Works matching DE "AZAINDOLES"

Results: 59

Indium Trichloride (InCl3) Catalyzed Synthesis of Fused 7-Azaindole Derivatives Using Domino Knoevenagel-Michael Reaction.

Published in:

Journal of the Chinese Chemical Society, 2016, v. 63, n. 4, p. 323, doi. 10.1002/jccs.201500540

By:

Dongare, Sakharam B.;
Chavan, Hemant V.;
Surwase, Datta N.;
Bhale, Pravin S.;
Mule, Yoginath B.;
Bandgar, Babasaheb P.

Publication type:

Article

Regioselective Functionalization of 7‐Azaindole by Controlled Annular Isomerism: The Directed Metalation‐Group Dance.

Published in:

Angewandte Chemie, 2019, v. 131, n. 22, p. 7391, doi. 10.1002/ange.201901724

By:

Dalziel, Michael E.;
Patel, Jignesh J.;
Kaye, Meagan K.;
Cosman, Jennifer L.;
Kitching, Matthew O.;
Snieckus, Victor

Publication type:

Article

Advances in Green Catalysis for the Synthesis of Medicinally Relevant N -Heterocycles.

Published in:

Catalysts (2073-4344), 2021, v. 11, n. 9, p. 1108, doi. 10.3390/catal11091108

By:

Santos, A. Sofia;
Raydan, Daniel;
Cunha, José C.;
Viduedo, Nuno;
Silva, Artur M. S.;
Marques, M. Manuel B.

Publication type:

Article

Crystal structure of 3- tert-butyl-7-azadioxindole, C11H14N2O2.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 4, p. 1069, doi. 10.1515/ncrs-2016-0054

By:

El-Hiti, Gamal A.;
Masmali, Ali M.;
Smith, Keith;
Hegazy, Amany S.;
Kariuki, Benson M.

Publication type:

Article

Synthetic approaches to site selective deuterium incorporation in a novel CRTh2 receptor antagonist clinical candidate.

Published in:

2014

By:

Sandham, David A.;
Page, Christopher J.

Publication type:

Other

Activation-free one-pot alkynylation-cyclization synthesis of 2-substituted 4-azaindoles and indoles.

Published in:

Chemistry of Heterocyclic Compounds, 2018, v. 54, n. 3, p. 334, doi. 10.1007/s10593-018-2269-z

By:

Lessing, Timo;
Müller, Thomas J. J.

Publication type:

Article

Synthesis of 5-chloro-7-azaindoles by Fischer reaction.

Published in:

Chemistry of Heterocyclic Compounds, 2017, v. 53, n. 2, p. 196, doi. 10.1007/s10593-017-2040-x

By:

Alekseyev, Roman;
Amirova, Sabina;
Terenin, Vladimir

Publication type:

Article

The Fischer Reaction in the Synthesis of 2,3-Disubstituted 7-Azaindoles*.

Published in:

Chemistry of Heterocyclic Compounds, 2014, v. 50, n. 9, p. 1305, doi. 10.1007/s10593-014-1593-1

By:

Alekseyev, R.;
Amirova, S.;
Kabanova, E.;
Terenin, V.

Publication type:

Article

Theoretical Studies on Azaindoles as Human Aurora B Kinase Inhibitors: Docking, Pharmacophore and ADMET Studies.

Published in:

Interdisciplinary Sciences: Computational Life Sciences, 2018, v. 10, n. 3, p. 486, doi. 10.1007/s12539-016-0205-4

By:

Vadlakonda, Rajashekar;
Nerella, Raghunandan;
Enaganti, Sreenivas

Publication type:

Article

Self-Assembling Azaindole Organogel for Organic Light-Emitting Devices (OLEDs).

Published in:

Advanced Functional Materials, 2017, v. 27, n. 41, p. n/a, doi. 10.1002/adfm.201702176

By:

Martín, Cristina;
Kennes, Koen;
Van der Auweraer, Mark;
Hofkens, Johan;
de Miguel, Gustavo;
García‐Frutos, Eva M.

Publication type:

Article

Hypervalent Fluoroiodane‐Triggered Synthesis of Fluoro‐Azabenzoxazepines and Azaindoles.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 20/21, p. 2615, doi. 10.1002/ejoc.201800129

By:

Brunner, Christoph;
Andries‐ulmer, Anna;
Kiefl, Gabriel M.;
Gulder, Tanja

Publication type:

Article

Dual Catalysis in Domino N-Benzylation/Intramolecular C-H Arylation: Regio- and Chemoselective Synthesis of Annelated Nitrogen Heterocycles.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 25, p. 5469, doi. 10.1002/ejoc.201402395

By:

Laha, Joydev K.;
Dayal, Neetu;
Singh, Swati;
Bhimpuria, Rohan

Publication type:

Article

Extending the Scope of the Aza-Fischer Synthesis of 4- and 6-Azaindoles.

