Works by Zalubovskis, Raivis

Results: 40

Sulfonamide‐incorporated bis(α‐aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X‐ray crystallographic studies.

Published in:

Archiv der Pharmazie, 2024, v. 357, n. 7, p. 1, doi. 10.1002/ardp.202400038

By:

Sobati, Marjan;
Abdoli, Morteza;
Angeli, Andrea;
Bonardi, Alessandro;
Ferraroni, Marta;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N -((4-Sulfamoylphenyl)carbamothioyl) Amides.

Published in:

Molecules, 2023, v. 28, n. 10, p. 4020, doi. 10.3390/molecules28104020

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Paoletti, Niccolò;
Aspatwar, Ashok;
Parkkila, Seppo;
Gratteri, Paola;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Synthesis and Carbonic Anhydrase I, II, IX, and XII Inhibition Studies with a Series of Cyclic Sulfonyl Guanidines.

Published in:

ChemMedChem, 2024, v. 19, n. 19, p. 1, doi. 10.1002/cmdc.202400197

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Design, Synthesis, and Bioactivity Evaluations of 3‐Methylenechroman‐2‐one Derivatives as Thioredoxin Reductase (TrxR) Inhibitors.

Published in:

ChemMedChem, 2024, v. 19, n. 3, p. 1, doi. 10.1002/cmdc.202300504

By:

Nikitjuka, Anna;
Ozola, Melita;
Krims‐Davis, Kristaps;
Žalubovskis, Raivis

Publication type:

Article

Front Cover: Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX (ChemMedChem 22/2023).

Published in:

ChemMedChem, 2023, v. 18, n. 22, p. 1, doi. 10.1002/cmdc.202300639

By:

Leitans, Janis;
Kazaks, Andris;
Bogans, Janis;
Supuran, Claudiu T.;
Akopjana, Inara;
Ivanova, Jekaterina;
Zalubovskis, Raivis;
Tars, Kaspars

Publication type:

Article

Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX.

Published in:

ChemMedChem, 2023, v. 18, n. 22, p. 1, doi. 10.1002/cmdc.202300454

By:

Leitans, Janis;
Kazaks, Andris;
Bogans, Janis;
Supuran, Claudiu T.;
Akopjana, Inara;
Ivanova, Jekaterina;
Zalubovskis, Raivis;
Tars, Kaspars

Publication type:

Article

Corrigendum: Asparagusic Acid – A Unique Approach toward Effective Cellular Uptake of Therapeutics: Application, Biological Targets, and Chemical Properties.

Published in:

ChemMedChem, 2023, v. 18, n. 19, p. 1, doi. 10.1002/cmdc.202300425

By:

Ņikitjuka, Anna;
Žalubovskis, Raivis

Publication type:

Article

Asparagusic Acid – A Unique Approach toward Effective Cellular Uptake of Therapeutics: Application, Biological Targets, and Chemical Properties.

Published in:

ChemMedChem, 2023, v. 18, n. 17, p. 1, doi. 10.1002/cmdc.202300143

By:

Ņikitjuka, Anna;
Žalubovskis, Raivis

Publication type:

Article

Inhibition Studies on Carbonic Anhydrase Isoforms I, II, IX, and XII with a Series of Sulfaguanidines.

Published in:

ChemMedChem, 2023, v. 18, n. 6, p. 1, doi. 10.1002/cmdc.202200658

By:

Abdoli, Morteza;
De Luca, Viviana;
Capasso, Clemente;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Surface Functionalization of ITO for Dual-Mode Hypoxia-Associated Cancer Biomarker Detection.

Published in:

Biosensors (2079-6374), 2025, v. 15, n. 3, p. 186, doi. 10.3390/bios15030186

By:

Zutis, Edmunds;
Paidere, Gunita;
Ruska, Rihards;
Freimanis, Toms;
Cipa, Janis;
Zalubovskis, Raivis;
Elksne, Maira;
Tars, Kaspars;
Kazaks, Andris;
Leitans, Janis;
Sarakovskis, Anatolijs;
Anspoks, Andris

Publication type:

Article

Benzenesulfonamides Incorporating Hydantoin Moieties Effectively Inhibit Eukaryoticand Human Carbonic Anhydrases.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 22, p. 14115, doi. 10.3390/ijms232214115

By:

Abdoli, Morteza;
De Luca, Viviana;
Capasso, Clemente;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 10, p. 412, doi. 10.3390/metabo10100412

By:

Angeli, Andrea;
Carta, Fabrizio;
Nocentini, Alessio;
Winum, Jean-Yves;
Zalubovskis, Raivis;
Akdemir, Atilla;
Onnis, Valentina;
Eldehna, Wagdy M.;
Capasso, Clemente;
Simone, Giuseppina De;
Monti, Simona Maria;
Carradori, Simone;
Donald, William A.;
Dedhar, Shoukat;
Supuran, Claudiu T.

