Works by Volcho, Konstantin P.


Results: 55
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    Structure-Based Design, Synthesis, and Biological Evaluation of the Cage–Amide Derived Orthopox Virus Replication Inhibitors.

    Published in:
    Viruses (1999-4915), 2023, v. 15, n. 1, p. 29, doi. 10.3390/v15010029
    By:
    • Mozhaitsev, Evgenii S.;
    • Suslov, Evgeniy V.;
    • Rastrepaeva, Daria A.;
    • Yarovaya, Olga I.;
    • Borisevich, Sophia S.;
    • Khamitov, Edward M.;
    • Kolybalov, Dmitry S.;
    • Arkhipov, Sergey G.;
    • Bormotov, Nikolai I.;
    • Shishkina, Larisa N.;
    • Serova, Olga A.;
    • Brunilin, Roman V.;
    • Vernigora, Andrey A.;
    • Nawrozkij, Maxim B.;
    • Agafonov, Alexander P.;
    • Maksyutov, Rinat A.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    Key Enzymes of the Serotonergic System – Tryptophan Hydroxylase 2 and Monoamine Oxidase A – In the Brain of Rats Selectively Bred for a Reaction toward Humans: Effects of Benzopentathiepin TC-2153.

    Published in:
    Biochemistry (00062979), 2024, v. 89, n. 6, p. 1109, doi. 10.1134/S0006297924060105
    By:
    • Moskaliuk, Vitalii S.;
    • Kozhemyakina, Rimma V.;
    • Khomenko, Tatyana M.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Kulikov, Alexander V.;
    • Naumenko, Vladimir S.;
    • Kulikova, Elizabeth A.
    Publication type:
    Article
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    Biotransformation of (–)-Isopulegol by Rhodococcus rhodochrous.

    Published in:
    Pharmaceuticals (14248247), 2022, v. 15, n. 8, p. 964, doi. 10.3390/ph15080964
    By:
    • Ivshina, Irina B.;
    • Luchnikova, Natalia A.;
    • Maltseva, Polina Yu.;
    • Ilyina, Irina V.;
    • Volcho, Konstantin P.;
    • Gatilov, Yurii V.;
    • Korchagina, Dina V.;
    • Kostrikina, Nadezhda A.;
    • Sorokin, Vladimir V.;
    • Mulyukin, Andrey L.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    Rational Design of New Monoterpene-Containing Azoles and Their Antifungal Activity.

    Published in:
    Antibiotics (2079-6382), 2023, v. 12, n. 5, p. 818, doi. 10.3390/antibiotics12050818
    By:
    • Li-Zhulanov, Nikolai S.;
    • Zaikova, Nadezhda P.;
    • Sari, Suat;
    • Gülmez, Dolunay;
    • Sabuncuoğlu, Suna;
    • Ozadali-Sari, Keriman;
    • Arikan-Akdagli, Sevtap;
    • Nefedov, Andrey A.;
    • Rybalova, Tatyana V.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    MPTP-Treated Zebrafish Recapitulate 'Late-Stage' Parkinson's-like Cognitive Decline.

    Published in:
    Toxics, 2022, v. 10, n. 2, p. N.PAG, doi. 10.3390/toxics10020069
    By:
    • Bashirzade, Alim A. O.;
    • Cheresiz, Sergey V.;
    • Belova, Alisa S.;
    • Drobkov, Alexey V.;
    • Korotaeva, Anastasiia D.;
    • Azizi-Arani, Soheil;
    • Azimirad, Amirhossein;
    • Odle, Eric;
    • Gild, Emma-Yanina V.;
    • Ardashov, Oleg V.;
    • Volcho, Konstantin P.;
    • Bozhko, Dmitrii V.;
    • Myrov, Vladislav O.;
    • Kolchanova, Sofia M.;
    • Polovian, Aleksander I.;
    • Galumov, Georgii K.;
    • Salakhutdinov, Nariman F.;
    • Amstislavskaya, Tamara G.;
    • Kalueff, Allan V.
    Publication type:
    Article
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    Identification and Study of the Action Mechanism of Small Compound That Inhibits Replication of Respiratory Syncytial Virus.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 16, p. 12933, doi. 10.3390/ijms241612933
    By:
    • Shtro, Anna A.;
    • Klabukov, Artem M.;
    • Garshinina, Anzhelika V.;
    • Galochkina, Anastasia V.;
    • Nikolaeva, Yulia V.;
    • Khomenko, Tatyana M.;
    • Bobkov, Danila E.;
    • Lozhkov, Aleksey A.;
    • Sivak, Konstantin V.;
    • Yakovlev, Kirill S.;
    • Komissarov, Andrey B.;
    • Borisevich, Sophia S.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.
    Publication type:
    Article
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    New 5-Hydroxycoumarin-Based Tyrosyl-DNA Phosphodiesterase I Inhibitors Sensitize Tumor Cell Line to Topotecan.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 11, p. 9155, doi. 10.3390/ijms24119155
    By:
    • Khomenko, Tatyana M.;
    • Zakharenko, Alexandra L.;
    • Kornienko, Tatyana E.;
    • Chepanova, Arina A.;
    • Dyrkheeva, Nadezhda S.;
    • Artemova, Anastasia O.;
    • Korchagina, Dina V.;
    • Achara, Chigozie;
    • Curtis, Anthony;
    • Reynisson, Jóhannes;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    Novel TDP1 Inhibitors: Disubstituted Thiazolidine-2,4-Diones Containing Monoterpene Moieties.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 4, p. 3834, doi. 10.3390/ijms24043834
    By:
    • Ivankin, Dmitry I.;
    • Kornienko, Tatyana E.;
    • Mikhailova, Marina A.;
    • Dyrkheeva, Nadezhda S.;
    • Zakharenko, Alexandra L.;
    • Achara, Chigozie;
    • Reynisson, Jóhannes;
    • Golyshev, Victor M.;
    • Luzina, Olga A.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    The First Berberine-Based Inhibitors of Tyrosyl-DNA Phosphodiesterase 1 (Tdp1), an Important DNA Repair Enzyme.