Published in:

European Journal of Organic Chemistry, 2013, v. 2013, n. 16, p. 3328, doi. 10.1002/ejoc.201300167

By:

Thomae, David;
Jeanty, Matthieu;
Coste, Jérome;
Guillaumet, Gérald;
Suzenet, Franck

Publication type:

Article

Synthesis and Characterization of Two New Mononuclear Complexes of Cobalt(II) with 7-Azaindole.

Published in:

Journal of Chemical Crystallography, 2017, v. 47, n. 1/2, p. 22, doi. 10.1007/s10870-017-0676-0

By:

Przyojski, Jacob;
Arman, Hadi;
Myers, Nicole;
Walmsley, Judith

Publication type:

Article

Structure and intermolecular vibrations of 7-azaindole-water 2:1 complex in a supersonic jet expansion: Laser-induced fluorescence spectroscopy and quantum chemistry calculation.

Published in:

Journal of Chemical Sciences, 2012, v. 124, n. 1, p. 131, doi. 10.1007/s12039-011-0200-6

By:

HAZRA, MONTU;
MUKHERJEE, MOITRAYEE;
RAMANATHAN, V;
CHAKRABORTY, TAPAS

Publication type:

Article

Palladium-catalyzed heteroannulation approach to 7-azatryptophan with a Schöllkopf chiral auxiliary.

Published in:

Bulletin of the Korean Chemical Society, 2015, v. 36, n. 5, p. 1546, doi. 10.1002/bkcs.10287

By:

Gee, Moon Bae;
Kim, Tae Seung;
Yum, Eul Kgun

Publication type:

Article

2,3,4-Trioxo-1-(1H-pyrrolo[2,3-b]pyridin-7-ium-7yl)-cyclobutan-1-ide.

Published in:

Molbank, 2018, v. 2018, n. 4, p. M1026, doi. 10.3390/M1026

By:

Lande, Duc Hoàng;
Kunick, Conrad;
Grünefeld, Johann

Publication type:

Article

A theoretical and optical spectroscopic study of the mechanism of a tautomeric transformation in the 7-azaindole dimer and the 7-azaindole complex with a water molecule.

Published in:

Journal of Structural Chemistry, 2017, v. 58, n. 2, p. 226, doi. 10.1134/S0022476617020020

By:

Ten, G.;
Glukhova, O.;
Slepchenkov, M.;
Shcherbakova, N.;
Baranov, V.

Publication type:

Article

7-Azaindole in the Gas Phase: Absorption, Luminescence, and the Mechanism of Long-Lived Luminescence.

Published in:

Journal of Applied Spectroscopy, 2018, v. 85, n. 5, p. 850, doi. 10.1007/s10812-018-0728-z

By:

Sukhodola, A. A.

Publication type:

Article

The Xanthate Route to Indolines, Indoles, and their Aza Congeners.

Published in:

Chemistry - A European Journal, 2020, v. 26, n. 56, p. 12689, doi. 10.1002/chem.202001341

By:

Zard, Samir Z.

Publication type:

Article

Intramolecular Oxidative Arylations in 7-Azaindoles and Pyrroles: Revamping the Synthesis of Fused N-Heterocycle Tethered Fluorenes.

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 9, p. 2044, doi. 10.1002/chem.201604192

By:

Laha, Joydev K.;
Bhimpuria, Rohan A.;
Hunjan, Mandeep Kaur

Publication type:

Article

Rhodium-Catalyzed Hydrogen-Releasing ortho-Alkenylation of 7-Azaindoles.

Published in:

Chemistry - A European Journal, 2016, v. 22, n. 50, p. 17926, doi. 10.1002/chem.201603887

By:

Li, Wei‐Huan;
Wu, Lin;
Li, Shuai‐Shuai;
Liu, Chen‐Fei;
Zhang, Guo‐Tai;
Dong, Lin

Publication type:

Article

Frontispiece: Rhodium-Catalyzed Hydrogen-Releasing ortho-Alkenylation of 7-Azaindoles.

