Works matching DE "ANTINEOPLASTIC agent synthesis"

Results: 138

Synthesis of a Regioisomer of β-Lapachone and Analogs as Potent Antitumor Agents.

Published in:

Helvetica Chimica Acta, 2015, v. 98, n. 1, p. 128, doi. 10.1002/hlca.201400160

By:

Ding, Qunshan;
Zhang, Yan;
Shen, Zhenhua;
Song, Chuanjun;
Chang, Junbiao

Publication type:

Article

Current understanding of synergistic interplay of chitosan nanoparticles and anticancer drugs: merits and challenges.

Published in:

Applied Microbiology & Biotechnology, 2015, v. 99, n. 5, p. 2055, doi. 10.1007/s00253-015-6384-9

By:

Kandra, Prameela;
Kalangi, Hemalatha

Publication type:

Article

A diaryl-linked [Pd 2 L 4 ] metallosupramolecular architecture: synthesis, structures and cisplatin binding studies.

Published in:

Supramolecular Chemistry, 2015, v. 27, n. 11/12, p. 734, doi. 10.1080/10610278.2015.1063633

By:

Kim, Tae Y.;
Lucas, Nigel T.;
Crowley, James D.

Publication type:

Article

MicroRNA-574-3p, identified by microRNA library-based functional screening, modulates tamoxifen response in breast cancer.

Published in:

Scientific Reports, 2015, p. 7641, doi. 10.1038/srep07641

By:

Ujihira, T.;
Ikeda, K.;
Suzuki, T.;
Yamaga, R.;
Sato, W.;
Horie-Inoue, K.;
Shigekawa, T.;
Osaki, A.;
Saeki, T.;
Okamoto, K.;
Takeda, S.;
Inoue, S.

Publication type:

Article

Synthesis and pharmacological evaluation of isoxazole derivatives containing 1,2,4-triazole Moiety.

Published in:

Marmara Pharmaceutical Journal, 2012, v. 16, n. 2, p. 134

By:

Khanage, Shantaram;
Mohite, Popat;
Pandhare, Ramdas;
Raju, Appala

Publication type:

Article

Synthesis and evaluation of cytotoxic activities of some 1,4-disubstituted thiosemicarbazides, 2,5-disubstituted-1,3,4-thiadiazoles and 1,2,4-triazole-5-thiones derived from benzilic acid hydrazide.

Published in:

Marmara Pharmaceutical Journal, 2012, v. 16, n. 1, p. 56

By:

Çoruh, Işıl;
Rollas, Sevim;
Özbaş Turan, Suna;
Akbuğa, Jülide

Publication type:

Article

Synthesis and Evaluation of Flavanones as Anticancer Agents.

Published in:

Indian Journal of Pharmaceutical Sciences, 2014, v. 76, n. 2, p. 163

By:

MURTI, Y.;
MISHRA, P.

Publication type:

Article

Effect of pantoprazole to enhance activity of docetaxel against human tumour xenografts by inhibiting autophagy.

Published in:

British Journal of Cancer, 2015, v. 112, n. 5, p. 832, doi. 10.1038/bjc.2015.17

By:

Tan, Q;
Joshua, A M;
Saggar, J K;
Yu, M;
Wang, M;
Kanga, N;
Zhang, J Y;
Chen, X;
Wouters, B G;
Tannock, I F

Publication type:

Article

MDM2 is an important prognostic and predictive factor for platin-pemetrexed therapy in malignant pleural mesotheliomas and deregulation of P14/ARF (encoded by CDKN2A) seems to contribute to an MDM2-driven inactivation of P53.

Published in:

British Journal of Cancer, 2015, v. 112, n. 5, p. 883, doi. 10.1038/bjc.2015.27

By:

Walter, R F H;
Mairinger, F D;
Ting, S;
Vollbrecht, C;
Mairinger, T;
Theegarten, D;
Christoph, D C;
Schmid, K W;
Wohlschlaeger, J

Publication type:

Article

Synthesis and Characterization of trans-Dichlorotetrakis(imidazole)cobalt(III) Chloride: A New Cobalt(III) Coordination Complex with Potential Prodrug Properties.

Published in:

Bioinorganic Chemistry & Applications, 2018, p. 1, doi. 10.1155/2018/4560757

By:

Hart, Kaila F.;
Joe, Natalie S.;
Miller, Rebecca M.;
Nash, Hannah P.;
Blake, David J.;
Morris, Aimee M.

Publication type:

Article

Double crosslinked chitosan and gelatin submicronic capsules entrapping aminoacid derivatives with potential antitumoral activity.