    Published in:
    International Journal of Molecular Sciences, 2020, v. 21, n. 19, p. 7162, doi. 10.3390/ijms21197162
    By:
    • Gladkova, Elizaveta D.;
    • Nechepurenko, Ivan V.;
    • Bredikhin, Roman A.;
    • Chepanova, Arina A.;
    • Zakharenko, Alexandra L.;
    • Luzina, Olga A.;
    • Ilina, Ekaterina S.;
    • Dyrkheeva, Nadezhda S.;
    • Mamontova, Evgeniya M.;
    • Anarbaev, Rashid O.;
    • Reynisson, Jóhannes;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    Promising New Inhibitors of Tyrosyl-DNA Phosphodiesterase I (Tdp 1) Combining 4-Arylcoumarin and Monoterpenoid Moieties as Components of Complex Antitumor Therapy.

    Published in:
    International Journal of Molecular Sciences, 2020, v. 21, n. 1, p. 126, doi. 10.3390/ijms21010126
    By:
    • Khomenko, Tatyana M.;
    • Zakharenko, Alexandra L.;
    • Chepanova, Arina A.;
    • Ilina, Ekaterina S.;
    • Zakharova, Olga D.;
    • Kaledin, Vasily I.;
    • Nikolin, Valeriy P.;
    • Popova, Nelly A.;
    • Korchagina, Dina V.;
    • Reynisson, Jóhannes;
    • Chand, Raina;
    • Ayine-Tora, Daniel M.;
    • Patel, Jinal;
    • Leung, Ivanhoe K. H.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    The Development of Tyrosyl-DNA Phosphodiesterase 1 Inhibitors. Combination of Monoterpene and Adamantine Moieties via Amide or Thioamide Bridges.

    Published in:
    Applied Sciences (2076-3417), 2019, v. 9, n. 13, p. 2767, doi. 10.3390/app9132767
    By:
    • Chepanova, Arina A.;
    • Mozhaitsev, Evgenii S.;
    • Munkuev, Aldar A.;
    • Suslov, Evgeniy V.;
    • Korchagina, Dina V.;
    • Zakharova, Olga D.;
    • Zakharenko, Alexandra L.;
    • Patel, Jinal;
    • Ayine-Tora, Daniel M.;
    • Reynisson, Jóhannes;
    • Leung, Ivanhoe K. H.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    New Hybrid Compounds Combining Fragments of Usnic Acid and Monoterpenoids for Effective Tyrosyl-DNA Phosphodiesterase 1 Inhibition.

    Published in:
    Biomolecules (2218-273X), 2021, v. 11, n. 7, p. 973, doi. 10.3390/biom11070973
    By:
    • Dyrkheeva, Nadezhda S.;
    • Filimonov, Aleksandr S.;
    • Luzina, Olga A.;
    • Zakharenko, Alexandra L.;
    • Ilina, Ekaterina S.;
    • Malakhova, Anastasia A.;
    • Medvedev, Sergey P.;
    • Reynisson, Jóhannes;
    • Volcho, Konstantin P.;
    • Zakian, Suren M.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    Sulfide, Sulfoxide, and Sulfone Derivatives of Usnic Acid as Inhibitors of Human TDP1 and TDP2 Enzymes.