Published in:

Chemistry - A European Journal, 2016, v. 22, n. 50, p. n/a, doi. 10.1002/chem.201685061

By:

Li, Wei‐Huan;
Wu, Lin;
Li, Shuai‐Shuai;
Liu, Chen‐Fei;
Zhang, Guo‐Tai;
Dong, Lin

Publication type:

Article

A THEORETICAL STUDY ON PROTON-GAIN BEHAVIORS OF SOME AZAINDOLE DERIVATIVES.

Published in:

Anadolu University of Sciences & Technology - B: Theoretical Sciences, 2011, v. 1, n. 2, p. 149

By:

ÇALIŞ, Sevgül;
BERBER, Halil;
UYSAL, Ülkü Dilek;
ÖĞRETİR, Cemil

Publication type:

Article

Flexible Analogues of Azaindole DYRK1A Inhibitors Elicit Cytotoxicity in Glioblastoma Cells*.

Published in:

Australian Journal of Chemistry, 2018, v. 71, n. 10, p. 789, doi. 10.1071/CH18251

By:

Zhou, Qingqing;
Reekie, Tristan A.;
Abbassi, Ramzi H.;
Venkata, Dinesh Indurthi;
Font, Josep S.;
Ryan, Renae M.;
Rendina, Louis M.;
Munoz, Lenka;
Kassiou, Michael

Publication type:

Article

Using a Johnson‐Claisen Rearrangement Strategy to Construct Azaindoles – A Streamlined and Concise Route for the Commercial Process of Fevipiprant.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 31, p. 4490, doi. 10.1002/ejoc.202100686

By:

Mathes, Christian;
Riss, Bernard;
Rüegger, Ueli;
Hueber, Lukas;
Dedic, Darija;
Fei, Zhongbo;
den Reijer, Carolien;
Königsberger, Kurt;
Napp, Matthias;
Schlama, Thierry;
Dempsey, Glen;
Lustenberger, Philipp

Publication type:

Article

The Rho kinase inhibitor azaindole-1 has long-acting vasodilator activity in the pulmonary vascular bed of the intact chest rat.

Published in:

Canadian Journal of Physiology & Pharmacology, 2012, v. 90, n. 7, p. 825, doi. 10.1139/Y2012-061

By:

Pankey, Edward A.;
Byun, Ryuk J.;
Smith II, William B.;
Bhartiya, Manish;
Bueno, Franklin R.;
Badejo, Adeleke M.;
Stasch, Johannes-Peter;
Murthy, Subramanyam N.;
Nossaman, Bobby D.;
Kadowitz, Philip J.

Publication type:

Article

Synthesis of Novel Fluorinated 11 H-Azaindolo[3,2- c]isoquinolines.

Published in:

Journal of Heterocyclic Chemistry, 2013, v. 50, n. 3, p. 513, doi. 10.1002/jhet.1511

By:

Atmakur, Krishnaiah;
Emmadi, Narender Reddy;
Balasubramanian, Sridhar

Publication type:

Article

Iodoindazoles with Selective Magnesiation at Position 3: A Route to Highly Functionalized Indazoles.

Published in:

Chemistry - A European Journal, 2016, v. 22, n. 13, p. 4440, doi. 10.1002/chem.201504828

By:

Lam, Bao Vy;
Berhault, Yohann;
Stiebing, Silvia;
Fossey, Christine;
Cailly, Thomas;
Collot, Valérie;
Fabis, Frédéric

Publication type:

Article

Synthesis of Indazoles and Azaindazoles by Intramolecular Aerobic Oxidative CN Coupling under Transition-Metal-Free Conditions.

Published in:

Chemistry - A European Journal, 2014, v. 20, n. 14, p. 3932, doi. 10.1002/chem.201304923

By:

Hu, Jiantao;
Xu, Huacheng;
Nie, Pengju;
Xie, Xiaobo;
Nie, Zongxiu;
Rao, Yu

Publication type:

Article

Azaindoles as Zinc-Binding Small-Molecule Inhibitors of the JAMM Protease CSN5.

Published in:

Angewandte Chemie, 2017, v. 129, n. 5, p. 1314, doi. 10.1002/ange.201608672

By:

Altmann, Eva;
Erbel, Paul;
Renatus, Martin;
Schaefer, Michael;
Schlierf, Anita;
Druet, Adelaide;
Kieffer, Laurence;
Sorge, Mickael;
Pfister, Keith;
Hassiepen, Ulrich;
Jones, Matthew;
Ruedisser, Simon;
Ostermeier, Daniela;
Martoglio, Bruno;
Jefferson, Anne B.;
Quancard, Jean

Publication type:

Article

Asymmetric Hydrogenation of Azaindoles: Chemo- and Enantioselective Reduction of Fused Aromatic Ring Systems Consisting of Two Heteroarenes.