Published in:

Journal of Materials Science, 2012, v. 47, n. 23, p. 8223, doi. 10.1007/s10853-012-6719-1

By:

Moise, Mihaela;
Şunel, Valeriu;
Holban, Mihaela;
Popa, Marcel;
Desbrieres, Jacques;
Peptu, Cristian;
Lionte, Cătălina

Publication type:

Article

Correction to: Lipophilic gold(I) complexes with 1,3,4-oxadiazol-2-thione or 1,3-thiazolidine-2-thione moieties: synthesis and their cytotoxic and antimicrobial activities.

Published in:

2017

By:

Almeida, Angelina;
Oliveira, Bruno;
Castro, Pedro;
Mendonça, Camille;
Furtado, Ricardo;
Nicolella, Heloiza;
Silva, Vânia;
Diniz, Cláudio;
Tavares, Denise;
Silva, Heveline;
Almeida, Mauro

Publication type:

Erratum

Anti-proliferative effect of Fe(III) complexed with 1-(2-hydroxy-3-methoxybenzaldehyde)-4-aminosalicylhydrazone in HepG2 cells.

Published in:

BioMetals, 2015, v. 28, n. 4, p. 669, doi. 10.1007/s10534-015-9852-x

By:

Fukushima, Takeshi;
Taniguchi, Erina;
Yamada, Hiroshi;
Kato, Kiyomasa;
Shimizu, Ayako;
Nishiguchi, Yoshikazu;
Onozato, Mayu;
Ichiba, Hideaki;
Azuma, Yutaro

Publication type:

Article

Cyclopropanol intermediates in the synthesis of the C-C fragment of laulimalides.

Published in:

Russian Journal of Organic Chemistry, 2016, v. 52, n. 3, p. 355, doi. 10.1134/S1070428016030118

By:

Mineeva, I.

Publication type:

Article

Synthesis and study of antitumor activity of tetraethyl 2-(2′,2′,6′,6′-Tetramethylpiperidin-4′-ylamino)ethylidene-1,1-bisphosphonate.

Published in:

Doklady Chemistry, 2014, v. 457, n. 1, p. 137, doi. 10.1134/S0012500814070064

By:

Grigor'ev, I.;
Morozov, D.;
Svyatchenko, V.;
Kiselev, N.;
Loktev, V.;
Luk'yanets, E.;
Vorozhtsov, G.

Publication type:

Article

Total Synthesis, Configuration, and Biological Evaluation of Anguinomycin C.

Published in:

Asian Journal of Control, 2013, v. 15, n. 6, p. 8707, doi. 10.1002/anie.200703134

By:

Bonazzi, Simone;
Güttinger, Stephan;
Zemp, Ivo;
Kutay, Ulrike;
Gademann, Karl

Publication type:

Article

Aryl sulfonate based anticancer alkylating agents.

Published in:

Pakistan Journal of Pharmaceutical Sciences, 2018, v. 31, p. 1081

By:

Sheikh, Hamdullah Khadim;
Arshad, Tanzila;
Kanwal, Ghazala

Publication type:

Article

Evaluation of cytotoxic and antiviral activities of aqueous leaves extracts of different plants against foot and mouth disease virus infection in farming animals.

Published in:

Pakistan Journal of Pharmaceutical Sciences, 2017, v. 30, n. 6, p. 2167

By:

Younus, Ishrat;
Ashraf, Muhammad;
Fatima, Anab;
Altaf, Imran;
Javeed, Aqeel

Publication type:

Article

The newly synthesized anticancer drug HUHS1015 is useful for treatment of human gastric cancer.

Published in:

Cancer Chemotherapy & Pharmacology, 2015, v. 75, n. 3, p. 527, doi. 10.1007/s00280-014-2661-z

By:

Kaku, Yoshiko;
Tsuchiya, Ayako;
Kanno, Takeshi;
Nakao, Shuhei;
Shimizu, Tadashi;
Tanaka, Akito;
Nishizaki, Tomoyuki

Publication type:

Article

Synthesis and biological evaluation of aziridin-1-yl oxime-based vorinostat analogs as anticancer agents.

Published in:

Chemistry of Heterocyclic Compounds, 2015, v. 51, n. 7, p. 647, doi. 10.1007/s10593-015-1752-z

By:

Nikitjuka, Anna;
Shestakova, Irina;
Romanchikova, Nadezhda;
Jirgensons, Aigars

Publication type:

Article

Scalable and green process for the synthesis of anticancer drug lenalidomide.