Publication type:

Article

Off-Stoichiometry Thiol-Ene Surface Functionalization: Example with Gold Nanoparticles.

Published in:

Materials (1996-1944), 2024, v. 17, n. 24, p. 6135, doi. 10.3390/ma17246135

By:

Ruska, Rihards;
Sarakovskis, Anatolijs;
Zutis, Edmunds;
Paidere, Gunita;
Vozny, Igor;
Cipa, Janis;
Gabrusenoks, Jevgenijs;
Freimanis, Toms;
Zalubovskis, Raivis;
Anspoks, Andris

Publication type:

Article

Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide–hydantoin hybrids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2335927

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Gratteri, Paola;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2249267

By:

Balašova, Anastasija;
Pustenko, Aleksandrs;
Nocentini, Alessio;
Vullo, Daniela;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

2-((1H-Benzo[d]imidazol-2-yl)amino)benzo[d]thiazole-6-sulphonamides: a class of carbonic anhydrase II and VII-selective inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2174981

By:

Abdoli, Morteza;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2170370

By:

Ivanova, Jekaterīna;
Abdoli, Morteza;
Nocentini, Alessio;
Žalubovskis, Raivis;
Supuran, Claudiu T.

Publication type:

Article

Novel thiazolone-benzenesulphonamide inhibitors of human and bacterial carbonic anhydrases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2163243

By:

Abdoli, Morteza;
De Luca, Viviana;
Capasso, Clemente;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Selected strategies to fight pathogenic bacteria.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2155816

By:

Plotniece, Aiva;
Sobolev, Arkadij;
Supuran, Claudiu T.;
Carta, Fabrizio;
Björkling, Fredrik;
Franzyk, Henrik;
Yli-Kauhaluoma, Jari;
Augustyns, Koen;
Cos, Paul;
De Vooght, Linda;
Govaerts, Matthias;
Aizawa, Juliana;
Tammela, Päivi;
Žalubovskis, Raivis

Publication type:

Article

Investigation of novel alkyl/benzyl (4-sulphamoylphenyl)carbamimidothioates as carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2152811

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 216, doi. 10.1080/14756366.2022.2143496

By:

Pustenko, Aleksandrs;
Balašova, Anastasija;
Nocentini, Alessio;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

1,2,3-Benzoxathiazine-2,2-dioxides – effective inhibitors of human carbonic anhydrases.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 225, doi. 10.1080/14756366.2022.2142787

By:

Ivanova, Jekaterina;
Abdoli, Morteza;
Nocentini, Alessio;
Žalubovskis, Raivis;
Supuran, Claudiu T.

Publication type:

Article

4-Cyanamidobenzenesulfonamide derivatives: a novel class of human and bacterial carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 156, doi. 10.1080/14756366.2022.2138367

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 561, doi. 10.1080/14756366.2021.1882453

By:

Nocentini, Alessio;
Angeli, Andrea;
Carta, Fabrizio;
Winum, Jean-Yves;
Zalubovskis, Raivis;
Carradori, Simone;
Capasso, Clemente;
Donald, William A.;
Supuran, Claudiu T.

Publication type:

Article

The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1011, doi. 10.1080/14756366.2020.1752201

By:

Pustenko, Aleksandrs;
Nocentini, Alessio;
Gratteri, Paola;
Bonardi, Alessandro;
Vozny, Igor;
Žalubovskis, Raivis;
Supuran, Claudiu T.

Publication type:

Article

Combining carbonic anhydrase and thioredoxin reductase inhibitory motifs within a single molecule dramatically increases its cytotoxicity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 665, doi. 10.1080/14756366.2020.1734800

By:

Krasavin, Mikhail;
Sharonova, Tatiana;
Sharoyko, Vladimir;
Zhukovsky, Daniil;
Kalinin, Stanislav;
Žalubovskis, Raivis;
Tennikova, Tatiana;
Supuran, Claudiu T.

Publication type:

Article

7-Acylamino-3H-1,2-benzoxathiepine 2,2-dioxides as new isoform-selective carbonic anhydrase IX and XII inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 650, doi. 10.1080/14756366.2020.1722658

By:

Pustenko, Aleksandrs;
Nocentini, Alessio;
Balašova, Anastasija;
Krasavin, Mikhail;
Žalubovskis, Raivis;
Supuran, Claudiu T.

Publication type:

Article

Sulfocoumarins as dual inhibitors of human carbonic anhydrase isoforms IX/XII and of human thioredoxin reductase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 506, doi. 10.1080/14756366.2020.1712596

By:

Krasavin, Mikhail;
Žalubovskis, Raivis;
Grandāne, Aiga;
Domračeva, Ilona;
Zhmurov, Petr;
Supuran, Claudiu T.