Published in:

Angewandte Chemie, 2016, v. 128, n. 39, p. 12038, doi. 10.1002/ange.201606083

By:

Makida, Yusuke;
Saita, Masahiro;
Kuramoto, Takahiro;
Ishizuka, Kentaro;
Kuwano, Ryoichi

Publication type:

Article

Electrochemical C−H/N−H Functionalization for the Synthesis of Highly Functionalized (Aza)indoles.

Published in:

Angewandte Chemie, 2016, v. 128, n. 32, p. 9314, doi. 10.1002/ange.201602616

By:

Hou, Zhong ‐ Wei;
Mao, Zhong ‐ Yi;
Zhao, Huai ‐ Bo;
Melcamu, Yared Yohannes;
Lu, Xin;
Song, Jinshuai;
Xu, Hai ‐ Chao

Publication type:

Article

A Designed Amide as an Aldol Donor in the Direct Catalytic Asymmetric Aldol Reaction.

Published in:

Angewandte Chemie, 2014, v. 126, n. 24, p. 6264, doi. 10.1002/ange.201403118

By:

Weidner, Karin;
Kumagai, Naoya;
Shibasaki, Masakatsu

Publication type:

Article

Theoretical Analysis of the Fluorescence Spectra of 7-Azaindole and Its Tautomer.

Published in:

Optics & Spectroscopy, 2016, v. 120, n. 3, p. 359, doi. 10.1134/S0030400X16030255

By:

Ten, G.;
Glukhova, O.;
Slepchenkov, M.;
Baranov, V.

Publication type:

Article

Palladium Nanocatalysts for Cascade C−N Cross‐Coupling/Heck Reaction.

Published in:

Asian Journal of Organic Chemistry, 2021, v. 10, n. 4, p. 872, doi. 10.1002/ajoc.202100077

By:

Rodriguez‐Oliva, Ivan;
Losada‐Garcia, Noelia;
Santos, A. Sofia;
Marques, M. Manuel B.;
Palomo, Jose M.

Publication type:

Article

Selenium‐Electrocatalytic Cyclization of 2‐Vinylanilides towards Indoles of Peptide Labeling.

Published in:

Chemistry - An Asian Journal, 2022, v. 17, n. 20, p. 1, doi. 10.1002/asia.202200762

By:

Zeng, Shaogao;
Fang, Songlin;
Cai, Haiping;
Wang, Dong;
Liu, Weiliang;
Hu, Xinwei;
Sun, Pinghua;
Ruan, Zhixiong

Publication type:

Article

A Convenient One-Pot Route to Screw-Shaped [5]Azahelicenes via Rhodium(III)-Catalyzed Multiple C−H Bond Activation.

Published in:

Chemistry - An Asian Journal, 2017, v. 12, n. 4, p. 415, doi. 10.1002/asia.201601744

By:

Li, Shuai ‐ Shuai;
Liu, Chen ‐ Fei;
Zhang, Guo ‐ Tai;
Xia, Ying ‐ Qi;
Li, Wei ‐ Huan;
Dong, Lin

Publication type:

Article

Scalable synthesis and properties of 7-methyl-4-azaindole.

Published in:

Heterocyclic Communications, 2017, v. 23, n. 6, p. 449, doi. 10.1515/hc-2017-0180

By:

Subota, Andrii I.;
Volochnyuk, Dmitriy M.;
Gorlova, Alina O.;
Grygorenko, Oleksandr O.

Publication type:

Article

Rhodium-Catalyzed Tandem Annulation Reactions of 7-Azaindoles with Electron-Deficient Olefins via Double CH Activation.

Published in:

Advanced Synthesis & Catalysis, 2016, v. 358, n. 10, p. 1595, doi. 10.1002/adsc.201600112

By:

Li, Shuai ‐ Shuai;
Lin, Hui;
Liu, Chen ‐ Fei;
Xia, Ying ‐ Qi;
Zhang, Xiao ‐ Mei;
Dong, Lin

Publication type:

Article

G-quadruplex binding properties of a potent PARP-1 inhibitor derived from 7-azaindole-1-carboxamide.