Published in:

Chemistry of Heterocyclic Compounds, 2015, v. 51, n. 2, p. 133, doi. 10.1007/s10593-015-1670-0

By:

Ponomaryov, Yuri;
Krasikova, Valeria;
Lebedev, Anton;
Chernyak, Dmitri;
Varacheva, Larisa;
Chernobroviy, Alexandr

Publication type:

Article

Macrocyclic complexes: synthesis, characterization, antitumor and DNA binding studies.

Published in:

Nucleosides, Nucleotides & Nucleic Acids, 2018, v. 37, n. 9, p. 498, doi. 10.1080/15257770.2018.1498515

By:

Lamani, Devappa S.;
Badiger, S. G.;
Venugopala Reddy, K. R.;
Bhojya Naik, H. S.

Publication type:

Article

Synthesis and anticancer activity of new [(Indolyl)pyrazolyl]-1,3,4-oxadiazole thioglycosides and acyclic nucleoside analogs.

Published in:

Nucleosides, Nucleotides & Nucleic Acids, 2017, v. 36, n. 7, p. 474, doi. 10.1080/15257770.2017.1327665

By:

El-Sayed, Wael A.;
El-Sofany, Walaa I.;
Hussein, Hoda A. R.;
Fathy, Nahed M.

Publication type:

Article

SYNTHESIS, SPECTRAL CHARACTERIZATION AND ANTICANCER EVALUATION OF NEW DIAZENYL SCHIFF BASE DERIVATIVES.

Published in:

Indian Drugs, 2017, v. 54, n. 2, p. 20, doi. 10.53879/id.54.02.10877

By:

Sarangi, P. K. N.;
Sahoo, J.;
Paidesetty, S. K.;
Mohanta, G. P.

Publication type:

Article

Ribonucleolytic activity of mycoplasmas.

Published in:

Microbiology (00262617), 2014, v. 83, n. 3, p. 247, doi. 10.1134/S0026261714030072

By:

Ilinskaya, O.;
Sokurenko, Yu.;
Ul'yanova, V.;
Vershinina, V.;
Zelenikhin, P.;
Kolpakov, A.;
Medvedeva, E.;
Baranova, N.;
Davydova, M.;
Muzykantov, A.;
Chernova, O.;
Chernov, V.

Publication type:

Article

Synthesis and Mode of Action Studies on Iridium(I)–NHC Anticancer Drug Candidates.

Published in:

European Journal of Inorganic Chemistry, 2018, v. 2018, n. 20/21, p. 2461, doi. 10.1002/ejic.201800225

By:

Gothe, Yvonne;
Romero‐canelón, Isolda;
Marzo, Tiziano;
Sadler, Peter J.;
Messori, Luigi;
Metzler‐nolte, Nils

Publication type:

Article

Cytotoxic Vanadium Complexes of Branched [ONNO]-Type Diamine Bis(phenolato) Ligands.

Published in:

European Journal of Inorganic Chemistry, 2017, v. 2017, n. 12, p. 1807, doi. 10.1002/ejic.201601276

By:

Nahari, Gilad;
Reytman, Lilia;
Vendier, Laure;
Tshuva, Edit Y.;
Lorber, Christian

Publication type:

Article

Mitochondria-Targeting Iron(III) Catecholates for Photoactivated Anticancer Activity under Red Light.

Published in:

European Journal of Inorganic Chemistry, 2016, v. 2016, n. 7, p. 1002, doi. 10.1002/ejic.201501105

By:

Basu, Uttara;
Pant, Ila;
Kondaiah, Paturu;
Chakravarty, Akhil R.

Publication type:

Article

Synthesis, Characterization, and Biological Properties of Osmium-Based Tamoxifen Derivatives - Comparison with Their Homologues in the Iron and Ruthenium Series.

Published in:

European Journal of Inorganic Chemistry, 2015, v. 2015, n. 25, p. 4217, doi. 10.1002/ejic.201500770

By:

Lee, Hui Zhi Shirley;
Buriez, Olivier;
Chau, François;
Labbé, Eric;
Ganguly, Rakesh;
Amatore, Christian;
Jaouen, Gérard;
Vessières, Anne;
Leong, Weng Kee;
Top, Siden

Publication type:

Article

Substitution-Modulated Anticancer Activity of Half-Sandwich Ruthenium(II) Complexes with Heterocyclic Ancillary Ligands.

Published in:

European Journal of Inorganic Chemistry, 2014, v. 2014, n. 22, p. 3536, doi. 10.1002/ejic.201402205

By:

Mitra, Raja;
Samuelson, Ashoka G.

Publication type:

Article

Synthesis and Biological Evaluation of 7-Deoxy-Epothilone Analogues.