Publication type:

Article

Aryl derivatives of 3H-1,2-benzoxathiepine 2,2-dioxide as carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 245, doi. 10.1080/14756366.2019.1695795

By:

Pustenko, Aleksandrs;
Nocentini, Alessio;
Balašova, Anastasija;
Alafeefy, Ahmed;
Krasavin, Mikhail;
Žalubovskis, Raivis;
Supuran, Claudiu T.

Publication type:

Article

Design, synthesis, and biological evaluation of novel derivatives of dithiodiglycolic acid prepared via oxidative coupling of thiols.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 665, doi. 10.1080/14756366.2019.1575372

By:

Bakulina, Olga;
Bannykh, Anton;
Jovanović, Mirna;
Domračeva, Ilona;
Podolski-Renić, Ana;
Žalubovskis, Raivis;
Pešić, Milica;
Dar'in, Dmitry;
Krasavin, Mikhail

Publication type:

Article

Symmetric molecules with 1,4-triazole moieties as potent inhibitors of tumour-associated lactate dehydrogenase-A.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 147, doi. 10.1080/14756366.2017.1404593

By:

Altamimi, Abdul-Malek S.;
Alafeefy, Ahmed M.;
Balode, Agnese;
Vozny, Igor;
Pustenko, Aleksandrs;
El Shikh, Mohey Eldin;
Alasmary, Fatmah A. S.;
Abdel-Gawad, Sherif A.;
Žalubovskis, Raivis

Publication type:

Article

3 H -1,2-benzoxathiepine 2,2-dioxides: a new class of isoform-selective carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 767, doi. 10.1080/14756366.2017.1316720

By:

Pustenko, Aleksandrs;
Stepanovs, Dmitrijs;
Žalubovskis, Raivis;
Vullo, Daniela;
Kazaks, Andris;
Leitans, Janis;
Tars, Kaspars;
Supuran, Claudiu T.

Publication type:

Article

5-Membered cyclic hydroxamic acids as HDAC inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 2, p. 216, doi. 10.3109/14756366.2014.912214

By:

Mutule, Ilze;
Borovika, Diana;
Rozenberga, Elina;
Romanchikova, Nadezhda;
Zalubovskis, Raivis;
Shestakova, Irina;
Trapencieris, Peteris

Publication type:

Article

May 1,2-Dithiolane-4-carboxylic Acid and Its Derivatives Serve as a Specific Thioredoxin Reductase 1 Inhibitor?

Published in:

Molecules, 2023, v. 28, n. 18, p. 6647, doi. 10.3390/molecules28186647

By:

Nikitjuka, Anna;
Krims-Davis, Kristaps;
Kaņepe-Lapsa, Iveta;
Ozola, Melita;
Žalubovskis, Raivis

Publication type:

Article

Synthetic Methods toward Phosphacoumarins (microreview).

Published in:

2022

By:

Balašova, Anastasija;
Žalubovskis, Raivis

Publication type:

Editorial

Recent advances in sultone synthesis (microreview).

Published in:

Chemistry of Heterocyclic Compounds, 2017, v. 53, n. 12, p. 1283, doi. 10.1007/s10593-018-2208-z

By:

Pustenko, Aleksandrs;
Žalubovskis, Raivis

Publication type:

Article

Derivatives of 2-aziridinyl ketones and aziridinyl-2-carboxylates (microreview).

Published in:

Chemistry of Heterocyclic Compounds, 2016, v. 52, n. 8, p. 535, doi. 10.1007/s10593-016-1925-4

By:

Ivanova, Jekaterīna;
Žalubovskis, Raivis

Publication type:

Article

In a search for selective inhibitors of carbonic anhydrases: coumarin and its bioisosteres - synthesis and derivatization.

Published in:

Chemistry of Heterocyclic Compounds, 2015, v. 51, n. 7, p. 607, doi. 10.1007/s10593-015-1748-8

By:

Žalubovskis, Raivis

Publication type:

Article

Hydrophobic substituents of the phenylmethylsulfamide moiety can be used for the development of new selective carbonic anhydrase inhibitors.

Published in:

2014

By:

De Simone, Giuseppina;
Pizika, Ginta;
Monti, Simona Maria;
Di Fiore, Anna;
Ivanova, Jekaterina;
Vozny, Igor;
Trapencieris, Peteris;
Zalubovskis, Raivis;
Supuran, Claudiu T;
Alterio, Vincenzo

Publication type:

Journal Article

Tiocianāta un cilvēka ogļskābes anhidrāzes II mijiedarbības kvantu ķīmisks pētījums.

Published in:

Material Science & Applied Chemistry, 2013, n. 27, p. 22

By:

Fleišers, Mendels;
Žalubovskis, Raivis;
Šmidlers, Andulis;
Jansone, Daina

Publication type:

Article