Published in:

Scientific Reports, 2021, v. 11, n. 1, p. 1, doi. 10.1038/s41598-021-83474-9

By:

Dallavalle, Sabrina;
Musso, Loana;
Artali, Roberto;
Aviñó, Anna;
Scaglioni, Leonardo;
Eritja, Ramon;
Gargallo, Raimundo;
Mazzini, Stefania

Publication type:

Article

Unlocking New Prenylation Modes: Azaindoles as a New Substrate Class for Indole Prenyltransferases.

Published in:

ChemCatChem, 2023, v. 15, n. 19, p. 1, doi. 10.1002/cctc.202300650

By:

Gardner, Eric D.;
Johnson, Bryce P.;
Dimas, Dustin A.;
McClurg, Heather E.;
Severance, Zachary C.;
Burgett, Anthony W.;
Singh, Shanteri

Publication type:

Article

Synthesis of Diverse 1,4‐(Azaindole)[60]fullerenes via Transition‐Metal Free Three‐Component Coupling Reaction of Azaindoles, C60, and Bromoalkanes/Triphenylamines†.

Published in:

Chinese Journal of Chemistry, 2023, v. 41, n. 22, p. 2975, doi. 10.1002/cjoc.202300292

By:

Huang, Xinmin;
Liu, Zi‐Zheng;
Cheng, Jia‐Qi;
Cao, Cheng‐Yu;
Li, Peng‐Cheng;
Xuan, Jun;
Li, Fei

Publication type:

Article

Base‐Promoted Formylation and N‐Difluoromethylation of Azaindoles with Ethyl Bromodifluoroacetate as a Carbon Source.

Published in:

Chinese Journal of Chemistry, 2021, v. 39, n. 6, p. 1477, doi. 10.1002/cjoc.202100008

By:

Li, Yang;
Sun, Ning;
Zhang, Cai‐Lin;
Hao, Meng

Publication type:

Article

Effects of Aromatic Stabilization Energies on Photochromism of New Asymmetrical Azaindole-Containing Diarylethenes.

Published in:

Chinese Journal of Chemistry, 2015, v. 33, n. 7, p. 785, doi. 10.1002/cjoc.201500110

By:

Sun, Zhiyuan;
Zhang, Congcong;
Li, Hui;
Fan, Congbin;
Liu, Gang;
Pu, Shouzhi

Publication type:

Article

Azaindoles as Zinc-Binding Small-Molecule Inhibitors of the JAMM Protease CSN5.

Published in:

Angewandte Chemie International Edition, 2017, v. 56, n. 5, p. 1294, doi. 10.1002/anie.201608672

By:

Altmann, Eva;
Erbel, Paul;
Renatus, Martin;
Schaefer, Michael;
Schlierf, Anita;
Druet, Adelaide;
Kieffer, Laurence;
Sorge, Mickael;
Pfister, Keith;
Hassiepen, Ulrich;
Jones, Matthew;
Ruedisser, Simon;
Ostermeier, Daniela;
Martoglio, Bruno;
Jefferson, Anne B.;
Quancard, Jean

Publication type:

Article

Asymmetric Hydrogenation of Azaindoles: Chemo- and Enantioselective Reduction of Fused Aromatic Ring Systems Consisting of Two Heteroarenes.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 39, p. 11859, doi. 10.1002/anie.201606083

By:

Makida, Yusuke;
Saita, Masahiro;
Kuramoto, Takahiro;
Ishizuka, Kentaro;
Kuwano, Ryoichi

Publication type:

Article

Electrochemical C−H/N−H Functionalization for the Synthesis of Highly Functionalized (Aza)indoles.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 32, p. 9168, doi. 10.1002/anie.201602616

By:

Hou, Zhong-Wei;
Mao, Zhong-Yi;
Zhao, Huai-Bo;
Melcamu, Yared Yohannes;
Lu, Xin;
Song, Jinshuai;
Xu, Hai-Chao

Publication type:

Article

Preparation of Functionalized Indoles and Azaindoles by the Intramolecular Copper-Mediated Carbomagnesiation of Ynamides.

Published in:

Angewandte Chemie International Edition, 2013, v. 52, n. 38, p. 10084, doi. 10.1002/anie.201304380

By:

Frischmuth, Annette;
Knochel, Paul

Publication type:

Article

Full Functionalization of the 7-Azaindole Scaffold by Selective Metalation and Sulfoxide/Magnesium Exchange.

Published in:

Angewandte Chemie International Edition, 2013, v. 52, n. 38, p. 10093, doi. 10.1002/anie.201303490

By:

Barl, Nadja M.;
Sansiaume-Dagousset, Elodie;
Karaghiosoff, Konstantin;
Knochel, Paul

Publication type:

Article