Published in:

International Journal of Molecular Sciences, 2017, v. 18, n. 3, p. 648, doi. 10.3390/ijms18030648

By:

Woods, Laura M.;
Arico, Joseph W.;
Frein, Jeffrey D.;
Sackett, Dan L.;
Taylor, Richard E.

Publication type:

Article

D-Amino Acid Position Influences the Anticancer Activity of Galaxamide Analogs: An Apoptotic Mechanism Study.

Published in:

International Journal of Molecular Sciences, 2017, v. 18, n. 3, p. 544, doi. 10.3390/ijms18030544

By:

Bai, Defa;
Siming Yu;
Shenghui Zhong;
Bingxin Zhao;
Shaoling Qiu;
Jianwei Chen;
Lunagariya, Jignesh;
Xiaojian Liao;
Shihai Xu

Publication type:

Article

A Series of New Ligustrazine-Triterpenes Derivatives as Anti-Tumor Agents: Design, Synthesis, and Biological Evaluation.

Published in:

International Journal of Molecular Sciences, 2015, v. 16, n. 9, p. 21035, doi. 10.3390/ijms160921035

By:

Bing Xu;
Fuhao Chu;
Yuzhong Zhang;
Xiaobo Wang;
Qiang Li;
Wei Liu;
Xin Xu;
Yanyi Xing;
Jing Chen;
Penglong Wang;
Haimin Lei

Publication type:

Article

Efficient Synthesis of a Maghemite/Gold Hybrid Nanoparticle System as a Magnetic Carrier for the Transport of Platinum-Based Metallotherapeutics.

Published in:

International Journal of Molecular Sciences, 2015, v. 16, n. 1, p. 2034, doi. 10.3390/ijms16012034

By:

Štarha, Pavel;
Smola, David;
Tuček, Jiří;
Trávníček, Zdeněk

Publication type:

Article

Synthesis, Docking and Biological Activities of Novel Hybrids Celecoxib and Anthraquinone Analogs as Potent Cytotoxic Agents.

Published in:

International Journal of Molecular Sciences, 2014, v. 15, n. 12, p. 22580, doi. 10.3390/ijms151222580

By:

Almutairi, Maha S.;
Hegazy, Gehan H.;
Haiba, Mogedda E.;
Ali, Hamed I.;
Khalifa, Nagy M.;
Soliman, Abd El-mohsen M.

Publication type:

Article

Self-activated DNA cleavage of a water-soluble mononuclear Cu(II) complex with polyquinolinyl ligand.

Published in:

Journal of Coordination Chemistry, 2014, v. 67, n. 22, p. 3598, doi. 10.1080/00958972.2014.973867

By:

Li, Jun-Ling;
Jiang, Lin;
Li, Si-Tong;
Tian, Jin-Lei;
Gu, Wen;
Liu, Xin;
Yan, Shi-Ping

Publication type:

Article

A new dinuclear Ag(I)– N -heterocyclic carbene complex derived from para -xylyl linked bis -imidazolium salt: synthesis, crystal structure, and in vitro anticancer studies.

Published in:

Journal of Coordination Chemistry, 2013, v. 66, n. 15, p. 2679, doi. 10.1080/00958972.2013.813492

By:

Haque, Rosenani A.;
Nasri, Siti Fatimah;
Iqbal, Muhammad Adnan

Publication type:

Article

Structure elucidation of 3-[1-(6-methoxy-2-naphtyl)ethyl]-6-(2,4-dichlorophenyl)-7H-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazine, C23H18Cl2N4OS from synchrotron X-ray powder diffraction.

Published in:

Powder Diffraction, 2017, v. 32, n. 4, p. 271, doi. 10.1017/S0885715617001099

By:

Gündoğdu, Gülsüm;
Aytaç, Sevim Peri;
Müller, Melanie;
Tozkoparan, Birsen;
Kaynak, Filiz Betül

Publication type:

Article

Synthesis and biological evaluation of Combretastatin A-4 derivatives containing a 3'-O-substituted carbonic ether moiety as potential antitumor agents.

Published in:

Chemistry Central Journal, 2013, v. 7, n. 1, p. 1, doi. 10.1186/1752-153X-7-179

By:

Mingyi Ma;
Longru Sun;
Hongxiang Lou;
Mei Ji

Publication type:

Article

Mechanistic studies of DepR in regulating FK228 biosynthesis in Chromobacterium violaceum no. 968.

