Works matching DE "BENZENESULFONAMIDES"
Results: 249
Antiparkinsonian activity of selective MAO-B inhibitors of different chemical structures.
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- Research Results in Pharmacology, 2024, v. 10, n. 4, p. 129, doi. 10.18413/rrpharmacology.10.540
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- Article
A Further Decrease in the Catalyst Loading for the Palladium-Catalyzed Direct Intramolecular Arylation of Amides and Sulfonamides.
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- 2015
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- Publication type:
- Other
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201407
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- Article
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2188147
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- Article
Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2185762
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- Article
Diversely N-substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N-nitrosulfonamides.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2178430
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- Article
Dependence on linkers' flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 2765, doi. 10.1080/14756366.2022.2130285
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- Article
Benzenesulfonamides with different rigidity-conferring linkers as carbonic anhydrase inhibitors: an insight into the antiproliferative effect on glioblastoma, pancreatic, and breast cancer cells.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1857, doi. 10.1080/14756366.2022.2091557
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- Article
4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 994, doi. 10.1080/14756366.2022.2055553
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- Article
4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1568, doi. 10.1080/14756366.2022.2080816
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- Article
Investigation of pesticides on honey bee carbonic anhydrase inhibition.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1923, doi. 10.1080/14756366.2020.1835885
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- Article
Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamides as carbonic anhydrase isoforms I and II inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1457, doi. 10.1080/14756366.2019.1652282
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- Article
Appraisal of anti-protozoan activity of nitroaromatic benzenesulfonamides inhibiting carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1164, doi. 10.1080/14756366.2019.1626375
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- Article
Carbonic anhydrase inhibition with a series of novel benzenesulfonamide-triazole conjugates.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1565, doi. 10.1080/14756366.2018.1513927
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- Article
Synthesis, carbonic anhydrase I and II inhibition studies of the 1,3,5-trisubstituted-pyrazolines.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 189, doi. 10.1080/14756366.2016.1244533
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- Article
Designing, synthesis and bioactivities of 4-[3-(4-hydroxyphenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]benzenesulfonamides.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 169, doi. 10.1080/14756366.2016.1243536
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- Article
3D QSAR studies, pharmacophore modeling, and virtual screening of diarylpyrazole–benzenesulfonamide derivatives as a template to obtain new inhibitors, using human carbonic anhydrase II as a model protein.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 688, doi. 10.1080/14756366.2016.1241781
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- Article
Selective inhibition of human carbonic anhydrase IX in Xenopus oocytes and MDA-MB-231 breast cancer cells.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 38, doi. 10.1080/14756366.2016.1217854
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- Article
Study of reactivity of cyanoacetohydrazonoethyl- N -ethyl- N -methyl benzenesulfonamide: preparation of novel anticancer and antimicrobial active heterocyclic benzenesulfonamide derivatives and their molecular docking against dihydrofolate reductase.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 7, doi. 10.1080/14756366.2016.1217851
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- Article
Synthesis and bioactivity studies on new 4-(3-(4-Substitutedphenyl)-3a,4-dihydro-3 H -indeno[1,2-c]pyrazol-2-yl) benzenesulfonamides.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1619, doi. 10.3109/14756366.2016.1160077
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- Article
Design, synthesis and biological evaluation of N -(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 174, doi. 10.1080/14756366.2016.1197221
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- Article
Synthesis and carbonic anhydrase inhibitory activities of new thienyl-substituted pyrazoline benzenesulfonamides.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 1, doi. 10.1080/14756366.2016.1181627
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- Article
Synthesis of 4-(2-substituted hydrazinyl)benzenesulfonamides and their carbonic anhydrase inhibitory effects.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 4, p. 568, doi. 10.3109/14756366.2015.1047359
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- Article
Synthesis and inhibition potency of novel ureido benzenesulfonamides incorporating GABA as tumor-associated carbonic anhydrase IX and XII inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 2, p. 205, doi. 10.3109/14756366.2015.1014477
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- Article
Fluorinated pyrrolidines and piperidines incorporating tertiary benzenesulfonamide moieties are selective carbonic anhydrase II inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 5, p. 737, doi. 10.3109/14756366.2014.963072
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- Article
Exploring QSARs of some benzenesulfonamides incorporating cyanoacrylamide moieties as a carbonic anhydrase inhibitors (specifically against tumor-associated isoforms IX and XII).
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 4, p. 519, doi. 10.3109/14756366.2014.948435
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- Article
Carbonic Anhydrase Isoenzymes I and II Inhibition Potentials of Leiotulus dasyanthus (K. Koch) Pimenov&Ostr. and Ferulago pauciradiata Boiss.&Heldr. (Apiaceae).
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- Bezmialem Science, 2021, v. 9, n. 2, p. 153, doi. 10.14235/bas.galenos.2020.4127
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- Article
Recent insights about pyrrolidine core skeletons in pharmacology.
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- Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1239658
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- Article
Carbonic anhydrase inhibition by antiviral drugs in vitro and in silico.
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- Journal of Molecular Recognition, 2023, v. 36, n. 12, p. 1, doi. 10.1002/jmr.3063
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- Article
Investigation of the effects of some pesticides on carbonic anhydrase isoenzymes.
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- Journal of Molecular Recognition, 2023, v. 36, n. 9, p. 1, doi. 10.1002/jmr.3048
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- Article
Biological activity and molecular docking studies of some N‐phenylsulfonamides against cholinesterases and carbonic anhydrase isoenzymes.
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- Journal of Molecular Recognition, 2022, v. 35, n. 10, p. 1, doi. 10.1002/jmr.2982
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- Article
Synthesis of Azasugar-Sulfonamide conjugates and their Evaluation as Inhibitors of Carbonic Anhydrases: the Azasugar Approach to Selectivity.
