • Bilotta, Maria Teresa;
    • Fionda, Cinzia;
    • Zingoni, Alessandra;
    • Soriani, Alessandra;
    • Vulpis, Elisabetta;
    • Borrelli, Cristiana;
    • Zitti, Beatrice;
    • Petrucci, Maria Teresa;
    • Ricciardi, Maria Rosaria;
    • Molfetta, Rosa;
    • Paolini, Rossella;
    • Santoni, Angela;
    • Cippitelli, Marco
    Publication type:
    Article
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    BRD4: an effective target for organ fibrosis.

    Published in:
    Biomarker Research, 2024, v. 12, n. 1, p. 1, doi. 10.1186/s40364-024-00641-6
    By:
    • Wei, Qun;
    • Gan, Cailing;
    • Sun, Meng;
    • Xie, Yuting;
    • Liu, Hongyao;
    • Xue, Taixiong;
    • Deng, Conghui;
    • Mo, Chunheng;
    • Ye, Tinghong
    Publication type:
    Article
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