Published in:

PLoS ONE, 2018, v. 13, n. 3, p. 1, doi. 10.1371/journal.pone.0196173

By:

Qiao, Yongjian;
Tong, Tiantian;
Xue, Jiao;
Lin, Wenjing;
Deng, Zixin;
Cheng, Yi-Qiang;
Zhu, Dongqing

Publication type:

Article

Synthesis and Εvaluation of Αnticancer Αctivity in Cells of Novel Stoichiometric Pegylated Fullerene-Doxorubicin Conjugates.

Published in:

Pharmaceutical Research, 2015, v. 32, n. 5, p. 1676, doi. 10.1007/s11095-014-1566-1

By:

Magoulas, George;
Bantzi, Marina;
Messari, Danai;
Voulgari, Efstathia;
Gialeli, Chrisostomi;
Barbouri, Despoina;
Giannis, Athanassios;
Karamanos, Nikos;
Papaioannou, Dionissios;
Avgoustakis, Konstantinos

Publication type:

Article

A Concise and Practical Semisynthesis of Ecteinascidin 743 and (–)-Jorumycin.

Published in:

European Journal of Organic Chemistry, 2017, v. 2017, n. 5, p. 975, doi. 10.1002/ejoc.201601409

By:

Xu, Shanghu;
Wang, Guan;
Zhu, Jinjin;
Shen, Chuang;
Yang, Zhezhou;
Yu, Jun;
Li, Zhong;
Lin, Tanghuan;
Sun, Xun;
Zhang, Fuli

Publication type:

Article

Improved Strategy for the Synthesis of the Anticancer Agent Culicinin D.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 28, p. 6341, doi. 10.1002/ejoc.201500872

By:

Stach, Michaela;
Weidkamp, Andreas J.;
Yang, Sung‐Hyun;
Hung, Kuo‐yuan;
Furkert, Daniel P.;
Harris, Paul W. R.;
Smaill, Jeff B.;
Patterson, Adam V.;
Brimble, Margaret A.

Publication type:

Article

Divergent and Concise Syntheses of Spiroisoxazolines: First Total Synthesis of 11-Deoxyfistularin-3.

Published in:

European Journal of Organic Chemistry, 2015, v. 2015, n. 23, p. 5159, doi. 10.1002/ejoc.201500603

By:

Das, Prasanta;
Hamme II, Ashton T.

Publication type:

Article

Diversity-Oriented Synthesis of Calothrixins and Ellipticines.

Published in:

European Journal of Organic Chemistry, 2014, v. 2014, n. 31, p. 6953, doi. 10.1002/ejoc.201402837

By:

Dethe, Dattatraya H.;
Murhade, Ganesh M.

Publication type:

Article

A20 suppresses hepatocellular carcinoma proliferation and metastasis through inhibition of Twist1 expression.

Published in:

Molecular Cancer, 2015, v. 14, n. 1, p. 1, doi. 10.1186/s12943-015-0454-6

By:

Haiyang Chen;
Liang Hu;
Zaili Luo;
Jian Zhang;
Cunzhen Zhang;
Bijun Qiu;
Liwei Dong;
Yexiong Tan;
Jin Ding;
Shanhua Tang;
Feng Shen;
Zhong Li;
Hongyang Wang

Publication type:

Article

Anticancer drugs: A one-two punch for KRAS-driven cancer.

Published in:

Nature Reviews Drug Discovery, 2015, v. 14, n. 9, p. 600, doi. 10.1038/nrd4710

By:

Cully, Megan

Publication type:

Article

Preparation of Diaminedicarboxyplatinum (II) Functionalized Single-Wall Carbon Nanotube via Bingel Reaction as a Novel Cytotoxic Agent.

Published in:

Iranian Journal of Pharmaceutical Research, 2016, v. 15, n. 4, p. 753

By:

Irannejad, Saeed;
Amini, Mohsen;
Modanlookordi, Mona;
Shokrzadeh, Mohammad;
Irannejad, Hamid

Publication type:

Article

Design and Synthesis of Pyrrolo[2,1-a]Isoquinoline-Based Derivatives as New Cytotoxic Agents.

Published in:

Iranian Journal of Pharmaceutical Research, 2016, v. 15, n. 4, p. 743

By:

Kakhki, Samaneh;
Shahosseini, Soraya;
Zarghi, Afshin

Publication type:

Article

Assessment of the Cytotoxic Effect of a Series of 1,4-Dihydropyridine Derivatives Against Human Cancer Cells.

Published in:

Iranian Journal of Pharmaceutical Research, 2016, v. 15, n. 3, p. 413

By:

Razzaghi-Asla, Nima;
Miri, Ramin;
Firuzi, Omidreza

Publication type:

Article