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- Language & Linguistics Compass, 2021, v. 15, n. 5, p. 2604, doi. 10.1002/ejoc.202100250
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- Article
Isolation and identification of a novel sildenafil analogue adulterant in herbal products.
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- Food Additives & Contaminants. Part A: Chemistry, Analysis, Control, Exposure & Risk Assessment, 2017, v. 34, n. 3, p. 330, doi. 10.1080/19440049.2016.1272137
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- Article
Synthesis, docking study and biological evaluation of some new thiourea derivatives bearing benzenesulfonamide moiety.
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- Chemistry Central Journal, 2017, v. 11, n. 1, p. 1, doi. 10.1186/s13065-017-0271-7
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- Article
Design, synthesis and anticancer activity of some novel thioureido-benzenesulfonamides incorporated biologically active moieties.
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- Chemistry Central Journal, 2016, v. 10, n. 1, p. 1, doi. 10.1186/s13065-016-0161-4
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- Article
Novel chloroquinoline derivatives incorporating biologically active benzenesulfonamide moiety: synthesis, cytotoxic activity and molecular docking.
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- Chemistry Central Journal, 2016, v. 10, n. 1, p. 1, doi. 10.1186/s13065-016-0164-1
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- Article
Disposable screen printed sensor for the electrochemical detection of methamphetamine in undiluted saliva.
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- Chemistry Central Journal, 2016, v. 10, n. 1, p. 1, doi. 10.1186/s13065-016-0147-2
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- Article
Thiazide and other Cl-benzenesulfonamide-bearing clinical drug affinities for human carbonic anhydrases.
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- PLoS ONE, 2021, v. 16, n. 6, p. 1, doi. 10.1371/journal.pone.0253608
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- Article
Co-detection of isoprenaline and paracetamol in biological and pharmaceutical media by a feather-like La3+/ZnO nano-flowers and N-(ferrocenylmethylidene)fluoren-2-amine-modified carbon paste electrode: analysis of a novel sensor.
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- Journal of the Iranian Chemical Society, 2020, v. 17, n. 6, p. 1447, doi. 10.1007/s13738-020-01870-w
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- Article
Synthesis, characterization, lipoxygenase inhibitory activity and in silico molecular docking of biaryl bis(benzenesulfonamide) and indol-3-yl-hydrazide derivatives.
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- Journal of the Iranian Chemical Society, 2015, v. 12, n. 6, p. 1123, doi. 10.1007/s13738-014-0573-9
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- Article
Expedient synthesis of novel coumarin-based sulfonamides.
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- Journal of the Iranian Chemical Society, 2015, v. 12, n. 3, p. 379, doi. 10.1007/s13738-014-0494-7
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- Publication type:
- Article
Synthesis of Azasugar-Sulfonamide conjugates and their Evaluation as Inhibitors of Carbonic Anhydrases: the Azasugar Approach to Selectivity.
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- European Journal of Organic Chemistry, 2021, v. 2021, n. 18, p. 2604, doi. 10.1002/ejoc.202100250
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- Article
Iron‐Catalyzed Electrophilic Amination of Sodium Sulfinates with Anthranils.
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- European Journal of Organic Chemistry, 2021, v. 2021, n. 9, p. 1466, doi. 10.1002/ejoc.202100010
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- Article
Synthesis of Tetrahydroquinoline-Embedded Bridged Benzothiaoxazepine-1,1-dioxides.
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- European Journal of Organic Chemistry, 2017, v. 2017, n. 45, p. 6671, doi. 10.1002/ejoc.201701152
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- Article
LSN2424100: a novel, potent orexin-2 receptor antagonist with selectivity over orexin-1 receptors and activity in an animal model predictive of antidepressant-like efficacy.
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- Frontiers in Neuroscience, 2014, v. 8, p. 1, doi. 10.3389/fnins.2014.00005
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- Article
The crystal structure of ((E)-2,4-dibromo-6-(((5-(nitro)-2-oxidophenyl)imino)methyl)phenolato-κ<sup>3</sup>N,O,O′)tris(pyridine-κN)manganese(II), C<sub>28</sub>H<sub>21</sub>Br<sub>2</sub>MnN<sub>5</sub>O<sub>4</sub>.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2023, v. 238, n. 1, p. 27, doi. 10.1515/ncrs-2022-0425
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- Article
Crystal structure of 5-methyl-3,3-diphenyl-1-tosyl-1,2,3,4-tetrahydropyridine, C<sub>25</sub>H<sub>25</sub>NO<sub>2</sub>S.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2018, v. 233, n. 3, p. 457, doi. 10.1515/ncrs-2017-0350
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- Article
The crystal structure of <italic>N</italic>-((3,5-di-<italic>tert</italic>-butyl-4-hydroxyphenyl)(phenyl)methyl)-4-methylbenzenesulfonamide, C<sub>28</sub>H<sub>35</sub>N<sub>3</sub>S.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2018, v. 233, n. 2, p. 259, doi. 10.1515/ncrs-2017-0257
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- Article
Crystal structure of 4-((4,4-dimethyl-2, 6-dioxocyclohexylidine)methylamino)- N-(3,4-dimethylisoxazol-5-yl)benzenesulfonamide, C<sub>20</sub>H<sub>23</sub>N<sub>3</sub>O<sub>5</sub>S.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 4, p. 1117, doi. 10.1515/ncrs-2016-0082
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- Article
Crystal structure of ( Z)-4-(4-oxopent-2-en-2-ylamino)benzenesulfonamide, C<sub>11</sub>H<sub>14</sub>N<sub>2</sub>O<sub>3</sub>S.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 867, doi. 10.1515/ncrs-2015-0297
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- Article