    Published in:
    Chemistry (2624-8549), 2024, v. 6, n. 6, p. 1658, doi. 10.3390/chemistry6060101
    By:
    • Filimonov, Aleksandr S.;
    • Mikhailova, Marina A.;
    • Dyrkheeva, Nadezhda S.;
    • Chernyshova, Irina A.;
    • Kornienko, Tatyana E.;
    • Naumenko, Konstantin A.;
    • Anarbaev, Rashid O.;
    • Nefedov, Andrey A.;
    • Achara, Chigozie;
    • Curtis, Anthony D. M.;
    • Luzina, Olga A.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.;
    • Reynisson, Jóhannes
    Publication type:
    Article
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    Novel Peptide–Drug Conjugates with Dual Anticancer Activity.

    Published in:
    International Journal of Molecular Sciences, 2024, v. 25, n. 22, p. 12411, doi. 10.3390/ijms252212411
    By:
    • O'Flaherty, Siobhán;
    • Luzina, Olga A.;
    • Dyrkheeva, Nadezhda S.;
    • Krier, Ysaline;
    • Leprince, Jérôme;
    • Zakharenko, Alexandra L.;
    • Pokrovsky, Mikhail A.;
    • Pokrovsky, Andrey G.;
    • Lavrik, Olga I.;
    • Salakhutdinov, Nariman F.;
    • Varbanov, Mihayl;
    • Devocelle, Marc;
    • Volcho, Konstantin P.
    Publication type:
    Article
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    Stereoselectivity Inversion by Water Addition in the −SO<sub>3</sub>H‐catalyzed Tandem Prins‐Ritter Reaction for Synthesis of 4‐amidotetrahydropyran Derivatives.

    Published in:
    ChemCatChem, 2020, v. 12, n. 9, p. 2605, doi. 10.1002/cctc.202000070
    By:
    • Sidorenko, Alexander Yu.;
    • Li‐Zhulanov, Nikolai S.;
    • Mäki‐Arvela, Päivi;
    • Sandberg, Thomas;
    • Kravtsova, Anna V.;
    • Peixoto, Andreia F.;
    • Freire, Cristina;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Agabekov, Vladimir E.;
    • Murzin, Dmitry Yu.
    Publication type:
    Article
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    A Newly Identified Monoterpenoid-Based Small Molecule Able to Support the Survival of Primary Cultured Dopamine Neurons and Alleviate MPTP-Induced Toxicity In Vivo.

    Published in:
    Molecules, 2022, v. 27, n. 23, p. 8286, doi. 10.3390/molecules27238286
    By:
    • Kotliarova, Anastasiia;
    • Podturkina, Alexandra V.;
    • Pavlova, Alla V.;
    • Gorina, Daria S.;
    • Lastovka, Anastasiya V.;
    • Ardashov, Oleg V.;
    • Rogachev, Artem D.;
    • Izyurov, Arseniy E.;
    • Arefieva, Alla B.;
    • Kulikov, Alexander V.;
    • Tolstikova, Tatyana G.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Sidorova, Yulia
    Publication type:
    Article
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    Adamantane-Monoterpenoid Conjugates Linked via Heterocyclic Linkers Enhance the Cytotoxic Effect of Topotecan.

    Published in:
    Molecules, 2022, v. 27, n. 11, p. 3374, doi. 10.3390/molecules27113374
    By:
    • Munkuev, Aldar A.;
    • Dyrkheeva, Nadezhda S.;
    • Kornienko, Tatyana E.;
    • Ilina, Ekaterina S.;
    • Ivankin, Dmitry I.;
    • Suslov, Evgeniy V.;
    • Korchagina, Dina V.;
    • Gatilov, Yuriy V.;
    • Zakharenko, Alexandra L.;
    • Malakhova, Anastasia A.;
    • Reynisson, Jóhannes;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.
    Publication type:
    Article
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    Design, Synthesis, and Biological Investigation of Novel Classes of 3-Carene-Derived Potent Inhibitors of TDP1.

    Published in:
    Molecules, 2020, v. 25, n. 15, p. 3496, doi. 10.3390/molecules25153496
    By:
    • Il'ina, Irina V.;
    • Dyrkheeva, Nadezhda S.;
    • Zakharenko, Alexandra L.;
    • Sidorenko, Alexander Yu.;
    • Li-Zhulanov, Nikolay S.;
    • Korchagina, Dina V.;
    • Chand, Raina;
    • Ayine-Tora, Daniel M.;
    • Chepanova, Arina A.;
    • Zakharova, Olga D.;
    • Ilina, Ekaterina S.;
    • Reynisson, Jóhannes;
    • Malakhova, Anastasia A.;
    • Medvedev, Sergey P.;
    • Zakian, Suren M.;
    • Volcho, Konstantin P.;
    • Salakhutdinov, Nariman F.;
    • Lavrik, Olga I.;
    • Sippl, Wolfgang;
    • Sousa, Maria Emília de
    Publication type:
    Article